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    New pyrazolyl acrylic acid derivatives, useful as systemic fungicides for plant and material protection
    71.
    发明公开
    New pyrazolyl acrylic acid derivatives, useful as systemic fungicides for plant and material protection 失效
    Pyrazolylacrylsäure-Derivate，verwendbar als systemische Fungiziden in Pflanzen- und Materialschutz。

    公开(公告)号：EP0433899A1

    公开(公告)日：1991-06-26

    申请号：EP90124128.1

    申请日：1990-12-13

    申请人： Mitsubishi Chemical Corporation

    发明人： Oda, Masatsugu, Ryoka-dai-ni ,  Sakaki, Toshiro ,  Kikutake, Kuzuhiko

    IPC分类号： C07D231/18 ,  A01N43/56 ,  C07D401/12 ,  C07D417/12 ,  C07D405/12 ,  A01N43/40 ,  A01N43/78 ,  A01N43/08 ,  A01N43/16 ,  A01N43/28

    CPC分类号： C07D401/12 ,  C07D231/18 ,  C07D405/12 ,  C07D417/12

    摘要： A pyrazolyl acrylic acid derivative having plant fungicidal activity of formula (I):
    wherein:

    R 1 and R 2 are independently hydrogen or C 1 - C s alkyl;
    A is a group of the formula:
    wherein X is independently hydrogen; halogen, cyano; nitro; C 1 - C 1 o alkyl, C 2 - C 11 alkenyl, C 1 - C 1 o alkoxy, C 2 - C 11 alkenyloxy, C 2 - C 11 alkynyloxy, C 2 - C 11 alkylcarbonyl or C 2 - C 11 alkylcarbonyloxy optionally substituted with one or more substituents selected from halogen, nitro, cyano, trifluoromethyl and C 1 - C s alkoxy; or C 7 - C 13 arylcarbonyl, C 4 - Cs cycloalkylcarbonyloxy, C 7 - C 13 arylcarbonyloxy, C 6 = C 12 aryl, C 6 - C 12 aryloxy, C 2 - C 13 heteroaryl having 1 - 3 heteroatom(s) selected from oxygen, sulfur, and nitrogen, C 2 -C 13 heteroaryloxy having 1 - 3 heteroatom(s) selected from oxygen, sulfur, and nitrogen, C 7 - C 12 aralkyl or C 7 - C 12 aralkyloxy optionally substitutes with one or more substituents selected from halogen, nitro, cyano, trifluoromethyl, C 1 - C 5 alkyl, and C 1 - Cs alkoxy; m is 1 or 2; and n is a integer of 1 - 5; or two Xs may form a fused ring together with the benzene ring or thiazole ring to which they are attached; and
    B is methoxycarbonyl or cyano.

    摘要翻译： 具有式（I）的植物杀真菌活性的吡唑基丙烯酸衍生物：其中：R 1和R 2独立地为氢或C 1 -C 5烷基; A是下式的基团：其中X独立地是氢; 卤素，氰基; 硝基; C 1 -C 10烷基，C 2 -C 11烯基，C 1 -C 10烷氧基，C 2 -C 11链烯氧基，C 2 -C 11炔氧基，C 2 -C 11烷基羰基或任选被一个或多个选自卤素，硝基，氰基，三氟甲基的取代基取代的C 2 -C 11烷基羰基氧基 和C 1 -C 5烷氧基; -C 13芳基羰基氧基，C 6 = C 12芳基，C 6 -C 12芳氧基，具有1-3个选自氧，硫和氮的杂原子的C 2 -C 13杂芳基，具有1-3个选自氧的杂原子的C 2 -C 13杂芳氧基 ，硫和氮，C7-C12芳烷基或C7-C12芳烷氧基任选地与一个或多个选自卤素，硝基，氰基，三氟甲基，C 1 -C 5烷基和C 1 -C 5烷氧基的取代基取代; m为1或2; n为1〜5的整数。 或两个X可以与它们所连接的苯环或噻唑环一起形成稠环; B是甲氧基羰基或氰基。 H

    Pyrazole amides and insecticide and miticide containing them as active ingredient
    72.
    发明公开
    Pyrazole amides and insecticide and miticide containing them as active ingredient 失效
    吡唑酰胺和二恶嗪。

    公开(公告)号：EP0365925A1

    公开(公告)日：1990-05-02

    申请号：EP89118914.4

    申请日：1989-10-11

    申请人： Mitsubishi Chemical Corporation

    发明人： Okada, Itaru ,  Okui, Shuko ,  Yamaura, Mabuko ,  Takahashi, Yoji

    IPC分类号： C07D231/16 ,  A01N43/56 ,  C07D231/14 ,  C07D231/18 ,  C07D231/54 ,  C07D231/56 ,  C07D401/12 ,  C07D405/12 ,  A01N43/40 ,  A01N43/08

    CPC分类号： C07D231/54 ,  C07D231/14 ,  C07D231/16 ,  C07D231/18 ,  C07D231/56 ,  C07D401/12 ,  C07D405/12

    摘要： Pyrazole amide represented by the following formula (I):
    where R¹ represents alkyl; R² represents hydrogen atom, alkyl, cyclopropyl, alkoxy or alkylcarbonyloxy; X represents hydrogen, halogen, alkyl, alkoxy, haloalkoxy, alkylcarbonyloxy group or hydroxy group; R² and X may combine together to form
    in which R⁹ represents hydrogen or alkyl; one of R³, R⁴ and R⁵ is hydrogen and the others represent independently hydrogen, halogen, alkyl, haloalkyl, cycloalkyl, alkoxy, haloalkoxy, amino, alkylamino, dialkylamino, alkoxy­ carbonylamino, alkylthio, alkylsulfinyl, alkylsulfonyl, alkoxycarbonyl, alkylcarbonyl, nitro, cyano, hydroxymethyl, alkoxyalkyl or alkoxyalkoxyalkyl; R³ and R⁴ may combine together to form
    in which R¹⁰ and R¹¹ represent independently hydrogen or alkyl; one of R⁶ and R⁷ represents hydrogen and the other represents hydrogen, alkyl, alkoxy or halogen; Y represents oxygen, sulfur, sulfinyl, sulfonyl or carbonyl; B represents -CH- or nitrogen; R⁸ represents hydrogen or methyl and Z represents oxygen or sulfur, with the proviso that all of R³, R⁴ and R⁵ are not hydrogen atoms when Y is oxygen and B is -CH-, and an insecticidal and miticidal composition containing the pyrazole amide as an active ingredient are described.
    The pyrazole amide according to the present invention shows excellent insecticidal and miticidal activities.

    摘要翻译： 由下式（I）表示的吡唑酰胺：其中R 1表示烷基的 R 2表示氢原子，烷基，环丙基，烷氧基或烷基羰基氧基; X表示氢，卤素，烷基，烷氧基，卤代烷氧基，烷基羰基氧基或羟基; R 2和X可以结合在一起形成其中R 9表示氢或烷基的 R 3，R 4和R 5之一是氢，其余的代表氢，卤素，烷基，卤代烷基，环烷基，烷氧基，卤代烷氧基，氨基，烷基氨基，二烷基氨基，烷氧羰基氨基，烷硫基，烷基亚磺酰基， 烷基磺酰基，烷氧基羰基，烷基羰基，硝基，氰基，羟甲基，烷氧基烷基或烷氧基烷氧基烷基; R 3和R 4可以结合在一起形成其中R 1，O和R 1独立地代表氢或烷基的 R 6和R 7中的一个表示氢，另一个表示氢，烷基，烷氧基或卤素; Y表示氧，硫，亚磺酰基，磺酰基或羰基; B表示-CH-或氮; R 8表示氢或甲基，Z表示氧或硫，条件是当Y为氧且B为-CH-时，R 3，R 4和R 5全部不为氢原子， 并描述了含有吡唑酰胺作为活性成分的杀虫和杀螨组合物。 根据本发明的吡唑酰胺显示出优异的杀虫和杀螨活性。

    N-phenylpyrazol-4-yl ether derivatives
    73.
    发明公开
    N-phenylpyrazol-4-yl ether derivatives 失效
    N-苯基吡唑-4-基醚。

    公开(公告)号：EP0350311A1

    公开(公告)日：1990-01-10

    申请号：EP89306885.8

    申请日：1989-07-06

    申请人： RHONE-POULENC AGRICULTURE LIMITED

    发明人： Hatton, Leslie Roy ,  Hawkins, David William ,  Pennicard, Richard Glyn ,  Roberts, David Alan

    IPC分类号： C07D231/18 ,  A01N43/56

    CPC分类号： C07D231/18 ,  A01N43/56

    摘要： An N-phenylpyrazol-4-yl ether derivative of the formula:
    wherein R¹ represents halogen, alkyl or alkoxy unsubstituted or substituted by halogen, alkylthio or alkylsulphinyl substituted by one or more halogen atoms, nitro, cyano, or alkylsulphonyl unsubstituted or substituted by halogen and n is 1 to 5, R³ represents hydrogen, halogen, cyano, nitro or alkyl group R² which may be unsubstituted or substituted by halogen, R⁴ represents alkyl, alkenyl or alkynyl which is substituted by halogen, R⁵ represents hydrogen or an amino group wherein R⁶ and R⁷ represent hydrogen, alkyl, formyl or alkanoyl (or R⁶ and R⁷ together form a 5 or 6 membered cyclic imide) which may be unsubstituted or substituted by halogen, or alkoxycarbonyl unsubstituted or substituted by halogen, or R⁵ represents alkoxymethyleneamino unsubstituted or substituted on methylene by alkyl, or represents halogen, or pyrrol-1-yl, pyrazol-1-yl, 1,2,3-triazol-1-yl, 1,2,4-triazol-4-yl, piperidino, pyrrolidino, morpholino or N-alkylpiperazino optionally substituted by alkyl or phenyl and pesticidally acceptable acid addition salts thereof, possess arthropodicidal, nematocidal, anthelmintic and anti-protozoal activity.

    摘要翻译： 硝基，氰基或卤素取代的被卤素，烷硫基或烷基亚磺酰基取代的烷基或烷氧基，其中R 1表示卤素，被卤素取代或被卤素取代的烷基或烷氧基， 未被取代或被卤素取代的烷基磺酰基，n为1至5，R 3表示氢，卤素，氰基，硝基或可以被未取代或被卤素取代的烷基R 2，R 4表示烷基，烯基或 被卤素取代的炔基，R 5表示氢或氨基，其中R 6和R 7表示氢，烷基，甲酰基或烷酰基（或R 6和R 7一起形成5 或6元环酰亚胺），其可以是未取代的或被卤素取代的烷氧基羰基，或被卤素取代的烷氧基羰基，或者R 5表示未取代或未被取代或被亚烷基取代的烷基，或表示卤素或吡咯-1-基，吡唑 -1-基，1,2,3-三唑-1-基，1,2,4-三唑-4-基，哌啶子基，吡咯基 任选被烷基或苯基取代的烟酰基，吗啉代或N-烷基哌嗪基及其农药可接受的酸加成盐，具有节肢动物杀线虫，杀线虫，驱肠虫和抗原生动物活性。

    Method for preparing pyrazolecarboxylic acid and derivatives
    74.
    发明公开
    Method for preparing pyrazolecarboxylic acid and derivatives 失效
    Verfahren zur Herstellung vonPyrazolkarbonsäureund Derivaten。

    公开(公告)号：EP0350176A2

    公开(公告)日：1990-01-10

    申请号：EP89306182.0

    申请日：1989-06-19

    申请人： NISSAN CHEMICAL INDUSTRIES, LIMITED

    发明人： Takigawa, Shinichiro Central Research Institute ,  Shinke, Shuzo c/o Central Research Institute

    IPC分类号： C07D231/16 ,  C07D231/14 ,  C07D231/18 ,  C07D401/04 ,  C07D231/38 ,  C07D231/22 ,  A01N43/56 ,  A01N43/40

    CPC分类号： C07D231/38 ,  C07D231/14 ,  C07D231/16 ,  C07D231/18 ,  C07D231/22 ,  C07D401/04

    摘要： There is disclosed a process for preparing a pyrazolecarbo­xylic acid derivative represented by the formula (II):
    wherein Y and Z each represent a hydrogen atom, a halogen atom, a nitro group, a cyano group, COOR₁, NR₁R₂, CONR₁R₂, SR₁, SO₂NR₁R₂, SO₂R₃, R₃CO, OR₄, CHX₂ or CX₃; A represents a hydrogen atom, an alkyl group having 1 to 4 carbon atoms, a substituted or unsubsti­tuted phenyl group, a substituted or unsubstituted pyridyl group or OR₅; where R₁ and R₂ each represent a hydrogen atom or an alkyl group having 1 to 10 carbon atoms; R₃ represents an alkyl group having 1 to 10 carbon atoms; R₄ represents a hydrogen atom, an alkyl group having 1 to 10 carbon atoms, a substi­tuted or unsubstituted phenyl group, CHF₂, CF₃ or CF₃CH₂; R₅ represents an alkyl group having 1 to 10 carbon atoms; and X represents a halogen atom,
    which comprises oxidizing a pyrazole compound represented by the formula (I):
    wherein Y, Z and A have the same meanings as defined above,
    with an oxygen-containing gas in the presence of a metal compound catalyst.

    摘要翻译： 公开了制备式（II）表示的吡唑羧酸衍生物的方法：其中Y和Z各自表示氢原子，卤素原子，硝基，氰基，COOR1，NR1R2，CONR1R2， SR1，SO2NR1R2，SO2R3，R3CO，OR4，CHX2或CX3; A表示氢原子，具有1至4个碳原子的烷基，取代或未取代的苯基，取代或未取代的吡啶基或OR 5; 其中R 1和R 2各自表示氢原子或具有1至10个碳原子的烷基; R3表示碳原子数1〜10的烷基， R 4表示氢原子，碳原子数1〜10的烷基，取代或未取代的苯基，CHF 2，CF 3或CF 3 CH 2; R5表示碳原子数1〜10的烷基。 X表示卤素原子，其包括在金属存在下用含氧气体氧化由式（I）表示的吡唑化合物：其中Y，Z和A具有与上述相同的含义。 复合催化剂。

    Herbicidal pyrazole derivatives
    76.
    发明公开
    Herbicidal pyrazole derivatives 失效
    除草剂吡唑衍生物

    公开(公告)号：EP0138527A3

    公开(公告)日：1987-06-03

    申请号：EP84306807

    申请日：1984-10-05

    申请人： NIPPON KAYAKU KABUSHIKI KAISHA

    发明人： Yanagi, Mikio ,  Yamada, Osamu ,  Futatsuya, Fumio ,  Shida, Atsuhiko

    IPC分类号： C07D231/56 ,  C07D231/54 ,  C07D231/16 ,  C07D231/18 ,  A01N43/56

    CPC分类号： C07D231/56 ,  A01N43/56 ,  C07D231/16 ,  C07D231/18 ,  C07D231/22 ,  C07D231/54

    摘要： Pyrazole derivatives, for use as herbicides, have the formula (I):
    wherein
    R 1 represents hydrogen, halogen or methyl; R 2 represents hydrogen, halogen, nitro, methyl, cyano, carboxy, (C 1 to C 8 )-alkoxy or (C 1 to C 4 )-alkoxycarbonyl; R 3 represents hydroxy, amino, (C 3 or C 4 )-alkenyloxy, (C 3 or C 4 )-alkynyloxy, (C 1 to C4)-alkoxy-(C 1 to C 4 )-alkoxy, (C 1 to C 4 )-alkylthio, (C 3 or C 4 )-alkenylamino, (C 1 to C 4 )-alkylsulfonylamino, (C 1 or C 2 )-alkoxy-(C 1 or C 2 )-alkylamino, -O-N=C-(CH 3 ) 2 , anilino, benzylamino, morpholino, (C 1 to C 6 )-alkoxy unsubstituted or substituted by (C 1 to C 4 )-alkoxycarbonyl, (C 1 to C 4 )-mono- or di-alkylamino group in which the or each alkyl group is unsubstituted or substituted by hydroxy or carboxy, or -OM wherein M represents an alkali metal, alkaline earth metal, ammonium or (C 1 to C 4 )-alkylammonium; R 4 represents halogen, methyl, (C 1 to C 4 )-alkoxy, -S(O) m -R 5 wherein m is 0, 1 or 2 and R 5 represents (C 1 to C 4 )-alkyl; X represents hydrogen, halogen, (C 1 to C 4 )-alkyl, (C 1 to C 4 )-alkylthio or (Ci to C 4 )-alkylsulfonyl; and Y represents (C 1 to C 4 )-alkyl or X and Y taken together with the atoms to which they are attached form a cyclopentyl or cyclohexyl ring unsubstituted or substituted with one or more methyl group.

    摘要翻译： 用作除草剂的吡唑衍生物具有式（I）：其中R 1表示氢，卤素或甲基的; R 2表示氢，卤素，硝基，甲基，氰基，羧基，（C 1至C 8） - 烷氧基或（C 1至C 4） - 烷氧基羰基; R 3表示羟基，氨基，（C 3或C 4） - 炔氧基，C 3或C 4） - 炔氧基，（C 1 -C 4） - 烷氧基 - （C 1至C 4） - 烷氧基，（C 1至C 4） - 烷硫基，（C 3 或（C 1 -C 4） - 烷基磺酰基氨基，（C 1或C 2） - 烷氧基 - （C 1或C 2） - 烷基氨基，-ON = C-（CH 3）2，苯胺基，苄基氨基，吗啉代，（C 1至C 6） ） - 未取代或被（C1-C4） - 烷氧基羰基，（C1-C4） - 单 - 或二 - 烷基氨基取代的烷氧基，其中每个烷基未被取代或被羟基或羧基取代，或-OM，其中M表示 碱金属，碱土金属，铵或（C1至C4） - 烷基铵; R 4表示卤素，甲基，（C 1至C 4） - 烷氧基，-S（O）m -R 5，其中m为0,1或2，R 5表示（C 1至C 4） - 烷基; X表示氢，卤素，（C1-C4） - 烷基，（C1-C4） - 烷硫基或（C1-C4） - 烷基磺酰基; Y表示（C1-C4） - 烷基或X和Y与它们所连接的原子一起形成未被取代或被一个或多个甲基取代的环戊基或环己基环。