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1.发明授权DERIVATIVES OF 1-N-AZACYCLOALKYL-3-PHENOXYPROPANE USEFUL FOR THE PREPARATION OF PSYCHOTROPIC MEDICAMENTS 有权用于生产精神药品的1-N-氮杂环烷基-3-苯氧合适的衍生物
公开(公告)号：EP1874746B1
公开(公告)日：2015-11-18
申请号：EP06744550.2
申请日：2006-04-25
申请人： BIOPROJET
发明人： BERTRAND, Isabelle , CAPET, Marc , LECOMTE, Jeanne-Marie , LEVOIN, Nicolas , LIGNEAU, Xavier , POUPARDIN-OLIVIER, Olivia , ROBERT, Philippe , SCHWARTZ, Jean-Charles , LABEEUW, Olivier
IPC分类号： C07D295/088 , C07D213/30 , C07D211/68 , C07D333/16 , C07D211/14 , C07D401/10 , A61K31/40 , A61K31/44 , A61K31/381 , A61K31/5377
CPC分类号： C07D213/30 , C07D207/20 , C07D207/30 , C07D207/335 , C07D211/22 , C07D211/42 , C07D211/46 , C07D211/68 , C07D211/70 , C07D213/61 , C07D213/64 , C07D213/89 , C07D231/12 , C07D295/088 , C07D295/192 , C07D333/16 , C07D333/20 , C07D401/12 , C07D401/14 , C07D409/12 , C07D413/12
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公开(公告)号：EP1874747A1
公开(公告)日：2008-01-09
申请号：EP06744570.0
申请日：2006-04-26
申请人： BIOPROJET
发明人： BERTRAND, Isabelle , CAPET, Marc , LECOMTE, Jeanne-Marie , LEVOIN, Nicolas , LIGNEAU, Xavier , POUPARDIN-OLIVIER, Olivia , ROBERT, Philippe , SCHWARTZ, Jean-Charles
IPC分类号： C07D295/088 , C07D307/79 , C07D317/54 , C07D319/18 , A61K31/40 , A61K31/445 , A61P25/00
CPC分类号： C07D295/088 , C07D307/79 , C07D317/54 , C07D319/18
摘要： The present patent application concerns new compounds of formula (I) with R1 and R2 taken together with the nitrogen atom to which they are attached, form a saturated nitrogen-containing ring, A is a saturated C1 -4 alkylene and B a C3-4 alkylene or alkenylene chain; their preparation and their use as a H3 receptor ligand for treating e.g. CNS disorders like Alzheimer's disease.
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公开(公告)号：EP3486243A1
公开(公告)日：2019-05-22
申请号：EP18206553.2
申请日：2018-11-15
申请人： Bioprojet
发明人： BERREBI-BERTRAND, Isabelle , BILLOT, Xavier , CALMELS, Thierry , CAPET, Marc , KRIEF, Stéphane , LABEEUW, Olivier , LECOMTE, Jeanne-Marie , LEVOIN, Nicolas , LIGNEAU, Xavier , ROBERT, Philippe , SCHWARTZ, Jean-Charles
IPC分类号： C07D401/12 , A61K31/4439 , A61P37/08
摘要： The present application concerns novel benzimidazole enantiomeric derivatives, their process of preparation and their therapeutical uses as dual H1 and H4 receptor ligands
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公开(公告)号：EP2621916A1
公开(公告)日：2013-08-07
申请号：EP11761383.6
申请日：2011-09-27
申请人： BIOPROJET
发明人： BERREBI-BERTRAND, Isabelle , BILLOT, Xavier , CALMELS, Thierry , CAPET, Marc , DANVY, Denis , KRIEF, Stéphane , LABEEUW, Olivier , LECOMTE, Jeanne-Marie , LEVOIN, Nicolas , LIGNEAU, Xavier , ROBERT, Philippe , SCHWARTZ, Jean-Charles
IPC分类号： C07D401/12 , C07D405/14 , C07D417/12 , C07D417/14 , A61K31/4439 , A61P37/08
CPC分类号： C07D417/14 , A61K31/428 , A61K31/454 , A61K31/4545 , A61K31/496 , A61K31/506 , A61K31/5377 , A61K45/06 , C07D401/04 , C07D401/12 , C07D401/14 , C07D405/14 , C07D417/04 , C07D417/12
摘要： The present patent application concerns new Iigands of the H4-receptor of formula (I), their process of preparation and their therapeutic use.
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公开(公告)号：EP3486243B1
公开(公告)日：2020-04-15
申请号：EP18206553.2
申请日：2018-11-15
申请人： Bioprojet
发明人： BERREBI-BERTRAND, Isabelle , BILLOT, Xavier , CALMELS, Thierry , CAPET, Marc , KRIEF, Stéphane , LABEEUW, Olivier , LECOMTE, Jeanne-Marie , LEVOIN, Nicolas , LIGNEAU, Xavier , ROBERT, Philippe , SCHWARTZ, Jean-Charles
IPC分类号： C07D401/12 , A61K31/4439 , A61P37/08
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公开(公告)号：EP2038268B1
公开(公告)日：2015-11-04
申请号：EP07766572.7
申请日：2007-06-21
申请人： BIOPROJET
发明人： CAPET, Marc , DANVY, Denis , LEVOIN, Nicolas , BERREBI-BERTRAND, Isabelle , CALMELS, Thierry , ROBERT, Philippe , LECOMTE, Jeanne-Marie , SCHWARTZ, Jean-Charles , LIGNEAU, Xavier
IPC分类号： C07D295/12 , A61K31/495 , A61P25/00 , C07D211/26 , C07D295/14 , C07D295/10 , C07D307/24 , C07D211/70 , C07D211/60 , C07D213/74 , C07D217/02 , C07D239/42 , C07D215/40
CPC分类号： C07D213/74 , C07D211/26 , C07D211/60 , C07D211/70 , C07D215/40 , C07D217/02 , C07D239/42 , C07D295/10 , C07D295/112 , C07D295/135 , C07D295/14 , C07D295/155 , C07D307/24
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公开(公告)号：EP2038268A2
公开(公告)日：2009-03-25
申请号：EP07766572.7
申请日：2007-06-21
申请人： BIOPROJET
发明人： CAPET, Marc , DANVY, Denis , LEVOIN, Nicolas , BERREBI-BERTRAND, Isabelle , CALMELS, Thierry , ROBERT, Philippe , LECOMTE, Jeanne-Marie , SCHWARTZ, Jean-Charles , LIGNEAU, Xavier
IPC分类号： C07D295/12 , A61K31/495 , A61P25/00 , C07D211/26 , C07D295/14 , C07D295/10 , C07D307/24 , C07D211/70 , C07D211/60 , C07D213/74 , C07D217/02 , C07D239/42 , C07D215/40
CPC分类号： C07D213/74 , C07D211/26 , C07D211/60 , C07D211/70 , C07D215/40 , C07D217/02 , C07D239/42 , C07D295/10 , C07D295/112 , C07D295/135 , C07D295/14 , C07D295/155 , C07D307/24
摘要： The invention relates to compounds of the general formula (I): to the process for preparing them, and to the use thereof as a therapeutic agent.
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公开(公告)号：EP2621916B1
公开(公告)日：2016-02-10
申请号：EP11761383.6
申请日：2011-09-27
申请人： BIOPROJET
发明人： BERREBI-BERTRAND, Isabelle , BILLOT, Xavier , CALMELS, Thierry , CAPET, Marc , DANVY, Denis , KRIEF, Stéphane , LABEEUW, Olivier , LECOMTE, Jeanne-Marie , LEVOIN, Nicolas , LIGNEAU, Xavier , ROBERT, Philippe , SCHWARTZ, Jean-Charles
IPC分类号： C07D401/12 , C07D405/14 , C07D417/12 , C07D417/14 , A61K31/4439 , A61P37/08
CPC分类号： C07D417/14 , A61K31/428 , A61K31/454 , A61K31/4545 , A61K31/496 , A61K31/506 , A61K31/5377 , A61K45/06 , C07D401/04 , C07D401/12 , C07D401/14 , C07D405/14 , C07D417/04 , C07D417/12
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公开(公告)号：EP2170850B1
公开(公告)日：2014-09-24
申请号：EP08761078.8
申请日：2008-06-16
发明人： CAPET, Marc , LEVOIN, Nicolas , BERREBI-BERTRAND, Isabelle , ROBERT, Philippe , SCHWARTZ, Jean-Charles , LECOMTE, Jeanne-Marie , ARADHYE, Jayraj Dilipbhai , PILLAI, Muthukumaran Natarajan , PANCHAL, Bhavesh Mohanbhai , JIVANI, Jignesh Kantilal , SAMANTA, Biswajit c/o SUN PHARMA ADVANCED RESEARCH CENTRE , PAL, Ranjan Kumar c/o SUN PHARMA ADVANCED RESEARCH CENTRE , THENNATI, Rajamannar c/o SUN PHARMA ADVANCED RESEARCH CENTRE
IPC分类号： C07D271/06 , C07D413/10 , C07D413/14 , A61K31/4245 , A61P29/00 , A61P37/06
CPC分类号： C07D413/10 , C07D271/06 , C07D413/14
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公开(公告)号：EP2170850A1
公开(公告)日：2010-04-07
申请号：EP08761078.8
申请日：2008-06-16
发明人： CAPET, Marc , LEVOIN, Nicolas , BERREBI-BERTRAND, Isabelle , ROBERT, Philippe , SCHWARTZ, Jean-Charles , LECOMTE, Jeanne-Marie , ARADHYE, Jayraj Dilipbhai , PILLAI, Muthukumaran Natarajan , PANCHAL, Bhavesh Mohanbhai , JIVANI, Jignesh Kantilal , SAMANTA, Biswajit , PAL, Ranjan Kumar , THENNATI, Rajamannar
IPC分类号： C07D271/06 , C07D413/10 , C07D413/14 , A61K31/4245 , A61P29/00 , A61P37/06
CPC分类号： C07D413/10 , C07D271/06 , C07D413/14
摘要： The present invention relates to new compounds of formula (I) possessing agonistic activity at sphingosine-1 -phosphate (S1 P) receptors, their process of preparation and their use as immunosuppressive agents. The invention is also directed to pharmaceutical compositions containing these compounds and use of these compounds for treatment/prevention of immune mediated diseases and conditions or inflammatory diseases and conditions.
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