Oligosaccharide derivatives and process for producing the same
    2.
    发明授权
    Oligosaccharide derivatives and process for producing the same 失效
    寡糖衍生物及其制备方法

    公开(公告)号:US06518249B1

    公开(公告)日:2003-02-11

    申请号:US09485978

    申请日:2000-02-18

    IPC分类号: A61K3170

    CPC分类号: C07H15/04

    摘要: An oligosaccharide derivative, at higher homogeneity than fucose polysaccharide and rhamnose polysaccharide and with greater antiulcer effects, which is represented by the following general formula: Y—OCH(CH2NHR)2 wherein, Y represents an oligofucose or oligorhamnose at a polymerization number of 2 to 20, where the hydroxyl groups may or may not be partially modified in the form of sulfate ester, and R represents phenyl group, a higher alkylphenyl group, a higher alkyl group or —(CH2)n—NHX wherein n is an integer of 1 to 10 and X represents a higher alkanoyl group or an alkylamino group.

    摘要翻译: 一种低聚糖衍生物,其比岩藻糖多糖和鼠李糖多糖具有更高的均一性,并且具有较大的抗溃疡作用,其由以下通式表示:其中Y表示聚合数为2至20的寡聚核糖或寡鼠李糖,其中羟基可以 或可以不以硫酸酯的形式部分修饰,R代表苯基,高级烷基苯基,高级烷基或 - (CH2)n-NHX,其中n为1至10的整数,X表示较高的 烷酰基或烷基氨基。

    Pyrimidine derivatives
    6.
    发明授权
    Pyrimidine derivatives 失效
    嘧啶衍生物

    公开(公告)号:US5455355A

    公开(公告)日:1995-10-03

    申请号:US186165

    申请日:1994-01-25

    摘要: A pyrimidine herbicide derivative having the formula, ##STR1## wherein A is C.sub.3 -C.sub.6 oxacycloalkyl, C.sub.3 -C.sub.6 oxacycloalkyl substituted with at least one member selected from the group consisting of C.sub.1 -C.sub.6 alkyl and halogen, C.sub.2 -C.sub.6 oxacycloalkyl C.sub.1 -C.sub.6 alkyl, C.sub.2 -C.sub.6 oxacycloalkyl C.sub.1 -C.sub.6 alkyl substituted with at least one member selected from the group consisting of C.sub.1 -C.sub.6 alkyl and halogen, C.sub.3 -C.sub.5 dioxacycloalykyl, C.sub.3 -C.sub.5 dioxacycloalkyl substituted with at least one member selected from the group consisting of C.sub.1 -C.sub.6 alkyl and halogen, C.sub.3 -C.sub.5 dioxacycloalkyl C.sub.1 -C.sub.6 alkyl or C.sub.3 -C.sub.5 dioxacycloalkyl C.sub.1 -C.sub.6 alkyl substituted with at least one member selected from the group consisting of C.sub.1 -C.sub.6 alkyl and halogen;each of R.sup.1 and R.sup.2, which may be the same or different, is C.sub.1 -C.sub.6 alkyl, C.sub.1 -C.sub.6 alkoxy, halo C.sub.1 -C.sub.6 alkoxy or halogen;X is oxygen or sulfur;Z is nitrogen or CY.sup.4 ;and Y.sup.1-4 are described in the specification.

    摘要翻译: 具有下式的嘧啶除草剂衍生物,其中A是C3-C6氧杂环烷基,被至少一种选自C1-C6烷基和卤素的C3-C6氧杂环烷基,C2-C6氧杂环烷基C1 -C 1-6烷基,被选自C 1 -C 6烷基和卤素中的至少一种取代的C 2 -C 6环烷基C 1 -C 6烷基,C 3 -C 5二氧环烷基,被至少一种选自下列基团的C 3 -C 5二氧杂环烷基 由C 1 -C 6烷基和卤素组成,C 3 -C 5二氧杂环烷基C 1 -C 6烷基或被选自C 1 -C 6烷基和卤素中的至少一种取代的C 3 -C 5二氧杂环烷基C 1 -C 6烷基; 可以相同或不同的R 1和R 2各自为C 1 -C 6烷基,C 1 -C 6烷氧基,卤代C 1 -C 6烷氧基或卤素; X是氧或硫; Z是氮或CY4; 和Y1-4在说明书中描述。

    Herbicidal composition
    7.
    发明授权
    Herbicidal composition 失效
    除草成分

    公开(公告)号:US5312798A

    公开(公告)日:1994-05-17

    申请号:US944084

    申请日:1992-09-11

    CPC分类号: A01N43/78 A01N47/18

    摘要: There is disclosed a herbicidal composition comprising as active ingredients a herbicidally effective amount of (a) an iminothiazoline compound of the formula: ##STR1## wherein R.sup.1 is halogen, halo(C.sub.1 -C.sub.2)alkyl, halo(C.sub.1 -C.sub.2)alkoxy or halo(C.sub.1 -C.sub.2)alkylthio; R.sup.2 is C.sub.1 -c.sub.2 alkyl, chroline, bromine or iodine; R.sup.3 is C.sub.1 -C.sub.6 alkyl, C.sub.3 -C.sub.6 cycloalkyl, C.sub.3 -C.sub.6 cycloalkoxy or C.sub.1 -C.sub.6 alkoxy, all of which are optionally substituted with at least one substituent selected from halogen, C.sub.1 -C.sub.2 alkyl and C.sub.1 -C.sub.2 alkoxy; R.sup.4 is hydrogen or halogen; and (b) at least one of herbicidal triazine compounds, herbicidal uracil compounds, herbicidal urea compounds, herbicidal dinitro aniline compounds, norflurazon, dimethazon, imazaquin and imazethapyr. Also disclosed is a method for controlling undesired weeds by use of the herbicidal composition.

    摘要翻译: 公开了除草组合物,其包含除草有效量的(a)下式的亚氨基噻唑啉化合物:其中R 1是卤素,卤代(C 1 -C 2)烷基,卤代(C 1 -C 2)烷氧基或卤素 (C1-C2)烷硫基; R2是C1-C2烷基,氯原子,溴或碘; R3是C1-C6烷基,C3-C6环烷基,C3-C6环烷氧基或C1-C6烷氧基,它们全部被至少一个选自卤素,C 1 -C 2烷基和C 1 -C 2烷氧基的取代基取代; R4是氢或卤素; 和(b)至少一种除草三嗪化合物,除草尿嘧啶化合物,除草脲化合物,除草二硝基苯胺化合物,诺氟拉津,二甲基噻唑,咪唑啉酮和咪草烟。 还公开了通过使用除草组合物来控制不需要的杂草的方法。

    Iminothiazolines, their production and use as herbicides
    9.
    发明授权
    Iminothiazolines, their production and use as herbicides 失效
    异噻唑啉,其生产和用作除草剂

    公开(公告)号:US5292715A

    公开(公告)日:1994-03-08

    申请号:US936516

    申请日:1992-08-28

    摘要: There is disclosed an iminothiazoline compound of the formula: ##STR1## wherein R.sup.1 is halogen, halo(lower)alkyl, halo(lower)alkoxy or halo(lower)alkylthio; R.sup.2 is methyl, ethyl, chlorine, bromine or iodine; R.sup.3 is lower alkyl, lower cycloalkyl, lower alkoxy, lower cycloalkoxy, lower alkylamino, phenylamino or phenyl, all of which are optionally substituted with at least one substituent selected from halogen, lower alkyl, lower alkoxy, halo(lower)alkyl, lower cycloalkyl and lower cycloalkoxy; and R.sup.4 is hydrogen or halogen. Also disclosed are a process for producing this compound, a herbicidal composition comprising this compound as an active ingredient, and a method for controlling undesired weeds by use of this compound as a herbicide.

    摘要翻译: 公开了下式的亚氨基噻唑啉化合物:(*化学结构*)(I)其中R1是卤素,卤代(低级)烷基,卤代(低级)烷氧基或卤代(低级)烷硫基; R2是甲基,乙基,氯,溴或碘; R3是低级烷基,低级环烷基,低级烷氧基,低级环烷氧基,低级烷基氨基,苯基氨基或苯基,它们全部被至少一个选自卤素,低级烷基,低级烷氧基,卤代(低级)烷基,低级环烷基 和低级环烷氧基; R4是氢或卤素。 还公开了制备该化合物的方法,包含该化合物作为活性成分的除草组合物,以及通过使用该化合物作为除草剂来控制不需要的杂草的方法。

    Herbicidal composition
comprising2-[7-fluoro-3,4-dihydro-3-oxo-4-(2-pyropynyl)-2H-1,4-benzoxazi
n-6-yl]-4,5,6,7-tetrahydro-1H-isoindole-1,3(2H)-dione and either
glufosinate or bialaphos
    10.
    发明授权
    Herbicidal composition comprising2-[7-fluoro-3,4-dihydro-3-oxo-4-(2-pyropynyl)-2H-1,4-benzoxazi n-6-yl]-4,5,6,7-tetrahydro-1H-isoindole-1,3(2H)-dione and either glufosinate or bialaphos 失效
    除草组合物包含2- [7-氟-3,4-二氢-3-氧代-4-(2-吡啶基)-2H-1,4-苯并恶嗪-6-基] -4,5,6,7-四氢 - 1H-异吲哚-1,3(2H) - 二酮和草铵膦或双丙二酸

    公开(公告)号:US5173103A

    公开(公告)日:1992-12-22

    申请号:US841277

    申请日:1992-02-26

    IPC分类号: A01N57/20

    CPC分类号: A01N57/20

    摘要: A herbicidal composition which comprises a herbicidally effective amount of the combinations of (a) 2-[7-fluoro-3,4-dihydro-3-oxo-4-(2-propynyl)-2H-1,4-benzoxazin-6-yl]-4,5,6,7-tetrahydro-1H-isoindole-1,3(2H)-dione and (b) at least one of (2-amino-4-methylphosphinobutyryl)alanylalanine and its salt (bialaphos) and DL-homoalanin-4-yl(methyl)phosphinic acid and its salt (glufosinate), and an inert carrier or diluent. The composition exerts synergistic herbicidal activity.

    摘要翻译: 一种除草组合物,其包含除草有效量的(a)2- [7-氟-3,4-二氢-3-氧代-4-(2-丙炔基)-2H-1,4-苯并恶嗪-6 - 基] -4,5,6,7-四氢-1H-异吲哚-1,3(2H) - 二酮和(b)至少一种(2-氨基-4-甲基膦酰基丁酰基)丙氨酰丙氨酸及其盐(双亚硫磷) 和DL-高丙氨酸-4-基(甲基)次膦酸及其盐(草铵膦)和惰性载体或稀释剂。 该组合物具有协同的除草活性。