5-Oxo-2,5-dihydro-1,2,4-triazines
    4.
    发明授权
    5-Oxo-2,5-dihydro-1,2,4-triazines 失效
    5-氧代-2,5-二氢-1,2,4-三嗪

    公开(公告)号:US4451283A

    公开(公告)日:1984-05-29

    申请号:US281776

    申请日:1981-07-09

    CPC分类号: C07D253/075 A01N43/707

    摘要: A herbicidal composition which comprises at least one of triazine compounds of the formula: ##STR1## wherein R.sup.1 is a C.sub.1 -C.sub.4 alkyl group or an amino group, R.sup.2 is a C.sub.1 -C.sub.4 alkoxy group, a C.sub.1 -C.sub.4 alkylthio group or a di(C.sub.1 -C.sub.4) alkylamino group and R.sup.3 is a cyclo(C.sub.3 -C.sub.7) alkyl group, a tertiary C.sub.4 -C.sub.5 alkyl group, an adamantyl group or a group of the formula: ##STR2## (in which R is a halogen atom, a C.sub.1 -C.sub.4 alkyl group, a C.sub.1 -C.sub.4 alkoxy group, a nitro group or a trihalomethyl group and n is an integer of 0 to 2) in a herbicidally effective amount and an inert carrier or diluent.

    摘要翻译: 一种除草组合物,其包含下式的三嗪化合物中的至少一种:其中R 1是C 1 -C 4烷基或氨基,R 2是C 1 -C 4烷氧基,C 1 -C 4烷硫基 或二(C1-C4)烷基氨基,R3是环(C3-C7)烷基,叔C4-C5烷基,金刚烷基或下式的基团:其中R是 卤素原子,C 1 -C 4烷基,C 1 -C 4烷氧基,硝基或三卤代甲基,n为0〜2的整数),除了有效量的惰性载体或稀释剂。

    Thiazolidin-4-one derivatives and acid addition salts thereof useful for
treating PAF mediated diseases
    6.
    发明授权
    Thiazolidin-4-one derivatives and acid addition salts thereof useful for treating PAF mediated diseases 失效
    噻唑烷-4-酮衍生物及其适用于治疗PAF介导性疾病的酸添加物

    公开(公告)号:US5106860A

    公开(公告)日:1992-04-21

    申请号:US624566

    申请日:1990-12-10

    IPC分类号: C07D417/04

    CPC分类号: C07D417/04

    摘要: Thiazolidin-4-one derivative represented by the following general formula (I) and acid addition salts thereof ##STR1## wherein; R.sup.1 and R.sup.2 are the same or different and denote each(i) a residue represented by the general formula--A--R.sup.4 wherein, A denotes a single bond, C.sub.1 -C.sub.8 alkylene, C.sub.2 -C.sub.8 alkenylene, or C.sub.2 -C.sub.8 alkynylene and R.sup.4 denotes hydrogen, C.sub.1 -C.sub.12 alkyl, C.sub.2 -C.sub.8 alkenyl, C.sub.3 -C.sub.8 cycloalkyl, or C.sub.1 -C.sub.6 haloalkyl,or(ii) a residue represented by the general formula ##STR2## wherein, B denotes a single bond or C.sub.1 -C.sub.6 alkylene, R.sup.5 denotes hydrogen, C.sub.1 -C.sub.6 alkyl, C.sub.2 -C.sub.8 alkenyl, C.sub.3 -C.sub.8 cycloalkyl, substituted silyl, or substituted or unsubstituted aryl, n and n' denote each an integer of 2 to 4, m denotes an integer of 1 to 3, and m' denotes an integer of 0 to 2;R.sup.3 denotes hydrogen, C.sub.1 -C.sub.2 alkyl, allyl, 2-propynyl,or(c) the general formula--F--R.sup.9 wherein, F denotes C.sub.2 -C.sub.6 alkylene and R.sup.9 denotes a nitrogen-containing heterocyclic aromatic residue or an amino group represented by the general formula ##STR3## (R.sup.10 denotes hydrogen, C.sub.2 -C.sub.4 alkyl or C.sub.1 -C.sub.4 alkanoyl and R.sup.11 denotes hydrogen or C.sub.1 -C.sub.4 alkyl or R.sup.10 in combination with R.sup.11 denotes a 5- to 7-membered cyclic amino group which optionally contains other hetero atoms.Having selective PAF-antagonistic activities, these compounds are very useful as preventive and curative agents for PAF-induced diseases, for example, various kinds of inflammation, allergic diseases, circulatory diseases, and gastro-intestinal diseases.

    Thiazolidin-4-one derivatives useful for treating diseases caused by
platelet activating factor
    7.
    发明授权
    Thiazolidin-4-one derivatives useful for treating diseases caused by platelet activating factor 失效
    可用于治疗血小板活化因子引起的疾病的噻唑烷-4-酮衍生物

    公开(公告)号:US4992455A

    公开(公告)日:1991-02-12

    申请号:US196058

    申请日:1988-05-19

    IPC分类号: C07D417/04

    CPC分类号: C07D417/04

    摘要: Thiazolidin-4-one derivative represented by the folowing general formula (I) and acid addition salts thereof ##STR1## wherein; R.sup.1 and R.sup.2 are the same or different and denote each(i) a residue represented by the general formula--A--R.sup.4 wherein, A denotes a single bond, C.sub.1 -C.sub.8 alkylene, C.sub.2 -C.sub.8 alkenylene, or C.sub.2 -C.sub.8 alkynylene and R.sup.4 denotes hydrogen, C.sub.1 -C.sub.12 alkyl, C.sub.2 -C.sub.8 alkenyl, C.sub.3 -C.sub.8 cycloalkyl, or C.sub.1 -C.sub.6 haloalkyl, or(ii) a residue represented by the general formula{(CH.sub.2).sub.n O}.sub.m {(CH.sub.2).sub.n' O}B--R.sup.5 wherein, B denotes a single bond or C.sub.1 -C.sub.6 alkylene, R.sup.5 denotes hydrogen, C.sub.1 -C.sub.6 alkyl, C.sub.2 -C.sub.8 alkenyl, C.sub.3 -C.sub.8 cycloalkyl, substituted silyl, or substituted or unsubstituted aryl, n and n' denote each an integer of 2 to 4, m denotes an integer of 1 to 3, and m' denotes an integer of 0 to 2; andR.sup.3 denotes hydrogen, C.sub.1 -C.sub.2 alkyl, allyl, 2-propynyl, or a residue represented by(a) the general formula--CH.sub.2).sub.l R.sup.6 wherein, R.sup.6 denotes halogen, an aryl group substituted or unsubstituted by one or more hydroxy or C.sub.1 -C.sub.4 alkoxy groups, or a residue represented by the general formula --D--R.sup.7 (D denotes oxygen or sulfur and R.sup.7 denotes hydrogen, C.sub.1 -C.sub.4 alkyl, or C.sub.1 -C.sub.4 alkanol) and l denotes an integer of 2 to 4,(b) the general formula--CH.sub.2).sub.k CO--E--R.sup.8 wherein, E denotes oxygen, sulfur, imino, or C.sub.1 -C.sub.4 alkylimino, R.sup.8 denotes hydrogen or C.sub.1 -C.sub.4 alkyl, or --(E--R.sup.8) denotes a 5- to 7-membered cyclic amino group which optionally contains other hetero atoms, and k denotes an integer of 1 to 3, or(c) the general formula--F--R.sup.9 wherein, F denotes C.sub.2 -C.sub.6 alkylene and R.sup.9 denotes a nitrogen-containing heterocyclic aromatic residue or an amino group represented by the general formula ##STR2## (R.sup.10 denotes hydrogen, C.sub.1 -C.sub.4 alkyl, or C.sub.1 -C.sub.4 alkyl or R.sup.10 in combination with R.sup.11 denotes a 5- to 7-membered cyclic amino group which optionally contains other hetero atoms), with the proviso that, when R.sup.1 is hydrogen and R.sup.2 is methyl, R.sup.3 denotes hydrogen, C.sub.1 -C.sub.2 alkyl, 2-propynyl, or a residue represented by(a) the general formula--CH.sub.2).sub.l R.sup.6 wherein, R.sup.6 denotes halogen, an aryl group substituted or unsubstituted by one or more hydroxy or C.sub.1 -C.sub.4 alkoxy groups, or a residue represented by the general formula --D--R.sup.7 (D denotes oxygen or sulfur and R.sup.7 denotes hydrogen, C.sub.1 -C.sub.4 alkyl, or C.sub.1 -C.sub.4 alkanoyl) and l denotes an integer of 2 to 4,(b) the general formula--CH.sub.2).sub.k CO--E--R.sup.8 wherein, E denotes oxygen, sulfur, imino, or C.sub.1 -C.sub.4 alkylimino, R.sup.8 denotes hydrogen or C.sub.1 -C.sub.4 alkyl, or --(E--R.sup.8) denotes a 5- to 7-membered cyclic amino group which optionally contains other hetero atoms, and k denotes an integer of 1 to 3, or(c) the general formula--F--R.sup.9 wherein, F denotes C.sub.2 -C.sub.6 alkylene and R.sup.9 denotes a nitrogen-containing heterocyclic aromatic residue or an amino group represented by the general formula ##STR3## (R.sup.10 denotes hydrogen, C.sub.2 -C.sub.4 alkyl or C.sub.1 -C.sub.4 alkanoyl and R.sup.11 denotes hydrogen or C.sub.1 -C.sub.4 alkyl or R.sup.10 in combination with R.sup.11 denotes a 5- to 7-membered cyclic amino group which optionally contains other hetero atoms.Having selective PAF-antagonistic activities, these compounds are very useful as preventive and curative agents for PAF-induced diseases, for example, various kinds of inflammation, allergic diseases, circulatory diseases, and gastro-intestinal diseases.

    Insecticidal and acaricidal 3,5-dioxo-2,3,4,5-triazine compounds
    8.
    发明授权
    Insecticidal and acaricidal 3,5-dioxo-2,3,4,5-triazine compounds 失效
    杀虫剂和杀螨剂3,5-二氧代-2,3,4,5-三嗪化合物

    公开(公告)号:US4327094A

    公开(公告)日:1982-04-27

    申请号:US225749

    申请日:1981-01-16

    摘要: A carboxylate of the formula, ##STR1## wherein R.sub.1 is an allyl or propargyl group, R.sub.2 is a group of ##STR2## in which R.sub.3 is a hydrogen atom or a methyl group, and when R.sub.3 is a hydrogen atom, R.sub.4 is a group of ##STR3## (in which R.sub.7 is a chlorine, bromine or fluorine atom, or a methyl, vinyl, methoxycarbonyl or methoxymethyl group, R.sub.8 is a hydrogen, chlorine, bromine or fluorine atom or a methyl group), and when R.sub.3 is a methyl group, R.sub.4 is a methyl group, R.sub.5 is an isopropyl or cyclopropyl group, R.sub.6 is an alkyl group having 1 to 3 carbon atoms or alkoxy group having 1 to 3 carbon atoms, or a chlorine, bromine or fluorine atom, n is 1 or 2, and --(R.sub.6).sub.n may include a 3,4-methylenedioxy group, and its use as an insecticide and/or acaricide.

    摘要翻译: 下式的羧酸酯,其中R 1是烯丙基或炔丙基,R 2是其中R 3是氢原子或甲基的“IMAGE”基团,当R 3是氢原子时,R 4是基团 的化合物(其中R 7为氯,溴或氟原子,或甲基,乙烯基,甲氧基羰基或甲氧基甲基,R 8为氢,氯,溴或氟原子或甲基),当R 3为 甲基,R4为甲基,R5为异丙基或环丙基,R6为碳原子数1〜3的烷基或碳原子数1〜3的烷氧基,或氯,溴或氟原子,n为1 或(2), - (R6)n可以包括3,4-亚甲二氧基,以及其作为杀虫剂和/或杀螨剂的用途。

    Process for producing pyridine compound
    9.
    发明授权
    Process for producing pyridine compound 有权
    制备吡啶化合物的方法

    公开(公告)号:US07157579B2

    公开(公告)日:2007-01-02

    申请号:US10486037

    申请日:2002-07-31

    IPC分类号: C07D401/12

    CPC分类号: C07D401/12

    摘要: The present invention provides a process for producing the pyridine compound [d]: [wherein R3 and R4 are as defined below], which has an excellent herbicidal activity, by making a pyridine compound [a]: [wherein R1 represents a C1–C6 alkoxy group, R3 represents a halogen atom, cyano group or nitro group, and R4 represents a hydrogen atom or halogen atom] react with an α-diazoester compound [f]: N2CHCOR1[f] [wherein R1 is defined above] in the presence of an acid.

    摘要翻译: 本发明提供一种制备吡啶化合物[d]的方法:其中R 3和R 4定义如下],其具有优异的除草活性,通过 制备吡啶化合物[a]:[其中R 1表示C 1 -C 6烷氧基,R 3表示卤素原子,氰基或硝基, SUP> 4 代表氢原子或卤素原子]与α-重氮化合物[f]反应:<?in-line-formula description =“In-line formula”end =“lead”?> N < &lt;&lt; 1&lt; 1&gt; [f] <?in-line-formula description =“In-line Formulas”end =“tail”?> [其中R 1, SUP>如上定义]在酸的存在下。

    Herbicidal composition
    10.
    发明授权
    Herbicidal composition 失效
    除草成分

    公开(公告)号:US5312798A

    公开(公告)日:1994-05-17

    申请号:US944084

    申请日:1992-09-11

    CPC分类号: A01N43/78 A01N47/18

    摘要: There is disclosed a herbicidal composition comprising as active ingredients a herbicidally effective amount of (a) an iminothiazoline compound of the formula: ##STR1## wherein R.sup.1 is halogen, halo(C.sub.1 -C.sub.2)alkyl, halo(C.sub.1 -C.sub.2)alkoxy or halo(C.sub.1 -C.sub.2)alkylthio; R.sup.2 is C.sub.1 -c.sub.2 alkyl, chroline, bromine or iodine; R.sup.3 is C.sub.1 -C.sub.6 alkyl, C.sub.3 -C.sub.6 cycloalkyl, C.sub.3 -C.sub.6 cycloalkoxy or C.sub.1 -C.sub.6 alkoxy, all of which are optionally substituted with at least one substituent selected from halogen, C.sub.1 -C.sub.2 alkyl and C.sub.1 -C.sub.2 alkoxy; R.sup.4 is hydrogen or halogen; and (b) at least one of herbicidal triazine compounds, herbicidal uracil compounds, herbicidal urea compounds, herbicidal dinitro aniline compounds, norflurazon, dimethazon, imazaquin and imazethapyr. Also disclosed is a method for controlling undesired weeds by use of the herbicidal composition.

    摘要翻译: 公开了除草组合物,其包含除草有效量的(a)下式的亚氨基噻唑啉化合物:其中R 1是卤素,卤代(C 1 -C 2)烷基,卤代(C 1 -C 2)烷氧基或卤素 (C1-C2)烷硫基; R2是C1-C2烷基,氯原子,溴或碘; R3是C1-C6烷基,C3-C6环烷基,C3-C6环烷氧基或C1-C6烷氧基,它们全部被至少一个选自卤素,C 1 -C 2烷基和C 1 -C 2烷氧基的取代基取代; R4是氢或卤素; 和(b)至少一种除草三嗪化合物,除草尿嘧啶化合物,除草脲化合物,除草二硝基苯胺化合物,诺氟拉津,二甲基噻唑,咪唑啉酮和咪草烟。 还公开了通过使用除草组合物来控制不需要的杂草的方法。