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公开(公告)号:US3329571A
公开(公告)日:1967-07-04
申请号:US43020465
申请日:1965-02-03
Applicant: AMERICAN HOME PROD
Inventor: RICE LEONARD M , FREED MEIER E
IPC: A61K31/00 , C07D209/94
CPC classification number: C07D209/94 , A61K31/00
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12.Novel xanthene-9-carboxylic acid esters of hydroxyalkyl azaspiranes 失效
Title translation: 羟烷基氮杂环丙烷的新型呫吨-9-羧酸酯公开(公告)号:US3265702A
公开(公告)日:1966-08-09
申请号:US29413963
申请日:1963-07-10
Applicant: AMERICAN HOME PROD
Inventor: FREED MEIER E , RICE LEONARD M
IPC: C07D221/20 , C07D405/12
CPC classification number: C07D221/20 , C07D405/12
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13.N-aminoalkyl-2, 3-polymethylene-1h-benz[g] indoles and methods of preparing same 失效
Title translation: N-氨基烷基-2,3-聚亚甲基-1h - 苯并[g]吲哚及其制备方法公开(公告)号:US3218326A
公开(公告)日:1965-11-16
申请号:US25024663
申请日:1963-01-09
Applicant: AMERICAN HOME PROD
Inventor: RICE LEONARD M , FREED MEIER E , ELISABETH HERTZ
IPC: C07D209/94
CPC classification number: C07D209/94
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14.13-substituted 5, 6-dihydro-13h-dibenzo-[a, i] carbazoles 失效
Title translation: 13-取代的5,6-二氢-13h-二苯并[a,i]咔唑公开(公告)号:US3144461A
公开(公告)日:1964-08-11
申请号:US18794062
申请日:1962-04-16
Applicant: AMERICAN HOME PROD
Inventor: RICE LEONARD M , FREED MEIER E , ELISABETH HERTZ
IPC: C07D209/80
CPC classification number: C07D209/80
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公开(公告)号:US3062839A
公开(公告)日:1962-11-06
申请号:US81953859
申请日:1959-06-11
Applicant: AMERICAN HOME PROD
Inventor: VITHAL SHETTY BOLA , BRUCE WILLIAM F , FREED MEIER E
IPC: C07D307/52 , C07D307/54
CPC classification number: C07D307/54 , C07D307/52
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16.Nicotinic acid ester of certain hydroxyalkyleneimino-diacetamides 失效
Title translation: 某些羟基亚烷基亚氨基二乙酰胺的烟酸酯公开(公告)号:US2945041A
公开(公告)日:1960-07-12
申请号:US75363458
申请日:1958-08-07
Applicant: AMERICAN HOME PROD
Inventor: JOSEPH SEIFTER , HANSLICK ROY S , FREED MEIER E
IPC: C07D213/80
CPC classification number: C07D213/80
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17.5,6,7,8,9,10-Hexahydro-5-phenyl-5,9-methanobenzocycloocten-11-amines and related compounds 失效
Title translation: 5,6,7,8,9,10-六氢-5-苯基-5,9-甲基苯并环辛烯-11-胺及相关化合物公开(公告)号:US3917680A
公开(公告)日:1975-11-04
申请号:US42931673
申请日:1973-12-28
Applicant: AMERICAN HOME PROD
Inventor: POTOSKI JOHN R , FREED MEIER E
CPC classification number: C07C317/00 , C07C45/30 , C07C45/64 , C07C45/673 , C07C45/68 , C07C49/755
Abstract: 5,6,7,8,9,10-Hexahydro-5-phenyl-5,9-methanobenzocyclooctene-11amines, intermediates therefore and processes for their preparation are disclosed. The final products have analgesic activity.
Abstract translation: 5,6,7,8,9,10-六氢-5-苯基-5,9-甲基苯并环辛烯-11-胺,因此其中间体及其制备方法被公开。 最终产品具有止痛活性。
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18.4 5-dihydro-n-(4-phenyl-1-piperazinylcarbonyl-1h( 14)-diazepino (12-a)indole 失效
Title translation: 4,5-二氢-N-(4-苯基-1-哌嗪子基)-1H(14) - 二氮杂(12-A)吲哚公开(公告)号:US3641030A
公开(公告)日:1972-02-08
申请号:US3641030D
申请日:1968-10-21
Applicant: AMERICAN HOME PROD
Inventor: FREED MEIER E , HERTZ ELISABETH
IPC: C07D487/04 , C07D51/70
CPC classification number: C07D487/04
Abstract: THIS INVENTION CONCERNS TETRAHYDROPYRAZINOINDOLE-2-CARBOXAMIDES AND DIHYDRODIAZEPINOINDOLE-2-CARBOXAMIDES WHICH ARE PHARMACOLOGICALLY ACTIVE AS CENTRAL NERVOUS DEPRESSANTS.
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公开(公告)号:US3501481A
公开(公告)日:1970-03-17
申请号:US3501481D
申请日:1966-12-22
Applicant: AMERICAN HOME PROD
Inventor: ARCHIBALD JOHN L , FREED MEIER E
IPC: C07D455/03 , C07D471/04 , C07D33/38
CPC classification number: C07D455/00 , C07D471/04
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公开(公告)号:US3458515A
公开(公告)日:1969-07-29
申请号:US3458515D
申请日:1966-07-21
Applicant: AMERICAN HOME PROD
Inventor: ARCHIBALD JOHN L , FREED MEIER E
IPC: C07D207/32 , C07D207/335 , C07D207/337 , C07D57/00 , C07D27/22 , C07D51/00
CPC classification number: C07D207/335 , C07D207/337
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