3-[Benz(ox/thi)azol-7-yl]-1h-pyrimidine-2,4-diones
    14.
    发明授权
    3-[Benz(ox/thi)azol-7-yl]-1h-pyrimidine-2,4-diones 失效
    3- [Benz(ox / thi)azol-7-yl] -1h-嘧啶-2,4-二酮

    公开(公告)号:US06624119B1

    公开(公告)日:2003-09-23

    申请号:US09830961

    申请日:2001-05-03

    IPC分类号: C07D41304

    摘要: The invention relates to herbicidally effective 3-{benz(ox/thi)azol-7-yl}-1H-pyrimidine-2,4-diones of formula (I) wherein X=oxygen or sulphur, Y=oxygen or sulphur; Z=chemical bond, C1-C4-alkylene, O, S, SO, SO2; R1=H, NH2, C1-C6-alkyl, C1-C6-alkyl halide; R2=H, halogen, C1-C6-alkyl, C1-C6-alkyl halide, C1-C6-alkylthio, C1-C6-alkylsulfinyl or C1C6-alkylsulfonyl; R3=H, halogen, C1-C6-alkyl; R4=H, halogen; R5=CN, halogen, C1-C6-alkyl, C1-C6-alkyl halide, C1-C6-alkoxy or C1-C6-halogenalkoxy; R6=H, C3-C7-cycloalkyl containing a 3 to 7-membered saturated heterocyclyl and one or more oxygen and/or sulphur atoms, whereby each heterocyclic ring may contain a carbonyl or thiocarbonyl ring member. The invention also relates to the agriculturally usable salts of the compounds of formula (I).

    摘要翻译: 本发明涉及其中X =氧或硫,Y =氧或硫的式(I)的除草有效3- {苯并(ox / thi)唑-4-基} -1H-嘧啶-2,4-二酮; Z =化学键,C1-C4亚烷基,O,S,SO,SO2; R 1 = H,NH 2,C 1 -C 6 - 烷基,C 1 -C 6烷基卤化物; R 2 = H,卤素,C 1 -C 6烷基,C 1 -C 6烷基卤,C 1 -C 6烷硫基,C 1 -C 6烷基亚磺酰基或C 1 -C 6烷基磺酰基; R 3 = H,卤素,C 1 -C 6 - 烷基; R 4 = H,卤素; R 5 = CN,卤素,C 1 -C 6烷基,C 1 -C 6烷基卤化物,C 1 -C 6 - 烷氧基或C 1 -C 6卤代烷氧基; R 6 = H,含有3至7元饱和杂环基和一个或多个氧和/或硫原子的C 3 -C 7环烷基,其中每个杂环可以含有羰基或硫代羰基环成员。 本发明还涉及式(I)化合物的农业上可用的盐。

    Substituted 2-phenylpyridines as herbicides
    19.
    发明授权
    Substituted 2-phenylpyridines as herbicides 失效
    取代的2-苯基吡啶作为除草剂

    公开(公告)号:US6010980A

    公开(公告)日:2000-01-04

    申请号:US29994

    申请日:1998-03-13

    CPC分类号: C07D213/61 A01N43/40

    摘要: Substituted 2-phenylpyridines I and their salts ##STR1## where n=0, 1;R.sup.1 =halogen, C.sub.1 -C.sub.4 -haloalkyl;R.sup.2 and R.sup.3 =H, halogen;R.sup.4 =CN, halogen;R.sup.5 =--CO--O-(C.sub.1 -C.sub.4 -alkylene)-CO--OR.sup.6, --CO--O-(C.sub.1 -C.sub.4 -alkylene)-CO--N(R.sup.7)R.sup.8, --O-(C.sub.1 -C.sub.4 -alkylene)-CO--O-(C.sub.1 -C.sub.4 -alkylene)-CO--OR.sup.6, --O-(C.sub.1 -C.sub.4 -alkylene)-CO--O-(C.sub.1 -C.sub.4 -alkylene)-CO--N(R.sup.7) R.sup.8, --S-(C.sub.1 -C.sub.4 -alkylene)-CO--O-(C.sub.1 -C.sub.4 -alkylene)-CO--OR.sup.6 or --S-(C.sub.1 -C.sub.4 -alkylene)-CO--O-(C.sub.1 -C.sub.4 -alkylene)-CO--N(R.sup.7)R.sup.8 ;R.sup.6 =H, C.sub.1 -C.sub.4 -alkyl, C.sub.1 -C.sub.4 -alkoxy-C.sub.1 -C.sub.4 -alkyl, C.sub.2 -C.sub.4 -alkenyl, C.sub.3 -C.sub.4 -alkynyl;R.sup.7 =H, C.sub.1 -C.sub.4 -alkyl, carboxy-C.sub.1 -C.sub.4 -alkyl, C.sub.1 -C.sub.4 -alkoxycarbonyl-C.sub.1 -C.sub.4 -alkyl;R.sup.8 =H or C.sub.1 -C.sub.4 -alkyl,are used as herbicides and for the desiccation/defoliation of plants.

    摘要翻译: PCT No.PCT / EP96 / 03949 Sec。 371日期1998年3月13日 102(e)1998年3月13日PCT PCT 1996年9月9日PCT公布。 出版物WO97 / 11059 日期1997年3月27日取代的2-苯基吡啶I及其盐,其中n = 0,1; R1 =卤素,C1-C4卤代烷基; R2和R3 = H,卤素; R4 = CN,卤素; R5 = -CO-O-(C1-C4-亚烷基)-CO-OR6,-CO-O-(C1-C4-亚烷基)-CO-N(R7)R8,-O-(C1-C4-亚烷基) -CO-O-(C1-C4-亚烷基)-CO-OR6,-O-(C1-C4-亚烷基)-CO-O-(C1-C4-亚烷基)-CO-N(R7)R8,-S - (C1-C4-亚烷基)-CO-O-(C1-C4-亚烷基)-CO-OR6或-S-(C1-C4-亚烷基)-CO-O-(C1-C4-亚烷基) N(R 7)R 8; R6 = H,C1-C4-烷基,C1-C4-烷氧基-C1-C4-烷基,C2-C4-烯基,C3-C4-炔基; R7 = H,C1-C4-烷基,羧基-C1-C4-烷基,C1-C4-烷氧基羰基-C1-C4-烷基; R8 = H或C1-C4烷基,用作除草剂和用于植物的干燥/脱叶。

    Substituted (4-brompyrazole-3-yl) benzazoles

    公开(公告)号:US06482774B1

    公开(公告)日:2002-11-19

    申请号:US09673996

    申请日:2000-10-25

    IPC分类号: C07D41704

    摘要: Substituted (4-bromopyrazol-3-yl)benzazoles I and their salts where R1=H, C1-C4-alkyl, C1-C4-haloalkyl; R2=CN, Cl-C4-alkyl, C1-C4-haloalkyl, C1-C4-alkoxy, C1-C4-haloalkoxy, C1-C4-alkylthio, C1-C4-haloalkylthio, C1-C4-alkylsulfinyl, C1-C4-haloalkylsulfinyl, C1-C4-alkylsulfonyl, C1-C4-haloalkylsulfonyl; R4=H, halogen; R5=H, CN, halogen, C1-C4-alkyl, C1-C4-haloalkyl, C1-C4-alkoxy or C1-C4-haloalkoxy; Z=—N═C(XR6)—O— or —N═C(XR6)—S—, attached to &agr; via the nitrogen, oxygen or sulfur; X=a chemical bond, oxygen, sulfur, —S(O)—, —SO2—, —NH— or —N(R7)—; R6, R7=Cl-C6-alkyl, Cl-C6-haloalkyl, cyano-Cl-C4-alkyl, hydroxy-C1-C4-alkyl, C3-C6-alkenyl, cyano-C3-C6-alkenyl, C3-C6-haloalkenyl, C3-C6-alkynyl, cyano-C3-C6-alkynyl, C3-C6-haloalkynyl, C1-C4-alkoxy-C1-C4-alkyl, C1-C4-haloalkoxy-C1-C4-alkyl, C3-C4-alkenyloxy-C1-C4-alkyl, C3-C4-alkynyloxy-C1-C4-alkyl, C3-C8-cycloalkyloxy-C1-C4-alkyl, amino-Cl-C4-alkyl, C1-C4-alkylamino-C1-C4-alkyl, di(C1-C4-alkyl)amino-C1-C4-alkyl, Cl-C4-alkylthio-C1-C4-alkyl, C1-C4-haloalkylthio-C1-C4-alkyl, C3-C4-alkenylthio-C1-C4-alkyl, C3-C4-alkynylthio-C1-C4-alkyl, C1-C4-alkylsulfinyl-Cl-C4-alkyl, C1-C4-haloalkylsulfinyl-C1-C4-alkyl, C3-C4-alkenylsulfinyl-C1-C4-alkyl, C3-C4-alkynylsulfinyl-C1-C4-alkyl, C1-C4-alkylsulfonyl-C1-C4-alkyl, C1-C4-haloalkylsulfonyl-C1-C4-alkyl, C3-C4-alkenylsulfonyl-C1-C4-alkyl, C3-C4-alkynylsulfonyl-C1-C4-alkyl, hydroxycarbonyl-C1-C4-alkyl, C1-C4-alkoxycarbonyl-C1-C4-alkyl, which may carry a CN or C1-C4-alkoxycarbonyl group, C1-C4-alkylthiocarbonyl-C1-C4-alkyl, aminocarbonyl-C1-C4-alkyl, C1-C4-alkylaminocarbonyl-C1-C4-alkyl, di(C1-C4-alkyl)aminocarbonyl-C1-C4-alkyl, di(C1-C4-alkyl)-phosphonyl-C1-C4-alkyl, C1-C4-alkoxyimino-C1-C4-alkyl, C3-C4-alkenyloxyimino-C1-C4-alkyl, unsubstituted or substituted C3-C8-cycloalkyl, C3-C8-cycloalkyl-C1-C4-alkyl, phenyl, phenyl-C1-C4-alkyl, 3- to 7-membered heterocyclyl or heterocyclyl-C1-C4-alkyl, where each cycloalkyl and each heterocyclyl ring may contain a CO or CS ring member; if X=a chemical bond, —O—, —S—, —NH— or —N(R7)—, R6 may also be C1-C4-alkylcarbonyl, C1-C4-haloalkylcarbonyl, C1-C4-alkoxycarbonyl, C1-C4-alkylsulfonyl or C1-C4-haloalkylsulfonyl; if X=a chemical bond, R6 may furthermore be CN, SH, NH2, halogen, —CH2—CH(halogen)-R8, —CH═CH—R8 or —CH═C(halogen)-R8, where R8=COOH, C1-C4-alkoxycarbonyl, C1-C4-alkylthiocarbonyl, CONH2, C1-C4-alkylaminocarbonyl, di(C1-C4-alkyl)aminocarbonyl or di(C1-C4-alkyl)phosphonyl; or R6+R7=an unsubstituted or substituted 1,3-propylene, tetramethylene, pentamethylene or ethyleneoxyethylene chain. Use: As herbicides; for the desiccation/defoliation of plants.