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公开(公告)号:US20070219198A1
公开(公告)日:2007-09-20
申请号:US11703522
申请日:2007-02-07
申请人: Jason Xiang , Eddine Saiah , Steve Tam , John Mckew , Lihren Chen , Manus Ipek , Katherine Lee , Huan-Qiu Li , Jianchang Li , Wei Li , Tarek Mansour , Vipin Suri , Richard Vargas , Yuchuan Wu , Zhao-Kui Wan , Jinbo Lee , Eva Binnun , Douglas Wilson
发明人: Jason Xiang , Eddine Saiah , Steve Tam , John Mckew , Lihren Chen , Manus Ipek , Katherine Lee , Huan-Qiu Li , Jianchang Li , Wei Li , Tarek Mansour , Vipin Suri , Richard Vargas , Yuchuan Wu , Zhao-Kui Wan , Jinbo Lee , Eva Binnun , Douglas Wilson
IPC分类号: A61K31/5377 , A61K31/497 , A61K31/496 , C07D413/02 , C07D403/02 , C07D409/02
CPC分类号: C07D211/96 , C07D295/26 , C07D401/04 , C07D403/02 , C07D409/02 , C07D413/02
摘要: This invention relates to inhibiting 11βHSD1.
摘要翻译: 本发明涉及抑制11betaHSD1。
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公开(公告)号:US06825208B2
公开(公告)日:2004-11-30
申请号:US10223860
申请日:2002-08-20
申请人: Jinglan Zhou , Leslie Robinson , Nikolaus M. Gubernator , Eddine Saiah , Xu Bai , Xin Gu
发明人: Jinglan Zhou , Leslie Robinson , Nikolaus M. Gubernator , Eddine Saiah , Xu Bai , Xin Gu
IPC分类号: A61K31473
CPC分类号: C07D221/18
摘要: This invention relates generally to tetracyclic tetrahydroquinoline compounds, and analogues thereof, and pharmaceutically acceptable salt forms thereof, which are selective inhibitors of serine protease enzymes, especially factor VIIa; pharmaceutical compositions containing the same; and methods of using the same as anticoagulant agents for modulation of the coagulation cascade.
摘要翻译: 本发明一般涉及四环四氢喹啉化合物及其类似物及其药学上可接受的盐形式,其是丝氨酸蛋白酶,特别是因子VIIa的选择性抑制剂; 含有该组合物的药物组合物; 以及使用其作为抗凝血剂调节凝血级联的方法。
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公开(公告)号:US20110105509A1
公开(公告)日:2011-05-05
申请号:US12938479
申请日:2010-11-03
申请人: Neelu Kaila , Eddine Saiah , Bruce Christopher Follows , Adrian Huang , Kristin Marie Janz , Michael Dennis Lowe , Alessandro Fabio Moretto , Jennifer Romanic Thomason , Tarek Suhayl Mansour , Cara Margaret May Williams
发明人: Neelu Kaila , Eddine Saiah , Bruce Christopher Follows , Adrian Huang , Kristin Marie Janz , Michael Dennis Lowe , Alessandro Fabio Moretto , Jennifer Romanic Thomason , Tarek Suhayl Mansour , Cara Margaret May Williams
IPC分类号: A61K31/502 , C07D403/04 , A61K31/501 , C07D401/06 , A61K31/4439 , C07D403/14 , C07D403/06 , A61K31/4725 , C07D417/14 , C07D401/14 , A61P11/00 , A61P1/00 , A61P17/00 , A61P29/00 , A61P37/06 , A61P37/08 , C12N5/02
CPC分类号: C07D403/04 , C07D401/04 , C07D401/06 , C07D401/14 , C07D403/06 , C07D403/14 , C07D417/14
摘要: Disclosed are compounds of Formula (I): which are useful as antagonists of the CRTH2 receptors. Pharmaceutical compositions containing compounds of Formula (I) and the use of compounds of Formula (I) to treat diseases or disorders that are responsive to inhibition of the binding of endogenous ligands to the CRTH2 receptor are also disclosed. Methods for preparing and using these compounds are further described.
摘要翻译: 公开了式(I)的化合物:其可用作CRTH2受体的拮抗剂。 还公开了含有式(I)化合物和式(I)化合物用于治疗对抑制内源性配体与CRTH2受体的结合有反应的疾病或病症的药物组合物。 进一步描述制备和使用这些化合物的方法。
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公开(公告)号:US07632838B2
公开(公告)日:2009-12-15
申请号:US11703522
申请日:2007-02-07
申请人: Jason Shaoyun Xiang , Eddine Saiah , Steve Y. Tam , John C. Mckew , Lihren Chen , Manus Ipek , Huan-Qiu Li , Jianchang Li , Wei Li , Tarek Suhayl Mansour , Vipin Suri , Yuchuan Wu , Zhao-Kui Wan , Jinbo Lee , Eva Binnun , Douglas P. Wilson
发明人: Jason Shaoyun Xiang , Eddine Saiah , Steve Y. Tam , John C. Mckew , Lihren Chen , Manus Ipek , Huan-Qiu Li , Jianchang Li , Wei Li , Tarek Suhayl Mansour , Vipin Suri , Yuchuan Wu , Zhao-Kui Wan , Jinbo Lee , Eva Binnun , Douglas P. Wilson
IPC分类号: A61K31/4965 , C07D241/04 , C07D295/00
CPC分类号: C07D211/96 , C07D295/26 , C07D401/04 , C07D403/02 , C07D409/02 , C07D413/02
摘要: This invention relates to inhibiting 11βHSD1.
摘要翻译: 本发明涉及抑制11betaHSD1。
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公开(公告)号:US20080188659A1
公开(公告)日:2008-08-07
申请号:US12027412
申请日:2008-02-07
申请人: Eddine Saiah , Huan-Qiu Li , Adrian Huang
发明人: Eddine Saiah , Huan-Qiu Li , Adrian Huang
IPC分类号: C07D241/04 , C07C311/16 , C07C311/21 , C07D211/60
CPC分类号: C07D241/04 , C07C231/12 , C07C303/40 , C07C2601/14 , C07C311/37 , C07C311/53 , C07C237/30
摘要: This invention relates to methods for preparing halogenated amines.
摘要翻译: 本发明涉及制备卤代胺的方法。
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公开(公告)号:US20100029648A1
公开(公告)日:2010-02-04
申请号:US12539232
申请日:2009-08-11
申请人: Jason Shaoyun Xiang , Eddine Saiah , Steve Y. Tam , John C. McKew , Lihren Chen , Manus Ipek , Katherine Lee , Huan-Qiu Li , Jianchang Li , Wei Li , Tarek Suhayl Mansour , Vipin Suri , Richard Vargas , Yuchuan Wu , Zhao-Kui Wan , Jinbo Lee , Eva Binnun , Douglas P. Wilson
发明人: Jason Shaoyun Xiang , Eddine Saiah , Steve Y. Tam , John C. McKew , Lihren Chen , Manus Ipek , Katherine Lee , Huan-Qiu Li , Jianchang Li , Wei Li , Tarek Suhayl Mansour , Vipin Suri , Richard Vargas , Yuchuan Wu , Zhao-Kui Wan , Jinbo Lee , Eva Binnun , Douglas P. Wilson
IPC分类号: A61K31/5377 , A61K31/497 , A61K31/4965 , A61K31/4545
CPC分类号: C07D211/96 , C07D295/26 , C07D401/04 , C07D403/02 , C07D409/02 , C07D413/02
摘要: This invention relates to inhibiting 11βHSD1.
摘要翻译: 本发明涉及抑制11betaHSD1。
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