1,2,3,6-tetrahydro-5-nitro-pyrimidine derivatives
    111.
    发明授权
    1,2,3,6-tetrahydro-5-nitro-pyrimidine derivatives 失效
    1,2,3,6-四氢-5-硝基 - 嘧啶衍生物

    公开(公告)号:US4831036A

    公开(公告)日:1989-05-16

    申请号:US52102

    申请日:1987-05-18

    CPC分类号: C07D487/04 A01N43/90

    摘要: New 1,2,3,6-tetrahydro-5-nitro-pyrimidine derivatives of the formula ##STR1## in which n represents the numbers 0, 1 or 2,R.sup.1 represents hydrogen or optionally substituted radicals from the series comprising alkyl, alkenyl, alkinyl, aralkyl and hetarylalkyl, andR.sup.2 represents dialkylamino, alkoxy, alkenyloxy, aralkoxy or optionally substituted radicals from the series comprising alkyl, alkenyl, alkinyl, cycloalkyl, aralkyl and hetarylalkyl,and their acid addition salts have been found.It has furthermore been found that these 1,2,3,6-tetrahydro-5-nitor-pyrimidine derivatives have unexpectedly high activity as insecticides, nematicides and ectoparasiticides.

    摘要翻译: 新的具有式“IMAGE”的1,2,3,6-四氢-5-硝基 - 嘧啶衍生物,其中n表示数字0,1或2,R 1表示氢或任选取代的基团,其包含烷基,烯基, 烷基,芳烷基和杂芳基烷基,并且R2表示二烷基氨基,烷氧基,烯氧基,芳烷氧基或任选被取代的基团,包括烷基,烯基,炔基,环烷基,芳烷基和杂芳基烷基,及其酸加成盐。 此外已经发现,这些1,2,3,6-四氢-5-硝基 - 嘧啶衍生物作为杀虫剂,杀线虫剂和外寄生虫杀螨剂具有出人意料的高活性。

    4-haloalkylthio-5-amino-1-arylpyrazoles, composition containing them,
and insecticidal and acaricidal method of using them
    112.
    发明授权
    4-haloalkylthio-5-amino-1-arylpyrazoles, composition containing them, and insecticidal and acaricidal method of using them 失效
    4-卤代烷硫基-5-氨基-1-芳基吡唑,含有它们的组合物,以及使用它们的杀虫和杀螨方法

    公开(公告)号:US4771066A

    公开(公告)日:1988-09-13

    申请号:US13741

    申请日:1987-02-12

    摘要: Insecticidally and acarididally active 1-arylpyrazoles of the formula ##STR1## in which R.sup.1 represents hydrogen, alkyl or halogen alkyl,R.sup.2 represents alkyl, alkenyl, alkinyl, cycloalkyl, halogenoalkyl, halogenoalkenyl, alkoxyalkyl, alkylthioalkyl, alkylsulphinylalkyl, alkylsulphonylalkyl, optionally substituted aralkyl or optionally substituted aryl,R.sup.3 represents alkyl, alkenyl, alkinyl, halogenoalkyl, halogenoalkenyl, alkoxyalkyl, alkylthioalkyl, cycloalkyl or optionally substituted aralkyl,R.sup.4 represents alkyl, alkenyl, alkinyl, halogenoalkyl, halogenoalkenyl, alkoxyalkyl, alkylthioalkyl, cycloalkyl or optionally substituted aralkyl, and, in addition, also represents hydrogen in the case where R.sup.3 does not simultaneously represent unsubstituted alkyl, orR.sup.3 and R.sup.4, together with the nitrogen atom to which they are bound, represent a saturated heterocycle, which can optionally contain further heteroatoms,Ar represents in each case optionally substituted phenyl or pyridyl, andn represents a number 0, 1 or 2.

    摘要翻译: 具有式“IMAGE”的杀虫和杀螨活性1-芳基吡唑其中R1代表氢,烷基或卤素烷基,R2代表烷基,烯基,炔基,环烷基,卤代烷基,卤代烯基,烷氧基烷基,烷硫基烷基,烷基亚磺酰基烷基,烷基磺酰基烷基,任选取代的芳烷基或 任选取代的芳基,R 3表示烷基,烯基,炔基,卤代烷基,卤代烯基,烷氧基烷基,烷硫基烷基,环烷基或任选取代的芳烷基,R 4表示烷基,烯基,炔基,卤代烷基,卤代烯基,烷氧基烷基,烷硫基烷基,环烷基或任选取代的芳烷基, 此外,在R3不同时表示未取代的烷基的情况下也表示氢,或者R 3和R 4与它们所连接的氮原子一起代表饱和的杂环,其可以任选地含有另外的杂原子,Ar表示每个 任选取代的苯基或吡啶基,n表示 数字0,1或2。

    Substituted 3,4-hetaryl-pyrazolines
    115.
    发明授权
    Substituted 3,4-hetaryl-pyrazolines 失效
    取代的3,4-二杂芳基吡唑啉

    公开(公告)号:US5502070A

    公开(公告)日:1996-03-26

    申请号:US129923

    申请日:1993-09-30

    摘要: The present invention relates to new substituted 3,4-hetaryl-pyrazolines of the general formula (I) ##STR1## in which R.sup.1 represents an unsaturated five- or six-membered optionally substituted and optionally benzo-fused heterocyclic ring containing 1 to 4 nitrogen atoms, or represents an optionally substituted heterocyclic ring from the series comprising ##STR2## X represents oxygen or sulphur and Het represents an optionally substituted and/or optionally fused heterocyclic ring,processes for their preparation and their use as agents for combating pests.

    摘要翻译: 本发明涉及通式(I)的新的取代的3,4-杂芳基 - 吡唑啉,其中含有1至4个氮原子的5或6元任选取代的和任选的苯并稠合杂环,或表示任选取代的杂环 包含 X的系列的环表示氧或硫,Het表示任选取代的和/或任选稠合的杂环,其制备方法及其用作防治害虫的试剂。