公开(公告)号：WO2011043568A2

公开(公告)日：2011-04-14

申请号：PCT/KR2010/006760

申请日：2010-10-04

Applicant: LG LIFE SCIENCES LTD. ,  SONG, Jeong Uk ,  KIM, Geun Tae ,  CHOI, Sung Pil ,  JUNG, Cheol Kyu ,  PARK, Deok Seong ,  CHOI, Eun Sil ,  KIM, Tae Hun ,  PARK, Hyun Jung ,  PARK, Wan Su ,  PARK, Heui Sul ,  KOO, Ki Chul ,  ARTEMOV, Vasily

Inventor： SONG, Jeong Uk ,  KIM, Geun Tae ,  CHOI, Sung Pil ,  JUNG, Cheol Kyu ,  PARK, Deok Seong ,  CHOI, Eun Sil ,  KIM, Tae Hun ,  PARK, Hyun Jung ,  PARK, Wan Su ,  PARK, Heui Sul ,  KOO, Ki Chul ,  ARTEMOV, Vasily

IPC: C07D403/02 ,  C07D209/04 ,  A61K31/40 ,  A61P3/10

CPC classification number: C07D403/04 ,  C07D401/04 ,  C07D405/14 ,  C07D409/04

Abstract: The present invention relates to novel compounds which are effective as an inhibitor for xanthine oxidase, a process for preparing the same, and a pharmaceutical composition comprising a therapeutically effective amount of the same.

Abstract translation: 本发明涉及作为黄嘌呤氧化酶抑制剂有效的新化合物，其制备方法和含有治疗有效量的药物组合物。

公开(公告)号：WO2010027236A3

公开(公告)日：2010-06-17

申请号：PCT/KR2009005073

申请日：2009-09-08

Applicant: LG LIFE SCIENCES LTD ,  LEE CHANG SEOK ,  LEE TAE HEE ,  YOON SOOK KYUNG ,  CHOI JEUNG SOON ,  JANG YONG JIN ,  KIM SUNG WOOK ,  CHANG HYE KYUNG ,  PARK MI JEONG ,  KIM TAE HUN ,  AHN YOUNG HA ,  PARK HEE DONG ,  PARK HYUN JUNG ,  LIM DONG CHUL ,  LEE JOO YOUN ,  LEE SUNG HACK ,  PARK WAN SU ,  OH YEONG SOO

Inventor： LEE CHANG SEOK ,  LEE TAE HEE ,  YOON SOOK KYUNG ,  CHOI JEUNG SOON ,  JANG YONG JIN ,  KIM SUNG WOOK ,  CHANG HYE KYUNG ,  PARK MI JEONG ,  KIM TAE HUN ,  AHN YOUNG HA ,  PARK HEE DONG ,  PARK HYUN JUNG ,  LIM DONG CHUL ,  LEE JOO YOUN ,  LEE SUNG HACK ,  PARK WAN SU ,  OH YEONG SOO

IPC: C07D495/04

CPC classification number: C07D495/04 ,  C07D519/00

Abstract: The present invention relates to a fused heterocyclic compound having the Formula 1, which is useful as a platelet aggregation inhibitor, a method for preparing the same, and a pharmaceutical composition for inhibiting platelet aggregation comprising the same.

Abstract translation: 本发明涉及用作血小板聚集抑制剂的具有式1的稠合杂环化合物，其制备方法和包含其的血小板聚集抑制药物组合物。

公开(公告)号：WO2011043568A3

公开(公告)日：2011-09-29

申请号：PCT/KR2010006760

申请日：2010-10-04

Applicant: LG LIFE SCIENCES LTD ,  SONG JEONG UK ,  KIM GEUN TAE ,  CHOI SUNG PIL ,  JUNG CHEOL KYU ,  PARK DEOK SEONG ,  CHOI EUN SIL ,  KIM TAE HUN ,  PARK HYUN JUNG ,  PARK WAN SU ,  PARK HEUI SUL ,  KOO KI CHUL ,  ARTEMOV VASILY

Inventor： SONG JEONG UK ,  KIM GEUN TAE ,  CHOI SUNG PIL ,  JUNG CHEOL KYU ,  PARK DEOK SEONG ,  CHOI EUN SIL ,  KIM TAE HUN ,  PARK HYUN JUNG ,  PARK WAN SU ,  PARK HEUI SUL ,  KOO KI CHUL ,  ARTEMOV VASILY

IPC: C07D403/02 ,  A61K31/40 ,  A61P3/10 ,  C07D209/04

CPC classification number: C07D403/04 ,  C07D401/04 ,  C07D405/14 ,  C07D409/04

Abstract: The present invention relates to novel compounds which are effective as an inhibitor for xanthine oxidase, a process for preparing the same, and a pharmaceutical composition comprising a therapeutically effective amount of the same.

Abstract translation: 本发明涉及作为黄嘌呤氧化酶抑制剂有效的新化合物，其制备方法以及包含治疗有效量的药物组合物。

公开(公告)号：WO2010027236A2

公开(公告)日：2010-03-11

申请号：PCT/KR2009/005073

申请日：2009-09-08

Applicant: LG LIFE SCIENCES LTD. ,  LEE, Chang Seok ,  LEE, Tae Hee ,  YOON, Sook Kyung ,  CHOI, Jeung Soon ,  JANG, Yong Jin ,  KIM, Sung Wook ,  CHANG, Hye Kyung ,  PARK, Mi Jeong ,  KIM, Tae Hun ,  AHN, Young Ha ,  PARK, Hee Dong ,  PARK, Hyun Jung ,  LIM, Dong Chul ,  LEE, Joo Youn ,  LEE, Sung Hack ,  PARK, Wan Su ,  OH, Yeong Soo

Inventor： LEE, Chang Seok ,  LEE, Tae Hee ,  YOON, Sook Kyung ,  CHOI, Jeung Soon ,  JANG, Yong Jin ,  KIM, Sung Wook ,  CHANG, Hye Kyung ,  PARK, Mi Jeong ,  KIM, Tae Hun ,  AHN, Young Ha ,  PARK, Hee Dong ,  PARK, Hyun Jung ,  LIM, Dong Chul ,  LEE, Joo Youn ,  LEE, Sung Hack ,  PARK, Wan Su ,  OH, Yeong Soo

IPC: C07D495/04

CPC classification number: C07D495/04 ,  C07D519/00

Abstract: The present invention relates to a fused heterocyclic compound having the Formula 1, which is useful as a platelet aggregation inhibitor, a method for preparing the same, and a pharmaceutical composition for inhibiting platelet aggregation comprising the same.

Abstract translation: 本发明涉及具有式1的稠合杂环化合物，其可用作血小板聚集抑制剂，其制备方法和包含其的用于抑制血小板聚集的药物组合物。

公开(公告)号：WO2009082134A3

公开(公告)日：2009-09-24

申请号：PCT/KR2008007543

申请日：2008-12-19

Applicant: LG LIFE SCIENCES LTD ,  LEE CHANG-SEOK ,  YIM HYEON JOO ,  KIM KYOUNG-HEE ,  LEE JAEICK ,  LEE SUNG-HACK ,  LEE KYU WOONG ,  LEE HEE BONG ,  PARK WAN SU ,  MIN CHANGHEE

Inventor： LEE CHANG-SEOK ,  YIM HYEON JOO ,  KIM KYOUNG-HEE ,  LEE JAEICK ,  LEE SUNG-HACK ,  LEE KYU WOONG ,  LEE HEE BONG ,  PARK WAN SU ,  MIN CHANGHEE

IPC: C07D471/04

CPC classification number: C07D471/04

Abstract: Disclosed herein are novel compounds of Formula (1) as defined in the specification having excellent inhibitory activity against dipeptidyl peptidase-IV (DPP-IV), methods of preparing the same and pharmaceutical compositions comprising the same as an active agent.

Abstract translation: 本文公开了如本说明书中所定义的具有优异的抗二肽基肽酶-IV（DPP-IV）抑制活性的式（1）化合物，其制备方法和包含其作为活性剂的药物组合物。

公开(公告)号：WO2009082134A2

公开(公告)日：2009-07-02

申请号：PCT/KR2008/007543

申请日：2008-12-19

Applicant: LG LIFE SCIENCES, LTD. ,  LEE, Chang-Seok ,  YIM, Hyeon Joo ,  KIM, Kyoung-Hee ,  LEE, Jaeick ,  LEE, Sung-Hack ,  LEE, Kyu Woong ,  LEE, Hee Bong ,  PARK, Wan Su ,  MIN, Changhee

Inventor： LEE, Chang-Seok ,  YIM, Hyeon Joo ,  KIM, Kyoung-Hee ,  LEE, Jaeick ,  LEE, Sung-Hack ,  LEE, Kyu Woong ,  LEE, Hee Bong ,  PARK, Wan Su ,  MIN, Changhee

IPC: C07D471/04

CPC classification number: C07D471/04

Abstract: Disclosed herein are novel compounds of Formula (1) as defined in the specification having excellent inhibitory activity against dipeptidyl peptidase-IV (DPP-IV), methods of preparing the same and pharmaceutical compositions comprising the same as an active agent.

Abstract translation: 本文公开的是具有对二肽基肽酶-IV（DPP-IV）具有优异抑制活性的本说明书中定义的新颖的式（1）化合物，其制备方法和包含其作为活性剂的药物组合物。