公开(公告)号：US06143745A

公开(公告)日：2000-11-07

申请号：US171524

申请日：1998-10-21

申请人： Karl Eicken ,  Eberhard Ammermann ,  Siegfried Strathmann ,  Gisela Lorenz ,  Harald Kohle ,  Gunter Retzlaff

发明人： Karl Eicken ,  Eberhard Ammermann ,  Siegfried Strathmann ,  Gisela Lorenz ,  Harald Kohle ,  Gunter Retzlaff

IPC分类号： A01N43/56 ,  A01N43/58 ,  A01N43/40

CPC分类号： A01N43/56 ,  A01N43/58

摘要： Compositions for controlling harmful fungi, containing in a solid or liquid carrier pyridaben of the formula: ##STR1## or fenpyroximate of the formula: ##STR2## or tebufenpyrad of the formula: ##STR3## and at least one amide compound of the following formula I:A--CO--NR.sup.1 R.sup.2 (I)where the substituents have the meanings indicated in the description, and methods for controlling harmful fungi using compositions of this type are described.

摘要翻译： PCT No.PCT / EP97 / 02037 371日期：1998年10月21日 102（e）日期1998年10月21日PCT 1997年4月22日PCT PCT。 公开号WO97 / 39630 PCT 日期1997年10月30日用于控制有效真菌的组合物，其含有下式的固体或液体载体哒哒啶：下式的咪苯并哒嗪或下式的替泊芬吡啶：和至少一种下式I的酰胺化合物：A-CO -NR1R2（I）其中取代基具有说明书中指出的含义，并且描述了使用这种类型的组合物来控制有害真菌的方法。

公开(公告)号：US6130224A

公开(公告)日：2000-10-10

申请号：US29629

申请日：1998-03-04

申请人： Karl Eicken ,  Harald Kohle ,  Gunter Retzlaff ,  Eberhard Ammermann ,  Gisela Lorenz ,  Siegfried Strathmann

发明人： Karl Eicken ,  Harald Kohle ,  Gunter Retzlaff ,  Eberhard Ammermann ,  Gisela Lorenz ,  Siegfried Strathmann

IPC分类号： A01N43/40 ,  A01N43/54

CPC分类号： A01N43/54

摘要： The present invention relates to composiitons for controlling harmful fungi which comprise, as active ingredients, fenazaquin and at least one amide compound of the formula IA--CO--NR.sup.1 R.sup.2 Iwhere A, R.sup.1 and R.sup.2 have the meanings given in the description. The compositions according to the invention are particularly useful for controlling botrytis.

摘要翻译： PCT No.PCT / EP96 / 03861 Sec。 371日期：1998年3月4日 102（e）1998年3月4日PCT PCT 1996年9月5日PCT公布。 公开号WO97 / 08952 日期1997年3月13日本发明涉及用于控制有害真菌的组合物，其包含作为活性成分的灭草醌和至少一种式I A-CO-NR1R2I的酰胺化合物，其中A，R 1和R 2具有在说明书中给出的含义 。 根据本发明的组合物特别可用于控制葡萄孢菌。

公开(公告)号：US20080027085A1

公开(公告)日：2008-01-31

申请号：US11632342

申请日：2005-07-22

申请人： Wassilios Grammenos ,  Thomas Grote ,  Carsten Blettner ,  Markus Gewehr ,  Udo Hunger ,  Bernd Muller ,  Joachim Rheinheimer ,  Peter Schafer ,  Frank Schieweck ,  Anja Schwogler ,  Ulrich Schofl ,  Harald Kohle ,  Siegfried Strathmann ,  Maria Scherer ,  Reinhard Stierl ,  Jan Rether

发明人： Wassilios Grammenos ,  Thomas Grote ,  Carsten Blettner ,  Markus Gewehr ,  Udo Hunger ,  Bernd Muller ,  Joachim Rheinheimer ,  Peter Schafer ,  Frank Schieweck ,  Anja Schwogler ,  Ulrich Schofl ,  Harald Kohle ,  Siegfried Strathmann ,  Maria Scherer ,  Reinhard Stierl ,  Jan Rether

IPC分类号： A01N43/54 ,  A01P3/00 ,  C07D471/00

CPC分类号： C07D401/04

摘要： The invention relates to 2-(pyridin-2-yl)-pyrimidine compounds of general formula (I) and their use for controlling pathogenic fungi and as plant protection products that, as an active constituent, contain compounds of this type, whereby: k represents 0, 1, 2, 3; m represents 0, 1, 2, 3, 4 or 5; n represents 1, 2, 3, 4 or 5; R1, independent of one another, represents halogen, OH, CN, NO2, C1-C4 alkyl, C1-C4 alkyl halide, C1-C4 alkoxy, C1-C4 alkoxy halide, C2-C4 alkenyl, C2-C4 alkynyl, C3-C8 cycloalkyl, C1-C4 alkoxy-C1-C4 alkyl, amino, phenoxy, which is optionally substituted by halogen or C1-C4 alkyl, NHR, NR2, C(Ra)═N—ORb, S(═O)pA1 or C(═O)A2, or two radicals R1 bound to adjacent carbon atoms can, together, also represent a group —O-Alk-O—, wherein Alk represents a linear or branched C1-C4 alkylene, and 1, 2, 3 or 4 hydrogen atoms can also be replaced by halogen; R2 represents C1-C4 alkyl halide, C1-C4 alkoxy, C1-C4 alkoxy halide, hydroxy, halogen, CN or NO2; whereby R2 can also represent hydrogen or C1-C4 alkyl when at least one of the three following conditions is fulfilled: n represents 3, 4 or 5; k represents 1, 2 or 3; if m is not equal to 0, at least one of the radicals R1 represents a radical that differs from halogen, C1-C4 alkyl, C1-C4 alkoxy and C1-C4 alkyl halide, and; R3 represents C1-C4 alkyl.

公开(公告)号：US20080262000A1

公开(公告)日：2008-10-23

申请号：US11884412

申请日：2006-02-14

申请人： Peter Schafer ,  Udo Hunger ,  Maria Scherer ,  Harald Kohle ,  Helmut Schiffer ,  Thomas Grote ,  Jochen Dietz ,  Wassilios Grammenos ,  Jan Klaas Lohmann ,  Bernd Muller ,  Joachim Rheinheimer ,  Frank Schieweck ,  Anja Schwogler

发明人： Peter Schafer ,  Udo Hunger ,  Maria Scherer ,  Harald Kohle ,  Helmut Schiffer ,  Thomas Grote ,  Jochen Dietz ,  Wassilios Grammenos ,  Jan Klaas Lohmann ,  Bernd Muller ,  Joachim Rheinheimer ,  Frank Schieweck ,  Anja Schwogler

IPC分类号： A01N43/90 ,  C07D487/04 ,  A01P3/00

CPC分类号： C07D487/04

摘要： 5-Alkoxyalkyl-6-alkyl-7-aminoazolopyrimidines of the formula I in which the substituents are defined as follows: R1 is alkyl, cycloalkyl, alkenyl, alkynyl, alkoxyalkyl, cyanoalkyl, and benzyloxyalkyl, where the groups in the aliphatic or aromatic moiety may be unsubstituted or may have substitution by from one to three groups Ra: Ra is halogen, cyano, nitro, hydroxy, cycloalkyl, alkoxy, alkylthio, and NRARB; RA, RB are hydrogen and alkyl; R2 is alkoxyalkyl, phenoxyalkyl, alkylthioalkyl, and phenylthioalkyl, which groups may have no substitution or may have substitution according to the description; R3 is hydrogen and alkyl; A is N and C—RA; processes for preparation of these compounds, compositions comprising them, and their use for controlling phytopathogenic harmful fungi.

摘要翻译： 式I的5-烷氧基烷基-6-烷基-7-氨基偶氮嘧啶，其中取代基定义如下：R 1是烷基，环烷基，烯基，炔基，烷氧基烷基，氰基烷基和苄氧基烷基，其中 脂族或芳族部分中的基团可以是未取代的或可以具有一至三个基团的取代基：R a是卤素，氰基，硝基，羟基，环烷基 ，烷氧基，烷硫基和NR A R B， R A，B B是氢和烷基; R 2是烷氧基烷基，苯氧基烷基，烷硫基烷基和苯硫基烷基，该基团可以不具有取代基或可以根据描述进行取代; R 3是氢和烷基; A是N和C-R A; 制备这些化合物的方法，包含它们的组合物及其用于控制​​植物病原性有害真菌的用途。

公开(公告)号：US20060172887A1

公开(公告)日：2006-08-03

申请号：US11230454

申请日：2005-09-21

申请人： Harald Kohle ,  Uwe Conrath ,  Kai Sechaus ,  Matthias Niedenbrock ,  Marco-Antonio Tavares-Rodrigues ,  Waldemar Sanchez ,  Edson Begliomini ,  Claudio Oliveira

发明人： Harald Kohle ,  Uwe Conrath ,  Kai Sechaus ,  Matthias Niedenbrock ,  Marco-Antonio Tavares-Rodrigues ,  Waldemar Sanchez ,  Edson Begliomini ,  Claudio Oliveira

IPC分类号： A01N25/26 ,  A01N43/40 ,  A01N43/36 ,  A01N37/12 ,  A01N37/10 ,  A01N37/44

CPC分类号： A01N47/24 ,  A01N25/00 ,  A01N37/36 ,  A01N37/38 ,  A01N37/50 ,  A01N37/52 ,  A01N43/40 ,  A01N43/54 ,  A01N43/88 ,  A01N2300/00

摘要： A method of inducing virus tolerance of plants which comprises treating the plants, the soil or seeds with an effective amount of a compound of the formula I in which X is halogen, alkyl or trifluoromethyl; m is 0 or 1; Q is C(═CH—CH3)—COOCH3, C(═CH—OCH3)—COOCH3, C(═N—OCH3)—CONHCH3, C(═N—OCH3)—COOCH3, N(—OCH3)—COOCH3, or a group Q1 wherein # denotes the bond to the phenyl ring; A is —0—B, —CH2O—B, —OCH2—B, —CH2S—B, —CH═CH—B, —C═C—B, —CH2O—N═C(R1)—B, —CH2S—N═C(R1)—B, —CH2O—N═C(R1)—CH═CH—B, or —CH2O—N═C(R1)—C(R2)═N—R3, where B is phenyl, naphthyl, 5- or 6-membered hetaryl or 5- or 6-membered hetero-cyclyl, containing one to three N atoms and/or one O or S atom or one or two O and/or S atoms, the ring systems being unsubstituted or substituted as defined in the description; R1 is hydrogen, cyano, alkyl, haloalkyl, cycloalkyl, alkoxy, or alkylthio; R2 is phenyl, phenylcarbonyl, phenylsulfonyl, 5- or 6-membered hetaryl, 5- or 6-membered hetarylcarbonyl or 5- or 6-membered hetarylsulfonyl, the ring systems being unsubstituted or substituted by one to three radicals RB, C1-C10-alkyl, C3-C6-cycloalkyl, C2-C10-alkenyl, C2-C10-alkynyl, C1-C10-alkyl-carbonyl, C2-C10-alkenylcarbonyl, C3-C10-alkenylcarbonyl, C1-C10alkyl-sulfonyl, or C(═NORA)—RB, the hydrocarbon radicals of these groups being unsubstituted or substituted as defined in the description; R3 is hydrogen, C1-C6-alkyl, C2-C6-alkenyl, C2-C6-alkynyl, the hydrocarbon radicals of these groups being unsubstituted or substituted as defined in the description; which is taken up by the plants or seeds, during the first six weeks of the growth period of the plants or germination of the seeds.

公开(公告)号：US20090011935A1

公开(公告)日：2009-01-08

申请号：US12279309

申请日：2007-03-02

申请人： Harald Kohle ,  Ted R. Bardinelli ,  Marco-Antonio Tavares-Rodrigues

发明人： Harald Kohle ,  Ted R. Bardinelli ,  Marco-Antonio Tavares-Rodrigues

IPC分类号： A01N43/40 ,  A01N43/64 ,  A01N43/48

CPC分类号： A01N43/54 ,  A01N37/36 ,  A01N37/38 ,  A01N37/50 ,  A01N43/40 ,  A01N43/653 ,  A01N47/24 ,  A01N61/00 ,  A01N2300/00

摘要： A method of inducing tolerance of plants against bacterioses which comprises treating the plants, the soil or seeds with an effective amount of a combination of a compound of the formula I in which the variables have the meaning as set forth in the description, and a second active compound as defined in the description; which is taken up by the plants or seeds.

摘要翻译： 诱导植物对细菌的耐受性的方法，其包括用有效量的式I化合物的组合处理植物，土壤或种子，其中变量具有如说明书中所述的含义，第二 活性化合物，如说明书中所定义; 这被植物或种子摄取。

公开(公告)号：US20080207455A1

公开(公告)日：2008-08-28

申请号：US11885360

申请日：2006-03-01

申请人： Peter Schafer ,  Udo Hunger ,  Maria Scherer ,  Harald Kohle ,  Helmut Schiffer ,  Thomas Grote ,  Jochen Dietz ,  Wassilios Grammenos ,  Jan Klaas Lohmann ,  Bernd Muller ,  Joachim Rheinheimer ,  Frank Schieweck ,  Anja Schwogler

发明人： Peter Schafer ,  Udo Hunger ,  Maria Scherer ,  Harald Kohle ,  Helmut Schiffer ,  Thomas Grote ,  Jochen Dietz ,  Wassilios Grammenos ,  Jan Klaas Lohmann ,  Bernd Muller ,  Joachim Rheinheimer ,  Frank Schieweck ,  Anja Schwogler

IPC分类号： A01N43/50 ,  C07D487/04 ,  A01P3/00

CPC分类号： C07D487/04

摘要： 5,6-Dialkyl-7-aminoazolopyrimidines of the formula I in which the substituents are as defined below: R1 is alkyl or alkoxyalkyl, where the aliphatic groups may be substituted as defined in the description; R2 is CHRxCH3, cyclopropyl, CH═CH2 or CH2CH═CH2; Rx is hydrogen, CH3 or CH2CH3 or halomethyl; A is N or CH; R3 is methyl, and, if A is CH, additionally hydrogen; processes and intermediates for preparing these compounds, compositions comprising them and their use for controlling phytopathogenic harmful fungi. 5,6-Dialkyl-7aminoazolopyrimidines, their preparation and their use for controlling harmful fungi, and compositions comprising these compounds

摘要翻译： 其中取代基如下定义的式I的5,6-二烷基-7-氨基偶氮嘧啶：R 1是烷基或烷氧基烷基，其中脂族基团可以如说明书中所定义的取代; R 2是CHR x CH 3，环丙基，CH-CH 2或CH 2， CH 2 CH 2; R x是氢，CH 3或CH 2 CH 3或卤代甲基; A是N或CH; R 3是甲基，并且如果A是CH，另外是氢; 制备这些化合物的方法和中间体，包含它们的组合物及其用于控制​​植物病原性有害真菌的用途。 5,6-二烷基-7氨基偶氮嘧啶，它们的制备及其用于控制​​有害真菌的用途，以及包含这些化合物的组合物

公开(公告)号：US20050090402A1

公开(公告)日：2005-04-28

申请号：US10495928

申请日：2002-11-21

申请人： Reinhold Dieing ,  Lysander Chrisstoffels ,  Rainer Berghaus ,  Oskar Schmidt ,  Harald Kohle ,  Michael Gotsche ,  Reiner Kober

发明人： Reinhold Dieing ,  Lysander Chrisstoffels ,  Rainer Berghaus ,  Oskar Schmidt ,  Harald Kohle ,  Michael Gotsche ,  Reiner Kober

IPC分类号： A01N61/00 ,  A01N25/10 ,  A01N25/30 ,  A01N27/00 ,  A01N37/06 ,  A01N43/88

CPC分类号： A01N25/30 ,  A01N25/10 ,  A01N43/88 ,  A01N2300/00

摘要： The present invention relates to the use of specific amphiphilic copolymers as synergistic adjuvant for agrotechnical applications. Suitable agrotechnical compositions are also described. Thus, the addition of such copolymers makes possible an accelerated uptake of active ingredients by the plant. The copolymers or salts thereof to be used comprise monomer units (i) based on at least one olefin and/or at least one vinyl ether, (ii) based on at least one ethylenically unsaturated dicarboxylic acid and/or at least one ethylenically unsaturated dicarboxylic acid derivative, and, optionally (iii) based on at least one further copolymerizable comonomer.

摘要翻译： 本发明涉及特定两亲共聚物作为农业技术应用的协同佐剂的用途。 还描述了合适的农业组合物。 因此，添加这种共聚物使得植物能够加速活性成分的吸收。 所使用的共聚物或其盐包括基于至少一种烯烃和/或至少一种乙烯基醚的单体单元（i），（ii）基于至少一种烯属不饱和二羧酸和/或至少一种烯属不饱和二羧酸 酸衍生物，和任选地（iii）基于至少一种其它可共聚共聚单体。

公开(公告)号：US20090143416A1

公开(公告)日：2009-06-04

申请号：US12223029

申请日：2007-03-06

申请人： Harald Kohle ,  Ted R. Bardinelli ,  Marco-Antonio Tavares-Rodrigues

发明人： Harald Kohle ,  Ted R. Bardinelli ,  Marco-Antonio Tavares-Rodrigues

IPC分类号： A61K31/4152 ,  A61K31/4196 ,  A61P37/04 ,  A61K31/505

CPC分类号： A01N47/24 ,  A01N37/50 ,  A01N43/40 ,  A01N43/54 ,  A01N43/76 ,  A01N43/88 ,  A01N47/14 ,  A01N47/34 ,  A01N55/00 ,  A01N59/20 ,  A01N63/04 ,  A01N2300/00

摘要： A method of inducing tolerance of plants against bacterioses which comprises treating the plants, the soil or seeds with an effective amount of a combination of a compound of the formula I in which X is halogen, alkyl or trifluoromethyl; m is 0 or 1; Q is C(═CH—CH3)—COOCH3, C(═CH—OCH3)—COOCH3, C(═N—OCH3)—CONHCH3, C(═N—OCH3)—COOCH3, N(—OCH3)—COOCH3, or a group Q1  wherein # denotes the bond to the phenyl ring; A is —O—B, —CH2O—B, —OCH2—B, —CH2S—B, —CH═CH—B, —C≡C—B, —CH2O—N═C(R1)—B, —CH2S—N═C(R1)—B, —CH2O—N═C(R1)—CH═CH—B, or —CH2O—N═C(R1)—C(R2)═N—OR3, where B is phenyl, naphthyl, 5- or 6-membered hetaryl or 5- or 6-membered heterocyclyl, containing one to three N atoms and/or one O or S atom or one or two O and/or S atoms, the ring systems being unsubstituted or substituted as defined in the description; R1 is hydrogen, cyano, alkyl, haloalkyl, cycloalkyl, alkoxy, or alkylthio; R2 is phenyl, phenylcarbonyl, phenylsulfonyl, 5- or 6-membered hetaryl, 5- or 6-membered hetarylcarbonyl or 5- or 6-membered hetarylsulfonyl, the ring systems being unsubstituted or substituted by one to three radicals Ra, C1-C10-alkyl, C3-C6-cycloalkyl, C2-C10-alkenyl, C2-C10-alkynyl, C1-C10-alkyl-carbonyl, C2-C10-alkenylcarbonyl, C3-C10-alkynylcarbonyl, C1-C10-alkyl-sulfonyl, or C(═NORA)—RB, the hydrocarbon radicals of these groups being unsubstituted or substituted as defined in the description; R3 is hydrogen, C1-C6-alkyl, C2-C6-alkenyl, C2-C6-alkynyl, the hydrocarbon radicals of these groups being unsubstituted or substituted as defined in the description; and a second active compound as defined in the description; which is taken up by the plants or seeds.

摘要翻译： 诱导植物对细菌的耐受性的方法，其包括用有效量的式I化合物（其中X为卤素，烷基或三氟甲基）的化合物处理植物，土壤或种子; m为0或1; C（-CH-CH 3）-COOCH 3，C（-CH-OCH 3）-COOCH 3，C（-N-OCH 3）-CONHCH 3，C（-N-OCH 3）-COOCH 3，N（-OCH 3） 或其中＃表示与苯环的键的基团Q1; A是-OB，-CH2O-B，-OCH2-B，-CH2S-B，-CH-CH-B，-C≡CB，-CH2O-NC（R1）-B，-CH2S-NC（R1） B，-CH2O-NC（R1）-CH-CH-B或-CH2O-NC（R1）-C（R2）-N-OR3，其中B是苯基，萘基，5-或6-元杂芳基或5 - 或6-元杂环基，其含有一至三个N原子和/或一个O或S原子或一个或两个O和/或S原子，所述环系是未被描述的或如说明书中所定义的取代; R 1是氢，氰基，烷基，卤代烷基，环烷基，烷氧基或烷硫基; R 2是苯基，苯基羰基，苯基磺酰基，5-或6-元杂芳基，5-或6-元杂芳基羰基或5-或6-元杂芳基磺酰基，该环系是未被取代的或被1-3个基团取代， 烷基，C 3 -C 6 - 环烷基，C 2 -C 10 - 烯基，C 2 -C 10 - 炔基，C 1 -C 10 - 烷基 - 羰基，C 2 -C 10 - 烯基羰基，C 3 -C 10 - 炔基羰基，C 1 -C 10 - 烷基磺酰基或C （-NORA）-RB，这些基团的烃基是未被描述的或如说明书中所定义的取代基; R 3是氢，C 1 -C 6 - 烷基，C 2 -C 6 - 烯基，C 2 -C 6 - 炔基，这些基团的烃基是未被取代或如说明书中所定义的取代; 和如说明书中定义的第二活性化合物; 这被植物或种子摄取。

公开(公告)号：US20080188493A1

公开(公告)日：2008-08-07

申请号：US11885332

申请日：2006-03-01

申请人： Peter Schäfer ,  Udo Hunger ,  Maria Scherer ,  Harald Kohle ,  Helmut Schiffer ,  Thomas Grote ,  Jochen Dietz ,  Wassilios Grammenos ,  Jan Klaas Lohmann ,  Bernd Muller ,  Joachim Rheinheimer ,  Frank Schieweck ,  Anja Schwogler

发明人： Peter Schäfer ,  Udo Hunger ,  Maria Scherer ,  Harald Kohle ,  Helmut Schiffer ,  Thomas Grote ,  Jochen Dietz ,  Wassilios Grammenos ,  Jan Klaas Lohmann ,  Bernd Muller ,  Joachim Rheinheimer ,  Frank Schieweck ,  Anja Schwogler

IPC分类号： A01N43/90 ,  C07D487/04 ,  A01N25/26 ,  A01P3/00

CPC分类号： C07D487/04 ,  A01N43/90

摘要： 5,6-Dialkyl-7-aminoazolopyrimidines of the formula I in which the substituents are as defined below: R1 is haloalkyl, haloalkoxyalkyl, alkoxyhaloalkyl, alkenyl, haloalkenyl, alkynyl oder haloalkynyl; R2 is alkyl, alkoxyalkyl, alkenyl or alkynyl; where R1 and/or R2 may be substituted according to the description; A is N or CH, and R3 is CH3 and, if A is CH, additionally hydrogen; processes and intermediates for preparing these compounds, compositions comprising them and their use for controlling phytopathogenic harmful fungi.

摘要翻译： 其中取代基如下定义的式I的5,6-二烷基-7-氨基偶氮嘧啶：R 1是卤代烷基，卤代烷氧基烷基，烷氧基卤代烷基，烯基，卤代烯基，炔基，卤代炔基; R 2是烷基，烷氧基烷基，烯基或炔基; 其中R 1和/或R 2可以根据描述被取代; A是N或CH，R 3是CH 3，并且如果A是CH，另外是氢; 制备这些化合物的方法和中间体，包含它们的组合物及其用于控制​​植物病原性有害真菌的用途。