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    2-HETEROARYLCARBONSÄUREAMIDE
    6.
    发明公开
    2-HETEROARYLCARBONSÄUREAMIDE 有权

    公开(公告)号：EP1515967A1

    公开(公告)日：2005-03-23

    申请号：EP03732517.2

    申请日：2003-06-02

    申请人： Bayer HealthCare AG

    发明人： LUITHLE, Joachim ,  BÖSS, Frank-Gerhard ,  ERB, Christina ,  HAFNER, Frank-Thorsten ,  SCHNIZLER, Katrin ,  FLESSNER, Timo ,  VAN KAMPEN, Marja ,  VAN DER STAAY, Franz-Josef

    IPC分类号： C07D453/02 ,  A61K31/439 ,  A61P25/00

    CPC分类号： C07D453/02

    摘要： The invention relates to the novel 2-heteroaryl carboxamides according to formula (I), wherein R represents 1-aza-bicyclo [2.2.2]oct-3-yl, which is optionally replaced via the nitrogen atom by a group selected from the family C1-C4 alkyl, benzyl and oxy, A represents oxygen or sulfur, the ring B represents benzo or pyrido that are optionally replaced by the groups from the family of halogen, cyano, formyl, trifluoromethyl, trifluoromethoxy, nitro, amino, C1-C6 alkyl and C1-C6 alkoxy, E represents C=C, aryl and heteroaryl, wherein aryl and heteroaryl may be replaced by groups from the family of halogen, cyano, trifluoromethyl, trifluoromethoxy, nitro, amino, C1-C6 alkoxy and C1-C6 alkyl, and to the solvents, salts or solvents of salts of said compounds. The invention also relates to the use of said compounds in the production of drugs for the treatment and/or the prophylaxis of diseases and for improving perception, power of concentration, learning power and/or retentiveness of memory.

    2-HETEROARYLCARBONSÄUREAMIDE
    8.
    发明授权
    2-HETEROARYLCARBONSÄUREAMIDE 有权
    2 - 杂芳基羧酰胺

    公开(公告)号：EP1515967B1

    公开(公告)日：2006-11-02

    申请号：EP03732517.2

    申请日：2003-06-02

    申请人： Bayer HealthCare AG

    发明人： LUITHLE, Joachim ,  BÖSS, Frank-Gerhard ,  ERB, Christina ,  HAFNER, Frank-Thorsten ,  SCHNIZLER, Katrin ,  FLESSNER, Timo ,  VAN KAMPEN, Marja ,  VAN DER STAAY, Franz-Josef

    IPC分类号： C07D453/02 ,  A61K31/439 ,  A61P25/00

    CPC分类号： C07D453/02

    摘要： The invention relates to the novel 2-heteroaryl carboxamides according to formula (I), wherein R represents 1-aza-bicyclo [2.2.2]oct-3-yl, which is optionally replaced via the nitrogen atom by a group selected from the family C1-C4 alkyl, benzyl and oxy, A represents oxygen or sulfur, the ring B represents benzo or pyrido that are optionally replaced by the groups from the family of halogen, cyano, formyl, trifluoromethyl, trifluoromethoxy, nitro, amino, C1-C6 alkyl and C1-C6 alkoxy, E represents C=C, aryl and heteroaryl, wherein aryl and heteroaryl may be replaced by groups from the family of halogen, cyano, trifluoromethyl, trifluoromethoxy, nitro, amino, C1-C6 alkoxy and C1-C6 alkyl, and to the solvents, salts or solvents of salts of said compounds. The invention also relates to the use of said compounds in the production of drugs for the treatment and/or the prophylaxis of diseases and for improving perception, power of concentration, learning power and/or retentiveness of memory.