公开(公告)号：US20070149400A1

公开(公告)日：2007-06-28

申请号：US10582934

申请日：2004-12-15

申请人： Jordi Tormo i Blasco ,  Carsten Biettner ,  Bernd Muller ,  Markus Gewehr ,  Wassilios Grammenos ,  Thomas Grote ,  Joachim Rheinheimer ,  Peter Schafer ,  Frank Schieweck ,  Anja Schwogler ,  Oliver Wagner ,  Maria Scherer ,  Siegfried Strathmann ,  Ulrich Schofl ,  Reinhard Stierl

发明人： Jordi Tormo i Blasco ,  Carsten Biettner ,  Bernd Muller ,  Markus Gewehr ,  Wassilios Grammenos ,  Thomas Grote ,  Joachim Rheinheimer ,  Peter Schafer ,  Frank Schieweck ,  Anja Schwogler ,  Oliver Wagner ,  Maria Scherer ,  Siegfried Strathmann ,  Ulrich Schofl ,  Reinhard Stierl

IPC分类号： A01N43/90 ,  C07D487/04

CPC分类号： C07D487/04 ,  A01N43/90

摘要： Substituted triazolopyrimidines of the formula I in which the substituents are as defined below: L is hydrogen, chlorine or bromine; R1, R2 are hydrogen, alkyl, haloalkyl, cycloalkyl, halocycloalkyl, alkenyl, haloalkenyl, cycloalkenyl, halocycloalkenyl, alkynyl, haloalkynyl or phenyl, naphthyl or a five- or six-membered saturated, partially unsaturated or aromatic heterocycle which contains one to four heteroatoms from the group consisting of O, N and S, R1 and R2 together with the nitrogen atom to which they are attached may also form a five- or six-membered heterocyclyl or heteroaryl which is attached via N and may contain a further heteroatom from the group consisting of O, N and S as ring member and/or may be substituted as defined in the description; R3 is alkyl, haloalkyl, alkenyl, haloalkenyl, alkynyl, haloalkynyl, cycloalkyl, halocycloalkyl or phenylalkyl; R1, R2 and/or R3 may be substituted as defined in the description; X is halogen, cyano, alkyl, haloalkyl, alkoxy or haloalkoxy; processes and intermediates for preparing these compounds, compositions comprising them and their use for controlling phytopathogenic harmful fungi.

摘要翻译： 取代基如下定义的式I的取代三唑并嘧啶：L是氢，氯或溴; R 1，R 2是氢，烷基，卤代烷基，环烷基，卤代环烷基，烯基，卤代烯基，环烯基，卤代环烯基，炔基，卤代炔基或苯基，萘基或五或 含有一至四个由O，N和S杂原子组成的组的六元饱和，部分不饱和或芳族杂环，R 1和R 2连同氮 它们所连接的原子也可以形成通过N连接的五元或六元杂环基或杂芳基，并且可以含有作为环成员的O，N和S中的另外的杂原子和/或可被取代为 在说明书中定义; R 3是烷基，卤代烷基，烯基，卤代烯基，炔基，卤代炔基，环烷基，卤代环烷基或苯基烷基; R 1，R 2和/或R 3可以如说明书中所定义的取代; X是卤素，氰基，烷基，卤代烷基，烷氧基或卤代烷氧基; 制备这些化合物的方法和中间体，包含它们的组合物及其用于控制​​植物病原性有害真菌的用途。

公开(公告)号：US20060258685A1

公开(公告)日：2006-11-16

申请号：US10558251

申请日：2004-05-27

申请人： Olivier Wagner ,  Thomas Grote ,  Carsten Blettner ,  Markus Gewehr ,  Wassilios Grammenos ,  Andreas Gypser ,  Bernd Muller ,  Joachim Rheinheimer ,  Peter Schafer ,  Frank Schieweck ,  Anja Schwogler ,  Jordi Blasco ,  Alan Akers ,  John-Bryan Speakman ,  Michael Rack ,  Reinhard Stierl ,  Maria Scherer ,  Ulrich Schofl ,  Siegfried Strathmann

发明人： Olivier Wagner ,  Thomas Grote ,  Carsten Blettner ,  Markus Gewehr ,  Wassilios Grammenos ,  Andreas Gypser ,  Bernd Muller ,  Joachim Rheinheimer ,  Peter Schafer ,  Frank Schieweck ,  Anja Schwogler ,  Jordi Blasco ,  Alan Akers ,  John-Bryan Speakman ,  Michael Rack ,  Reinhard Stierl ,  Maria Scherer ,  Ulrich Schofl ,  Siegfried Strathmann

IPC分类号： A61K31/519 ,  C07D487/04

CPC分类号： C07D487/04 ,  A01N43/90

摘要： The invention relates to substituted pyrazolopyrimidines of formula (I) wherein the substituents have the following designations: L represents halogen, alkyl, halogenalkyl, alkenyl, alkoxy, amino, NHR, NR2, cyano, S(═O)nA1 or C(═O)A2, R representing alkyl or alkylcarbonyl, A1 representing hydrogen, hydroxy, alkyl, alkylamino or dialkylamino, n representing 0, 1 or 2, and A2 representing alkenyl, alkoxy, halogenalkoxy or one of the groups cited for A1; m represents 0 or 1 to 5; R1 represents alkyl, halogenalkyl, cycloalkyl, halogencycloalkyl, alkenyl, alkadienyl, halogenalkenyl, cycloalkenyl, alkinyl, halogenalkinyl or cycloalkinyl, phenyl, naphthyl, or a five-membered to ten-membered saturated, partially unsaturated or aromatic heterocycle containing between one and four heteroatoms from the group O, N or S; and R2 represents hydrogen or one of the groups cited for R1. Together with the nitrogen atom to which they are bonded, R1 and R2 can form a five-membered to six-membered ring that can be interrupted by an atom from the groups O, N and S, and R1 and/or R2 can also be substituted according to the description. Furthermore, in formula (I): X represents halogen, cyano, OH, alkyl, alkoxy or halogenalkoxy; Y represents a five-membered to ten-membered saturated, partially unsaturated or aromatic heterocycle according to the description, or a group X or another group according to the description; p represents 1 or 2, the groups Y being potentially different when p=2; and p represents 0, when X is according to the description. The invention also relates to methods and intermediate products for producing said compounds, agents containing the same, and the use thereof for controlling phytopathogenic fungi.

公开(公告)号：US20070117852A1

公开(公告)日：2007-05-24

申请号：US10582040

申请日：2004-12-22

申请人： Markus Gewehr ,  Bernd Muller ,  Thomas Grote ,  Wassilios Grammenos ,  Jordi Tormo i Blasco ,  Anja Schwogler ,  Joachim Rheinheimer ,  Carsten Blettner ,  Peter Schafer ,  Frank Schieweck ,  Oliver Wagner ,  John-Bryan Speakman ,  Jan Rether ,  Siegfried Strathmann ,  Reinhard Stierl

发明人： Markus Gewehr ,  Bernd Muller ,  Thomas Grote ,  Wassilios Grammenos ,  Jordi Tormo i Blasco ,  Anja Schwogler ,  Joachim Rheinheimer ,  Carsten Blettner ,  Peter Schafer ,  Frank Schieweck ,  Oliver Wagner ,  John-Bryan Speakman ,  Jan Rether ,  Siegfried Strathmann ,  Reinhard Stierl

IPC分类号： A01N43/56 ,  A01N43/40 ,  A01N43/78 ,  C07D213/24

CPC分类号： C07D213/82 ,  A01N43/40 ,  A01N43/56 ,  A01N43/78 ,  A01N47/48 ,  C07C251/38 ,  C07D207/34 ,  C07D231/14 ,  C07D263/34 ,  C07D277/56 ,  C07D279/12 ,  C07D307/30 ,  C07D307/54 ,  C07D307/71 ,  C07D333/38

摘要： The present invention relates to (hetero)cyclylcarboxanilides of the formula I, in which n is 0, 1, 2, 3 or 4; and m is 1, 2 or 3, Y is oxygen or sulfur; A is unsubstituted or substituted phenyl or is an at least monounsaturated, unsubstituted or substituted 5- or 6-membered heterocycle, R1, R2, R3m, R4m, R5 and R6 are as defined in claim 1, and their agriculturally useful salts. Moreover, the present invention relates to the use of the (hetero)cyclylcarboxanilides of the formula I and their agriculturally useful salts as fungicides, and to crop protection compositions comprising these compounds.

摘要翻译： 本发明涉及式（I）的（杂）环己基甲酰苯胺，其中n为0,1,2,3或4; m为1,2或3，Y为氧或硫; A是未取代或取代的苯基，或至少是一个不饱和的，未取代的或取代的5元或6元杂环，R 1，R 2，R 3， R 4，R 5，R 5和R 6如权利要求1所定义，及其农业上有用的盐。 此外，本发明涉及式I的（杂）环己基甲酰苯胺及其农业上有用的盐作为杀真菌剂，以及包含这些化合物的作物保护组合物的用途。

公开(公告)号：US20080032889A1

公开(公告)日：2008-02-07

申请号：US11630558

申请日：2005-06-14

申请人： Carsten Blettner ,  Markus Gewehr ,  Wassilios Grammenos ,  Thomas Grote ,  Udo Hunger ,  Bernd Muller ,  Matthias Niedenbruck ,  Joachim Rheinheimer ,  Peter Schafer ,  Frank Schieweck ,  Anja Schwogler ,  Oliver Wagner ,  Barbara Nave ,  Maria Scherer ,  Siegfried Strathmann ,  Ulrich Schofl ,  Reinhard Stierl

发明人： Carsten Blettner ,  Markus Gewehr ,  Wassilios Grammenos ,  Thomas Grote ,  Udo Hunger ,  Bernd Muller ,  Matthias Niedenbruck ,  Joachim Rheinheimer ,  Peter Schafer ,  Frank Schieweck ,  Anja Schwogler ,  Oliver Wagner ,  Barbara Nave ,  Maria Scherer ,  Siegfried Strathmann ,  Ulrich Schofl ,  Reinhard Stierl

IPC分类号： A01N43/90 ,  A01C1/06 ,  C07D487/04

CPC分类号： A01N43/90 ,  C07D487/04

摘要： Substituted triazolopyrimidines of the formula I in which the substituents are as defined below: R1 is alkyl, halocycloalkyl, alkenyl, cycloalkyl, cycloalkenyl, halocycloalkenyl, alkynyl, haloalkynyl or naphthyl, or a five- or six-membered saturated, partially unsaturated or aromatic heterocycle comprising one to four heteroatoms from the group consisting of O, N and S, R2 is hydrogen, alkyl or one of the groups mentioned under R1; R1 and/or R2 may carry one to four identical or different groups Ra: Ra is chlorine, bromine, iodine, cyano, nitro, hydroxyl, alkyl, alkylcarbonyl, cycloalkyl, alkoxy, haloalkoxy, alkoxycarbonyl, alkylthio, alkylamino, dialkyl-amino, alkenyl, cycloalkenyl, alkenyloxy, haloalkenyloxy, alkynyl, halo-alkynyl, alkynyloxy, haloalkynyloxy, cycloalkoxy, cycloalkenyloxy, oxyalkylenoxy, naphthyl, a five- to ten-membered saturated, partially unsaturated or aromatic heterocycle comprising one to four heteroatoms from the group consisting of O, N and S, where these aliphatic, alicyclic or aromatic groups for their part may be substituted according to the description; and X is halogen; processes for preparing these compounds, compositions comprising them and their use for controlling phytopathogenic harmful fungi.

摘要翻译： 取代基如下定义的式I的取代三唑并嘧啶：R 1是烷基，卤代环烷基，烯基，环烷基，环烯基，卤代环烯基，炔基，卤代炔基或萘基，或五或六元环， 包含一至四个由O，N和S组成的组的杂原子的2-元饱和的，部分不饱和的或芳族的杂环，R 2是氢，烷基或R 1上提到的基团之一， / SUP>; R 1和/或R 2可以携带一至四个相同或不同的基团R a是：R a是 氯，溴，碘，氰基，硝基，羟基，烷基，烷基羰基，环烷基，烷氧基，卤代烷氧基，烷氧基羰基，烷硫基，烷基氨基，二烷基氨基，烯基，环烯基，烯氧基，卤代烯氧基，炔基，卤代炔基，炔氧基，卤代炔氧基， 环烷氧基，环烯氧基，氧亚烷基氧基，萘基，五至十元饱和的部分不饱和或芳族杂环，其包含一至四个由O，N和S组成的组的杂原子，其中这些脂族，脂环族或芳族基团可以 根据描述进行替代; X为卤素; 制备这些化合物的方法，包含它们的组合物及其用于控制​​植物病原性有害真菌的用途。

公开(公告)号：US20070208038A1

公开(公告)日：2007-09-06

申请号：US10594738

申请日：2005-03-26

申请人： Carsten Blettner ,  Markus Gewehr ,  Wassilios Grammenos ,  Thomas Grote ,  Udo Hunger ,  Bernd Muller ,  Matthias Niedenbruck ,  Joachim Rheinheimer ,  Peter Schafer ,  Frank Schieweck ,  Anja Schwogler ,  Oliver Wagner ,  Michael Rack ,  Barbara Nave ,  Maria Scherer ,  Siegfried Strathmann ,  Ulrich Schofl ,  Reinhard Stierl

发明人： Carsten Blettner ,  Markus Gewehr ,  Wassilios Grammenos ,  Thomas Grote ,  Udo Hunger ,  Bernd Muller ,  Matthias Niedenbruck ,  Joachim Rheinheimer ,  Peter Schafer ,  Frank Schieweck ,  Anja Schwogler ,  Oliver Wagner ,  Michael Rack ,  Barbara Nave ,  Maria Scherer ,  Siegfried Strathmann ,  Ulrich Schofl ,  Reinhard Stierl

IPC分类号： A61K31/519 ,  C07D487/04 ,  A01N43/90

CPC分类号： A01N43/90 ,  C07D487/04

摘要： 6-(2-Fluorophenyl)-triazolopyrimidines of the formula I in which the substituents are as defined below: R1 is C4-C8-alkyl, C4-C8-haloalkyl, substituted C3-C8-cycloalkyl, C3-C8-halocycloalkyl, C5-C8-alkenyl, C2-C8-haloalkenyl, C3-C6-cycloalkenyl, C3-C6-halocycloalkenyl, C2-C8-alkynyl, C2-C8-haloalkynyl or phenyl, naphthyl, or a five- or six-membered saturated, partially unsaturated or aromatic heterocycle which contains one to four heteroatoms from the group consisting of O, N and S, R2 is hydrogen, C1-C3-alkyl or one of the groups mentioned under R1, R1 and R2 together with the nitrogen atom to which they are attached may also form a five- or six-membered heterocyclyl or heteroaryl which is attached via N and contain one to three further heteroatoms from the group consisting of O, N and S as ring member, except for piperidin-1-yl optionally substituted by methyl groups; R1 and/or R2 may be substituted according to the description; L1 is chlorine or fluorine; L2 is hydrogen, is, if L1 is fluorine, also fluorine; X is alkyl; processes for preparing these compounds, compositions comprising them and their use for controlling phytopathogenic harmful fungi.

公开(公告)号：US20070142404A1

公开(公告)日：2007-06-21

申请号：US10590924

申请日：2005-03-29

申请人： Carsten Blettner ,  Markus Gewehr ,  Wassilios Grammenos ,  Thomas Grote ,  Udo Hunger ,  Bernd Muller ,  Matthias Niedenbruck ,  Joachim Rheinheimer ,  Peter Schafer ,  Frank Schieweck ,  Anja Schwogler ,  Oliver Wagner ,  Michael Rack ,  Barbara Nave ,  Maria Scherer ,  Siegfried Strathmann ,  Ulrich Schofl ,  Reinhard Stierl

发明人： Carsten Blettner ,  Markus Gewehr ,  Wassilios Grammenos ,  Thomas Grote ,  Udo Hunger ,  Bernd Muller ,  Matthias Niedenbruck ,  Joachim Rheinheimer ,  Peter Schafer ,  Frank Schieweck ,  Anja Schwogler ,  Oliver Wagner ,  Michael Rack ,  Barbara Nave ,  Maria Scherer ,  Siegfried Strathmann ,  Ulrich Schofl ,  Reinhard Stierl

IPC分类号： A61K31/519 ,  C07D487/04

CPC分类号： A01N43/90 ,  C07D487/04

摘要： 6-(2,6-Dichlorophenyl)triazolopyrimidines of the formula I in which the substituents are as defined below: R1, R2 are hydrogen, alkyl, haloalkyl, cycloalkyl, halocycloalkyl, alkenyl, haloalkenyl, cycloalkenyl, halocycloalkenyl, alkynyl, haloalkynyl or phenyl, naphthyl, or a five- or six-membered saturated, partially unsaturated or aromatic heterocycle which contains one to four heteroatoms from the group consisting of O, N and S, R1 and R2 together with the nitrogen atom to which they are attached may also form a five- or six-membered heterocyclyl or heteroaryl which is attached via N and may contain one to three further heteroatoms from the group consisting of O, N and S as ring member and which is substituted according to the description; X is alkyl, cyano, alkoxy, haloalkoxy, alkenyloxy or haloalkenyloxy; processes for preparing these compounds, compositions comprising them and their use for controlling phytopathogenic harmful fungi.

摘要翻译： 其中取代基如下定义的式I的6-（2,6-二氯苯基）三唑并嘧啶：R 1，R 2是氢，烷基，卤代烷基，环烷基 ，卤代环烷基，烯基，卤代烯基，环烯基，卤代环烯基，炔基，卤代炔基或苯基，萘基或五元或六元饱和的部分不饱和或芳族杂环，其含有一至四个由O，N和S组成的组的杂原子 R 1和R 2连同它们所连接的氮原子一起也可以形成通过N连接的五元或六元杂环基或杂芳基，并且可以 含有一个至三个由O，N和S组成的组的另外的杂原子作为环成员，并且根据描述被取代; X是烷基，氰基，烷氧基，卤代烷氧基，烯氧基或卤代烯氧基; 制备这些化合物的方法，包含它们的组合物及其用于控制​​植物病原性有害真菌的用途。

公开(公告)号：US20080176831A1

公开(公告)日：2008-07-24

申请号：US11596891

申请日：2005-05-17

申请人： Anja Schwogler ,  Frank Schieweck ,  Joachim Rheinheimer ,  Markus Gewehr ,  Bernd Muller ,  Thomas Grote ,  Wassilios Grammenos ,  Udo Hunger ,  Carsten Blettner ,  Peter Schafer ,  Oliver Wagner ,  Reinhard Stierl ,  Ulrich Schofl ,  Siegfried Strathmann ,  Maria Scherer

发明人： Anja Schwogler ,  Frank Schieweck ,  Joachim Rheinheimer ,  Markus Gewehr ,  Bernd Muller ,  Thomas Grote ,  Wassilios Grammenos ,  Udo Hunger ,  Carsten Blettner ,  Peter Schafer ,  Oliver Wagner ,  Reinhard Stierl ,  Ulrich Schofl ,  Siegfried Strathmann ,  Maria Scherer

IPC分类号： A01N43/46 ,  C07D403/04 ,  A01N43/54 ,  A01P7/00 ,  A01P3/00 ,  A01N43/58

CPC分类号： C07D401/04 ,  C07D403/04

摘要： The invention relates to 2-substituted pyrimidines of the formula I in which the index n and the substituents L and R1 to R3 are as defined in the description and X is a group —CH—Ra, —N— or —S—; R1 may be hydrogen, halogen, C1-C6-alkyl, C1-C6-alkoxy, cyano or C1-C6-alkoxycarbonyl; Rb is hydrogen, C1-C6-alkyl or C3-C6-cycloalkyl; T is a group —CH—Ra—; p is an integer from 1 to 4; Y is a group —CH—Ra— or —N—Rb o is 0 or 1; Z is O, S or a group N(Rc) Rc is hydrogen, C1-C6-alkyl or C1-C6-alkoxy, and to processes for their preparation, to pesticidal compositions comprising them and to their use as pesticides.

摘要翻译： 本发明涉及式I的2-取代嘧啶，其中指数n和取代基L和R 1至R 3如在说明书中所定义，X是 基团-CH-R a，N - 或-S-; R 1可以是氢，卤素，C 1 -C 6 - 烷基，C 1 -C 3 > 6个 - 烷氧基，氰基或C 1 -C 6 - 烷氧基羰基; R b是氢，C 1 -C 6 - 烷基或C 3 -C 6 - 环烷基; T是基团-CH-R a， p是1至4的整数; Y是基团-CH-R a - 或-N-R b是0或1; Z是O，S或基团N（R c）R c是氢，C 1 -C 6 烷基或C 1 -C 6 - 烷氧基，并且其制备方法，包含它们的杀虫组合物及其作为农药的用途。

公开(公告)号：US20070179061A1

公开(公告)日：2007-08-02

申请号：US10590368

申请日：2005-03-08

申请人： Jordi Blasco ,  Carsten Blettner ,  Bernd Muller ,  Markus Gewehr ,  Wassilios Grammenos ,  Thomas Grote ,  Joachim Rheinheimer ,  Peter Schafer ,  Frank Schieweck ,  Anja Schwogler ,  Oliver Wagner ,  Matthias Niedenbruck ,  Maria Scherer ,  Siegfried Strathmann ,  Ulrich Schofl ,  Reinhard Stierl

发明人： Jordi Blasco ,  Carsten Blettner ,  Bernd Muller ,  Markus Gewehr ,  Wassilios Grammenos ,  Thomas Grote ,  Joachim Rheinheimer ,  Peter Schafer ,  Frank Schieweck ,  Anja Schwogler ,  Oliver Wagner ,  Matthias Niedenbruck ,  Maria Scherer ,  Siegfried Strathmann ,  Ulrich Schofl ,  Reinhard Stierl

IPC分类号： A01N43/54 ,  C07D487/08

CPC分类号： C07D487/04

摘要： The invention relates to 5,6-dialkyl-7-amino-triazolopyrimidines of formula (I), in which the substituents are defined as follows: R1 represents alkyl or alkoxyalkyl; R2 represents alkyl, R1 and/or R2 being substituted according to the description. The invention also relates to a method for producing said compounds, to agents containing the latter and to their use for controlling plant-pathogenic fungi.

摘要翻译： 本发明涉及式（I）的5,6-二烷基-7-氨基 - 三唑并嘧啶，其中取代基定义如下：R 1表示烷基或烷氧基烷基; R 2表示根据描述被取代的烷基，R 1和/或R 2 O 2。 本发明还涉及一种生产所述化合物的方法，含有后者的药剂及其用于控制​​植物致病真菌的用途。

公开(公告)号：US20080248952A1

公开(公告)日：2008-10-09

申请号：US11631004

申请日：2005-07-06

申请人： Carsten Blettner ,  Markus Gewehr ,  Wassilios Grammenos ,  Thomas Grote ,  Udo Hunger ,  Bernd Muller ,  Matthias Niedenbruck ,  Joachim Rheinheimer ,  Peter Schafer ,  Frank Schieweck ,  Anja Schwogler ,  Oliver Wagner ,  Barbara Nave ,  Maria Scherer ,  Siegfried Strathmann ,  Ulrich Schofl ,  Reinhard Stierl

发明人： Carsten Blettner ,  Markus Gewehr ,  Wassilios Grammenos ,  Thomas Grote ,  Udo Hunger ,  Bernd Muller ,  Matthias Niedenbruck ,  Joachim Rheinheimer ,  Peter Schafer ,  Frank Schieweck ,  Anja Schwogler ,  Oliver Wagner ,  Barbara Nave ,  Maria Scherer ,  Siegfried Strathmann ,  Ulrich Schofl ,  Reinhard Stierl

IPC分类号： C07D487/04 ,  A01N43/90 ,  A01N25/00

CPC分类号： A01N43/90 ,  C07D487/04

摘要： Substituted triazolopyrimidines of the formula I in which the substituents are as defined below: R1 is alkyl, haloalkyl, cycloalkyl, halocycloalkyl, alkenyl, haloalkenyl, cycloalkenyl, halocycloalkenyl, alkynyl, haloalkynyl or phenyl, naphthyl, or a five- or six-membered saturated, partially unsaturated or aromatic heterocycle comprising one to four heteroatoms from the group consisting of O, N and S, R2 is hydrogen or a group R1, R1 and R2 together with the nitrogen atom, to which they are attached, may also form a five- or six-membered heterocyclyl or heteroaryl which is attached via N and which may comprise one to three further heteroatoms from the groups consisting of O, N and S as ring member and/or may be substituted according to the description; L is fluorine, chlorine or methyl; X is cyano, C1-C4-alkyl, C1-C4-alkoxy or C1-C2-haloalkoxy, where X is not methyl if R1 and R2 together are n-pentylene or 3-methyl-n-pentylene and L is fluorine, or R1 and R2 together are 3-methyl-n-pentylene and L is chlorine; processes and intermediates for preparing these compounds, compositions comprising them and their use for controlling phytopathogenic harmful fungi.

摘要翻译： 取代基如下定义：式I的取代三唑并嘧啶：R 1是烷基，卤代烷基，环烷基，卤代环烷基，烯基，卤代烯基，环烯基，卤代环烯基，炔基， 包含一至四个由O，N和S组成的组的杂原子的五或六元饱和的部分不饱和或芳族杂环，R 2是氢或基团R 1， R 1，R 2和R 2与它们所连接的氮原子一起也可以形成五元或六元杂环基或杂芳基，它们是 通过N连接并且其可以包含一个至三个由O，N和S组成的基团的另外的杂原子作为环成员和/或可以根据描述被取代; L是氟，氯或甲基; X是氰基，C 1 -C 4 - 烷基，C 1 -C 4 - 烷氧基或C 1 -C 4 - 如果R 1和R 2一起都是正 - 亚戊基，其中X不是甲基，其中X不是甲基 或3-甲基 - 正戊烯，L是氟，R 1和R 2一起是3-甲基 - 正戊烯，L是氯; 制备这些化合物的方法和中间体，包含它们的组合物及其用于控制​​植物病原性有害真菌的用途。

公开(公告)号：US20070197389A1

公开(公告)日：2007-08-23

申请号：US10589496

申请日：2005-02-24

申请人： Anja Schwogler ,  Markus Gewehr ,  Bernd Muller ,  Thomas Grote ,  Wassilios Grammenos ,  Jordi Blasco ,  Joachim Rheinheimer ,  Carsten Blettner ,  Peter Schafer ,  Frank Schieweck ,  Oliver Wagner ,  Reinhard Stierl ,  Ulrich Schofl ,  Siegfried Strathmann ,  Maria Scherer

发明人： Anja Schwogler ,  Markus Gewehr ,  Bernd Muller ,  Thomas Grote ,  Wassilios Grammenos ,  Jordi Blasco ,  Joachim Rheinheimer ,  Carsten Blettner ,  Peter Schafer ,  Frank Schieweck ,  Oliver Wagner ,  Reinhard Stierl ,  Ulrich Schofl ,  Siegfried Strathmann ,  Maria Scherer

IPC分类号： A01N43/713 ,  C07D487/02

CPC分类号： C07D487/04

摘要： The invention relates to azolopyrimidine compounds of general formula (I), wherein A represents N or C—R6; X and Y, independent of one another, represent a chemical compound or oxygen, sulphur or a group N—R7; the variables R1, R2, R3, R4, R5, R6 and R7 have the meanings cited in the claims and the description. The invention also relates to tautomers of compounds of formula (I) and to the agriculturally compatible salts of compounds (I) and of the tautomers thereof. The invention further relates to the use of azolopyrimidine compounds of general formula (I), to the tautomers thereof and to the agriculturally compatible salts thereof which are used to combat phytopathogenic fungi, and to a method for combating phytopathogenic fungi and means for combating fungi, said means containing at least one compound of general formula (I), a tautomer of formula (I) and/or an agriculturally compatible salt thereof or the tautomer thereof and at least one liquid or solid carrier medium.

摘要翻译： 本发明涉及通式（I）的偶氮嘧啶化合物，其中A代表N或C-R 6; X和Y彼此独立地表示化合物或氧，硫或基团N-R 7; 变量R 1，R 2，R 3，R 4，R 5，...，SUP >，R 6和R 7具有权利要求书和说明书中引用的含义。 本发明还涉及式（I）化合物和化合物（I）的农业相容盐及其互变异构体的互变异构体。 本发明还涉及通式（I）的偶氮嘧啶化合物与其互变异构体及其与植物致病真菌的农业相容盐的用途，以及用于防治植物病原性真菌的方法和对抗真菌的方法， 所述方法含有至少一种通式（I）的化合物，式（I）的互变异构体和/或其农业上相容的盐或其互变异构体和至少一种液体或固体载体介质。