摘要:
Compounds having the formula ##STR1## wherein R is lower alkoxy or alkyl having from 1 to 6 carbon atoms, and preferably 1 to 3 carbon atoms and most preferably 1 carbon atom, R.sub.1 is lower alkoxy having from 1 to 6 carbon atoms, preferably 2 to 4 carbon atoms, and most preferably 2 carbon atoms, have shown utility as insecticides and miticides.
摘要:
Compounds of formula ##STR1## wherein Y, R.sub.1, R.sub.2, Het, X and n have the meanings reported in the description, processes for their preparation and pharmaceutical compositions which contain them as active ingredients are described. The compounds of formula I are useful in the treatment of cardiovascular diseases.
摘要:
Intramolecular nucleophilic displacement compound or a precursor thereof wherefrom during photographic processing a photographically useful group can be split off, said intramolecular nucleophilic displacement compound or precursor thereof corresponding to the following general structure (I): ##STR1## wherein Nu.sup.1 represents a nucelophilic group e.g. HO, H.sub.2 N or Hs, or a precursor of such nucleophilic group e.g. an oxidized nucleophilic group e.g. O.dbd. or HN.dbd., or RO wherein R is an alkyl, an acyl, an aryl or a trialkylsilanyl group, which groups may be substituted, the said nucleophilic group or precursor thereof being located in adjacent position to C(R.sup.1 R.sup.2) so as to make possible elimination of PUG through a nucleophilic displacement reaction;Ar represents an aryl group or a heteroaryl group (e.g. pyridine), which groups may be substituted by one or more mono-atomic or poly-atomic groups, e.g. alkyl groups, nitro groups, cyano groups, carboxy groups, or by sibstituents which, when in adjacent positions on the ring, together form a ring fused with the (hetero)aryl group, e.g. a benzene ring, a cyclohexane ring, a heteroannulated ring; Ar may comprise as substituent e.g. another nucleophilic group Nu.sup.2 (same as or different from Nu.sup.1);each of R.sup.1 and R.sup.2 (same or different) represents hydrogen or an alkyl, an aryl or an aralkyl group which groups each may be substituted;R.sup.3 represents an alkyl, an aralkyl, an alkyloxy, an aryloxy, an alkylthio, an arylthio, an amino group which groups each may be substituted, an oxy (O.sup.-) or a hydroxy group;PUG is a group containing a hetero atom (selected from among N, S and O) through which it is attached to the phosphor atom and producing a photographically useful activity after cleavage of the bond between the hetero atom and the phosphor atom.
摘要:
The present invention relates to a class of 5-haloalkyl-3-hydroxy-1-(C.sub.1-2 alkyl)pyrazoles useful as precursors for an active class of phenoxypyrazole herbicides.
摘要:
Compounds of the formula ##STR1## wherein Het is a heterocycle containing 2 to 3 nitrogen atoms;R is hydrogen, lower alkyl, alkoxy of 1 to 3 carbon atoms or halogen;Y is --SO.sub.3 H or ##STR2## R" is alkyl of 1 to 3 carbon atoms; and R' is straight or branched alkyl which may contain a heteroatom such as sulfur, oxygen or nitrogen; straight or branched alkenyl; cycloalkyl; alkyl-cycloalkyl; aryl; or aralkyl optionally substituted by lower alkyl, alkoxy of 1 to 3 carbon atoms or halogen; tautomers thereof, and non-toxic, pharmacologically acceptable acid addition salts thereof. The compounds as well as their salts are useful as anti-ulcerogenics and gastric acid secretion inhibitors.
摘要:
P-Xylylenediphosphonic acid groups connected through the aromatic ring to a variety of chromophores provide a class of novel dyes of the general formula ##STR1## wherein "Dye" represents the chromophore. These dyes may be covalently bonded to fibers and other substrates containing hydroxyl, amino, or thiol groups to form phosphonic acid esters or amides by reaction in the presence of a carbodiimide such as cyanamide or dicyandiamide.