2-(pyridin-2-yl)-pyrimidines and their use for controlling harmful fungi
    24.
    发明授权
    2-(pyridin-2-yl)-pyrimidines and their use for controlling harmful fungi 失效
    2-(吡啶-2-基) - 嘧啶及其用于控制​​有害真菌的用途

    公开(公告)号:US07786043B2

    公开(公告)日:2010-08-31

    申请号:US11632342

    申请日:2005-07-22

    CPC分类号: C07D401/04

    摘要: The invention relates to 2-(pyridin-2-yl)-pyrimidine compounds of general formula (I) and their use for controlling pathogenic fungi and as plant protection products that, as an active constituent, contain compounds of this type: In general formula (I), k represents 0, 1, 2, 3; m represents 0, 1, 2, 3, 4 or 5; n represents 1, 2, 3, 4 or 5; R1, independent of one another, represents halogen, OH, CN, NO2, C1-C4 alkyl, C1-C4 alkyl halide, C1-C4 alkoxy, C1-C4 alkoxy halide, C2-C4 alkenyl, C2-C4 alkynyl, C3-C8 cycloalkyl, C1-C4 alkoxy-C1-C4 alkyl, amino, phenoxy, which is optionally substituted by halogen or C1-C4 alkyl, NHR, NR2, C(Ra)═N—ORb, S(═O)pA1 or C(═O)A2, or two radicals R1 bound to adjacent carbon atoms can, together, also represent a group —O-Alk-O—, wherein Alk represents a linear or branched C1-C4 alkylene, and 1, 2, 3 or 4 hydrogen atoms can also be replaced by halogen; R2 represents C1-C4 alkyl halide, C1-C4 alkoxy, C1-C4 alkoxy halide, hydroxy, halogen, CN or NO2; whereby R2 can also represent hydrogen or C1-C4 alkyl when at least one of the three following conditions is fulfilled: n represents 3, 4 or 5; k represents 1, 2 or 3; if m is not equal to 0, at least one of the radicals R1 represents a radical that differs from halogen, C1-C4 alkyl, C1-C4 alkoxy and C1-C4 alkyl halide, and; R3 represents C1-C4 alkyl.

    摘要翻译: 本发明涉及通式(I)的2-(吡啶-2-基) - 嘧啶化合物及其用于控制​​致病真菌的用途,作为作为活性成分的植物保护产品含有这种化合物:通式 (I)中,k表示0,1,2,3; m表示0,1,2,3,4或5; n表示1,2,3,4或5; R 1彼此独立地表示卤素,OH,CN,NO 2,C 1 -C 4烷基,C 1 -C 4烷基卤,C 1 -C 4烷氧基,C 1 -C 4烷氧基卤化物,C 2 -C 4烯基,C 2 -C 4炔基, C8环烷基,C1-C4烷氧基-C1-C4烷基,氨基,苯氧基,其任选被卤素或C 1 -C 4烷基取代,NHR,NR 2,C(R a)= N-OR b,S(= O)p A1或C (ΟO)A2或与相邻碳原子结合的两个基团R1一起也可以代表基团-O-Alk-O-,其中Alk表示直链或支链C 1 -C 4亚烷基,和1,2,3或 4个氢原子也可以被卤素取代; R2代表C1-C4烷基卤,C1-C4烷氧基,C1-C4烷氧基卤化物,羟基,卤素,CN或NO2; 其中当满足以下三个条件中的至少一个时,R2还可以表示氢或C1-C4烷基:n表示3,4或5; k表示1,2或3; 如果m不等于0,则基团R1中的至少一个表示与卤素,C 1 -C 4烷基,C 1 -C 4烷氧基和C 1 -C 4烷基卤化物不同的基团, R3表示C1-C4烷基。

    Method For Enhancing The Effectiveness Of Ethaboxam
    26.
    发明申请
    Method For Enhancing The Effectiveness Of Ethaboxam 审中-公开
    提高乙异唑的有效性的方法

    公开(公告)号:US20080200334A1

    公开(公告)日:2008-08-21

    申请号:US11791191

    申请日:2005-11-23

    摘要: Method for enhancing the fungicidal effectiveness of a) ethaboxam of the formula I, which comprises applying the active compound I simultaneously, that is separately or together, with at least one active compound II from the group consisting of: b) dithiocarbamates, such as maneb, mancozeb, metam or metiram, sulfenic acid derivatives, such as captan or folpet, strobilurin derivatives, such as kresoxim-methyl or pyraclostrobin, cinnamides and analogs, such as dimethomorph or flumorph, or dithianon, famoxadone, cymoxanil, fluazinam, zoxamide, mefenoxam or chlorothalonil, N-(2-{4-[3-(4-chlorophenyl)prop-2-ynyloxy]-3-methoxyphenyl}ethyl)-2-methanesulfonylamino-3-methylbutyramide, N-(2-{4-[3-(4-chlorophenyl)prop-2-ynyloxy]-3-methoxyphenyl}ethyl)-2-ethanesulfonylamino-3-methylbutyramide or 5-chloro-7-(4-methylpiperidin-1-yl)-6-(2,4,6-trifluorophenyl)-[1,2,4]triazolo[1,5-a]pyrimidine in synergistically effective amounts, by spraying or dusting the seeds, the plants or the soils before or after sowing of the plants or before or after emergence of the plants, no polyoxyalkylene alkyl ether being used as adjuvants, novel synergistic mixtures of ethaboxam and also compositions comprising these mixtures, and the use of ethaboxam for preparing such mixtures.

    摘要翻译: 提高a)式I的ethaboxam的方法,其包括将活性化合物I同时与另一种或一起与至少一种活性化合物II一起施用,所述活性化合物II来自以下组中的至少一种活性化合物II:b)二硫代氨基甲酸盐,例如maneb ,代森锰锌,metam或metiram,磺酸衍生物,例如克虏伯或派生物,嗜球果伞形毒素衍生物,例如甲氧基甲基或嘧菌酯,肉桂酸酯和类似物,例如烯酰吗啉或氟吗啉,或二噻尼龙,恶唑酮,胞嘧啶,氟啶胺,唑酰胺, 或百菌清,N-(2- {4- [3-(4-氯苯基)丙-2-炔基氧基] -3-甲氧基苯基}乙基)-2-甲磺酰基氨基-3-甲基丁酰胺,N-(2- {4- [ 3-(4-氯苯基)丙-2-炔基氧基] -3-甲氧基苯基}乙基)-2-乙磺酰基氨基-3-甲基丁酰胺或5-氯-7-(4-甲基哌啶-1-基)-6-(2, 4,6-三氟苯基) - [1,2,4]三唑并[1,5-a]嘧啶,具有协同有效的量,通过在或之前喷洒或除尘种子,植物或土壤 r播种植物或在植物出现之前或之后,不使用聚氧亚烷基烷基醚作为佐剂,含有这些混合物的组合物的ethaboxam的新型协同混合物,以及使用ethaboxam制备这些混合物。

    7-Aminomethyl-1,2,4-Triazolo[1,5-A]Pyrimidine Compounds And Their Use For Controlling Pathogenic Fungi
    28.
    发明申请
    7-Aminomethyl-1,2,4-Triazolo[1,5-A]Pyrimidine Compounds And Their Use For Controlling Pathogenic Fungi 审中-公开
    7-氨基甲基-1,2,4-三唑并[1,5-A]嘧啶化合物及其用于控制​​致病真菌

    公开(公告)号:US20080076785A1

    公开(公告)日:2008-03-27

    申请号:US11663982

    申请日:2005-09-27

    IPC分类号: A01N43/54 A01P3/00 C07D239/70

    CPC分类号: A01N43/90 C07D487/04

    摘要: The invention relates to 7-aminomethyl-1,2,4-triazolo[1,5-a]pyrimidine compounds of general formula (I) and the agriculturally compatible salts of said compounds. In said formula: R1 and R2 represent hydrogen, alkyl, haloalkyl, alkoxy, cycloalkyl, bicycloalkyl, halocycloalkyl, alkenyl, alkadienyl, haloalkenyl, cycloalkenyl, halocycloalkenyl, alkynyl, haloalkynyl or phenyl, naphthyl, or a 5- or 6-membered saturated, partially unsaturated or aromatic heterocycle, containing 1 to 4 heteroatoms from the group containing O, N or S, or R1 and R2, together with the nitrogen atom to which they are bonded, can also form a five- or six-membered heterocyclyl or heteroaryl, which is bonded by means of N and can contain 1 to 3 additional heteroatoms from the group containing O, N and S as the ring member and can be substituted according to the description; R3 and R4 represent hydrogen, alkyl, haloalkyl, haloalkoxy, alkoxy, or alkoxyalkyl; X represents halogen, cyano, a 5- or 6-membered saturated, partially unsaturated or aromatic heterocycle, containing 1, 2 or 3 heteroatoms from the group containing O, N or S as the ring member, alkyl, alkoxy, alkenyl or alkynyl, whereby the latter 4 groups can be substituted according to the description; L is defined as cited in the claims and the description; and m represents 0, 1, 2, 3, 4 or 5. The invention also relates to the use of the triazolopyrimidine compounds of general formula (I) and their agriculturally compatible salts for controlling plant-pathogenic fungi, to a method for controlling plant-pathogenic fungi, containing at least one compound of general formula (I) and/or an agriculturally compatible salt of said compound and at least one liquid or solid carrier.

    摘要翻译: 本发明涉及通式(I)的7-氨基甲基-1,2,4-三唑并[1,5-a]嘧啶化合物和所述化合物的农业上相容的盐。 在所述式中:R 1和R 2表示氢,烷基,卤代烷基,烷氧基,环烷基,二环烷基,卤代环烷基,烯基,链烯基,卤代烯基,环烯基,卤代环烯基,炔基,卤代炔基或苯基,萘基或5-或6-元饱和, 部分不饱和或芳族杂环,含有1至4个含有O,N或S的杂原子,或R 1和R 2与它们所键合的氮原子一起也可以形成五元或六元杂环基或杂芳基 ,其通过N键合并且可以含有来自含有O,N和S的基团的1至3个另外的杂原子作为环成员,并且可以根据描述进行取代; R3和R4代表氢,烷基,卤代烷基,卤代烷氧基,烷氧基或烷氧基烷基; X代表卤素,氰基,含有1,2或3个杂原子的5-或6-元饱和的部分不饱和或芳族杂环,所述杂环含有作为环成员的O,N或S,烷基,烷氧基,烯基或炔基, 由此后4个组可以根据描述被替代; L定义为权利要求书和说明书中引用的; 和m表示0,1,2,3,4或5.本发明还涉及通式(I)的三唑并嘧啶化合物及其农业上相容的盐用于控制植物致病真菌的用途,用于控制植物的方法 致病真菌,含有至少一种通式(I)的化合物和/或所述化合物的农业上相容的盐和至少一种液体或固体载体。

    Fungicidal Mixtures
    29.
    发明申请
    Fungicidal Mixtures 审中-公开
    杀菌混合物

    公开(公告)号:US20080058352A1

    公开(公告)日:2008-03-06

    申请号:US10594268

    申请日:2005-03-22

    IPC分类号: A01N43/56 A01N43/78 A01N43/90

    CPC分类号: A01N43/90 A01N2300/00

    摘要: Fungicidal mixtures comprising, as active components, 1) the triazolopyrimidine derivative of the formula I and 2) an anilide of the formula II  in which the variables are as defined below: Ar is phenyl or a five- or six-membered aromatic heterocycle which contains one to four heteroatoms selected from the group consisting of O, N and S, where the cycles are unsubstituted or may be substituted by one to three groups R1: R1 is halogen, alkyl or haloalkyl; R is phenyl, alkyl, haloalkyl, alkoxy, haloalkoxy; Q is hydrogen, alkyl, haloalkyl, alkoxy, haloalkoxy; in a synergistically effective amount, methods for controlling harmful fungi using mixtures of the compound I with the compound II and the use of the compound I with the compound II for preparing such mixtures, and also compositions comprising these mixtures.

    摘要翻译: 作为活性组分的杀真菌混合物包括1)式I的三氮代嘧啶衍生物和2)式II的酰苯胺,其中变量如下所定义:Ar是苯基或五或六元芳族杂环,其含有 一至四个选自O,N和S的杂原子,其中循环是未取代的或可以被一至三个R 1取代:R 1是 卤素,烷基或卤代烷基; R是苯基,烷基,卤代烷基,烷氧基,卤代烷氧基; Q是氢,烷基,卤代烷基,烷氧基,卤代烷氧基; 协同有效量的方法,使用化合物I与化合物II的混合物来控制有害真菌,以及使用化合物I与化合物II制备这种混合物,以及包含这些混合物的组合物。

    Fungicidal Mixtures
    30.
    发明申请
    Fungicidal Mixtures 审中-公开
    杀菌混合物

    公开(公告)号:US20070197556A1

    公开(公告)日:2007-08-23

    申请号:US11579048

    申请日:2005-05-11

    摘要: Fungicidal mixtures, comprising, as active components, 1) the triazolopyrimidine derivative of the formula I and 2) at least one biphenylamide of the formula II in which the variables are as defined below: A is oxathiinyl or 5-membered heteroaryl which contains one to four nitrogen atoms or one to three nitrogen atoms and/or one sulfur or oxygen atom, where A may be substituted according to the description; R1 is hydrogen, alkyl, alkylcarbonyl or a group A which is attached via carbonyl; Ra, Rb are halogen, cyano, alkyl, haloalkyl, alkoxycarbonyl, alkoxy, haloalkoxy, alkylthio, alkylcarbonyl, formyl, alkylene or alkenylene which links two adjacent carbon atoms; m is 0, 1, 2, 3, 4 or 5; n is 0, 1 or 2; in a synergistically effective amount, methods for controlling harmful fungi using mixtures of the compound I with compound II and the use of the compound I with compounds II for preparing such mixtures, and also compositions comprising these mixtures.

    摘要翻译: 包含作为活性成分的杀真菌混合物,1)式I的三唑并嘧啶衍生物和2)至少一种式II的联苯酰胺,其中变量如下所定义:A是氧亚硫代基或5元杂芳基,其含有1至 四个氮原子或一至三个氮原子和/或一个硫或氧原子,其中A可以根据描述被取代; R 1是氢,烷基,烷基羰基或通过羰基连接的基团A; R 2是卤素,氰基,烷基,卤代烷基,烷氧基羰基,烷氧基,卤代烷氧基,烷硫基,烷基羰基,甲酰基,亚烷基或亚链烯基,其连接两个相邻的碳原子; m为0,1,2,3,4或5; n为0,1或2; 在协同有效量的情况下,使用化合物I与化合物II的混合物控制有害真菌的方法以及化合物I与化合物II用于制备此类混合物的用途,以及包含这些混合物的组合物。