Derivatives of dihydrotriazole, and herbicidal compositions containing
the same as an active ingredient
    2.
    发明授权
    Derivatives of dihydrotriazole, and herbicidal compositions containing the same as an active ingredient 失效
    二氢三唑衍生物和含有其作为活性成分的除草组合物

    公开(公告)号:US4902805A

    公开(公告)日:1990-02-20

    申请号:US820948

    申请日:1986-01-21

    摘要: Disclosed herein are a derivative of dihydrotriazole represented by the general formula (I): ##STR1## wherein R.sup.1 represents an amino group, lower alkoxy group, or lower alkyl amino group, R.sup.2 represents a hydrogen atom, halogen atom, or lower alkyl group and R.sup.3 represents a hydrogen atom, lower alkyl group, benzyl group, furyl group, phenyl group or phenyl group substituted with a halogen atom, hydroxyl group, carboxyl group, methoxycarbonyl group, lower alkyl group or lower alkoxy group, and a herbicidal composition containing as an active ingredient at least one of the derivatives of dihydrotriazole.

    摘要翻译: 本文公开了由通式(I)表示的二氢三唑衍生物:其中R 1表示氨基,低级烷氧基或低级烷基氨基,R 2表示氢原子,卤原子或低级 烷基,R 3表示氢原子,低级烷基,苄基,呋喃基,苯基或被卤素原子,羟基,羧基,甲氧基羰基,低级烷基或低级烷氧基取代的苯基,除草 组合物,其含有作为活性成分的二氢三唑衍生物中的至少一种。

    Herbicidal composition containing a derivative of 1,2,4-triazole as an
active ingredient
    4.
    发明授权
    Herbicidal composition containing a derivative of 1,2,4-triazole as an active ingredient 失效
    含有1,2,4-三唑衍生物作为活性成分的除草组合物

    公开(公告)号:US4795484A

    公开(公告)日:1989-01-03

    申请号:US858531

    申请日:1986-04-24

    IPC分类号: A01N43/653 C07D249/10

    CPC分类号: A01N43/653 C07D249/10

    摘要: Disclosed herein is herbicidal composition comprising a derivative of 1,2,4-triazole as an active ingredient, represented by the general formula (I): ##STR1## wherein R.sup.1 represents a hydrogen atom, a halogen atom or a C.sub.1 -C.sub.2) alkyl group; R.sup.2 represents a hydrogen atom, a halogen atom, a (C.sub.1 -C.sub.2) alkyl group fluoromethyl group (--CH.sub.2 F),3,3,3-trifluoropopyl group, methoxy group, cyano group, methoxymethyl group, methylthio group, methoxycarbonyl group or isopropoxycarbonyl group and R.sup.3 represents a thiocarbamoyl group or a group represented by the general formula (II): ##STR2## wherein R.sup.4 represents a hydrogen atom, a (C.sub.1 -C.sub.2) alkyl group or a hydroxy (C.sub.1 -C.sub.2) alkyl group and R.sup.5 represents a hydrogen atom, a C.sub.1 -C.sub.2) alkyl group, halogeno (C.sub.1 -C.sub.2) alkyl group, hydroxy (C.sub.1 -C.sub.2) alkyl group, cyanomethyl group, acetyl group, halogenoacetyl group, methoxyacetyl group, amino group, phenyl group, methoxy group, hydroxyl group, (C.sub.2 -C.sub.3) alkenyl group, halogeno (C.sub.2 -C.sub.3) alkenyl group, isopropylcarbonyl group, methylthiocarbamoyl group or 2-methoxyethyl group, the proviso that R.sup.2 is not a hydrogen atom, halogen atom or (C.sub.1 -C.sub.2) alkyl group when both of R.sup.4 and R.sup.5 represent hydrogen atoms, and herbicidally acceptable carrier(s) or diluent(s).

    摘要翻译: 本文公开了包含由通式(I)表示的1,2,4-三唑衍生物作为活性成分的除草组合物:其中R1表示氢原子,卤素原子或C1- C2)烷基; R2表示氢原子,卤素原子,(C1-C2)烷基氟甲基(-CH2F),3,3,3-三氟戊酰基,甲氧基,氰基,甲氧基甲基,甲硫基,甲氧基羰基或异丙氧基羰基 基团,R 3表示硫代氨基甲酰基或由通式(II)表示的基团:其中R 4表示氢原子,(C 1 -C 2)烷基或羟基(C 1 -C 2)烷基) R5为氢原子,C1-C2)烷基,卤代(C1-C2)烷基,羟基(C1-C2)烷基,氰基甲基,乙酰基,卤代乙酰基,甲氧基乙酰基,氨基,苯基 ,甲氧基,羟基,(C2-C3)烯基,卤代(C2-C3)烯基,异丙基羰基,甲硫基氨基甲酰基或2-甲氧基乙基,条件是R2不是氢原子,卤素原子或(C1 -C 2)烷基,当R4和R5都表示氢原子,除草可接受的载体或稀释剂( s)。

    Herbicidal tetrahydrobenzothiazolyl-1,3,5-triazinone derivatives and
compositions thereof
    6.
    发明授权
    Herbicidal tetrahydrobenzothiazolyl-1,3,5-triazinone derivatives and compositions thereof 失效
    除草四氢苯并噻唑基-1,3,5-三嗪酮衍生物及其组合物

    公开(公告)号:US4624698A

    公开(公告)日:1986-11-25

    申请号:US695178

    申请日:1985-01-25

    CPC分类号: C07D417/04 A01N43/78

    摘要: Disclosed herein is a derivative of tetrahydrobenzothiazolyl-1,3,5-triazinone represented by the formula (I): ##STR1## wherein R is a chemical group selected from the group consisting of 1-phenylethyl, 1-methylpropyl, 2-methylpropyl, allyl, 2-propynyl, cyclopropyl, cyclopentyl, phenyl, ethoxycarbonylmethyl, 2-tetrahydrofurylmethyl, 2-acetoxyethyl, 2-chloroethyl, 2-cyanoethyl, 2-hydroxyethyl, 2-methoxyethyl, 2,2-dimethoxyethyl, 2-(propionyloxy)ethyl, 2-(ethoxycarbonyl)ethyl, 2-(4-chlorobenzoyloxy)ethyl, 1-hydroxymethyl)propyl, 3-hydroxypropyl, 3-methoxypropyl, 3-acetoxypropyl, 3-morpholinopropyl and 3-(2-methylpiperidino)propyl, and a herbicidal composition containing the derivative as an active ingredient thereof.

    摘要翻译: 本文公开的是由式(I)表示的四氢苯并噻唑基-1,3,5-三嗪酮的衍生物:其中R是选自1-苯基乙基,1-甲基丙基,2- 甲基丙基,烯丙基,2-丙炔基,环丙基,环戊基,苯基,乙氧基羰基甲基,2-四氢呋喃基甲基,2-乙酰氧基乙基,2-氯乙基,2-氰基乙基,2-羟基乙基,2-甲氧基乙基,2,2-二甲氧基乙基,2-( 丙氧基)乙基,2-(乙氧基羰基)乙基,2-(4-氯苯甲酰氧基)乙基,1-羟基甲基)丙基,3-羟丙基,3-甲氧基丙基,3-乙酰氧基丙基,3-吗啉代丙基和3-(2-甲基哌啶子基) 和含有该衍生物作为其有效成分的除草组合物。

    Process for the manufacture of triazolecarboxamide
    9.
    发明授权
    Process for the manufacture of triazolecarboxamide 失效
    三唑甲酰胺的制备方法

    公开(公告)号:US5434268A

    公开(公告)日:1995-07-18

    申请号:US221688

    申请日:1994-03-31

    IPC分类号: C07D249/08 C07D249/10

    CPC分类号: C07D249/10

    摘要: A process for the manufacture of 1-(substituted or unsubstituted)phenyl-5-(substituted or unsubstituted)-phenyl-1H-1,2,4-triazole-3-carboxamide of the formula (I), which comprises heating 2-(substituted or unsubstituted)phenyl-4,5-oxazoledione 4-(substituted or unsubstituted)phenylhydrazone of the formula (II) and ammonia in water according to the following reaction formula, ##STR1## wherein A and B individually represent one or more substituted or unsubstituted phenyl groups. The target compound can be manufactured at a high purity and a high yield without using an organic solvent or an acidic compound.

    摘要翻译: 一种制备式(I)的1-(取代或未取代)苯基-5-(取代或未取代的) - 苯基-1H-1,2,4-三唑-3-甲酰胺的方法,该方法包括加热2- (II)的式(II)的(取代或未取代的)苯基-4,5-恶唑二酮4-(取代或未取代的)苯基腙和水中的氨,其中A和B各自表示一个 或更多取代或未取代的苯基。 目标化合物可以在不使用有机溶剂或酸性化合物的情况下以高纯度和高产率制造。

    Benzylether derivatives
    10.
    发明授权
    Benzylether derivatives 失效
    苄醚衍生物

    公开(公告)号:US5162583A

    公开(公告)日:1992-11-10

    申请号:US588996

    申请日:1990-09-27

    摘要: Disclosed herein are the derivative of benzyl ether represented by the formula (I) ##STR1## which is useful as an intermediate compound of the derivatives of 1,5-diphenyl-1H-1,2,4- triazole-3-carboxamide represented by the formula (II), ##STR2## wherein R is a straight-chain alkyl group having 1 to 10 carbon atoms which is non-substituted or substituted with 1 to 19 fluorine atoms, a branched alkyl group having 3 to 10 carbon atoms which is non-substituted or substituted with 1 to 19 fluorine atoms, a cyclic alkyl group having 3 to 10 carbon atoms, an alkyl group having 1 to 3 carbon atoms which is substituted with an alicyclic structure having 3 to 7 carbon atoms, a phenyl group or an aralkyl group having 7 to 9 carbon atoms; X.sup.1 is a halogen or an alkyl group having 1 to 3 carbon atoms; X.sup.2 is a hydrogen, a halogen or an alkyl group having 1 to 3 carbon atoms; Y.sup.1 is a hydrogen or a fluorine; Y.sup.2 is a hydrogen or a fluorine; and Z is a nitro group or an amino group.

    摘要翻译: 本文公开了由式(I)表示的苄基醚衍生物,其可用作1,5-二苯基-1H-1,2,4-三唑-3-基的衍生物的中间体化合物, 由式(II)表示的羧酰胺,其中R是未取代或被1〜19个氟原子取代的碳原子数为1〜10的直链烷基,具有3个 未取代或被1〜19个氟原子取代的10个碳原子,碳原子数3〜10的环状烷基,碳原子数1〜3的被碳数3〜7的脂环结构取代的烷基 原子,苯基或碳原子数为7〜9的芳烷基; X1是卤素或具有1至3个碳原子的烷基; X 2是氢,卤素或具有1至3个碳原子的烷基; Y1是氢或氟; Y2是氢或氟; Z为硝基或氨基。