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公开(公告)号：WO2004096235A8
公开(公告)日：2005-02-24
申请号：PCT/US2004013121
申请日：2004-04-26
Applicant: GILEAD SCIENCES INC , BOOJAMARA CONSTANTINE G , CANNIZZARO CARINA E , CHEN JAMES M , CHEN XIAOWU , CHO AESOP , CHONG LEE S , FARDIS MARIA , HUANG ALAN X , KIM CHOUNG X , KIRSCHBERG THORSTEN A , KRAWCZYK STEVEN , LEE CHRISTOPHER P , LIN KUEI-YING , MACKMAN RICHARD L , MARKEVITCH DAVID Y , NELSON PETER H , OARE DAVID , PRASAD VIDYA K , PYUN HYUNG-JUNG , RAY ADRIAN S , SWAMINATHAN SUNDARAMOORTHI , WATKINS WILL , ZHANG LIJUN
Inventor： BOOJAMARA CONSTANTINE G , CANNIZZARO CARINA E , CHEN JAMES M , CHEN XIAOWU , CHO AESOP , CHONG LEE S , FARDIS MARIA , HUANG ALAN X , KIM CHOUNG X , KIRSCHBERG THORSTEN A , KRAWCZYK STEVEN , LEE CHRISTOPHER P , LIN KUEI-YING , MACKMAN RICHARD L , MARKEVITCH DAVID Y , NELSON PETER H , OARE DAVID , PRASAD VIDYA K , PYUN HYUNG-JUNG , RAY ADRIAN S , SWAMINATHAN SUNDARAMOORTHI , WATKINS WILL , ZHANG LIJUN
IPC: A61K20060101 , A61K31/662 , C07D205/04 , C07D211/58 , C07D409/06 , C07D409/14 , C07D413/14 , C07D475/00 , C07D487/04 , C07F9/40 , C07F9/572 , C07F9/58 , C07F9/60 , C07F9/6503 , C07F9/6509 , C07F9/653 , C07F9/6539 , C07F9/655 , C07F9/6553 , C07F9/6561
CPC classification number: A61K31/662 , A61K47/548 , C07D205/04 , C07D211/58 , C07D239/94 , C07D409/06 , C07D409/14 , C07D413/14 , C07D475/00 , C07D487/04 , C07F9/4075 , C07F9/5728 , C07F9/582 , C07F9/588 , C07F9/60 , C07F9/65037 , C07F9/650941 , C07F9/653 , C07F9/6539 , C07F9/65515 , C07F9/655354 , C07F9/6561
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公开(公告)号：WO2005002626A3
公开(公告)日：2005-01-13
申请号：PCT/US2004/013283
申请日：2004-04-26
Applicant: GILEAD SCIENCES, INC. , BOOJAMRA, Constantine, G. , CANNIZZARO, Carina, E. , CHEN, James, M. , CHEN, Xiaowu , CHO, Aesop , CHONG, Lee, S. , DESAI, Manoj , FARDIS, Maria , GIBBS, Craig, S. , HIRSCHMANN, Ralph, F. , HUANG, Alan, X. , JIN, Haolun , KIM, Choung, U. , KIRSCHBERG, Thorsten, A. , KRAWCZYK, Steven , LEE, Christopher, P. , LEE, William, A. , LIN, Kuei-Ying , MACKMAN, Richard, L. , MARKEVITCH, David, Y. , NELSON, Peter, H. , OARE, David, A. , PRASAD, Vidya, K. , PYUN, Hyung-Jung , RAY, Adrian, S. , SHERLOCK, Rosemarie , SWAMINATHAN, Sundaramoorthi , WATKINS, William, J. , ZHANG, Jennifer, R. , ZHANG, Lijun
Inventor： BOOJAMRA, Constantine, G. , CANNIZZARO, Carina, E. , CHEN, James, M. , CHEN, Xiaowu , CHO, Aesop , CHONG, Lee, S. , DESAI, Manoj , FARDIS, Maria , GIBBS, Craig, S. , HIRSCHMANN, Ralph, F. , HUANG, Alan, X. , JIN, Haolun , KIM, Choung, U. , KIRSCHBERG, Thorsten, A. , KRAWCZYK, Steven , LEE, Christopher, P. , LEE, William, A. , LIN, Kuei-Ying , MACKMAN, Richard, L. , MARKEVITCH, David, Y. , NELSON, Peter, H. , OARE, David, A. , PRASAD, Vidya, K. , PYUN, Hyung-Jung , RAY, Adrian, S. , SHERLOCK, Rosemarie , SWAMINATHAN, Sundaramoorthi , WATKINS, William, J. , ZHANG, Jennifer, R. , ZHANG, Lijun
IPC: A61K47/48
Abstract: The invention is related to phosphorus substituted therapeutic agents, compositions containing such phosphorus substituted agents, and therapeutic methods that include the administration of such phosphorus substituted agents, as well as to processes and intermediates useful for preparing such agents.
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公开(公告)号：WO2008011116A3
公开(公告)日：2008-04-24
申请号：PCT/US2007016397
申请日：2007-07-19
Applicant: GILEAD SCIENCES INC , CANNIZZARO CARINA E , CHEN JAMES M , DESAI MANOJ C , MITCHELL MICHAEL L , SWAMINATHAN SUNDARAMOORTHI , XU LIANHONG
Inventor： CANNIZZARO CARINA E , CHEN JAMES M , DESAI MANOJ C , MITCHELL MICHAEL L , SWAMINATHAN SUNDARAMOORTHI , XU LIANHONG
IPC: C07D493/04 , A61K31/34 , A61K31/443 , A61P31/18 , C07D405/12 , C07D519/00
CPC classification number: C07D493/04 , C07D405/12 , C07D519/00
Abstract: The invention is related to compounds of Formula I: or a pharmaceutically acceptable salt, solvate, ester, and /or phosphonate thereof, compositions containing such compounds, and therapeutic methods that include the administration of such compounds.
Abstract translation: 本发明涉及式I化合物或其药学上可接受的盐，溶剂化物，酯和/或膦酸酯，含有这些化合物的组合物，以及包括给予这些化合物的治疗方法。
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公开(公告)号：WO2008011116A2
公开(公告)日：2008-01-24
申请号：PCT/US2007/016397
申请日：2007-07-19
Applicant: GILEAD SCIENCES, INC. , CANNIZZARO, Carina, E. , CHEN, James, M. , DESAI, Manoj, C. , MITCHELL, Michael, L. , SWAMINATHAN, Sundaramoorthi , XU, Lianhong
Inventor： CANNIZZARO, Carina, E. , CHEN, James, M. , DESAI, Manoj, C. , MITCHELL, Michael, L. , SWAMINATHAN, Sundaramoorthi , XU, Lianhong
CPC classification number: C07D493/04 , C07D405/12 , C07D519/00
Abstract: The invention is related to compounds of Formula I: or a pharmaceutically acceptable salt, solvate, ester, and /or phosphonate thereof, compositions containing such compounds, and therapeutic methods that include the administration of such compounds.
Abstract translation: 本发明涉及式I化合物或其药学上可接受的盐，溶剂合物，酯和/或膦酸盐，含有这些化合物的组合物，以及包括施用这些化合物的治疗方法。
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公开(公告)号：WO2004096234A3
公开(公告)日：2005-01-27
申请号：PCT/US2004013062
申请日：2004-04-26
Applicant: GILEAD SCIENCES INC , CANNIZZARO CARINA E , CHEN JAMES M , CHEN XIAOWU , CHO AESOP , CHONG LEE S , DESAI MANOJ , FARDIS MARIA , KIRSCHBERG THORSTEN A , MACKMAN RICHARD L , SWAMINATHAN SUNDARAMOORTHI , WATKINS WILL
Inventor： CANNIZZARO CARINA E , CHEN JAMES M , CHEN XIAOWU , CHO AESOP , CHONG LEE S , DESAI MANOJ , FARDIS MARIA , KIRSCHBERG THORSTEN A , MACKMAN RICHARD L , SWAMINATHAN SUNDARAMOORTHI , WATKINS WILL
IPC: A61K31/66 , A61K31/662 , A61K47/48 , C07F9/02 , C07F9/58 , C07F9/6561
CPC classification number: A61K31/662 , A61K47/54 , A61K47/548 , C07F9/588 , C07F9/6561
Abstract: The invention is related to phosphorus substituted kinase inhibitory compounds, compositions containing such compounds, and therapeutic methods that include the administration of such compounds, as well as to processes and intermediates useful for preparing such compounds.
Abstract translation: 本发明涉及磷取代的激酶抑制化合物，含有这些化合物的组合物，以及包括施用这些化合物的治疗方法以及可用于制备这些化合物的方法和中间体。
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Patent Agency Ranking
公开(公告)号：WO2004096236A2
公开(公告)日：2004-11-11
申请号：PCT/US2004/013143
申请日：2004-04-26
Applicant: GILEAD SCIENCES, INC. , CANNIZZARO, Carina, E. , CHEN, James, M. , CHEN, Xiaowu , CHO, Aesop , CHONG, Lee, S. , DESAI, Manoj , FARDIS, Maria , HUANG, Alan, X. , KIRSCHBERG, Thorsten, A. , LEE, Christopher, P. , MACKMAN, Richard, L. , NELSON, Peter, H. , PYUN, Hyung-Jung , RAY, Adrian, S. , SWAMINATHAN, Sundaramoorthi , WATKINS, Will , ZHANG, Jennifer, R.
Inventor： CANNIZZARO, Carina, E. , CHEN, James, M. , CHEN, Xiaowu , CHO, Aesop , CHONG, Lee, S. , DESAI, Manoj , FARDIS, Maria , HUANG, Alan, X. , KIRSCHBERG, Thorsten, A. , LEE, Christopher, P. , MACKMAN, Richard, L. , NELSON, Peter, H. , PYUN, Hyung-Jung , RAY, Adrian, S. , SWAMINATHAN, Sundaramoorthi , WATKINS, Will , ZHANG, Jennifer, R.
IPC: A61K31/662
CPC classification number: A61K31/662 , A61K47/548 , C07D205/04 , C07D211/58 , C07D409/06 , C07D409/14 , C07D413/14 , C07D475/00 , C07D487/04 , C07F9/4075 , C07F9/5728 , C07F9/582 , C07F9/588 , C07F9/60 , C07F9/65037 , C07F9/650941 , C07F9/653 , C07F9/6539 , C07F9/65515 , C07F9/655354 , C07F9/6561
Abstract: The invention is related to phosphonate substituted compounds having immuno-modulatory activity, compositions containing such compounds, and therapeutic methods that include the administration of such compounds, as well as to processes and intermediates useful for preparing such compounds.
Abstract translation: 本发明涉及具有免疫调节活性的膦酸酯取代的化合物，含有这些化合物的组合物，以及包括施用这些化合物的治疗方法以及可用于制备这些化合物的方法和中间体。
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公开(公告)号：WO2008011117A2
公开(公告)日：2008-01-24
申请号：PCT/US2007/016398
申请日：2007-07-19
Applicant: GILEAD SCIENCES, INC. , CANNIZZARO, Carina, E. , YANG, Zheng-Yu , DESAI, Manoj, C. , MITCHELL, Michael, L. , XU, Lianhong , SWAMINATHAN, Sundaramoorthi , CHEN, James, M.
Inventor： CANNIZZARO, Carina, E. , YANG, Zheng-Yu , DESAI, Manoj, C. , MITCHELL, Michael, L. , XU, Lianhong , SWAMINATHAN, Sundaramoorthi , CHEN, James, M.
IPC: C07D213/56 , C07D401/12 , C07D405/12 , C07D405/14 , C07D407/12 , C07D409/12
CPC classification number: C07D405/12 , C07D213/56 , C07D401/12 , C07D405/14 , C07D407/12 , C07D409/12 , C07D417/12 , C07D493/04 , C07F9/65583 , C07F9/65586 , C07F9/6561
Abstract: The invention is related to compounds of Formula I or a pharmaceutically acceptable salt, solvate, ester, and /or phosphonate thereof, compositions containing such compounds, and therapeutic methods that include the administration of such compounds.
Abstract translation: 本发明涉及式I化合物或其药学上可接受的盐，溶剂化物，酯和/或膦酸酯，含有这些化合物的组合物，以及包括给予这些化合物的治疗方法。 / p>
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公开(公告)号：WO2004096287A3
公开(公告)日：2005-05-06
申请号：PCT/US2004013064
申请日：2004-04-26
Applicant: GILEAD SCIENCES INC , CANNIZZARO CARINA E , CHEN JAMES M , CHEN XIAOWU , CHO AESOP , CHONG LEE S , FARDIS MARIA , KIRSCHBERG THORSTEN A , PYUN HYUNG-JUNG , WATKINS WILL , ZHANG JENNIFER R
Inventor： CANNIZZARO CARINA E , CHEN JAMES M , CHEN XIAOWU , CHO AESOP , CHONG LEE S , FARDIS MARIA , KIRSCHBERG THORSTEN A , PYUN HYUNG-JUNG , WATKINS WILL , ZHANG JENNIFER R
IPC: A61K31/662 , A61K31/675 , C07D205/04 , C07D211/58 , C07D409/06 , C07D409/14 , C07D413/14 , C07D475/00 , C07F9/40 , C07F9/572 , C07F9/58 , C07F9/60 , C07F9/6503 , C07F9/6509 , C07F9/653 , C07F9/6539 , C07F9/655 , C07F9/6553 , C07F9/6561
CPC classification number: C07F9/4075 , A61K31/662 , A61K47/548 , C07D205/04 , C07D211/58 , C07D409/06 , C07D409/14 , C07D413/14 , C07D475/00 , C07F9/5728 , C07F9/582 , C07F9/588 , C07F9/60 , C07F9/65037 , C07F9/650941 , C07F9/653 , C07F9/6539 , C07F9/65515 , C07F9/655354 , C07F9/6561
Abstract: The invention is related to phosphorus substituted IMPDH inhibitory compounds, compositions containing such compounds, and therapeutic methods that include the administration of such compounds, as well as to processes and intermediates useful for preparing such compounds.
Abstract translation: 本发明涉及磷取代的IMPDH抑制化合物，含有这些化合物的组合物，以及包括施用这些化合物的治疗方法以及可用于制备这些化合物的方法和中间体。
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公开(公告)号：WO2004100960A2
公开(公告)日：2004-11-25
申请号：PCT/US2004/013198
申请日：2004-04-26
Applicant: GILEAD SCIENCES, INC. , CANNIZZARO, Carina, E. , CHEN, James, M. , CHEN, Xiaowu , CHO, Aesop , CHONG, Lee, S. , FARDIS, Maria , GIBBS, Craig , HIRSCHMANN, Ralph, F. , KIRSCHBERG, Thorsten, A. , LEE, Christopher, P. , LIN, Kuei-Ying , MACKMAN, Richard, L. , NELSON, Peter, H. , OARE, David , PYUN, Hyung-Jung , RAY, Adrian, S. , SHERLOCK, Rosemarie , SWAMINATHAN, Sundaramoorthi , WATKINS, Will , ZHANG, Jennifer, R.
Inventor： CANNIZZARO, Carina, E. , CHEN, James, M. , CHEN, Xiaowu , CHO, Aesop , CHONG, Lee, S. , FARDIS, Maria , GIBBS, Craig , HIRSCHMANN, Ralph, F. , KIRSCHBERG, Thorsten, A. , LEE, Christopher, P. , LIN, Kuei-Ying , MACKMAN, Richard, L. , NELSON, Peter, H. , OARE, David , PYUN, Hyung-Jung , RAY, Adrian, S. , SHERLOCK, Rosemarie , SWAMINATHAN, Sundaramoorthi , WATKINS, Will , ZHANG, Jennifer, R.
IPC: A61K31/662
CPC classification number: A61K31/662 , A61K47/548 , C07D205/04 , C07D211/58 , C07D409/06 , C07D409/14 , C07D413/14 , C07D475/00 , C07D487/04 , C07F9/4075 , C07F9/5728 , C07F9/582 , C07F9/588 , C07F9/60 , C07F9/65037 , C07F9/650941 , C07F9/653 , C07F9/6539 , C07F9/65515 , C07F9/655354 , C07F9/6561 , C07F9/65616
Abstract: The invention is related to phosphorus substituted anti-inflammatory compounds, compositions containing such compounds, and therapeutic methods that include the administration of such compounds, as well as to processes and intermediates useful for preparing such compounds.
Abstract translation: 本发明涉及磷取代的抗炎化合物，含有这些化合物的组合物，以及包括施用这些化合物的治疗方法以及可用于制备这些化合物的方法和中间体。
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公开(公告)号：WO2004096286A2
公开(公告)日：2004-11-11
申请号：PCT/US2004/013063
申请日：2004-04-26
Applicant: GILEAD SCIENCES, INC. , BOOJAMARA, Constantine, G. , CANNIZZARO, Carina, E. , CHEN, James, M. , CHEN, Xiaowu , CHO, Aesop , CHONG, Lee, S. , FARDIS, Maria , JIN, Haolun , HIRSCHMANN, Ralph, F. , HUANG, Alan, X. , KIM, Choung, U. , KIRSCHBERG, Thorsten, A. , LEE, Christopher, P. , LEE, William, A. , MACKMAN, Richard, L. , MARKEVITCH, David, Y. , OARE, David , PRASAD, Vidya, K. , PYUN, Hyung-Jung , RAY, Adrian, S. , SHERLOCK, Rosemarie , SWAMINATHAN, Sundaramoorthi , WATKINS, Will , ZHANG, Jennifer, R.
Inventor： BOOJAMARA, Constantine, G. , CANNIZZARO, Carina, E. , CHEN, James, M. , CHEN, Xiaowu , CHO, Aesop , CHONG, Lee, S. , FARDIS, Maria , JIN, Haolun , HIRSCHMANN, Ralph, F. , HUANG, Alan, X. , KIM, Choung, U. , KIRSCHBERG, Thorsten, A. , LEE, Christopher, P. , LEE, William, A. , MACKMAN, Richard, L. , MARKEVITCH, David, Y. , OARE, David , PRASAD, Vidya, K. , PYUN, Hyung-Jung , RAY, Adrian, S. , SHERLOCK, Rosemarie , SWAMINATHAN, Sundaramoorthi , WATKINS, Will , ZHANG, Jennifer, R.
IPC: A61K47/48
CPC classification number: C07F9/65616 , A61K31/662 , A61K31/7072 , A61K31/7076 , A61K47/548 , C07D205/04 , C07D211/58 , C07D409/06 , C07D409/14 , C07D413/14 , C07D475/00 , C07F9/4075 , C07F9/5728 , C07F9/582 , C07F9/588 , C07F9/60 , C07F9/65037 , C07F9/650941 , C07F9/653 , C07F9/6539 , C07F9/65515 , C07F9/655354 , C07F9/6561 , C07H15/00 , C07H17/00 , C07H19/056 , C07H19/10 , C07H19/20 , C07H21/00 , Y02A50/393 , Y02A50/465
Abstract: The invention is related to phosphorus substituted compounds with antiviral activity, compositions containing such compounds, and therapeutic methods that include the administration of such compounds, as well as to processes and intermediates useful for preparing such compounds.
Abstract translation: 本发明涉及具有抗病毒活性的磷取代的化合物，含有这些化合物的组合物和包括施用这些化合物的治疗方法以及可用于制备这些化合物的方法和中间体。
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