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1.NICOTINAMIDE DERIVATIVES AS INHIBITORS OF H-PGDS AND THEIR USE FOR TREATING PROSTAGLANDIN D2 MEDIATED DISEASES 审中-公开
Title translation: 作为H-PGDS的抑制剂的NICOTINAMIDE衍生物及其用于治疗PROSTAGLANDIN D2介导的疾病的用途公开(公告)号:WO2008075172A3
公开(公告)日:2008-10-02
申请号:PCT/IB2007003928
申请日:2007-12-03
Applicant: PFIZER PROD INC , BLAKE TANISHA DANIELLE ROWE , HAMPER BRUCE CAMERON , HUANG WEI , KIEFER JAMES RICHARD JR , MOON JOSEPH BLAIR , NEAL BRADLEY E , OLSON KIRK LANG , PELC MATTHEW JAMES , SCHWEITZER BARBARA ANN , THORARENSEN ALTI , TRUJILLO JOHN I , TURNER STEVE R
Inventor: BLAKE TANISHA DANIELLE ROWE , HAMPER BRUCE CAMERON , HUANG WEI , KIEFER JAMES RICHARD JR , MOON JOSEPH BLAIR , NEAL BRADLEY E , OLSON KIRK LANG , PELC MATTHEW JAMES , SCHWEITZER BARBARA ANN , THORARENSEN ALTI , TRUJILLO JOHN I , TURNER STEVE R
IPC: C07D213/82 , A61P11/00 , C07D401/12 , C07D401/14 , C07D413/14 , C07D417/14 , C07D471/04
CPC classification number: C07D401/12 , C07D213/82 , C07D401/14 , C07D413/14 , C07D417/14 , C07D471/04 , C07D487/04
Abstract: The present invention relates to compounds of formula (I) and pharmaceutically acceptable salts and solvates thereof, wherein the substituents are as defined herein, compositions containing such compounds and the uses of such compounds for the treatment of various diseases and conditions such as asthma.
Abstract translation: 本发明涉及式(I)化合物及其药学上可接受的盐和溶剂合物,其中取代基如本文所定义,含有这些化合物的组合物以及这些化合物用于治疗各种疾病和病症例如哮喘的用途。
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2.NICOTINAMIDE DERIVATIVES AS INHIBITORS OF H-PGDS AND THEIR USE FOR TREATING PROSTAGLANDIN D2 MEDIATED DISEASES 审中-公开
Title translation: 作为H-PGDS的抑制剂的NICOTINAMIDE衍生物及其用于治疗PROSTAGLANDIN D2介导的疾病的用途公开(公告)号:WO2008104869A1
公开(公告)日:2008-09-04
申请号:PCT/IB2008/000467
申请日:2008-02-15
Applicant: PFIZER PRODUCTS INC. , BLAKE, Tanisha, Danielle, Rowe , HAMPER, Bruce, Cameron , HUANG, Wei , KIEFER, James, Richard, Jr. , MOON, Joseph, Blair , NEAL, Bradley, E. , OLSON, Kirk, Lang , PELC, Matthew, James , SCHWEITZER, Barbara, Ann , THORARENSEN, Atli , TRUJILLO, John, I. , TURNER, Steve, R.
Inventor: BLAKE, Tanisha, Danielle, Rowe , HAMPER, Bruce, Cameron , HUANG, Wei , KIEFER, James, Richard, Jr. , MOON, Joseph, Blair , NEAL, Bradley, E. , OLSON, Kirk, Lang , PELC, Matthew, James , SCHWEITZER, Barbara, Ann , THORARENSEN, Atli , TRUJILLO, John, I. , TURNER, Steve, R.
IPC: C07D401/12 , C07D401/14 , C07D413/14 , C07D417/14 , C07D471/04 , A61P11/00
CPC classification number: C07D401/12 , C07D401/02 , C07D401/14 , C07D413/14 , C07D417/14 , C07D471/04
Abstract: The present invention relates to compounds of formula (I), and pharmaceutically acceptable salts and solvates thereof, wherein the substituents are as defined herein, compositions containing such compounds and the uses of such compounds for the treatment of various diseases and conditions such as asthma.
Abstract translation: 本发明涉及式(I)化合物及其药学上可接受的盐和溶剂合物,其中取代基如本文所定义,含有这些化合物的组合物以及这些化合物用于治疗各种疾病和病症如哮喘的用途。
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公开(公告)号:WO2008075172A2
公开(公告)日:2008-06-26
申请号:PCT/IB2007/003928
申请日:2007-12-03
Applicant: PFIZER PRODUCTS INC. , BLAKE, Tanisha, Danielle, Rowe , HAMPER, Bruce, Cameron , HUANG, Wei , KIEFER, James, Richard, Jr. , MOON, Joseph, Blair , NEAL, Bradley, E. , OLSON, Kirk, Lang , PELC, Matthew, James , SCHWEITZER, Barbara, Ann , THORARENSEN, Alti , TRUJILLO, John, I. , TURNER, Steve, R.
Inventor: BLAKE, Tanisha, Danielle, Rowe , HAMPER, Bruce, Cameron , HUANG, Wei , KIEFER, James, Richard, Jr. , MOON, Joseph, Blair , NEAL, Bradley, E. , OLSON, Kirk, Lang , PELC, Matthew, James , SCHWEITZER, Barbara, Ann , THORARENSEN, Alti , TRUJILLO, John, I. , TURNER, Steve, R.
CPC classification number: C07D401/12 , C07D213/82 , C07D401/14 , C07D413/14 , C07D417/14 , C07D471/04 , C07D487/04
Abstract: The present invention relates to compounds of formula (I) and pharmaceutically acceptable salts and solvates thereof, wherein the substituents are as defined herein, compositions containing such compounds and the uses of such compounds for the treatment of various diseases and conditions such as asthma.
Abstract translation: 本发明涉及式(I)化合物及其药学上可接受的盐和溶剂合物,其中取代基如本文所定义,含有这些化合物的组合物以及这些化合物用于治疗各种疾病和病症例如哮喘的用途。
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