Avermectins and avermectin monosacharides substituted in the 4′-and 4″ position having pesticidal properties
    3.
    发明授权
    Avermectins and avermectin monosacharides substituted in the 4′-and 4″ position having pesticidal properties 有权
    在具有杀虫性的4'和4“位置取代的阿维菌素和阿维菌素单糖苷

    公开(公告)号:US07704961B2

    公开(公告)日:2010-04-27

    申请号:US10568715

    申请日:2004-08-27

    CPC分类号: A01N43/90 C07H19/01

    摘要: Described is a compound of the formula (I) wherein the bond between carbon atoms 22 and 23 is a single or double bond; m is 0 or 1; R1, is C1-C12alkyl, C3-C8cycloalkyl or C2-C12alkenyl; and either (A) R2 is —N(R3)R4, and (1) X is 0, wherein R3 is, for instance, hydrogen, unsubstituted or mono- to pentasubstituted C1-C12alkyl, and R4 is, for instance, mono- to pentasubstituted C1-C12alkyl, unsubstituted or mono- to pentasubstituted C3-C12cycloalkyl; or (2) X is S, wherein R3 is, for instance, hydrogen, unsubstituted or mono- to pentasubstituted C1-C12alkyl, and R4 is, for instance, hydrogen, unsubstituted or mono- to pentasubstituted C1-C12alkyl; or (3) X is 0 or S, wherein R3 and R4 together are, for instance, a three- to seven membered alkylene or a four- to seven-membered alkenylene bridge; or (B) R2 is OR5, X is 0 or S, wherein R5 is, for instance, C1-C12alkyl, mono- to pentasubstituted C1-C12alkyl; or, if appropriate, an E/Z isomer, E/Z isomer mixture and/or tautomer thereof, in each case in free form or in salt form; such a compound demonstrates pesticidal activity.

    摘要翻译: 描述了式(I)的化合物,其中碳原子22和23之间的键是单键或双键; m为0或1; R1是C1-C12烷基,C3-C8环烷基或C2-C12链烯基; (A)R 2是-N(R 3)R 4,和(1)X是0,其中R 3是例如氢,未被取代的或单取代到五取代的C 1 -C 12烷基,R 4是例如, 至五取代的C 1 -C 12烷基,未取代的或一至五取代的C 3 -C 12环烷基; 或(2)X为S,其中R 3为例如氢,未取代或单价至五价取代的C 1 -C 12烷基,R 4为例如氢,未取代或单价至五价取代的C 1 -C 12烷基; 或(3)X为0或S,其中R3和R4一起为例如三至七元亚烷基或四至七元亚烯基桥; 或(B)R 2是OR 5,X是0或S,其中R 5是例如C 1 -C 12烷基,一至五取代的C 1 -C 12烷基; 或者如果合适的话,E / Z异构体,E / Z异构体混合物和/或其互变异构体在每种情况下都是游离形式或盐形式; 这种化合物显示出杀虫活性。

    Chemical compounds
    4.
    发明授权
    Chemical compounds 失效
    化合物

    公开(公告)号:US08629284B2

    公开(公告)日:2014-01-14

    申请号:US13129063

    申请日:2009-10-27

    摘要: A compound of the formula I or where W, X and Y are for example each CH; R1 is H; R2 is halogen; and R6 is, for formula I, for example, OH, CN, C3-C8-cycloalkyl, C3-C8-cycloalkyl-C1-C6-alkyl, C2-C6-alkenyl, C2-C6-haloalkenyl, C2-C6-alkenyloxy, C2-C6-alkynyl, C2-C6-haloalkynyl, C2-C6-alkynyloxy, optionally substituted C1 to C3-alkyl, or optionally substituted C1-C6-alkoxy, or R6 is, for formula II, for example, CN, C3-C8-cycloalkyl, or optionally substituted C3-C6-alkyl; and/or salts thereof; and their use as as pesticidal agents.

    摘要翻译: 式I化合物或其中W,X和Y为例如CH; R1是H; R2是卤素; 对于式I,R 6为例如OH,CN,C 3 -C 8 - 环烷基,C 3 -C 8 - 环烷基-C 1 -C 6烷基,C 2 -C 6 - 烯基,C 2 -C 6 - 卤代烯基,C 2 -C 6 - 烯氧基 ,C 2 -C 6炔基,C 2 -C 6 - 卤代炔基,C 2 -C 6 - 炔氧基,任选取代的C 1至C 3 - 烷基或任选取代的C 1 -C 6 - 烷氧基,或R 6为式II,例如CN,C 3 -C 8 - 环烷基或任选取代的C 3 -C 6 - 烷基; 和/或其盐; 以及其作为杀虫剂的用途。

    INSECTICIDAL COMPOUNDS
    5.
    发明申请
    INSECTICIDAL COMPOUNDS 审中-公开
    杀虫剂化合物

    公开(公告)号:US20140005245A1

    公开(公告)日:2014-01-02

    申请号:US13984478

    申请日:2012-02-07

    IPC分类号: A01N43/647 C07D403/04

    CPC分类号: A01N43/647 C07D403/04

    摘要: The present invention relates to novel triazole derivatives of formula (I) having insecticidal activity, to processes and intermediates for preparing them, to insecticidal, acaricidal, nematicidal or molluscicidal compositions comprising them and to methods of using them to combat and control insect, acarine, nematode or mollusc pests wherein A1, A2, A3, A4, R1, R2, G1, Q1 and Q2 are as defined in claim 1; or salts or N— oxides thereof.

    摘要翻译: 本发明涉及具有杀虫活性的新颖的具有杀虫活性的式(I)的三唑衍生物,其制备方法和中间体,包含它们的杀虫,杀螨,杀线虫或杀软体动物的组合物以及使用它们来对抗和控制昆虫,螨类, 线虫或软体动物害虫,其中A1,A2,A3,A4,R1,R2,G1,Q1和Q2如权利要求1所定义; 或其盐或N-氧化物。

    3-amino-benzo [D] isothiazole dioxide derivatives and their use as pesticides
    7.
    发明授权
    3-amino-benzo [D] isothiazole dioxide derivatives and their use as pesticides 失效
    3-氨基 - 苯并[D]异噻唑二氧化物衍生物及其作为农药的用途

    公开(公告)号:US08563744B2

    公开(公告)日:2013-10-22

    申请号:US12993983

    申请日:2009-05-18

    IPC分类号: C07D275/06 A61K31/425

    CPC分类号: C07D275/06

    摘要: A compound of Formula (I) or Formula (II) where W is C—R3; X is C—R4; Y is C—R5; R1 and R6, independently of each other, is, for example, H, C1-C6-alkyl, C2-C6-alkenyl, C2-C6-alkynyl, C3-C8-cycloalkyl or C1-C6-alkyl-C(═O); R2 is H; and R3, R4 and R5, independently of each other, are, for example, H, halogen, cyano, nitro, C1-C6-alkyl, or C1-C6-haloalkyl; provided that in formula II R1 is H and R6 is as defined above; and in formula I that (a) at least one of R1 and R3 to R6 is other than hydrogen, (b) R3 or R4 is other than C1 when in each instance the remaining five groups of R1 to R6 are hydrogen, and (c) (i) R3 is other than methyl, (ii) R4 is other than C1, (iii) R5 is other than C1 and (iv) R3 is not C1 when R5 is methoxy, when in each instance (i) to (iv) R1 is H, R6 is MeC(═O), and remaining groups of R2 to R5 are hydrogen; and/or salts thereof; and their use as as pesticidal agents.

    摘要翻译: 式(I)或式(II)的化合物,其中W是C-R 3; X是C-R4; Y为C-R5; R 1和R 6彼此独立地是例如H,C 1 -C 6 - 烷基,C 2 -C 6 - 烯基,C 2 -C 6 - 炔基,C 3 -C 8 - 环烷基或C 1 -C 6 - 烷基-C(= O ); R2为H; 和R 3,R 4和R 5彼此独立地是例如H,卤素,氰基,硝基,C 1 -C 6烷基或C 1 -C 6卤代烷基; 条件是式Ⅱ中R 1为H且R 6如上定义; (a)R1和R3至R6中的至少一个不是氢,(b)R 3或R 4不同于C 1,当R 5至R 6的剩余五个基团为氢时,和(c )(i)R 3不是甲基,(ⅱ)R 4不是C 1,(ⅲ)R 5不是C 1,(ⅳ)当R 5是甲氧基时,R 3不是C 1,当(i)〜 )R1为H,R6为MeC(= O),R2至R5的其余基团为氢; 和/或其盐; 以及其作为杀虫剂的用途。

    INSECTICIDAL COMPOUNDS
    8.
    发明申请
    INSECTICIDAL COMPOUNDS 审中-公开
    杀虫剂化合物

    公开(公告)号:US20130253011A1

    公开(公告)日:2013-09-26

    申请号:US13991731

    申请日:2011-12-15

    IPC分类号: A01N43/647

    摘要: The present invention relates to novel triazole derivatives of formula (I) having insecticidal activity, to processes and intermediates for preparing them, to insecticidal, acaricidal, nematicidal or molluscicidal compositions comprising them and to methods of using them to combat and control insect, acarine, nematode or mollusc pests wherein A1, A2, A3, A4, R1, G1, Q1 and Q2 are as defined in claim 1; or salts or N-oxides thereof.

    摘要翻译: 本发明涉及具有杀虫活性的新颖的具有杀虫活性的式(I)三唑衍生物,其制备方法和中间体,包含它们的杀虫,杀螨,杀线虫或杀软体动物的组合物以及使用它们来对抗和控制昆虫,螨类, 线虫或软体动物害虫,其中A1,A2,A3,A4,R1,G1,Q1和Q2如权利要求1所定义; 或其盐或N-氧化物。

    Avermectin and avermectin monosaccharide substituted in the 4″- and 4″ position respectively
    10.
    发明授权
    Avermectin and avermectin monosaccharide substituted in the 4″- and 4″ position respectively 有权
    阿维菌素和阿维菌素单糖分别在4“和4”位置取代

    公开(公告)号:US07687470B2

    公开(公告)日:2010-03-30

    申请号:US10599671

    申请日:2005-03-09

    IPC分类号: A61K31/70 C07H17/08

    CPC分类号: A01N43/90 C07H19/01

    摘要: Avermectin and avermectin monosaccharaide compounds, derivatives, and compositions thereof are provided as well as processes for preparing such compounds, derivatives, and compositions. Intermediates in the preparation of avermectin and avermectin monosaccharaide derivatives and methods of controlling pests are also provided. The avermectin and avermectin monosaccharaide derivatives are demonstrated as useful in controlling pests, in particular pests that are harmful to crop plants and to its propagation materials, such as representatives of the class insecta, the order Acarina and the class nematede.

    摘要翻译: 提供阿维菌素和除虫菌素单糖化合物,其衍生物及其组合物以及制备这些化合物,衍生物和组合物的方法。 还提供了制备除虫菌素和除虫菌素单糖衍生物的中间体以及防治害虫的方法。 阿维菌素和除虫菌素单糖衍生物被证明可用于防治害虫,特别是对作物和其繁殖材料有害的害虫,例如类昆虫,螨类和螨类的代表。