Novel cyclobutane derivative
    5.
    发明公开
    Novel cyclobutane derivative 失效
    Cyclobutanderivate。

    公开(公告)号:EP0444597A1

    公开(公告)日:1991-09-04

    申请号:EP91102806.6

    申请日:1991-02-26

    CPC分类号: C07D263/26

    摘要: This invention relates to a cyclobutane derivative represented by the following general formula (I):

    wherein X represents a group represented by the formula

    (wherein R¹ represents an alkyl group having 1 to 5 carbon atoms or an aryl-substituted alkyl group wherein the alkyl group has 1 to 5 carbon atoms;
    R² represents a hydrogen atom, an alkyl group having 1 to 5 carbon atoms, a protected hydroxyalkyl group having 1 to 5 carbon atoms or a protected carboxyl group; and
    R³ and R⁴ independently represent each a hydrogen atom, an alkyl group having 1 to 5 carbon atoms, a protected hydroxyalkyl group having 1 to 5 carbon atoms, an alkoxy group having 1 to 5 carbon atoms or an aryl-substituted alkoxy group wherein the alkoxy group has 1 to 5 carbon atoms; or
    alternately R³ and R⁴ are bound together to thereby form a 3- to 30-membered carbocyclic or heterocyclic ring);
    A represents an optionally substituted polymethylene group having 2 to 5 carbon atoms;
    Y represents an oxygen or a sulfur atom; and
    Z represents an optionally substituted methylene group or an oxygen or a sulfur atom;
    which is expected to be useful as reagents, drugs, agricultural chemicals and perfumes as well as an intermediate for the preparation thereof.

    摘要翻译: 本发明涉及由以下通式(I)表示的环丁烷衍生物:其中X表示由式CHEM表示的基团(其中R 1表示具有1至5个碳原子的烷基或 芳基取代的烷基,其中烷基具有1至5个碳原子; R 2表示氢原子,具有1至5个碳原子的烷基,被保护的具有1至5个碳原子的羟烷基或被保护的羧基 R 3和R 4各自独立地表示氢原子,碳原子数1〜5的烷基,碳原子数1〜5的保护羟烷基,碳原子数1〜5的烷氧基或碳原子数1〜5的烷氧基 芳基取代的烷氧基,其中烷氧基具有1至5个碳原子;或者R 3和R 4交替结合在一起形成3-至30元碳环或杂环); A表示任选取代的具有2至5个碳原子的多亚甲基; Y表示氧或硫原子; Z表示任选取代的亚甲基或氧或硫原子; 预期其可用作试剂,药物,农药和香料以及其制备的中间体。

    BENZAMIDE DERIVATIVES, INSECTICIDES FOR AGRICULTURAL AND HORTICULTURAL USE AND USAGE THEREOF
    9.
    发明公开
    BENZAMIDE DERIVATIVES, INSECTICIDES FOR AGRICULTURAL AND HORTICULTURAL USE AND USAGE THEREOF 有权
    苯甲酰胺衍生物,杀虫剂FOR USE IN农业和花园区及其用途

    公开(公告)号:EP1195375A1

    公开(公告)日:2002-04-10

    申请号:EP00940822.0

    申请日:2000-06-23

    摘要: Benzamide derivatives represented by the general formula (I):
    and insecticides for agricultural and horticultural use and usage thereof, wherein Z 1 is O or S; R is H, (substituted) alkyl, or alkoxycarbonyl; X is halogeno, cyano, nitro, C 3 -C 6 (halo)cycloalkyl, (substituted) phenyl, a (substituted) heterocyclic group, or -A 1 -R 1 [wherein A 1 is -O-, -S-, -SO-, -SO2-, -C(=O)-, or -C(=NOR2)- (wherein R 2 is H, C 1 -C 6 (halo)alkyl, (substituted) phenylated C 1 -C 4 alkyl, or the like); and R 1 is halogeno, C 3 -C 6 cycloalkyl, C 3 -C 6 halocycloalkenyl, (substituted) phenyl, or the like]; n is 0 to 4; Y is halogeno, cyano, nitro, C 3 -C 6 halocycloalkyl, (substituted) phenyl, or the like; m is 1 to 5; Q is a heterocycle such as oxazoline; and B 1 to B 4 are each CH or N.

    摘要翻译: 由通式(I)表示的苯甲酰胺衍生物:和杀虫剂用于农业和园艺用途和用途,worinž<1>是O或S; R为H,(取代的)烷基,或烷氧羰; X是卤素,氰基,硝基,C3-C6(卤代)环烷基,(取代的)苯基,(取代的)杂环基,或-A <1> -R <1> a其中A <1>是-O - , - S-,-SO - , - SO 2 - ,-C(= O) - ,或-C(= NOR2) - (其中R <2> H,C1-C6(卤代)烷基,(取代的)苯基化C1 1 -C 4烷基,或类似物); 和R <1>是卤素,C3-C6环烷基,C3-C6卤代环烯基,(substituiertem)苯基,或likeÜ; n是0至4; Y为卤素,氰基,硝基,C3-C6卤代环烷基,(取代的)苯基,或类似物; m是1至5; Q是杂周期:如恶唑啉; 和B <1>到B <4>各自为CH或N.