Benzeneazo polynuclear aromatic or heteroaromatic amidine compounds
containing amidine substituents
    3.
    发明授权
    Benzeneazo polynuclear aromatic or heteroaromatic amidine compounds containing amidine substituents 失效
    含有脒取代基的苯并偶氮多核芳香族或杂芳族脒化合物

    公开(公告)号:US4619994A

    公开(公告)日:1986-10-28

    申请号:US759493

    申请日:1985-07-25

    摘要: A compound, useful as an anti-cancer drug or agent, having the formulaR.sub.1 --X--R.sub.2where X represents a polynuclear aromatic or heteroaromatic hydrocarbon having between two and four fused rings which may be substituted by hydroxyl, amino, alkylamino, alkoxy or halogeno, R.sub.1 represents: ##STR1## where y represents one member selected from: ##STR2## or alkylated derivatives thereof, and R.sub.2 represents hydrogen or R.sub.1, an acid addition salt of said compound, a nitrogen oxide derivative of said compound in the case where it contains a ring nitrogen atom or atoms, and a quaternary salt of said compound in the case where it contains a ring nitrogen atom or atoms.

    摘要翻译: 用作抗癌药物或药剂的化合物,其具有式R1-X-R2,其中X表示具有2-4个可被羟基,氨基,烷基氨基,烷氧基或烷氧基取代的稠合环的多核芳族或杂芳族烃 卤素,R1表示:其中y表示选自以下的一种:其中R 1表示氢或R 1,所述化合物的酸加成盐,所述化合物的氮氧化物衍生物, 它含有环氮原子或原子,并且在含有环氮原子或原子的情况下,所述化合物的季盐。

    Preparation of aromatic azoamines by
diazotization/coupling/rearrangement of aromatic amines
    4.
    发明授权
    Preparation of aromatic azoamines by diazotization/coupling/rearrangement of aromatic amines 失效
    通过芳香胺的重氮化/偶联/重排制备芳族偶氮胺

    公开(公告)号:US4275003A

    公开(公告)日:1981-06-23

    申请号:US876504

    申请日:1978-02-09

    CPC分类号: C09B37/00

    摘要: Aromatic azoamines are prepared by diazotizing an aromatic amine, coupling the diazonium salt with the aromatic amine, and rearranging the resulting aromatic diazoamine. The several reactions are effected in single stage by introducing vaporous nitrogen oxides to a reaction medium essentially consisting of the aromatic amine [.alpha.], a salt of the aromatic amine [.beta.], and water [.gamma.], with the percentage weight relationship existing among the components .alpha., .beta. and .gamma. being such that:10

    摘要翻译: 芳族偶氮胺通过将芳族胺重氮化,将重氮盐与芳族胺偶联并重排所得的芳族重氮胺来​​制备。 通过将气态氮氧化物引入到基本上由芳香族胺α,芳香族胺β的盐和水γ的反应介质中,在单个阶段中实现了几个反应,其中百分比重量关系存在于 组分α,β和γ使得:10 <70 13 <5 5

    Process for preparing diazonium salts of 3-amino-pyrazole
    5.
    发明授权
    Process for preparing diazonium salts of 3-amino-pyrazole 失效
    制备3-氨基 - 吡唑的重氮盐的方法

    公开(公告)号:US4268436A

    公开(公告)日:1981-05-19

    申请号:US41550

    申请日:1979-05-23

    CPC分类号: C07D231/38

    摘要: 3-Diazonium salts of pyrazole, useful as intermediates in the preparation of azo dyes are obtained by an oxidative diazotization of 3-amino-pyrazolines with nitrous acid or with nitrosyl-sulphuric acid. The 3-diazonium salts of pyrazole have the following structure: ##STR1## wherein: X is a radical --CO-- or --COO--,n is 0 or 1,R is hydrogen (in such case n is always 0), a normal or ramified alkyl C.sub.1 --C.sub.4, an aromatic or heterocyclic, optionally substituted, radical, in particular a phenyl radical having the structure: ##STR2## in which m may vary from 0 to 3 and substituents R.sub.3, either like or unlike one another for m>1, are alkyls C.sub.1 --C.sub.4 with linear or ramified chain, halogens, a cyano, nitro, sulphonic or carboxylic group, carboxyesters having a linear or ramified chain C.sub.1 --C.sub.4, alkoxyls having a linear or ramified chain C.sub.1 --C.sub.4, trifluoro-methyl groups, acylamino groups having a linear or ramified aliphatic chain C.sub.1 --C.sub.4, or sulphonamide groups of the type ##STR3## wherein substituents R.sub.4 and R.sub.5, like or unlike each other, are hydrogen, or linear or ramified aliphatic chains C.sub.1 --C.sub.4, andR.sub.1 and R.sub.2, either like or unlike each other, are hydrogen, linear or ramified aliphatic chains C.sub.1 --C.sub.4, or non-substituted or substituted benzene residues.

    摘要翻译: 通过用亚硝酸或亚硝酰基硫酸对3-氨基 - 吡唑啉进行氧化重氮化可以得到用作制备偶氮染料中的中间体的吡唑的3-重氮鎓盐。 吡唑的3-重氮盐具有以下结构:其中:X是-CO-或-COO-基团,n是0或1,R是氢(在这种情况下,n总是为0) ,正烷基或分支的烷基C1-C4,芳族或杂环的,任选取代的基团,特别是具有以下结构的苯基:其中m可以在0至3之间变化,并且取代基R3与或不同于一个 对于m> 1,另一个是具有直链或支链,卤素,氰基,硝基,磺酸或羧基的烷基C1-C4,具有直链或支链C 1 -C 4的烷基酯,具有直链或支链C1-C4 三氟甲基,具有线性或分枝的脂族链C1-C4的酰基氨基或类型“IMAGE”的磺酰胺基团,其中取代基R 4和R 5彼此相似或不同,为氢,或直链或分枝的脂族链C1 -C4和R1和R2彼此相似或不同,是氢,直链或分枝的脂族链C1-C4或n 取代或取代的苯残基。

    Drop-in type shifter with displaced shift stick
    10.
    发明授权
    Drop-in type shifter with displaced shift stick 失效
    带移位移位棒的插入式移位器

    公开(公告)号:US4515032A

    公开(公告)日:1985-05-07

    申请号:US429516

    申请日:1982-09-30

    申请人: Bruce E. Olmsted

    发明人: Bruce E. Olmsted

    摘要: A drop-in shifter for a manual transmission includes an elongated base, a shift stick mounted on the base for multi-axis movement and a depending gear actuating lever. An elongated rail is supported on the base by spaced bearings for rotational and lateral shifting movement. The shift stick has a lower end pivoted to the rail. The gear actuating lever is fixed to the rail at a point spaced from the shift stick. The lever extends through the base which is bolted to the transmission. Multi-axis movement of the shift stick is translated into multi-axis movement of the gear actuating lever through the bearings and rail.

    摘要翻译: 用于手动变速器的换档装置包括细长基座,安装在用于多轴运动的基座上的换档杆和从动齿轮致动杆。 细长轨道通过间隔开的轴承支撑在基座上,用于旋转和横向移动运动。 换档杆具有枢转到轨道的下端。 齿轮驱动杆在与换档杆间隔开的位置固定在轨道上。 杠杆延伸通过螺栓连接到变速器的基座。 换档杆的多轴运动通过轴承和导轨转换成齿轮传动杆的多轴运动。