公开(公告)号：US09162966B2

公开(公告)日：2015-10-20

申请号：US14213240

申请日：2014-03-14

Applicant: KUREHA CORPORATION

Inventor： Nobuyuki Araki ,  Toru Yamazaki ,  Nobuyuki Kusano ,  Eiyu Imai ,  Hisashi Kanno ,  Masaru Mori ,  Taiji Miyake

IPC: C07C61/06 ,  C07C67/31 ,  C07D405/06 ,  A01N37/10 ,  A01N43/50 ,  A01N43/653 ,  C07C201/12

CPC classification number: C07C67/31 ,  A01N37/10 ,  A01N43/50 ,  A01N43/653 ,  C07C201/12 ,  C07C2601/08 ,  C07D405/06

Abstract: A method of producing an azole derivative according to the invention represented by Formula (XI) wherein R1 denotes a C1-C6 alkyl group, a C2-C6 alkenyl group or a C2-C6 alkynyl group; R2 denotes a C1-C4 alkyl group; each Y denotes a halogen atom, a C1-C4 alkyl group, a C1-C4 haloalkyl group, a C1-C4 alkoxy group, a C1-C4 haloalkoxy group, a phenyl group, a cyano group or a nitro group; and m denotes 0 to 5; when m is 2 or more, each Y may be the same or different. As a result, an azole derivative contained as an active ingredient in an agro-horticultural agent having an excellent controlling effect on diseases can be provided.

Abstract translation: 制备式（Ⅺ）表示的本发明唑类衍生物的方法，其中R1表示C1-C6烷基，C2-C6链烯基或C2-C6炔基; R2表示C1-C4烷基; 每个Y表示卤素原子，C1-C4烷基，C1-C4卤代烷基，C1-C4烷氧基，C1-C4卤代烷氧基，苯基，氰基或硝基; m表示0〜5; 当m为2以上时，Y可以相同也可以不同。 结果，可以提供在对疾病具有优异控制作用的农业园艺剂中作为活性成分含有的唑衍生物。

公开(公告)号：US09145351B2

公开(公告)日：2015-09-29

申请号：US14213043

申请日：2014-03-14

Applicant: KUREHA CORPORATION

Inventor： Nobuyuki Araki ,  Toru Yamazaki ,  Nobuyuki Kusano ,  Eiyu Imai ,  Hisashi Kanno ,  Masaru Mori ,  Taiji Miyake

IPC: C07C61/06 ,  C07C67/31 ,  C07D405/06 ,  A01N37/10 ,  A01N43/50 ,  A01N43/653 ,  C07C201/12

CPC classification number: C07C67/31 ,  A01N37/10 ,  A01N43/50 ,  A01N43/653 ,  C07C201/12 ,  C07C2601/08 ,  C07D405/06

Abstract: An azole derivative according to the invention is represented by Formula (XI) wherein R1 denotes a C1-C6 alkyl group, a C2-C6 alkenyl group or a C2-C6 alkynyl group; R2 denotes a C1-C4 alkyl group; each Y denotes a halogen atom, a C1-C4 alkyl group, a C1-C4 haloalkyl group, a C1-C4 alkoxy group, a C1-C4 haloalkoxy group, a phenyl group, a cyano group or a nitro group; and m denotes 0 to 5; when m is 2 or more, each Y may be the same or different. As a result, an azole derivative contained as an active ingredient in an agro-horticultural agent having an excellent controlling effect on diseases can be provided.

Abstract translation: 根据本发明的唑衍​​生物由式（XI）表示，其中R1表示C1-C6烷基，C2-C6烯基或C2-C6炔基; R2表示C1-C4烷基; 每个Y表示卤素原子，C1-C4烷基，C1-C4卤代烷基，C1-C4烷氧基，C1-C4卤代烷氧基，苯基，氰基或硝基; m表示0〜5; 当m为2以上时，Y可以相同也可以不同。 结果，可以提供在对疾病具有优异控制作用的农业园艺剂中作为活性成分含有的唑衍生物。

公开(公告)号：US09440933B2

公开(公告)日：2016-09-13

申请号：US14691279

申请日：2015-04-20

Applicant: KUREHA CORPORATION

Inventor： Nobuyuki Araki ,  Taiji Miyake ,  Eiyu Imai ,  Emiko Obata

IPC: C07D249/08 ,  C07D249/12 ,  C07D233/56 ,  A01N43/653 ,  C07D233/60 ,  C07D405/06 ,  A01N43/50 ,  A01N43/80 ,  C07D405/04

CPC classification number: C07D249/12 ,  A01N43/50 ,  A01N43/653 ,  A01N43/80 ,  C07D233/56 ,  C07D233/60 ,  C07D249/08 ,  C07D405/04 ,  C07D405/06 ,  A01N25/04 ,  A01N25/28

Abstract: Provided is an azole derivative superior in disease-controlling activity contained as an active ingredient in agricultural or horticultural chemical agents.The azole derivative according to the present invention is represented by the following General Formula (I): (in Formula (I), R1 represents an unsubstituted or substituted C1-C6-alkyl group; R2 represents a carbonyl group-containing functional group, wherein the carbon atom in the carbonyl group is bound to the carbon atom in the cyclopentane ring substituted with R1 and to a hydrogen atom, a hydroxyl group, R3, OR3, or NR3R4; R3 and R4 each represent a C1-C6-alkyl group, a C2-C6-alkenyl group, or a C2-C6-alkynyl group; Y represents a halogen atom, a C1-C4-alkyl group, a C1-C4-haloalkyl group, a C1-C4-alkoxy group, a C1-C4-haloalkoxy group, a phenyl group, a cyano group, or a nitro group; m is 0 to 5; and A represents a nitrogen atom or a methine group).