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1.发明公开
公开(公告)号：EP4458807A1
公开(公告)日：2024-11-06
申请号：EP22916030.4
申请日：2022-12-26
发明人： HARA, Kenji , SUGIHARA, Kousuke , MASUDA, Tsuyoshi , YORIFUJI, Nobuyuki , TANAKA, Koji , FUJII, Kazuki , FUKATSU, Kosuke , TANAKA, Ryosuke
IPC分类号： C07C235/82 , A01N37/22 , A01N37/24 , A01N43/10 , A01N43/30 , A01N43/40 , A01N43/50 , A01N43/78 , A01N47/02 , A01P5/00 , A01P7/04 , A61K31/167 , A61K31/36 , A61K31/381 , A61K31/426 , A61K31/44 , A61K31/4402 , A61K31/505 , A61P33/14 , C07C317/40
摘要： In the production of crops in agriculture, horticulture and the like, the damage caused by insect pests and the like is still large, and the development of a novel pest control agent is desired in view of the factors such as the development of insect pests that are resistant to existing drugs, and the like.
The present invention provides compounds represented by the formula (1)
wherein X and Y are oxygen atoms or sulfur atoms, Z is a hydroxyl group or the like, R 1 and R 2 are hydrogen atoms and the like, R 3 is a substituted phenyl group or the like, and Q is a substituted phenyl group or the like, or salts thereof, pest control agents containing the compounds as active ingredients, and methods for use thereof.-
2.发明公开
公开(公告)号：EP4458817A1
公开(公告)日：2024-11-06
申请号：EP22916032.0
申请日：2022-12-26
发明人： HARA, Kenji , SUGIHARA, Kousuke , MASUDA, Tsuyoshi , TANAKA, Koji , YASUKOUCHI, Eiji , FUJII, Kazuki , FUKATSU, Kosuke , TANAKA, Ryosuke
IPC分类号： C07D309/32 , C07D405/04 , C07D405/12 , C07D407/04 , C07D407/12 , C07D409/12 , C07D491/107 , A01P5/00 , A01P7/04 , C07D311/96 , A01N43/10 , A01N43/16 , A01N43/40 , A01N43/56 , A01N47/02 , A01N47/16
摘要： In the production of crops in agriculture, horticulture and the like, the damage caused by insect pests and the like is still large, and the development of a novel pest control agent is desired in view of the factors such as the development of insect pests that are resistant to existing drugs, and the like.
The present invention provides compounds represented by the formula (1)
wherein X and Y are oxygen atoms or sulfur atoms, Z is a hydroxyl group or the like, R 1 is a hydrogen atom or the like, R 2 , R 3 and R 4 are hydrogen atoms and the like, and R 5 and Q are substituted phenyl groups and the like, or salts thereof, pest control agents containing the compounds as active ingredients, and methods for use thereof.-
3.发明公开
公开(公告)号：EP4458809A1
公开(公告)日：2024-11-06
申请号：EP22916029.6
申请日：2022-12-26
发明人： HARA, Kenji , SUGIHARA, Kousuke , MASUDA, Tsuyoshi , YASUKOUCHI, Eiji , TANAKA, Koji , FUJII, Kazuki , FUKATSU, Kosuke , TANAKA, Ryosuke
IPC分类号： C07D211/90 , A01N43/40 , A01N43/42 , A01N43/54 , A01N43/56 , A01N43/58 , A01N43/60 , A01N43/653 , A01N43/66 , A01N43/713 , A01N43/78 , A01N43/80 , A01N43/824 , A01N43/832 , A01N43/84 , A01N47/02 , A01P5/00 , A01P7/02 , A01P7/04 , A01P9/00 , A61K31/45
摘要： In the production of crops in agriculture, horticulture and the like, the damage caused by insect pests and the like is still large, and the development of a novel pest control agent is desired in view of the factors such as the development of insect pests that are resistant to existing drugs, and the like.
The present invention provides compounds represented by the formula (1)
wherein X and Y are oxygen atoms or sulfur atoms, Z is a hydroxyl group or the like, R 1 is an alkyl group or the like, R 2 and R 4 are substituted phenyl groups and the like, R 3 , R 5 and R 6 are hydrogen atoms and the like, and R 7 is a substituted phenyl group or the like, or salts thereof, pest control agents containing the compounds as active ingredients, and methods for use thereof.-
4.发明公开
公开(公告)号：EP4458811A1
公开(公告)日：2024-11-06
申请号：EP22916028.8
申请日：2022-12-26
发明人： ANDO, Akihiro , YONEMURA, Ikki , TANAKA, Koji , YAMADA, Takayuki , TANAKA, Ryosuke , FUJITA, Naoya , YOKOI, Taiki , YAMADA, Hiroto , MATSUI, Shunsuke , OIKAWA, Hinoki
IPC分类号： C07D237/24 , A01N43/58 , A01N43/60 , A01N43/76 , A01N43/78 , A01N43/80 , A01N43/836 , A01N43/90 , A01N47/02 , A01N47/16 , A01N47/38 , A01N55/10 , A01P5/00 , A01P7/02 , A01P7/04 , A01P9/00 , C07D401/04 , C07D401/12 , C07D401/14 , C07D403/04
摘要： For example, in agricultural and horticultural crop production, pests, etc. still cause heavy damage, and there is a demand for the development of novel agricultural and horticultural insecticidal agents due to factors such as the emergence of pests resistant to existing drugs. The present invention has found that a compound represented by the general formula (1):
wherein X and Y each represent an oxygen atom or a sulfur atom, Z represents a hydroxyl group or the like, R 1 represents an alkoxycarbonyl group or the like, R 2 represents a substituted phenyl group or the like, R 3 represents a hydrogen atom or the like, and R 4 represents a substituted phenyl group or the like, or a salt thereof exhibits a high insecticidal effect on pests, etc. in the agricultural and horticultural field, and provides an agricultural and horticultural insecticidal agent comprising the same as an active ingredient and a method for using the same.-
公开(公告)号：EP4174057A1
公开(公告)日：2023-05-03
申请号：EP21828251.5
申请日：2021-06-24
IPC分类号： C07D237/24 , A01P7/04 , A01M1/20 , C07D401/04 , A01N43/50
摘要： Crop production in agriculture, horticulture, and the like has still been significantly damaged by pests and the like, and pests that are resistant to existing drugs have appeared. Due to such concerns, it is desired to develop novel insecticidal agents and acaricides.
The present invention has found that a compound represented by general formula (1):
wherein X and Y represent an oxygen atom or a sulfur atom, R 1 represents a hydrogen atom or the like, R 2 represents a substituted phenyl group or the like, R 3 represents a hydrogen atom or the like, and R 4 represents a phenyl group or the like, or a salt thereof has a high insecticidal effect on pests in agriculture and horticulture, and the like. The present invention provides an agricultural and horticultural insecticidal agent containing the compound or a salt thereof as an active ingredient, and a method of use thereof.-
公开(公告)号：EP2891489B1
公开(公告)日：2018-01-10
申请号：EP13832194.8
申请日：2013-08-29
发明人： KITA, Kiyoshi , SUWA, Akiyuki , ODA, Masatsugu , TANAKA, Koji
IPC分类号： A61K31/166 , A61K31/415 , A61K31/44 , A61P33/00 , C07D213/74 , C07D231/16 , C07D231/18 , C07D231/12 , C07D231/20 , C07D213/643 , C07D213/64 , C07D213/61 , C07C317/32 , C07C323/62 , C07C235/60 , C07D401/04
CPC分类号： C07D401/04 , A61K31/166 , A61K31/415 , A61K31/44 , C07C233/69 , C07C235/46 , C07C235/60 , C07C317/32 , C07C323/42 , C07C323/62 , C07D213/56 , C07D213/61 , C07D213/643 , C07D213/74 , C07D231/12 , C07D231/16 , C07D231/18 , C07D231/20
摘要： An object of the present invention is to provide a novel endoparasite control agent as a parasiticide, an antiprotozoal or the like. Provided is an endoparasite control agent comprising a carboxamide derivative represented by the general formula (I): or a salt thereof as an active ingredient.
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7.发明公开N-2-(HETERO)ARYLETHYLCARBOXAMIDE DERIVATIVE, AND PEST-CONTROLLING AGENT COMPRISING THE SAME 审中-公开N-2-（HETERO）芳基乙酰胺衍生物和含有该化合物的防治虫剂
公开(公告)号：EP1997800A1
公开(公告)日：2008-12-03
申请号：EP07739169.6
申请日：2007-03-20
发明人： ODA, Masatsugu , MATSUZAKI, Yoshihiro , TANAKA, Koji , TAKIZAWA, Eiji , HASEBE, Motohiro , KUROKI, Nobutaka , SUWA, Akiyuki , OSHIMA, Kenji
IPC分类号： C07C233/66 , A01N37/18 , A01N43/08 , A01N43/10 , A01N43/32 , A01N43/40 , A01N43/56 , A01N43/60 , A01N43/78 , A01N47/02 , A01P3/00 , C07C233/65 , C07C233/73 , C07D213/82 , C07D231/14 , C07D241/24 , C07D277/20 , C07D277/56 , C07D307/56 , C07D327/06 , C07D333/38
CPC分类号： C07D241/24 , A01N37/18 , A01N37/40 , A01N43/08 , A01N43/10 , A01N43/32 , A01N43/40 , A01N43/56 , A01N43/60 , A01N43/78 , A01N47/02 , C07D213/82 , C07D231/14 , C07D277/20 , C07D277/56 , C07D307/56 , C07D327/06 , C07D333/38
摘要： An N-2-(hetero)arylethylcarboxamide derivative represented by the formula (I)
wherein R 1 and R 2 are each independently a hydrogen atom etc., R 3 and R 4 are each independently a hydrogen atom etc., each Y is independently a halogen atom; a (C 1 -C 6 )alkyl group optionally substituted by halogen atom(s) etc., n is an integer of 1 to 5, A is a specific substituted cyclic group, E is C-H; C-Y (Y is as defined above); or a nitrogen atom, a salt thereof, and a pest controlling agent containing the derivative or salt as an active ingredient show superior performance as compared to the prior art technique, and are useful particularly as plant disease controlling agents or nematocides having a broad control spectrum at a low dose.摘要翻译： 式（I）表示的N-2-（杂）芳基乙基甲酰胺衍生物，其中R1和R2各自独立地为氢原子等，R3和R4各自独立地为氢原子等，每个Y独立地为卤素原子; 任选被卤素原子等取代的（C 1 -C 6）烷基，n是1至5的整数，A是特定取代的环状基团，E是C-H; C-Y（Y如上所定义）; 或氮原子，其盐和含有该衍生物或盐作为活性成分的害虫防治剂与现有技术相比表现出优异的性能，并且特别用作植物病害防治剂或具有广谱防治谱的杀线虫剂 低剂量。
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8.发明公开ANTICANCER AGENT COMPRISING AMINOACETONITRILE COMPOUND AS ACTIVE INGREDIENT 审中-公开细菌对癌AMINOACETONITRILVERBINDUNG为活动
公开(公告)号：EP3043791A1
公开(公告)日：2016-07-20
申请号：EP14781682.1
申请日：2014-09-12
发明人： ANDOH, Nobuharu , SANPEI, Osamu , TOGA, Tetsuo , MORRIS, David Lawson , ASTON, Roger , TANAKA, Koji , HINO, Tomokazu
IPC分类号： A61K31/277 , A61K31/415 , A61P35/00
CPC分类号： A61K31/277 , A61K31/341 , A61K31/381 , A61K31/415 , A61K31/4196 , A61K31/42 , A61K31/421 , A61K31/4245 , A61K31/426 , A61K31/433 , A61K31/437 , A61K31/44 , A61K31/4965 , A61K31/505 , A61K31/5377 , A61K31/5383
摘要： wherein R1 is a hydrogen atom, an alkyl group and the like, R2, R3, and R4 are the same or different and each is a hydrogen atom, an alkyl group and the like, R5 and R6 are the same or different and each is a hydrogen atom, a halogen atom and the like, m is 0 or 1, R is a halogen atom, a cyano group, a nitro group, a phenyl group optionally substituted by an alkyl group and the like, an alkyl group and the like, Ar1 is a phenyl group, a naphthyl group, a pyridyl group, a pyrazolyl group, or the like, each of which is optionally substituted by a halogen atom, a cyano group, a nitro group, alkyl group and the like, and W is —O—, —S—, —SO2—, or —N(R7)—wherein R7 is a hydrogen atom, a (C1-C6) alkyl group and the like, or a pharmacologically acceptable salt thereof.
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公开(公告)号：EP2891492A1
公开(公告)日：2015-07-08
申请号：EP13833021.2
申请日：2013-08-29
发明人： KITA, Kiyoshi , SUWA, Akiyuki , ODA, Masatsugu , TANAKA, Koji
IPC分类号： A61K31/44 , A61K31/381 , A61K31/39 , A61K31/415 , A61K31/426 , A61K31/4965 , A61K31/505 , A61P33/00
CPC分类号： C07D401/12 , A61K31/381 , A61K31/39 , A61K31/415 , A61K31/426 , A61K31/44 , A61K31/4439 , A61K31/444 , A61K31/4965 , A61K31/497 , A61K31/505 , C07D213/82 , C07D231/14 , C07D239/28 , C07D241/24 , C07D277/56 , C07D307/68 , C07D327/06 , C07D333/38 , C07D401/00
摘要： An object of the present invention is to provide a novel endoparasite control agent as a parasiticide, an antiprotozoal or the like. Provided is an endoparasite control agent comprising a carboxamide derivative represented by the general formula (I):
(wherein Het represents a 5- or 6-membered heterocyclic group), or
a salt thereof as an active ingredient.摘要翻译： 本发明的一个目的是提供一种新的内寄生虫防治剂作为杀寄生虫剂，抗原生动物剂等。 本发明提供一种含有通式（I）所示的羧酰胺衍生物或其盐作为有效成分的内寄生物防除剂：（式中，Het表示5或6元杂环基）。
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公开(公告)号：EP2891489A1
公开(公告)日：2015-07-08
申请号：EP13832194.8
申请日：2013-08-29
发明人： KITA, Kiyoshi , SUWA, Akiyuki , ODA, Masatsugu , TANAKA, Koji
IPC分类号： A61K31/166 , A61K31/415 , A61K31/44 , A61P33/00
CPC分类号： C07D401/04 , A61K31/166 , A61K31/415 , A61K31/44 , C07C233/69 , C07C235/46 , C07C235/60 , C07C317/32 , C07C323/42 , C07C323/62 , C07D213/56 , C07D213/61 , C07D213/643 , C07D213/74 , C07D231/12 , C07D231/16 , C07D231/18 , C07D231/20
摘要： An object of the present invention is to provide a novel endoparasite control agent as a parasiticide, an antiprotozoal or the like. Provided is an endoparasite control agent comprising a carboxamide derivative represented by the general formula (I):
or
a salt thereof as an active ingredient.摘要翻译： 本发明的一个目的是提供一种新的内寄生虫防治剂作为杀寄生虫剂，抗原生动物剂等。 提供了一种内寄生物防治剂，其包含由通式（I）表示的甲酰胺衍生物或其盐作为活性成分。
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