公开(公告)号：US20150150257A1

公开(公告)日：2015-06-04

申请号：US14408174

申请日：2013-06-12

Applicant: BASF SE

Inventor： Sebastian Soergel ,  Daniel Saelinger ,  Christian Defieber ,  Juergen Langewald ,  Birgit Gockel ,  Egon Haden ,  Deborah L. Culberston ,  Koshi Gunjima

IPC: A01N43/58 ,  C07D403/12

CPC classification number: A01N43/58 ,  A01N37/22 ,  A01N43/36 ,  A01N43/56 ,  A01N43/653 ,  A01N43/78 ,  A01N43/88 ,  A01N47/18 ,  C07D403/12 ,  A01N37/46 ,  A01N47/02 ,  A01N47/24 ,  A01N51/00 ,  A01N2300/00

Abstract: The present invention relates to pesticidal mixtures comprising as active compounds 1) at least one pyrazole compound A selected from the compounds of formula I: wherein the variables have the meaning as defined in the description, and 2) at least one further compound B selected from the compounds of the following groups A.1, A.2, A.3, A.4, A.5, A.6, A.7, A.8, A.9, A.10, A.11, A.12, A.13, A.14, A.15, A.16, A.17, F.1, F.2, F.3, F.4, F.5, F.6, F.7, F.8, F.9, F.10 and F.11 as defined in the specification. The present invention also relates to novel pyrazole compounds of the formula I. The present invention also relates to methods and use of these mixtures and novel compounds for combating invertebrate pests such as insects, arachnids or nematodes in and on plants, and for protecting such plants being infested with pests, especially also for protecting plant propagation material as like seeds.

Abstract translation: 本发明涉及包含作为活性化合物的至少一种选自式I化合物的至少一种吡唑化合物A的农药混合物：其中变量具有如说明书中定义的含义，和2）至少一种其它化合物B，其选自 以下A.1，A.2，A.3，A.4，A.5，A.6，A.7，A.8，A.9，A.10，A.11， A.12，A.13，A.14，A.15，A.16，A.17，F.1，F.2，F.3，F.4，F.5，F.6，F 7，F.8，F.9，F.10和F.11。 本发明还涉及式I的新型吡唑化合物。本发明还涉及这些混合物和新化合物与植物中和植物上的昆虫，蜘蛛或线虫等无脊椎害虫相抗和保护这些植物的方法和用途 被害虫侵染，特别是用于保护植物繁殖材料，如同种子一样。

公开(公告)号：US11591293B2

公开(公告)日：2023-02-28

申请号：US17296683

申请日：2019-12-11

Applicant: BASF SE

Inventor： Volker Maywald ,  Roland Goetz ,  Daniel Saelinger ,  Birgit Gockel ,  Manfred Ehresmann ,  Markus Jegelka ,  Joaquim Henrique Teles

IPC: C07C263/10

Abstract: A method for manufacturing an isocyanate compound represented by formula (2) (2) wherein R1 represents a methyl group, an ethyl group, a cyclopropyl group, a chlorine atom, a bromine atom, or a methoxy group; and R2 represents an alkyl group having 1 to 6 carbon atoms, comprising reacting an aniline compound represented by formula (1) (1) wherein R1 and R2 are defined as above with a phosgene compound at a temperature of from 40° C. to the boiling point of the inert solvent in at least one kind of inert solvent.

公开(公告)号：US11440861B2

公开(公告)日：2022-09-13

申请号：US17295102

申请日：2019-11-25

Applicant: BASF SE

Inventor： Karsten Koerber ,  Michael Rack ,  Pascal Bindschaedler ,  Martin John McLaughlin ,  Birgit Gockel ,  Devendra Vyas ,  Sebastian Soergel

IPC: C07C17/35 ,  B01J21/18 ,  B01J23/44 ,  C07C25/08 ,  C07C245/20 ,  C07C37/045 ,  C07C39/30 ,  C07C17/093

Abstract: The invention relates to a process for the preparation of 5-bromo-1,3-dichloro-2-fluoro-benzene by diazotization and reduction of 6-bromo-2,4-dichloro-3-fluoro-aniline, which is obtained by bromination of 2,4-dichloro-3-fluoro-aniline, which is obtained by reduction of 1,3-dichloro-2-fluoro-4-nitro-benzene, and a process for preparing active compounds of formula V (Formula V) wherein the variables are defined in the specification by further transforming 5-bromo-1,3-dichloro-2-fluoro-benzene obtained from 2,4-dichloro-3-fluoro-aniline by the process according to the invention.

公开(公告)号：US20220024898A1

公开(公告)日：2022-01-27

申请号：US17311403

申请日：2020-01-10

Applicant: BASF SE

Inventor： Joachim Gebhardt ,  Martin Viertelhaus ,  Tiziana Chiodo ,  Michael Rack ,  Eric George Klauber ,  Wen Xu ,  Roland Goetz ,  Florian Vogt ,  Birgit Gockel ,  Sebastian Soergel

IPC: C07D403/12 ,  A01N43/58 ,  A01P7/04

Abstract: The present invention relates to a novel crystalline form of 1-(1,2-dimethylpropyl)-N-ethyl-5-methyl-N-pyridazin-4-yl-pyrazole-4-carboxamide recently assigned the common name dimpropyridaz. The invention also relates to the use of the crystalline form B for combating invertebrate pests and to formulations for plant protection which contain the crystalline form B of 1-(1,2-dimethylpropyl)-N-ethyl-5-methyl-N-pyridazin-4-yl-pyrazole-4-carboxamide. The crystalline form B according to the present invention can be identified by powder X-ray diffractometry on the basis of its powder X-ray diffraction diagram, hereinafter also termed powder X-ray diffraction pattern or PXRD pattern, of the polymorph form B recorded using Cu—Kα radiation (1.54178 Å) at 25° C. displays the 3 following reflections, quoted as 2θ values: 20.69±0.10°, 24.15±0.10° and 30.52±0.10°. In addition to these 3 reflections, the polymorph B of the present invention may display in such a PXRD pattern one or more, in particular at least 2, often at least 4, in particular at least 6 or at least 8 reflections and especially all of the reflections quoted hereinafter as 2θ values: 7.99±0.10°, 10.07±0.10°, 12.38±0.10°, 15.31±0.10°, 15.97±0.10°, 16.50±0.10°, 18.03±0.10°, 19.29±0.10°, 20.22±0.0.10°, 20.96±0.10°, 23.40±0.10°, 23.70±0.10°, 26.09±0.10°, 27.26±0.10° and 32.91±0.10°.

公开(公告)号：US20200178542A9

公开(公告)日：2020-06-11

申请号：US15754074

申请日：2016-08-08

Applicant: BASF SE

Inventor： Birgit Gockel ,  Joachim Dickhaut ,  Daniel Saelinger

IPC: A01N65/00 ,  A01H1/06 ,  A01H6/60

Abstract: A method for controlling pests of a cotton plant is disclosed. The method includes the step of contacting the cotton plant, parts of it, or its propagation material with components of the ginkgo tree selected from bilobalide, ginkgolide A, ginkgolide B, ginkgolide C, ginkgolide J, ginkgolide M, and mixtures thereof. The use of components of the ginkgo tree for controlling pests in a cotton plant, parts of it, or its propagation material, is also disclosed. A pesticide including one or more components of the ginkgo tree selected from bilobalide, ginkgolide A, ginkgolide B, ginkgolide C, ginkgolide J, and ginkgolide M is further disclosed.

公开(公告)号：US09955692B2

公开(公告)日：2018-05-01

申请号：US15114974

申请日：2015-01-30

Applicant: BASF SE

Inventor： Sebastian Soergel ,  Daniel Saelinger ,  Birgit Gockel

IPC: A01N43/58 ,  C07D403/12 ,  A01N43/36 ,  A01N43/56

CPC classification number: A01N43/58 ,  A01N43/36 ,  A01N43/56 ,  C07D403/12

Abstract: The present invention relates to novel pyrazoles of formula I. Moreover, the invention relates to processes and intermediates for preparing the pyrazoles of formula I, and also to active compound combinations comprising them, to compositions comprising them, and to their use for protecting growing plants from attack or infestation by invertebrate pests. Furthermore, the invention relates to methods of applying such compounds. The present invention also relates to seed comprising such compounds.

公开(公告)号：US09783523B2

公开(公告)日：2017-10-10

申请号：US15038272

申请日：2014-11-21

Applicant: BASF SE

Inventor： Nina Gertrud Bandur ,  Jochen Dietz ,  Matthias Pohlman ,  Martin John McLaughlin ,  Birgit Gockel ,  Karsten Körber ,  Wolfgang Von Deyn

IPC: C07D401/14 ,  C07D405/14 ,  C07D401/06 ,  C07D405/06 ,  C07D417/06 ,  C07D417/14 ,  C07D419/14 ,  A01N43/40 ,  A01N43/54 ,  A01N43/60 ,  A01N43/78 ,  A01N43/80 ,  A01N43/84 ,  A01N47/10 ,  C07D409/14 ,  C07D413/14

CPC classification number: C07D401/06 ,  A01N43/40 ,  A01N43/54 ,  A01N43/60 ,  A01N43/78 ,  A01N43/80 ,  A01N43/84 ,  A01N47/10 ,  C07D401/14 ,  C07D405/06 ,  C07D405/14 ,  C07D409/14 ,  C07D413/14 ,  C07D417/06 ,  C07D417/14 ,  C07D419/14

Abstract: The present invention relates to N-acylimino compound of formula (I): wherein X is O or S, in particular O; Y is a single bond, O, S or NR5; Het is a 5 or 6 membered carbon-bound or nitrogen-bound heterocyclic ring, W1-W2-W3-W4 represents a carbon chain group connected to N and C═N, and thus forming a saturated, unsaturated, or partially unsaturated 5 or 6 membered nitrogen containing heterocycle, wherein W1, W2, W3 and W4 each individually represent CRvRw; R1, R2 may be hydrogen, halogen, etc.; R3 may be hydrogen, CN, C1-C6-alkyl, etc.; R4 may be of hydrogen, C1-C6-alkyl, C2-C6-alkenyl, C2-C6-alkinyl, C3-C8-cycloalkyl, Q-phenyl, Q′-O-phenyl, Q′-S-phenyl, where the phenyl ring is optionally substituted with one or more, e.g. 1, 2, 3, 4 or 5 identical or different substituents R10, and the moieties Q-Het#, Q′-O-Het# and Q′-S-Het# where Het# represents a heterocyclic radical and where Q and Q′ are C1-C6-alkandiyl, C2-C6-alkendiyl, or C2-C6-alkyndiyl, and where Q may also be a single bond; R3 and R4 together may also may also a bivalent radical, selected from the group consisting of C2-C5-alkandiyl, C2-C5-alkendiyl, Q″-C1-C4-alkandiyl and Q″-C2-C4-alkendiyl, where Q″ is O or S. The invention also relates to the use of the N-acylimino heterocyclic compounds, their stereoisomers, their tautomers and their salts, for combating invertebrate pests. Furthermore the invention relates also to methods of combating invertebrate pests, which comprises applying such compounds.

公开(公告)号：US11591335B2

公开(公告)日：2023-02-28

申请号：US16612111

申请日：2018-05-07

Applicant: BASF SE

Inventor： Martin John Mclaughlin ,  Arun Narine ,  Wolfgang Von Deyn ,  Birgit Gockel

IPC: C07D487/04 ,  A01N43/90 ,  A01P7/04

Abstract: The present invention relates to compounds of formula I, wherein the variables are defined as given in the description and claims. The invention further relates to uses, processes and composition for compounds I.

公开(公告)号：US11142514B2

公开(公告)日：2021-10-12

申请号：US15764414

申请日：2016-09-29

Applicant: BASF SE

Inventor： Martin John McLaughlin ,  Karsten Koerber ,  Birgit Gockel ,  Wolfgang von Deyn

IPC: C07D401/06 ,  A01N43/54 ,  C07D417/06 ,  A01N25/02 ,  A01N25/08 ,  A01N61/00

Abstract: Provided herein are imino compounds of formula I and stereoisomers, tautomers and salts thereof. Further provided herein are agricultural and veterinary compositions including the compounds. Also provided herein are methods related to the use of these compounds, and the stereoisomers, tautomers and/or salts thereof, for combating invertebrate pests. Further provided herein are methods for combating invertebrate pests, wherein the methods include applying such compounds, steroisomers, tautomers, and salts.

公开(公告)号：US10961226B2

公开(公告)日：2021-03-30

申请号：US16347414

申请日：2017-10-27

Applicant: BASF SE

Inventor： Eric George Klauber ,  Birgit Gockel ,  Sebastian Soergel ,  Roland Goetz ,  Henricus Maria Martinus Bastiaans ,  Jochen Dietz ,  Joachim Gebhardt

IPC: C07D403/12 ,  A01N43/58

Abstract: The present invention relates to a process for the purification of pyrazolpyridazines of formula I wherein the variables are as defined in the specification, by adding HCl to a solution of the pyrazolpyridazine in an inert solvent under non-aqueous conditions, effecting crystallization of the HCl-salt, isolating the resulting precipitate.