公开(公告)号：US07632820B2

公开(公告)日：2009-12-15

申请号：US10543638

申请日：2004-01-30

申请人： Thomas Pitterna ,  Peter Maienfisch ,  Fiona Murphy Kessabi ,  Jerome Cassayre ,  Laura Quaranta ,  Pierre Jung

发明人： Thomas Pitterna ,  Peter Maienfisch ,  Fiona Murphy Kessabi ,  Jerome Cassayre ,  Laura Quaranta ,  Pierre Jung

IPC分类号： A01N43/04 ,  A61K31/40 ,  A61K31/335 ,  A61K31/70 ,  A61K31/397 ,  A61K31/445 ,  A61K31/44 ,  A01N43/38

CPC分类号： A01N43/90 ,  C07H17/08

摘要： Disclosed are compounds of the formulain which n is 0 or 1; X—Y is —CH═CH— or —CH2—CH2—; Z is —C(═O)—, —C(═S)— or —SO2—; R1 is C1-C12alkyl, C3-C8cycloalkyl or C2-C12alkenyl; and R2 is R3-Z-, R3—O-Z-, R4 or -Z-N(R6)(R7); Q is O or —N—R5; R3 and R4 are for example H, C1C12alkyl, C2-C12alkenyl, C2-C12alkynyl, C3-C12zcycloalkyl, C5-C12cycloalkenyl, aryl or heterocyclyl; R5 is for example H, C1-C8alkyl, hydroxy-C1-C8alkyl, C3-C8cycloalkyl, C2-C8alkenyl, C2-C8alkynyl, phenyl or benzyl; R6 and R7 are for example, H, unsubstituted or mono- to pentasubstituted C1-C12alkyl, unsubstituted or mono- to pentasubstituted C2-C12alkenyl or, if appropriate, an E/Z isomer, E/Z isomer mixture and/or tautomer thereof, in each case in free form or in salt form, are useful as pesticides.

摘要翻译： 公开了n为0或1的甲醛化合物; X-Y是-CH-CH-或-CH 2 -CH 2 - ; Z是-C（-O） - ， - C（-S） - 或-SO 2 - ; R1是C1-C12烷基，C3-C8环烷基或C2-C12链烯基; R2为R3-Z-，R3-O-Z-，R4或-Z-N（R6）（R7）; Q是O或-N-R5; R 3和R 4例如是H，C 1 -C 12烷基，C 2 -C 12烯基，C 2 -C 12炔基，C 3 -C 12环烷基，C 5 -C 12环烯基，芳基或杂环基; R5是例如H，C1-C8烷基，羟基-C1-C8烷基，C3-C8环烷基，C2-C8链烯基，C2-C8炔基，苯基或苄基; R 6和R 7为例如未取代的或未被取代的一价或五价取代的C 1 -C 12烷基，未被取代的或一至五取代的C 2 -C 12链烯基或（如果合适的话）E / Z异构体，E / Z异构体混合物和/或其互变异构体， 在每种情况下以游离形式或盐形式，都可用作农药。

公开(公告)号：US20060166824A1

公开(公告)日：2006-07-27

申请号：US10543638

申请日：2004-01-30

申请人： Thomas Pitterna ,  Peter Maienfisch ,  Fiona Murphy Kessabi ,  Jerome Cassayre ,  Laura Quaranta ,  Pierre Jung

发明人： Thomas Pitterna ,  Peter Maienfisch ,  Fiona Murphy Kessabi ,  Jerome Cassayre ,  Laura Quaranta ,  Pierre Jung

IPC分类号： A01N43/04 ,  A61K31/7048

CPC分类号： A01N43/90 ,  C07H17/08

摘要： Disclosed are compounds of the formula in which n is 0 or 1; X—Y is —CH═CH— or —CH2—CH2—; Z is —C(═O)—, —C(═S)— or —S02—; R1 is C1-C12alkyl, C3-C8cycloalkyl or C2-C12alkenyl; and R2 is R3-Z-, R3—O-Z-, R4 or -Z-N(R6)(R7); Q is O or —N—R5; R3 and R4 are for example H, C1C12alkyl, C2-C12alkenyl, C2-C12alkynyl, C3-C12zcycloalkyl, C5-C12cycloalkenyl, aryl or heterocyclyl; R5 is for example H, C1-C8alkyl, hydroxy-C1-C8alkyl, C3-C8cycloalkyl, C2-C8alkenyl, C2-C8alkynyl, phenyl or benzyl; R6 and R7 are for example, H, unsubstituted or mono- to pentasubstituted C1-C12alkyl, unsubstituted or mono- to pentasubstituted C2-C12alkenyl or, if appropriate, an E/Z isomer, E/Z isomer mixture and/or tautomer thereof, in each case in free form or in salt form, are useful as pesticides.

摘要翻译： 公开了下式的化合物，其中n为0或1; X-Y是-CH-CH-或-CH 2 -CH 2 - 。 Z是-C（-O） - ， - C（-S） - 或-SO 2 - 。 R 1是C 1 -C 12烷基，C 3 -C 8烷基，C 1 -C 12烷基，C 3 -C 12烷基， 环烷基或C 2 -C 12 - 烯基; 和R 2是R 3 -Z-，R 3 -OZ-，R 4或-ZN（ R 6）（R 7）; Q是O或-N-R 5; R 3和R 4是例如H，C 1 -C 12烷基，C 2， C 1 -C 12亚烷基，C 2 -C 12炔基，C 3 -C 12链烯基，C 2 -C 12亚炔基，C 3 -C 12亚烷基， 12个环烷基，C 5 -C 12环烯基，芳基或杂环基; R 5是例如H，C 1 -C 8烷基，羟基-C 1 -C 3 C 1 -C 8烷基，C 3 -C 8环烷基，C 2 -C 8链烯基，C 1 -C 8烷基， C 2 -C 8炔基，苯基或苄基; R 6和R 7是例如H，未取代的或一至五取代的C 1 -C 12 - 烷基，未取代的或一至五取代的C 2 -C 12链烯基，或者如果合适的话，E / Z异构体，E / Z异构体混合物和/或其互变异构体， 在每种情况下以游离形式或盐形式，都可用作农药。

公开(公告)号：US08263566B2

公开(公告)日：2012-09-11

申请号：US13117292

申请日：2011-05-27

申请人： Peter Maienfisch ,  Fiona Murphy Kessabi ,  Jerome Cassayre ,  Laura Quaranta ,  Thomas Pitterna ,  Ottmar Franz Hueter ,  Pierre Jung

发明人： Peter Maienfisch ,  Fiona Murphy Kessabi ,  Jerome Cassayre ,  Laura Quaranta ,  Thomas Pitterna ,  Ottmar Franz Hueter ,  Pierre Jung

IPC分类号： A61K31/70 ,  C07H17/04

CPC分类号： C07H17/08 ,  A61K31/7042

摘要： What is described are a compound of the formula wherein n is 0 or 1; A-B is —CH═CH— or —CH2—CH2—; R1 is C1-C12-alkyl, C3-C8-cycloalkyl or C2-C12-alkenyl; R2 is for example C1-C12-alkyl, C2-C12-alkenyl or C2-C12-alkinyl; which are optionally substituted with one to five substituents selected from the group consisting of OH, halogen, CN, —N3, —NO2, C3-C8-Cycloalkyl, norbornylenyl-, C3-C8-Cycloalkenyl; C3-C8-halocycloalkyl, C1-C12-alkoxy, C1-C6-alkoxy-C1-C6-alkoxy, C3-C8-cycloalkoxy, C1-C12-haloalkoxy, C1-C12-alkylthio, C3-C8-cycloalkylthio, C1-C12-haloalkylthio, C1-C12-alkylsulfinyl, C3-C8-cycloalkylsulfinyl, C1-C12-haloalkylsulfinyl, C3-C8-halocycloalkylsulfinyl, C1-C12-alkylsulfonyl, C3-C8-cycloalkylsulfonyl, C1-C12-haloalkylsulfonyl, C3-C8-halocycloalkylsulfonyl, —NR4R6, —X—C(═Y)—R4, —X—C(═Y)—Z—R4, —P(═O)(OC1-C6-alkyl)2, aryl, heterocyclyl, aryloxy, arylthio and heterocyclyloxy; R3 is for example H, C1-C12-alkyl or C1-C12-alkyl which is optionally substituted and, where applicable, to E/Z isomers, mixtures of E/Z isomers and/or tautomers, in each case in free form or in salt form; a process for preparing and using these compounds and their tautomers; pesticides whose active compound is selected from these compounds and their tautomers; and a process for preparing these compounds and compositions, and the use of these compounds and compositions.

摘要翻译： 描述的是下式的化合物，其中n是0或1; A-B是-CH = CH-或-CH 2 -CH 2 - ; R1是C1-C12-烷基，C3-C8-环烷基或C2-C12-烯基; R2是例如C1-C12-烷基，C2-C12-烯基或C2-C12-炔基; 其任选被一至五个选自OH，卤素，CN，-N 3，-NO 2，C 3 -C 8 - 环烷基，降冰片基 - ，C 3 -C 8 - 环烯基的取代基取代; C 3 -C 8卤代环烷基，C 1 -C 12烷氧基，C 1 -C 6烷氧基-C 1 -C 6 - 烷氧基，C 3 -C 8环烷氧基，C 1 -C 12卤代烷氧基，C 1 -C 12烷硫基，C 3 -C 8环烷硫基， C 1 -C 12烷基亚磺酰基，C 3 -C 8环烷基亚磺酰基，C 1 -C 12卤代烷基亚磺酰基，C 3 -C 8卤代环烷基亚磺酰基，C 1 -C 12烷基磺酰基，C 3 -C 8环烷基磺酰基，C 1 -C 12卤代烷基磺酰基， 卤代环烷基磺酰基，-NR4R6，-X-C（= Y）-R4，-X-C（= Y）-Z-R4，-P（= O）（OC1-C6-烷基）2，芳基，杂环基，芳氧基， 芳硫基和杂环氧基; R3是例如任选取代的H，C 1 -C 12 - 烷基或C 1 -C 12 - 烷基，并且在适用的情况下，E / Z异构体，E / Z异构体和/或互变异构体的混合物，在每种情况下为游离形式或 盐形式; 一种制备和使用这些化合物及其互变异构体的方法; 活性化合物选自这些化合物及其互变异构体的农药; 以及制备这些化合物和组合物的方法，以及这些化合物和组合物的用途。

公开(公告)号：US07521429B2

公开(公告)日：2009-04-21

申请号：US10560390

申请日：2004-06-15

申请人： Thomas Pitterna ,  Pierre Jung ,  Fiona Murphy Kessabi ,  Jerome Cassayre ,  Laura Quaranta ,  Ottmar Franz Hueter

发明人： Thomas Pitterna ,  Pierre Jung ,  Fiona Murphy Kessabi ,  Jerome Cassayre ,  Laura Quaranta ,  Ottmar Franz Hueter

IPC分类号： A61K31/70 ,  C07H17/08

CPC分类号： C07H19/01 ,  C07H17/08

摘要： A compound of formula (I) wherein the bond between carbon atoms 22 and 23 may be a single or a double bond; R1 is C1-C12alkyl, C3-C8cycloalkyl, or C2-C12alkenyl; R2 and R3 are, for example, independently of each other hydrogen, C1-C12alkyl, C3-C12cycloalkyl, C2-C12alkenyl, C2-C12alkynyl, aryl or heteroaryl; and, where applicable, to E/Z isomers, mixtures of E/Z isomers, diastereomers and/or tautomers, in each case in free form or in salt form; pesticidal compositions in which the active ingredient has been selected from those compounds and their tautomers; and a method of controlling pests using those compositions are described.

摘要翻译： 式（I）的化合物，其中碳原子22和23之间的键可以是单键或双键; R1是C1-C12烷基，C3-C8环烷基或C2-C12链烯基; R 2和R 3例如彼此独立地为氢，C 1 -C 12烷基，C 3 -C 12环烷基，C 2 -C 12烯基，C 2 -C 12炔基，芳基或杂芳基; 在适用的情况下，E / Z异构体，E / Z异构体，非对映异构体和/或互变异构体的混合物，在每种情况下为游离形式或盐形式; 其中活性成分选自那些化合物及其互变异构体的杀虫组合物; 并描述了使用这些组合物来控制害虫的方法。

公开(公告)号：US07378399B2

公开(公告)日：2008-05-27

申请号：US10544274

申请日：2004-02-03

申请人： Jerome Cassayre ,  Hans Tobler ,  Thomas Pitterna ,  Peter Maienfisch ,  Fiona Murphy Kessabi ,  Laura Quaranta ,  Ottmar Franz Hueter

发明人： Jerome Cassayre ,  Hans Tobler ,  Thomas Pitterna ,  Peter Maienfisch ,  Fiona Murphy Kessabi ,  Laura Quaranta ,  Ottmar Franz Hueter

IPC分类号： A01N43/04 ,  A01N43/00 ,  A01N43/40 ,  A01N43/02 ,  A01N43/16 ,  A61K31/40 ,  A61K31/38 ,  A61K31/335 ,  A61K31/35 ,  A61K31/70 ,  A61K31/397 ,  A61K31/445 ,  A61K31/44 ,  A01N43/38 ,  A01N31/40

CPC分类号： C07H17/08

摘要： What is described are a compound of the formula (I) Wherein A-B is —CH═CH— or —CH2—CH2—; n is 0 or 1; R1, is C1-C12alkyl, C3-C8cycloalkyl or C2-C12alkenyl; R2 and R3 for instance are either, (i) independently from each other for instance -Q, —C(═Y)-Q, or —C(═Y)—O-Q; or (ii) together form with the nitrogen atom to which they are bound a three- to seven-membered ring, (iii) together are ═C(R4)R5; R4 and R5 are, independently from each other, for instance -Q, —C(═Y)-Q, or —C(═Y)—O-Q; Y is O or S; Q is for instance H or unsubstituted or mono- to pentasubstituted C1-C12alkyl; or, if appropriate, an E/Z isomer, E/Z isomer mixture and/or tautomer thereof; a process for preparing these compounds, their isomers and tautomers and the use of these compounds, their isomers and tautomers; pesticidal compositions whose active compound is selected from these compounds and their tautomers; intermediates for the preparation of the said compounds of the formula (I), methods for the preparation of the compounds of the formula (I), and a method for controlling pests using these compositions

摘要翻译： 描述的是式（I）的化合物，其中A-B是-CH-CH-或-CH 2 -CH 2 - 。 n为0或1; R 1是C 1 -C 12烷基，C 3 -C 8烷基，C 3 -C 12烷基，C 3 -C 12烷基，C 3 -C 12烷基， >环烷基或C 2 -C 12 - 烯基; 例如，R 2和R 3是（i）彼此独立地例如-Q，-C（-Y）-Q或-C（ - Y）-OQ; 或（ii）与其结合的氮原子一起形成三至七元环，（iii）一起为-C（R 4）R 5 >; R 4和R 5各自独立地为例如-Q，-C（-Y）-Q或-C（-Y）-O-Q; Y为O或S; Q是例如H或未被取代或单取代或未取代的C 1 -C 12烷基; 或者，如果合适的话，E / Z异构体，E / Z异构体混合物和/或其互变异构体; 制备这些化合物，其异构体和互变异构体的方法以及这些化合物，其异构体和互变异构体的用途; 活性化合物选自这些化合物及其互变异构体的杀虫组合物; 用于制备所述式（I）化合物的中间体，式（I）化合物的制备方法和使用这些组合物来控制害虫的方法

公开(公告)号：US07781411B2

公开(公告)日：2010-08-24

申请号：US11574588

申请日：2005-08-19

申请人： Ottmar Franz Hueter ,  Thomas Pitterna ,  Pierre Jung ,  Fiona Murphy Kessabi ,  Laura Quaranta

发明人： Ottmar Franz Hueter ,  Thomas Pitterna ,  Pierre Jung ,  Fiona Murphy Kessabi ,  Laura Quaranta

IPC分类号： A61K31/70 ,  C07H17/08

CPC分类号： C07H17/08 ,  A01N43/90

摘要： Certain derivatives of avermectin, avermectin monosaccharide and avermectin aglycone, having on the 4″, 4′ or 13 position, respectively, a 6-membered cyclic acetal with a substituent on position 2, that are useful in controlling pests, in particular pests that are harmful to crop plants and to its propagation material, such as representatives of the class insecta, the order acarina and the class nematode, are provided.

摘要翻译： 除虫菌素，除虫菌素单糖和除虫菌素苷元的某些衍生物分别在4“，4”或13“位置上具有2位上具有取代基的6元环状缩醛，可用于防治害虫，特别是害虫 提供对作物和其繁殖材料有害的植物，如昆虫类，螨类和类线虫的代表。

公开(公告)号：US07687470B2

公开(公告)日：2010-03-30

申请号：US10599671

申请日：2005-03-09

申请人： Pierre Jung ,  Thomas Pitterna ,  Fiona Murphy Kessabi ,  Laura Quaranta ,  Ottmar Franz Hueter

发明人： Pierre Jung ,  Thomas Pitterna ,  Fiona Murphy Kessabi ,  Laura Quaranta ,  Ottmar Franz Hueter

IPC分类号： A61K31/70 ,  C07H17/08

CPC分类号： A01N43/90 ,  C07H19/01

摘要： Avermectin and avermectin monosaccharaide compounds, derivatives, and compositions thereof are provided as well as processes for preparing such compounds, derivatives, and compositions. Intermediates in the preparation of avermectin and avermectin monosaccharaide derivatives and methods of controlling pests are also provided. The avermectin and avermectin monosaccharaide derivatives are demonstrated as useful in controlling pests, in particular pests that are harmful to crop plants and to its propagation materials, such as representatives of the class insecta, the order Acarina and the class nematede.

摘要翻译： 提供阿维菌素和除虫菌素单糖化合物，其衍生物及其组合物以及制备这些化合物，衍生物和组合物的方法。 还提供了制备除虫菌素和除虫菌素单糖衍生物的中间体以及防治害虫的方法。 阿维菌素和除虫菌素单糖衍生物被证明可用于防治害虫，特别是对作物和其繁殖材料有害的害虫，例如类昆虫，螨类和螨类的代表。

公开(公告)号：US20080194498A1

公开(公告)日：2008-08-14

申请号：US10568715

申请日：2004-08-27

申请人： Fiona Murphy Kessabi ,  Thomas Pitterna ,  Peter Maienfisch ,  Jerome Cassayre ,  Laura Quaranta ,  Pierre Jung ,  Ottmar Franz Hueter

发明人： Fiona Murphy Kessabi ,  Thomas Pitterna ,  Peter Maienfisch ,  Jerome Cassayre ,  Laura Quaranta ,  Pierre Jung ,  Ottmar Franz Hueter

IPC分类号： A01N43/90 ,  C07H17/08 ,  A01P17/00

CPC分类号： A01N43/90 ,  C07H19/01

摘要： Described is a compound of the formula (1) wherein the bond between carbon atoms 22 and 23 is a single or double bond; m is 0 or 1; R1, is C1-C12alkyl, C3-C8cycloalkyl or C2-C12alkenyl; and either (A) R2 is —N(R3)R4, and (1) X is 0, wherein R3 is, for instance, hydrogen, unsubstituted or mono- to pentasubstituted C1-C12alkyl, and R4 is, for instance, mono- to pentasubstituted C1-C12alkyl, unsubstituted or mono- to pentasubstituted C3-C12cycloalkyl; or (2) X is S, wherein R3 is, for instance, hydrogen, unsubstituted or mono- to pentasubstituted C1-C12alkyl, and R4 is, for instance, hydrogen, unsubstituted or mono- to pentasubstituted C1-C12alkyl; or (3) X is 0 or S, wherein R3 and R4 together are, for instance, a three- to seven membered alkylene or a four- to seven-membered alkenylene bridge; or (B) R2 is OR5, X is 0 or S, wherein R5 is, for instance, C1-C12alkyl, mono- to pentasubstituted C1-C12alkyl; or, if appropriate, an E/Z isomer, E/Z isomer mixture and/or tautomer thereof, in each case in free form or in salt form; such a compound demonstrates pesticidal activity.

摘要翻译： 描述了式（1）的化合物，其中碳原子22和23之间的键是单键或双键; m为0或1; R 1是C 1 -C 12烷基，C 3 -C 8烷基，C 3 -C 12烷基，C 3 -C 12烷基，C 3 -C 12烷基， >环烷基或C 2 -C 12 - 烯基; （A）R 2是-N（R 3）R 4，和（1）X是0，其中R _{3是例如氢，未取代的或一至五取代的C 1 -C 12烷基，R 4是氢， 是例如一至五取代的C 1 -C 12烷基，未取代或单取代或五取代的C 3 -C 12烷基， 12环烷基; 或（2）X是S，其中R 3是例如氢，未取代的或一至五取代的C 1 -C 12 - 烷基和R 4是例如氢，未取代的或一至五取代的C 1 -C 12烷基; 或（3）X为0或S，其中R 3和R 4一起为例如三至七元亚烷基或四至七元亚烷基， 多元亚烯基桥; 或（B）R 2是OR 5，X是0或S，其中R 5是例如C 1 C 1 -C 12烷基，一至五取代C 1 -C 12烷基; 或者如果合适的话，E / Z异构体，E / Z异构体混合物和/或其互变异构体在每种情况下都是游离形式或盐形式; 这种化合物显示出杀虫活性。}

公开(公告)号：US20060094600A1

公开(公告)日：2006-05-04

申请号：US10544281

申请日：2004-02-03

申请人： Laura Quaranta ,  Thomas Pitterna ,  Peter Maienfisch ,  Fiona Murphy Kessabi ,  Jerome Cassayre

发明人： Laura Quaranta ,  Thomas Pitterna ,  Peter Maienfisch ,  Fiona Murphy Kessabi ,  Jerome Cassayre

IPC分类号： A01N43/04 ,  A01N25/26 ,  C07H17/08

CPC分类号： C07H17/08 ,  A01N43/90

摘要： What is described are a compound of the formula (I) wherein the bond of atoms C22 and C23 is a single or double bond; m is 0 or 1; n is 0, 1 or 2; p is 0 or 1; R1 is C1-C12-alkyl, C3-C8-cycloalkyl or C2-C12alkenyl; R2 is for example H, C1-C12-alkyl, C1-C12-haloalkyl or C1-C12-hydroxyalkyl; or together with R4 form with the carbon to which they are bound for example a three- to seven-membered ring; R3 is for example H, C1-C12-alkyl, halogen, halo-C1-C2alkyl, CN, NO2 or C3-C8-cycloalkyl; R4 has the same meanings as R2; R5 and R6 independently of each other are for example H, C1-C12-alkyl, CN, NO2, OH, SH, halogen, halo-C1-C2alkyl or C3-C8cycloalkyl; or, if appropriate, an E/Z isomer, E/Z isomer mixture and/or tautomer thereof, in each case in free form or in salt form a process for preparing and using these compounds and their tautomers; pesticides whose active compound is selected from these compounds and their tautomers; and a process for preparing these compounds and compositions, and the use of these compounds and compositions.

摘要翻译： 描述的是式（I）的化合物，其中原子C 22和C 23的键是单键或双键; m为0或1; n为0,1或2; p为0或1; R 1是C 1 -C 12 - 烷基，C 3 -C 8亚烷基，C 3 -C 12 - 烷基，C 3 -C 12 - 环烷基或C 2 -C 12链烯基; R 2是例如H，C 1 -C 12 - 烷基，C 1 -C 3 - 12个 - 卤代烷基或C 1 -C 12 - 羟基烷基; 或与R 4 S形成的碳与它们所键合的碳例如为三至七元环; R 3是例如H，C 1 -C 12 - 烷基，卤素，卤素-C 1 - C 2 -C 12烷基，CN，NO 2或C 3 -C 8 - 环烷基; R 4具有与R 2'相同的含义; R 5和R 6彼此独立地是例如H，C 1 -C 12 - 烷基， CN，NO 2，OH，SH，卤素，卤代-C 1 -C 2烷基或C 3 - -C 8环烷基; 或者如果适用，E / Z异构体，E / Z异构体混合物和/或其互变异构体在每种情况下以游离形式或盐形成用于制备和使用这些化合物及其互变异构体的方法; 活性化合物选自这些化合物及其互变异构体的农药; 以及制备这些化合物和组合物的方法，以及这些化合物和组合物的用途。

公开(公告)号：US07737261B2

公开(公告)日：2010-06-15

申请号：US10539274

申请日：2003-12-19

申请人： Peter Maienfisch ,  Fiona Murphy Kessabi ,  Jérôme Cassayre ,  Laura Quaranta ,  Thomas Pitterna ,  Ottmar Franz Hueter ,  Pierre Jung

发明人： Peter Maienfisch ,  Fiona Murphy Kessabi ,  Jérôme Cassayre ,  Laura Quaranta ,  Thomas Pitterna ,  Ottmar Franz Hueter ,  Pierre Jung

IPC分类号： C07H17/04

CPC分类号： C07H17/08 ,  A61K31/7042

摘要： Avermectin B1 and avermectin B1 monosaccharide derivative compounds having an alkoxymethyl substituent in the 4″- or 4′-position; a process for preparing and using these compounds and their tautomers; pesticides whose active compound is selected from these compounds and their tautomers; and a process for preparing these compounds and compositions are provided.

摘要翻译： 在4“或4”位具有烷氧基甲基取代基的阿维菌素B1和除虫菌素B1单糖衍生物化合物; 一种制备和使用这些化合物及其互变异构体的方法; 活性化合物选自这些化合物及其互变异构体的农药; 并提供了这些化合物和组合物的制备方法。