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1.3,4-dihydro-3-amino-2H-1-benzopyrane and -benzothiopyrane derivatives as dopamine-beta-hydroxylase Inhibitors and methods of their preparation 有权
标题翻译: 3,4-二氢-3-氨基-2H-1-苯并吡喃和-benzothiopyran衍生物作为多巴胺-β-羟化酶抑制剂和它们的制备方法公开(公告)号:EP1908759B1
公开(公告)日:2012-03-21
申请号:EP07076123.4
申请日:2003-10-10
发明人: Learmonth, David Alexander , Soares da Silva, Patricio Manuel Vieira Araujo , Beliaev, Alexander
IPC分类号: C07D405/04 , A61K31/4164 , A61P43/00 , C07D409/04 , C07D233/84 , C07D311/58 , C07D335/06 , C07F7/18
CPC分类号: C07D405/04 , C07D233/84 , C07D409/04 , Y02P20/55
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2.Silyl-protected hydroxymethyl-carbamoylalkyl-ketones as intermediates in the preparation of dopamine-beta-hydroxylase inhibitors 有权
标题翻译: 甲硅烷基保护的羟甲基烷基氨基甲酮作为中间体在生产多巴胺β-羟化酶抑制剂的公开(公告)号:EP1914233B8
公开(公告)日:2011-04-13
申请号:EP07076122.6
申请日:2003-10-10
发明人: Learmonth, David Alexander , Soares Da Silva, Patricio Manuel Vieira Araujo , Beliaev, Alexander
IPC分类号: C07D405/04 , A61K31/4164 , A61P43/00 , C07D409/04 , C07D233/84 , C07F7/18 , C07D311/58
CPC分类号: C07D405/04 , C07D233/84 , C07D409/04 , Y02P20/55
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3.Imidazole deriviatives and their use as peripherally-selective inhibitors of dopamine-beta-hydroxylase 有权
标题翻译: 咪唑衍生物及其作为多巴胺β-羟化酶的外周选择性抑制剂的用途公开(公告)号:EP1408038B1
公开(公告)日:2008-08-06
申请号:EP03256420.5
申请日:2003-10-10
发明人: Learmonth, David Alexander , Soares Da Silva, Patricio Manuel Viera Araujo , Beliaev, Alexander
IPC分类号: C07D405/04 , A61K31/4164 , A61P43/00 , C07D409/04 , C07D233/84
CPC分类号: C07D405/04 , C07D233/84 , C07D409/04 , Y02P20/55
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4.Method of preparation of 3-(1,3-Dihydroimidazole-2-thione-1-yl)-chromanes and thiochromanes as dopamine-beta-hydroxylase inhibitors 有权
标题翻译: 制备作为多巴胺-β-羟化酶抑制剂的3-(1,3-二氢咪唑-2-硫酮-1-基) - 色满和硫代色菁的方法公开(公告)号:EP1911757B8
公开(公告)日:2011-05-25
申请号:EP07076124.2
申请日:2003-10-10
发明人: Learmonth, David Alexander , Soares da Silva, Patricio Manuel Vieira Araujo , Beliaev, Alexander
IPC分类号: C07D405/04 , A61K31/4164 , A61P43/00 , C07D409/04 , C07D233/84 , C07D311/58 , C07D335/06 , C07F7/18
CPC分类号: C07D405/04 , C07D233/84 , C07D409/04 , Y02P20/55
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5.Chromane and thiochromane-3-yl-1,3-dihydroimidazoles as inhibitors of dopamine-beta-hydroxylase and methods of their preparation 有权
标题翻译: 苯并二氢吡喃和二氢苯并噻喃-3-基-1,3-二氢咪唑它们的制备的多巴胺-β-羟化酶的抑制剂和方法公开(公告)号:EP1908760B1
公开(公告)日:2011-04-13
申请号:EP07076125.9
申请日:2003-10-10
发明人: Learmonth, David Alexander , Soares da Silva, Patricio Manuel Vieira Araujo , Beliaev, Alexander
IPC分类号: C07D405/04 , A61K31/4164 , A61P43/00 , C07D409/04 , C07D233/84 , C07D311/58 , C07D335/06 , C07F7/18
CPC分类号: C07D405/04 , C07D233/84 , C07D409/04 , Y02P20/55
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