公开(公告)号：WO2017025377A1

公开(公告)日：2017-02-16

申请号：PCT/EP2016/068365

申请日：2016-08-02

Applicant: BASF SE

Inventor： KLAUBER, Eric George ,  FRASSETTO, Timo ,  NIEMES, Reinhold ,  BAUER, Ralf ,  SCHROEDER, Jochen

IPC: C07D231/24 ,  C07D231/04

CPC classification number: C07D231/04 ,  C07D231/24

Abstract: The present invention relates to a process for preparing crystalline methyl N-[2-[[[1-(4-chlorophenyl)-1H-pyrazol-3-yl]oxy]methyl]phenyl]-N-methoxycarbamate (I), comprising a) reacting a compound of formula (II) with an alkylating agent in the presence of a base in the presence of a polar solvent selected from alcohols and ketons; b) the addition of water.

Abstract translation: 本发明涉及N- [2 - [[[1-（4-氯苯基）-1H-吡唑-3-基]氧基]甲基]苯基] -N-甲氧基氨基甲酸叔丁酯（I）的制备方法，包括 a）在碱存在下，在选自醇和酮的极性溶剂的存在下，使式（II）的化合物与烷基化剂反应; b）加水。

公开(公告)号：WO2015158518A1

公开(公告)日：2015-10-22

申请号：PCT/EP2015/056541

申请日：2015-03-26

Applicant: BASF SE

Inventor： WOLF, Bernd ,  RACK, Michael ,  MAYWALD, Volker ,  GÖTZ, Roland ,  FRASSETTO, Timo

IPC: C07D265/36

CPC classification number: C07D265/36

Abstract: The present invention relates to for manufacturing benzoxazinones of formula (I), characterized in that amino compounds of formula (II) are added to an acid; wherein the substituents are defined according to the specification.

Abstract translation: 本发明涉及制备式（I）的苯并恶嗪酮，其特征在于将式（II）的氨基化合物加入酸中; 其中取代基根据说明书定义。

公开(公告)号：WO2014202589A1

公开(公告)日：2014-12-24

申请号：PCT/EP2014/062695

申请日：2014-06-17

Applicant: BASF SE

Inventor： FRASSETTO, Timo ,  DOCHNAHL, Maximilian ,  RACK, Michael ,  MAYWALD, Volker ,  WOLF, Bernd ,  GÖTZ, Roland ,  MÜLHEIMS, Philip ,  HÄBERLE, Rudolf

IPC: C07D265/36 ,  C07C17/16

CPC classification number: C07D265/36 ,  C07C17/16 ,  C07D413/04 ,  C07C21/22

Abstract: The present invention relates to a process for manufacturing 4-propargylated amino- benzoxazinones of formula (I), comprising the following steps: step a) preparing propargyl chloride by reacting propargyl alcohol with thionyl chloride optionally in the presence of a catalyst; and step b) reacting the propargyl chloride prepared in step (a) with a NH-benzoxazinone of formula (II); wherein the variables are defined according to the description.

Abstract translation: 本发明涉及一种制备式（I）的4-炔丙基化 - 苯并恶嗪酮的方法，包括以下步骤：步骤a）任选地在催化剂存在下，将炔丙醇与亚硫酰氯反应制备炔丙基氯; 和步骤b）使步骤（a）中制备的炔丙基氯与式（II）的NH-苯并嗪酮反应; 其中根据描述定义变量。

公开(公告)号：WO2018149813A1

公开(公告)日：2018-08-23

申请号：PCT/EP2018/053522

申请日：2018-02-13

Applicant: BASF SE

Inventor： FRASSETTO, Timo ,  MAYER, Horst ,  KRAEMER, Siegfried

IPC: C07D231/14 ,  C07F9/50 ,  C07F9/54 ,  C07C201/12 ,  C07C205/19 ,  C07D241/24 ,  C07F5/02

Abstract: The present invention relates to a process for preparing substituted 2-nitrobiphenyls via Suzuki coupling using a palladium catalyst with specific phosphorus ligands and a solvent mixture containing water and an organic solvent which is at least partially miscible with water.

公开(公告)号：WO2018091338A1

公开(公告)日：2018-05-24

申请号：PCT/EP2017/078680

申请日：2017-11-09

Applicant: BASF SE

Inventor： MAYWALD, Volker ,  GOETZ, Roland ,  SAELINGER, Daniel ,  FRASSETTO, Timo ,  GROPP, Stefan

IPC: C07D231/22

Abstract: The present invention relates to a process to produce highly purified crystalline 1-(4-chlorophenyl)pyrazol-3-ol (I).

公开(公告)号：WO2014026928A1

公开(公告)日：2014-02-20

申请号：PCT/EP2013/066719

申请日：2013-08-09

Applicant: BASF SE ,  BASF SCHWEIZ AG

Inventor： DOCHNAHL, Maximilian ,  GÖTZ, Roland ,  GEBHARDT, Joachim ,  VOGELBACHER, Uwe Josef ,  FRASSETTO, Timo ,  RACK, Michael ,  MAYWALD, Volker ,  WOLF, Bernd

IPC: C07D413/04

CPC classification number: C07D413/04 ,  C07C335/28 ,  C07D265/36

Abstract: The present invention relates to a process for manufacturing benzoxazinones of formula (I), wherein the variables are defined according to the description, by reacting carbamates of formula (II) are reacted with carbamat-benzoxazinones of formula (III) in the presence of a base.

Abstract translation: 本发明涉及一种制备式（I）的苯并恶嗪酮的方法，其中根据描述定义变量，使式（II）的氨基甲酸酯与式（III）的氨基甲酸酯 - 苯并恶嗪酮反应，在 基础。

公开(公告)号：WO2014026893A1

公开(公告)日：2014-02-20

申请号：PCT/EP2013/066562

申请日：2013-08-07

Applicant: BASF SE ,  BASF SCHWEIZ AG

Inventor： DOCHNAHL, Maximilian ,  GöTZ, Roland ,  GEBHARDT, Joachim ,  VOGELBACHER, Uwe Josef ,  FRASSETTO, Timo ,  RACK, Michael ,  MAYWALD, Volker ,  WOLF, Bernd

IPC: C07D265/36 ,  C07D413/04

CPC classification number: C07D265/36 ,  C07D413/04

Abstract: The present invention relates to carbamat-benzoxazinones of formula (I), wherein the variables are defined according to the description, 5 as well as to a process for manufacturing carbamat-benzoxazinones of formula (I), and to the use of carbamat-benzoxazinones of formula (I) in manufacturing benzoxazinones of formula (X).

Abstract translation: 本发明涉及式（I）的氨基甲酰 - 苯并恶嗪酮，其中根据描述5定义变量，以及制备式（I）的氨基甲酰 - 苯并恶嗪酮的方法，以及使用氨基甲酰 - 苯并恶嗪酮 式（I）在制备式（X）的苯并恶嗪酮时。

公开(公告)号：WO2013092856A1

公开(公告)日：2013-06-27

申请号：PCT/EP2012/076373

申请日：2012-12-20

Applicant: BASF SE

Inventor： DOCHNAHL, Maximilian ,  RACK, Michael ,  KEIL, Michael ,  WOLF, Bernd ,  VOGELBACHER, Uwe, Josef ,  GEBHARDT, Joachim ,  FRASSETTO, Timo ,  MAYWALD, Volker

IPC: C07D265/36 ,  C07D413/04

CPC classification number: C07D265/36 ,  C07C231/12 ,  C07D413/04

Abstract: The present invention relates to a process for manufacturing a benzoxazinone of formula (I), by reacting a nitro compound of formula (II)with a reducing agent to obtain an amino compound of formula (III), and then reacting the amino compound of formula (III) with an acid; wherein the variables are defined according to the description, and benzoxazinone of formula (I).

Abstract translation: 本发明涉及式（I）的苯并恶嗪酮的制备方法，通式（II）的硝基化合物与还原剂反应得到式（III）的氨基化合物，然后使式 （III）与酸反应; 其中根据描述定义变量，和式（I）的苯并嗪酮。

公开(公告)号：WO2022078796A1

公开(公告)日：2022-04-21

申请号：PCT/EP2021/077255

申请日：2021-10-04

Applicant: BASF SE

Inventor： FRASSETTO, Timo ,  ALZNAUER, Christiane ,  VOGT, Florian ,  SHINDE, Harish ,  SAELINGER, Daniel ,  SUTORIS, Heinz Friedrich

IPC: C07C29/40 ,  C07C33/46

Abstract: The present invention relates to a process for the preparation of preparation α-alkyl-2- (trifluoromethyl)-benzyl alcohol.

公开(公告)号：WO2013178585A1

公开(公告)日：2013-12-05

申请号：PCT/EP2013/060866

申请日：2013-05-27

Applicant: BASF SE ,  BASF SCHWEIZ AG

Inventor： WITSCHEL, Matthias ,  KRAUS, Helmut ,  HUTZLER, Johannes ,  NEWTON, Trevor William ,  REINGRUBER, Rüdiger ,  FRASSETTO, Timo ,  PARRA RAPADO, Liliana ,  BESONG, Gilbert ,  RACK, Michael ,  KLOET, Andree van der ,  SEITZ, Thomas ,  LERCHL, Jens ,  KREUZ, Klaus ,  PASTERNAK, Maciej ,  EVANS, Richard Roger

IPC: C07D495/04 ,  A01N43/90 ,  A01P21/00 ,  A01P13/00

CPC classification number: A01N43/90 ,  C07D495/04

Abstract: The present invention provides a substituted pyridine compound of the formula (I) or an agriculturally suitable salt or N-oxide thereof, wherein the variables in the formula (I) are defined as in the description. Substituted pyridine compounds of formula (I) are useful as herbicides.

Abstract translation: 本发明提供式（I）的取代的吡啶化合物或其农业上合适的盐或N-氧化物，其中式（I）中的变量如描述中所定义。 取代的式（I）的吡啶化合物可用作除草剂。