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公开(公告)号：WO2005011700A1
公开(公告)日：2005-02-10
申请号：PCT/US2004/024340
申请日：2004-07-28
Applicant: SMITHKLINE BEECHAM CORPORATION , HEERDING, Dirk, A. , CLARK, Tammy, J. , DREWRY, David, H. , LEBER, Jack, Dale , SAFONOV, Igor , YAMASHITA, Dennis, S.
Inventor： HEERDING, Dirk, A. , CLARK, Tammy, J. , DREWRY, David, H. , LEBER, Jack, Dale , SAFONOV, Igor , YAMASHITA, Dennis, S.
IPC: A61K31/4965
CPC classification number: C07D471/04
Abstract: Invented are novel 1 H-imidazo[4,5-c]pyridin-2-yI compounds, the use of such compounds as inhibitors of protein kinase B activity and in the treatment of cancer and arthritis.
Abstract translation: 发明了新的1H-咪唑并[4,5-c]吡啶-2-基化合物，使用这些化合物作为蛋白激酶B活性的抑制剂和治疗癌症和关节炎。
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公开(公告)号：WO2009032652A1
公开(公告)日：2009-03-12
申请号：PCT/US2008/074371
申请日：2008-08-27
Applicant: SMITHKLINE BEECHAM CORPORATION , HEERDING, Dirk, A. , LIN, Hong , YAMASHITA, Dennis, A.
Inventor： HEERDING, Dirk, A. , LIN, Hong , YAMASHITA, Dennis, A.
IPC: A01N43/90 , A61K31/415 , A61K31/519
CPC classification number: C07D471/04
Abstract: Invented are novel substituted pyridine compounds, the use of such compounds as inhibitors of protein kinase B activity and in the treatment of cancer and arthritis.
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公开(公告)号：WO2007076423A2
公开(公告)日：2007-07-05
申请号：PCT/US2006/062453
申请日：2006-12-21
Applicant: SMITHKLINE BEECHAM CORPORATION , SEEFELD, Mark, Andrew , HAMAJIMA, Toshihiro , JUNG, David, Kendall , NAKAMURA, Hiroko , REID, Paul, R. , RENO, Michael, John , ROUSE, Meagan, B. , HEERDING, Dirk, A. , TANG, Jun , WANG, Jizhou
Inventor： SEEFELD, Mark, Andrew , HAMAJIMA, Toshihiro , JUNG, David, Kendall , NAKAMURA, Hiroko , REID, Paul, R. , RENO, Michael, John , ROUSE, Meagan, B. , HEERDING, Dirk, A. , TANG, Jun , WANG, Jizhou
IPC: A61K31/53 , A61K31/519
CPC classification number: C07D471/04 , C07D487/04
Abstract: Invented are novel thiophene compounds, the use of such compounds as inhibitors of protein kinase B activity and in the treatment of cancer and arthritis.
Abstract translation: 发明的是新颖的噻吩化合物，这些化合物作为蛋白激酶B活性抑制剂的用途以及治疗癌症和关节炎。
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公开(公告)号：WO2004054515A2
公开(公告)日：2004-07-01
申请号：PCT/US2003/039633
申请日：2003-12-12
Applicant: SMITHKLINE BEECHAM CORPORATION , HEERDING, Dirk, A. , PRICE, Alan, T. , SAFONOV, Igor
Inventor： HEERDING, Dirk, A. , PRICE, Alan, T. , SAFONOV, Igor
IPC: A61K
CPC classification number: C07D417/00 , C07D235/18
Abstract: Invented are non-peptide TPO mimetics. Also invented are novel processes and intermediates used in the preparation of the presently invented compounds. Also invented is a method of treating thrombocytopenia, in a mammal, including a human, in need thereof which comprises administering to such mammal an effective amount of a selected benzimidazole derivative.
Abstract translation: 本发明的是非肽TPO模拟物。 还发明了用于制备目前发明的化合物的新型方法和中间体。 还发明了一种治疗需要治疗的哺乳动物，包括人的血小板减少症的方法，该方法包括给这种哺乳动物施用有效量的所选苯并咪唑衍生物。
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公开(公告)号：WO2002072760A2
公开(公告)日：2002-09-19
申请号：PCT/US2002/006941
申请日：2002-03-07
Inventor： HEERDING, Dirk, A. , YUAN, Catherine, C. K.
IPC: C12N
CPC classification number: C07C217/60 , C07C255/54
Abstract: This invention relates to the novel PcrA helicase inhibitors useful as broad-spectrum antibacterials.
Abstract translation: 本发明涉及可用作广谱抗菌剂的新型PcrA解旋酶抑制剂。
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Patent Agency Ranking
公开(公告)号：WO2002072087A1
公开(公告)日：2002-09-19
申请号：PCT/US2002/006842
申请日：2002-03-07
Applicant: SMITHKLINE BEECHAM CORPORATION , HEERDING, Dirk, A.
Inventor： HEERDING, Dirk, A.
IPC: A61K31/40
CPC classification number: C07D207/14 , C07D207/12
Abstract: This invention relates to the novel PcrA helicase inhibitors useful as broad-spectrum antibacterials.
Abstract translation: 本发明涉及用作广谱抗菌剂的新型PcrA解旋酶抑制剂。
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公开(公告)号：WO2008098104A8
公开(公告)日：2008-08-14
申请号：PCT/US2008/053269
申请日：2008-02-07
Applicant: SMITHKLINE BEECHAM CORPORATION , SEEFELD, Mark, Andrew , ROUSE, Meagan, B. , HEERDING, Dirk, A. , PEACE, Simon , YAMASHITA, Dennis, S. , MCNULTY, Kenneth, C.
Inventor： SEEFELD, Mark, Andrew , ROUSE, Meagan, B. , HEERDING, Dirk, A. , PEACE, Simon , YAMASHITA, Dennis, S. , MCNULTY, Kenneth, C.
IPC: A61K31/12
Abstract: Invented are novel heterocyclic carboxamide compounds, the use of such compounds as inhibitors of protein kinase B activity and in the treatment of cancer and arthritis.
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公开(公告)号：WO2003103686A1
公开(公告)日：2003-12-18
申请号：PCT/US2003/017837
申请日：2003-06-06
Applicant: SMITHKLINE BEECHAM CORPORATION , HEERDING, Dirk, A.
Inventor： HEERDING, Dirk, A.
IPC: A61K31/655
CPC classification number: C07D417/12 , C07C205/56 , C07C229/44 , C07C243/20 , C07C2601/08 , C07D231/20 , C07D231/46 , C07F9/65031
Abstract: Invented are non-peptide TPO mimetics. Also invented are novel processes and intermediates used in the preparation of the presently invented compounds. Also invented is a method of treating thrombocytopenia, in a mammal, including a human, in need thereof which comprises administering to such mammal an effective amount of a selected hydroxy1-azobenzene derivative.
Abstract translation: 发明的是非肽TPO模拟物。 还发明了用于制备本发明化合物的新方法和中间体。 还发明了一种在有需要的哺乳动物（包括人）中治疗血小板减少症的方法，其包括向所述哺乳动物施用有效量的选择的羟基-1-偶氮苯衍生物。
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公开(公告)号：WO2002072760A3
公开(公告)日：2002-09-19
申请号：PCT/US2002/006941
申请日：2002-03-07
Inventor： HEERDING, Dirk, A. , YUAN, Catherine, C. K.
IPC: C07C215/20
Abstract: This invention relates to the novel PcrA helicase inhibitors useful as broad-spectrum antibacterials.
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公开(公告)号：WO2002060443A1
公开(公告)日：2002-08-08
申请号：PCT/US2001/049119
申请日：2001-12-17
Applicant: SMITHKLINE BEECHAM CORPORATION , HEERDING, Dirk, A.
Inventor： HEERDING, Dirk, A.
IPC: A61K31/425
CPC classification number: A61K31/428 , A61K31/426 , Y02A50/473
Abstract: This invention relates to novel thiazolidinediones and their use as anti-bacterials
Abstract translation: 本发明涉及新的噻唑烷二酮类化合物及其作为抗菌剂的用途
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