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公开(公告)号:US5413997A
公开(公告)日:1995-05-09
申请号:US7104
申请日:1993-01-21
申请人: Iwao Kinoshita , Daisuke Machii , Yasuo Onoda , Haruki Takai , Nobuo Kosaka , Katsuichi Shuto , Katsushige Gomi , Makoto Morimoto , Akio Ishii
发明人: Iwao Kinoshita , Daisuke Machii , Yasuo Onoda , Haruki Takai , Nobuo Kosaka , Katsuichi Shuto , Katsushige Gomi , Makoto Morimoto , Akio Ishii
IPC分类号: A61K31/09 , A61K31/135 , A61K31/165 , A61K31/365 , A61K31/38 , A61K31/381 , A61K31/395 , A61K31/40 , A61K31/425 , A61K31/426 , A61K31/428 , A61K31/44 , A61K31/4406 , A61K31/4427 , A61K31/47 , A61K31/472 , A61P3/00 , A61P9/00 , A61P19/10 , C07C217/58 , C07C217/60 , C07C233/11 , C07C233/25 , C07C233/26 , C07C233/29 , C07C233/60 , C07C233/65 , C07C233/75 , C07C235/44 , C07C235/46 , C07C235/54 , C07C235/56 , C07C235/64 , C07C237/32 , C07C237/40 , C07C323/42 , C07D207/09 , C07D211/58 , C07D213/74 , C07D213/75 , C07D213/82 , C07D215/06 , C07D217/04 , C07D221/20 , C07D223/20 , C07D225/08 , C07D277/20 , C07D277/44 , C07D277/46 , C07D277/82 , C07D295/096 , C07D295/10 , C07D295/112 , C07D295/13 , C07D295/135 , C07D295/192 , C07D295/205 , C07D307/00 , C07D311/00 , C07D333/20 , C07D333/38 , C07D401/04 , C07D413/04 , A01N43/00 , A01N33/02 , A01N43/40 , A01N43/62 , C07C43/21 , C07C211/45 , C07C229/42 , C07D215/28 , C07D215/36 , C07D215/38
CPC分类号: C07D213/75 , C07C217/58 , C07C217/60 , C07C233/25 , C07C233/26 , C07C233/29 , C07C233/60 , C07C233/75 , C07C235/44 , C07C235/56 , C07C235/64 , C07C237/40 , C07C323/42 , C07D211/58 , C07D213/74 , C07D215/06 , C07D217/04 , C07D221/20 , C07D225/08 , C07D277/46 , C07D277/82 , C07D295/096 , C07D295/112 , C07D295/13 , C07D295/135 , C07D295/192 , C07D295/205 , C07D307/00 , C07D333/20 , C07D333/38 , C07D413/04 , C07C2101/02 , C07C2101/08 , C07C2101/18 , C07C2102/08 , C07C2102/42 , C07C2103/18 , C07C2103/74
摘要: A triphenylmethane derivative represented by the following general formula: ##STR1## exhibits bone absorption inhibiting effects and is useful as a medicament for treating osteoporosis.
摘要翻译: 由以下通式表示的三苯甲烷衍生物:
表现出骨吸收抑制作用,可用作治疗骨质疏松症的药物。 -
公开(公告)号:US5510501A
公开(公告)日:1996-04-23
申请号:US256711
申请日:1994-07-21
申请人: Hirofumi Nakano , Noboru Fujii , Yoshinori Yamashita , Yutaka Saitoh , Tsutomu Agatsuma , Katsuhiko Ando , Yasushi Nishiie , Katsunori Kita , Naoki Morishima , Katsushige Gomi
发明人: Hirofumi Nakano , Noboru Fujii , Yoshinori Yamashita , Yutaka Saitoh , Tsutomu Agatsuma , Katsuhiko Ando , Yasushi Nishiie , Katsunori Kita , Naoki Morishima , Katsushige Gomi
IPC分类号: C07C50/38 , C07C305/22 , C07C305/26 , C12P29/00 , C07C49/423
CPC分类号: C07C305/26 , C07C305/22 , C07C50/38 , C12P29/00
摘要: The present invention relates to Saintopin derivatives represented by the following formula (I): ##STR1## wherein R.sup.1 is hydrogen and R.sup.2 is SO.sub.2 OH (UCE 1022), or R.sup.1 is acetyl and R.sup.2 is H (Saintopin E), which are useful as antibacterial and anti-tumor agents.
摘要翻译: PCT No.PCT / JP93 / 01680 Sec。 371日期:1994年7月21日 102(e)日期1994年7月21日PCT 1993年11月17日PCT公布。 公开号WO94 / 12458 日本6月9日,1994年。本发明涉及由下式(I)表示的Saintopin衍生物:其中R1是氢,R2是SO2OH(UCE1022),或R1是乙酰基,R2是H (Saintopin E),其可用作抗细菌剂和抗肿瘤剂。
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公开(公告)号:US5112867A
公开(公告)日:1992-05-12
申请号:US515873
申请日:1990-04-27
申请人: Iwao Kinoshita , Daisuke Machii , Yasuo Onoda , Haruki Takai , Nobuo Kasaka , Katsuichi Shuto , Katsushige Gomi , Makoto Morimoto , Akio Ishii
发明人: Iwao Kinoshita , Daisuke Machii , Yasuo Onoda , Haruki Takai , Nobuo Kasaka , Katsuichi Shuto , Katsushige Gomi , Makoto Morimoto , Akio Ishii
IPC分类号: A61K31/09 , A61K31/135 , A61K31/165 , A61K31/365 , A61K31/38 , A61K31/381 , A61K31/395 , A61K31/40 , A61K31/425 , A61K31/426 , A61K31/428 , A61K31/44 , A61K31/4406 , A61K31/4427 , A61K31/47 , A61K31/472 , A61P3/00 , A61P9/00 , A61P19/10 , C07C217/58 , C07C217/60 , C07C233/11 , C07C233/25 , C07C233/26 , C07C233/29 , C07C233/60 , C07C233/65 , C07C233/75 , C07C235/44 , C07C235/46 , C07C235/54 , C07C235/56 , C07C235/64 , C07C237/32 , C07C237/40 , C07C323/42 , C07D207/09 , C07D211/58 , C07D213/74 , C07D213/75 , C07D213/82 , C07D215/06 , C07D217/04 , C07D221/20 , C07D223/20 , C07D225/08 , C07D277/20 , C07D277/44 , C07D277/46 , C07D277/82 , C07D295/096 , C07D295/10 , C07D295/112 , C07D295/13 , C07D295/135 , C07D295/192 , C07D295/205 , C07D307/00 , C07D311/00 , C07D333/20 , C07D333/38 , C07D401/04 , C07D413/04
CPC分类号: C07D213/75 , C07C217/58 , C07C217/60 , C07C233/25 , C07C233/26 , C07C233/29 , C07C233/60 , C07C233/75 , C07C235/44 , C07C235/56 , C07C235/64 , C07C237/40 , C07C323/42 , C07D211/58 , C07D213/74 , C07D215/06 , C07D217/04 , C07D221/20 , C07D225/08 , C07D277/46 , C07D277/82 , C07D295/096 , C07D295/112 , C07D295/13 , C07D295/135 , C07D295/192 , C07D295/205 , C07D307/00 , C07D333/20 , C07D333/38 , C07D413/04 , C07C2101/02 , C07C2101/08 , C07C2101/18 , C07C2102/08 , C07C2102/42 , C07C2103/18 , C07C2103/74
摘要: A triphenylmethane derivative represented by the following general formula: ##STR1## exhibits born absorption inhibiting effects and is useful as a medicament for treating osteoporosis.
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公开(公告)号:US5189187A
公开(公告)日:1993-02-23
申请号:US903476
申请日:1992-06-24
申请人: Hirofumi Nakano , Shozo Kawada , Yoichi Uosaki , Yutaka Saito , Katsushige Gomi , Toshiaki Iwazaki
发明人: Hirofumi Nakano , Shozo Kawada , Yoichi Uosaki , Yutaka Saito , Katsushige Gomi , Toshiaki Iwazaki
IPC分类号: C07D303/32 , C07D407/06 , C07D493/10 , C12P17/02
CPC分类号: C07D407/06 , C07D303/32 , C07D493/10 , C12P17/02 , C12R1/465
摘要: A clerodane-type diterpene derivative, which has antibacterial and antitumor activities, as well as chemically equivalent tautomers thereof and a process for producing said derivative using a microorganism belonging to the genus Streptomyces.
摘要翻译: 具有抗细菌和抗肿瘤活性的氯化丹烷型二萜衍生物及其化学等效的互变异构体,以及使用属于链霉菌属的微生物来生产所述衍生物的方法。
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