公开(公告)号：US5683964A

公开(公告)日：1997-11-04

申请号：US504862

申请日：1995-07-20

申请人： Yoichi Kanda ,  Hideo Arabori ,  Masato Arahira ,  Tsutomu Sato

发明人： Yoichi Kanda ,  Hideo Arabori ,  Masato Arahira ,  Tsutomu Sato

IPC分类号： C07D491/18 ,  A01N47/36 ,  C07D403/12 ,  C07D521/00 ,  A01N43/54 ,  A01N43/66 ,  A01N43/68 ,  C07D251/42

CPC分类号： C07D521/00 ,  A01N47/36

摘要： An N-(substituted amino)imide derivative represented by the formula (I) is a novel compound which can be utilized as an effective ingredient of herbicidal compositions. ##STR1## wherein, R.sup.1 is hydrogen atom, C.sub.1 -C.sub.4 alkyl group, C.sub.7 -C.sub.9 aralkyl group, C.sub.1 -C.sub.4 haloalkyl group, (C.sub.1 -C.sub.4 alkyl)carbonyl group or (C.sub.1 -C.sub.4 alkyl)sulfonyl group; A represents a structure selected from the group consisting of the following formulas (A-1), (A-2), (A-3), (A-4) and (A-5) ##STR2## wherein R.sup.2 and R.sup.3 in the formula (A-1) are independently hydrogen atom or C.sub.1 -C.sub.4 alkyl group, but not R.sup.2 =R.sup.3 =H, R.sup.4 in the formula (A-4) is halogen atom, C.sub.1 -C.sub.4 alkyl group and/or nitro group, m is an integer of 0-4, the substituents of m not less than 2 being same or different; X.sup.1 and X.sup.2 are independently hydrogen atom, halogen atom, C.sub.1 -C.sub.4 alkyl group, C.sub.1 -C.sub.4 alkoxy group, C.sub.1 -C.sub.4 alkylthio group, C.sub.1 -C.sub.4 haloalkyl group, C.sub.1 -C.sub.4 haloalkoxy group, C.sub.1 -C.sub.4 haloalkylthio group, C.sub.2 -C.sub.4 alkoxyalkyl group, C.sub.2 -C.sub.4 thioalkoxyalkyl group or NR.sup.7 R.sup.8, wherein R.sup.7 and R.sup.8 are independently hydrogen atom, C.sub.1 -C.sub.4 alkyl group or C.sub.1 -C.sub.4 alkoxy group; and Z is nitrogen atom or CH.

摘要翻译： 由式（I）表示的N-（取代氨基）酰亚胺衍生物是可用作除草组合物的有效成分的新型化合物。 （Ⅰ）其中R1是氢原子，C1-C4烷基，C7-C9芳烷基，C1-C4卤代烷基，（C1-C4烷基）羰基或（C1-C4烷基）磺酰基; （A-1），（A-2），（A-3），（A-4）和（A-5）（A-1） （A-2）（A-3）（A-4）（A-4）（A-5）其中式（A-1）中的R 2和R 3独立地为氢原子或C 1 -C4烷基，但不是R2 = R3 = H，式（A-4）中的R4是卤素原子，C1-C4烷基和/或硝基，m是0-4的整数，m的取代基 不少于2个相同或不同; X1和X2独立地为氢原子，卤素原子，C1-C4烷基，C1-C4烷氧基，C1-C4烷硫基，C1-C4卤代烷基，C1-C4卤代烷氧基，C1-C4卤代烷硫基，C2-C4 烷氧基烷基，C 2 -C 4硫代烷氧基烷基或NR 7 R 8，其中R 7和R 8独立地为氢原子，C 1 -C 4烷基或C 1 -C 4烷氧基; Z是氮原子或CH。

公开(公告)号：US5604178A

公开(公告)日：1997-02-18

申请号：US323413

申请日：1994-10-14

申请人： Yoichi Kanda ,  Hideo Arabori ,  Masato Arahira ,  Tsutomu Sato

发明人： Yoichi Kanda ,  Hideo Arabori ,  Masato Arahira ,  Tsutomu Sato

IPC分类号： C07D403/12 ,  A01N43/50 ,  A01N43/64 ,  A01N47/36 ,  C07D207/50 ,  C07D403/04 ,  C07D521/00 ,  A01N43/66 ,  C07D251/42

CPC分类号： C07D521/00 ,  A01N47/36 ,  C07D207/50 ,  C07D403/04

摘要： This invention is to provide an N-(substituted amino)pyrrole derivative represented by the formula (I): which is used as an effective ingredient of herbicidal compositions: ##STR1## wherein R.sup.2, R.sup.3, R.sup.4 and R.sup.5 is independently hydrogen atom, halogen atom, C.sub.1 -C.sub.4 alkyl group, (C.sub.1 -C.sub.4 alkyl)carbonyl group, (C.sub.3 -C.sub.6 cycloalkyl) carbonyl group, (C.sub.1 -C.sub.4 haloalkyl)carbonyl group, (C.sub.3 -C.sub.5 alkenyl)carbonyl group, benzoyl group which may be substituted with 1-3 halogen atoms and/or C.sub.1 -C.sub.4 alkyl groups, N,N-[(di-C.sub.1 -C.sub.4 alkyl)amino]carbonyl group, (C.sub.1 -C.sub.4 alkoxy)carbonyl group, etc., X.sup.1 and X.sup.2 are independently hydrogen atom, halogen atom, C.sub.1 -C.sub.4 alkyl group, C.sub.1 -C.sub.4 alkoxy group, etc., and Z is nitrogen atom or CH.

摘要翻译： 本发明提供由式（I）表示的N-（取代氨基）吡咯衍生物：其用作除草组合物的有效成分：其中R2，R3，R4和R5独立地为氢 原子，卤素原子，C1-C4烷基，（C1-C4烷基）羰基，（C3-C6环烷基）羰基，（C1-C4卤代烷基）羰基，（C3-C5烯基）羰基，苯甲酰基 可以被1-3个卤素原子和/或C 1 -C 4烷基，N，N - [（二-C 1 -C 4烷基）氨基]羰基，（C 1 -C 4烷氧基）羰基等取代，X 1和 X2独立地为氢原子，卤素原子，C1-C4烷基，C1-C4烷氧基等，Z为氮原子或CH。

公开(公告)号：US4973353A

公开(公告)日：1990-11-27

申请号：US162699

申请日：1988-03-01

申请人： Takafumi Shida ,  Hideo Arabori ,  Takeo Watanabe ,  Yoshikazu Kubota ,  Isao Ichinose ,  Yoichi Kanda ,  Shiro Yamazaki ,  Hiroyasu Shinkawa

发明人： Takafumi Shida ,  Hideo Arabori ,  Takeo Watanabe ,  Yoshikazu Kubota ,  Isao Ichinose ,  Yoichi Kanda ,  Shiro Yamazaki ,  Hiroyasu Shinkawa

IPC分类号： A01N43/653 ,  C07C205/34 ,  C07C205/35 ,  C07C217/76 ,  C07D249/10

CPC分类号： C07C205/34 ,  A01N43/653 ,  C07C205/35 ,  C07C217/76 ,  C07D249/10

摘要： Disclosed herein is a derivative of 1,5-diphenyl-1H-1,2,4-triazole-3-carboxamide represented by the formula (I): ##STR1## wherein R is a straight-chain alkyl group having 1 to 10 carbon atoms which is non-substituted or substituted with 1 to 19 fluorine atoms, a branched alkyl group having 3 to 10 carbon atoms which is non-substituted or substituted with 1 to 19 fluorine atoms, a cyclic alkyl group having 3 to 10 carbon atoms, an alkyl group having 1 to 3 carbon atoms which is substituted with an alicyclic structure having 3 to 7 carbon atoms, a phenyl group or an aralkyl group having 7 to 9 carbon atoms; X.sup.1 is a halogen or an alkyl group having 1 to 3 carbon atoms; X.sup.2 is a hydrogen, a halogen or an alkyl group having 1 to 3 carbon atoms; Y.sup.1 is a hydrogen or a fluorine; and Y.sup.2 is a hydrogen or a fluorine, and the herbicidal compositions containing said derivatives as active ingredient therefor.The derivative of 1,5-diphenyl-1H-1,2,4-triazole-3-carboxamide represented by the formula (I) of the present invention is the compound having high herbicidal activity and also showing excellent selectivity for killing weeds alone without doing any serious harm to the crops such as rice, wheat and corn.

公开(公告)号：US4492597A

公开(公告)日：1985-01-08

申请号：US379944

申请日：1982-05-19

申请人： Katsumichi Aoki ,  Yoichi Kanda ,  Keigo Satake ,  Hiroyasu Shinkawa

发明人： Katsumichi Aoki ,  Yoichi Kanda ,  Keigo Satake ,  Hiroyasu Shinkawa

IPC分类号： A01N43/653 ,  C07D249/10 ,  A01N43/64

CPC分类号： C07D249/10 ,  A01N43/653

摘要： A compound of 1,5-disubstituted 1,2,4-triazole-3-carboxamide represented by the general formula; ##STR1## wherein R.sup.1 is alkyl of one to three carbon atoms, chloro, fluoro, iodo, trifluoromethyl or nitro, R.sup.2 is hydrogen, methyl or chloro, R.sup.3 is hydrogen or methyl is provided in the invention, which shows an excellent herbicidal activity.

摘要翻译： 由通式表示的1,5-二取代的1,2,4-三唑-3-甲酰胺的化合物; 其中R 1是1-3个碳原子的烷基，氯，氟，碘，三氟甲基或硝基，R 2是氢，甲基或氯，R 3是氢或甲基，其显示出优异的除草活性 。

公开(公告)号：US06200933B1

公开(公告)日：2001-03-13

申请号：US09331734

申请日：1999-08-09

申请人： Hisashi Kanno ,  Yoichi Kanda ,  Kazuhiko Sunagawa ,  Takayoshi Eizuka

发明人： Hisashi Kanno ,  Yoichi Kanda ,  Kazuhiko Sunagawa ,  Takayoshi Eizuka

IPC分类号： A01N4340

CPC分类号： C07D213/79 ,  A01N43/40

摘要： An agricultural or horticultural fungicide containing 6-(unsubstituted or substituted) phenoxy picolinic acid represented by the general formula (I), as an effective ingredient. wherein R is a halogen atom, a C1 to C4 alkyl group, a C1 to C4 haloalkyl group, a C1 to C4 alkoxy group, a C1 to C4 haloalkoxy group, a C1 to C4 alkylthio group, a C1 to C4 alkylamino group, a di(C1 to C4 alkyl)amino group or a C7 to C8 aralkyl(C1 to C4 alkyl)amino group; n2 is an integer of 0 to 3; Y is a C1 to C4 alkyl group, a C1 to C4 haloalkyl group, a C1 to C4 alkoxy group, a C1 to C4 haloalkoxy group, a C1 to C4 alkylthio group, a C1 to C4 haloalkylthio group or a halogen atom; and m is an integer of 0 to 5, and when m and n2 are not less than 2, Rs and Ys may be the same or different, respectively. The compound is useful as an effective ingredient of agricultural or horticultural fungicides.

摘要翻译： 一种含有由通式（I）表示的6-（未取代或取代的）苯氧基吡啶甲酸作为有效成分的农业或园艺杀真菌剂，其中R为卤素原子，C1至C4烷基，C1至C4卤代烷基， C1〜C4烷氧基，C1〜C4卤代烷氧基，C1〜C4烷硫基，C1〜C4烷基氨基，二（C1〜C4烷基）氨基或C7〜C8芳烷基（C1〜C4烷基） 氨基; n2为0〜3的整数，Y为C1〜C4烷基，C1〜C4卤代烷基，C1〜C4烷氧基，C1〜C4卤代烷氧基，C1〜C4烷硫基， C1〜C4卤代烷硫基或卤素原子; andm为0〜5的整数，当m和n2不小于2时，Rs和Y可以相同或不同。化合物可用作农业或园艺杀真菌剂的有效成分。

公开(公告)号：US5612287A

公开(公告)日：1997-03-18

申请号：US467441

申请日：1995-06-06

申请人： Yoichi Kanda ,  Hideo Arabori ,  Masato Arahira ,  Tsutomu Sato

发明人： Yoichi Kanda ,  Hideo Arabori ,  Masato Arahira ,  Tsutomu Sato

IPC分类号： C07D403/12 ,  A01N43/50 ,  A01N43/64 ,  A01N47/36 ,  C07D207/50 ,  C07D403/04 ,  C07D521/00 ,  A01N43/54

CPC分类号： C07D521/00 ,  A01N47/36 ,  C07D207/50 ,  C07D403/04

摘要： This invention is to provide an N-(substituted amino)pyrrole derivative represented by the formula (I): which is used as an effective ingredient of herbicidal compositions: ##STR1## wherein R.sup.2, R.sup.3, R.sup.4 and R.sup.5 is independently hydrogen atom halogen atom, C.sub.1 -C.sub.4 alkyl group, (C.sub.1 -C.sub.4 alkyl)carbonyl group, (C.sub.3 -C.sub.6 cycloalkyl)carbonyl group, (C.sub.1 -C.sub.4 haloalkyl)carbonyl group, (C.sub.3 -C.sub.5 alkenyl)carbonyl group, benzoyl group which may be substituted with 1-3 halogen atoms and/or C.sub.1 -C.sub.4 alkyl groups, N,N-[(di-C.sub.1 -C.sub.4 alkyl)amino]carbonyl group, (C.sub.1 -C.sub.4 alkoxy)carbonyl group, etc., X.sup.1 and X.sup.2 are independently hydrogen atom, halogen atom, C.sub.1 -C.sub.4 alkyl group, C.sub.1 -C.sub.4 alkoxy group, etc., and Z is nitrogen atom or CH.

摘要翻译： 本发明提供由式（I）表示的N-（取代氨基）吡咯衍生物：其用作除草组合物的有效成分：其中R2，R3，R4和R5独立地为氢 原子卤素原子，C1-C4烷基，（C1-C4烷基）羰基，（C3-C6环烷基）羰基，（C1-C4卤代烷基）羰基，（C3-C5烯基）羰基，苯甲酰基 被1-3个卤素原子和/或C1-C4烷基取代，N，N - [（二C1-C4烷基）氨基]羰基，（C1-C4烷氧基）羰基等，X1和X2 独立地为氢原子，卤素原子，C1-C4烷基，C1-C4烷氧基等，Z为氮原子或CH。

公开(公告)号：US5162583A

公开(公告)日：1992-11-10

申请号：US588996

申请日：1990-09-27

申请人： Takafumi Shida ,  Hideo Arabori ,  Takeo Watanabe ,  Yoshikazu Kubota ,  Isao Ichinose ,  Yoichi Kanda ,  Shiro Yamazaki ,  Hiroyasu Shinkawa

发明人： Takafumi Shida ,  Hideo Arabori ,  Takeo Watanabe ,  Yoshikazu Kubota ,  Isao Ichinose ,  Yoichi Kanda ,  Shiro Yamazaki ,  Hiroyasu Shinkawa

IPC分类号： A01N43/653 ,  C07C201/12 ,  C07C205/33 ,  C07C205/34 ,  C07C205/35 ,  C07C217/76 ,  C07D249/10

CPC分类号： A01N43/653 ,  C07C205/33 ,  C07C205/34 ,  C07C205/35 ,  C07C217/76 ,  C07D249/10

摘要： Disclosed herein are the derivative of benzyl ether represented by the formula (I) ##STR1## which is useful as an intermediate compound of the derivatives of 1,5-diphenyl-1H-1,2,4- triazole-3-carboxamide represented by the formula (II), ##STR2## wherein R is a straight-chain alkyl group having 1 to 10 carbon atoms which is non-substituted or substituted with 1 to 19 fluorine atoms, a branched alkyl group having 3 to 10 carbon atoms which is non-substituted or substituted with 1 to 19 fluorine atoms, a cyclic alkyl group having 3 to 10 carbon atoms, an alkyl group having 1 to 3 carbon atoms which is substituted with an alicyclic structure having 3 to 7 carbon atoms, a phenyl group or an aralkyl group having 7 to 9 carbon atoms; X.sup.1 is a halogen or an alkyl group having 1 to 3 carbon atoms; X.sup.2 is a hydrogen, a halogen or an alkyl group having 1 to 3 carbon atoms; Y.sup.1 is a hydrogen or a fluorine; Y.sup.2 is a hydrogen or a fluorine; and Z is a nitro group or an amino group.

摘要翻译： 本文公开了由式（I）表示的苄基醚衍生物，其可用作1,5-二苯基-1H-1,2,4-三唑-3-基的衍生物的中间体化合物， 由式（II）表示的羧酰胺，其中R是未取代或被1〜19个氟原子取代的碳原子数为1〜10的直链烷基，具有3个 未取代或被1〜19个氟原子取代的10个碳原子，碳原子数3〜10的环状烷基，碳原子数1〜3的被碳数3〜7的脂环结构取代的烷基 原子，苯基或碳原子数为7〜9的芳烷基; X1是卤素或具有1至3个碳原子的烷基; X 2是氢，卤素或具有1至3个碳原子的烷基; Y1是氢或氟; Y2是氢或氟; Z为硝基或氨基。

公开(公告)号：US4968345A

公开(公告)日：1990-11-06

申请号：US162934

申请日：1988-03-02

申请人： Takafumi Shida ,  Hideo Arabori ,  Takeo Watanabe ,  Yoichi Kanda ,  Shiro Yamazaki ,  Hiroyasu Shinkawa

发明人： Takafumi Shida ,  Hideo Arabori ,  Takeo Watanabe ,  Yoichi Kanda ,  Shiro Yamazaki ,  Hiroyasu Shinkawa

IPC分类号： A01N37/52 ,  C07C67/00 ,  C07C239/00 ,  C07C257/20 ,  C07C257/22

CPC分类号： A01N37/52

摘要： Disclosed herein is a phenylhydrazone derivative of oxamide represented by the formula (I): ##STR1## wherein R.sup.1 is straight-chain alkyl group having 2 to 10 carbon atoms, branched alkyl group or cyclic alkyl group having 3 to 10 carbon atoms, alkyl group having 1 to 3 carbon atoms which is substituted with an alicyclic structure having 3 to 7 carbon atoms, phenyl group, halogen-substituted phenyl group, aralkyl group having 7 to 9 carbon atoms, alkenyl group having 3 to 6 carbon atoms, alkyl group having 2 to 4 carbon atoms which is substituted with alkoxy group having 1 to 4 carbon atoms, or alkyl group having 2 to 10 carbon atoms which is substituted with 1 to 19 fluorine atoms; and R.sup.2 is hydrogen, fluorine, chlorine, methyl group or methoxy group, and a herbicidal composition containing the derivative as active ingredient. The phenylhydrazone derivative of oxamide represented by the formula (I) of the present invention shows a high herbicidal activity and also have an excellent selectivity allowing killing of weeds alone without doing any practical harm to the crops such as rice, wheat and corn.