公开(公告)号：US20050176736A1

公开(公告)日：2005-08-11

申请号：US10508409

申请日：2003-03-19

申请人： Jordi Tormo i Blasco ,  Carsten Blettner ,  Bernd Muller ,  Markus Gewehr ,  Wassilios Grammenos ,  Thomas Grote ,  Andreas Gypser ,  Joachim Rheinheimer ,  Peter Schafer ,  Frank Schieweck ,  Anja Schwogler ,  Eberhard Ammermann ,  Siegfried Strathmann ,  Gisela Lorenz ,  Reinhard Stierl ,  Ulrich Schofl

发明人： Jordi Tormo i Blasco ,  Carsten Blettner ,  Bernd Muller ,  Markus Gewehr ,  Wassilios Grammenos ,  Thomas Grote ,  Andreas Gypser ,  Joachim Rheinheimer ,  Peter Schafer ,  Frank Schieweck ,  Anja Schwogler ,  Eberhard Ammermann ,  Siegfried Strathmann ,  Gisela Lorenz ,  Reinhard Stierl ,  Ulrich Schofl

IPC分类号： A01N43/90 ,  C07C255/57 ,  C07D487/04 ,  A61K31/519

CPC分类号： C07D487/04 ,  A01N43/90 ,  C07C255/57

摘要： The invention relates to triazolopyrimidines of formula (I), in which the substituents are defined as follows: L1 represents cyano, S(═O)nA1 or C(═O)A2, wherein A1 stands for hydrogen, hydroxy, alkyl, alkylamino or dialkylamino; A2 stands for C1-C8 alkoxy, C1-C6 haloalkoxy or one of the groups named in A1; and n stands for 0, 1 or 2; L2, L3 represent hydrogen or halogen; L4, L5 represent hydrogen, halogen or alkyl; X represents halogen, cyano, alkyl, haloalkyl, alkoxy or haloalkoxy; R1 represents alkyl, haloalkyl, cycloalkyl, halocycloalkyl, alkenyl, alkadienyl, haloalkenyl, cycloalkenyl, alkynyl, haloalkynyl or cycloalkynyl, phenyl, naphthyl, or a five to ten-membered saturated, partially unsaturated or aromatic heterocyclus containing between one and four heteroatoms from the group containing O, N or S; R2 represents hydrogen or R1; R1 and R2 can form, together with the nitrogen atom to which they are bonded, a five or six-membered ring, which can be interrupted and/or substituted by an atom from the group O, N and S; whereby R1 and/or R2 can be substituted in accordance with the description. The invention also relates to methods and intermediate products for producing said compounds, to agents containing the latter and to the use of said compounds for combating harmful fungi.

摘要翻译： 本发明涉及式（I）的三唑并嘧啶，其中取代基定义如下：L 1表示氰基，S（-O）n A 1 或其中A 1代表氢，羟基，烷基，烷基氨基或二烷基氨基;或C（= O） A 2代表C 1 -C 8烷氧基，C 1 -C 6烷基，C 1 -C 6 - >卤代烷氧基或在A 中命名的基团之一; 而n代表0,1或2; L 2，L 3表示氢或卤素; L 4，L 5代表氢，卤素或烷基; X表示卤素，氰基，烷基，卤代烷基，烷氧基或卤代烷氧基; R 1表示烷基，卤代烷基，环烷基，卤代环烷基，烯基，链烯基，卤代烯基，环烯基，炔基，卤代炔基或环炔基，苯基，萘基或五至十元饱和，部分不饱和或芳族杂环 含有一个至四个来自含有O，N或S的基团的杂原子; R 2表示氢或R 1; R 1和R 2可以与它们所键合的氮原子一起形成五元或六元环，其可被中断和/或被 来自O，N和S族的原子; 其中R 1和/或R 2可以根据描述被取代。 本发明还涉及用于生产所述化合物的方法和中间产物，含有后者的试剂和所述化合物用于防治有害真菌的用途。

公开(公告)号：US07550471B2

公开(公告)日：2009-06-23

申请号：US10531981

申请日：2003-11-04

申请人： Jordi Tormo i Blasco ,  Carsten Blettner ,  Bernd Müller ,  Markus Gewehr ,  Wassilios Grammenos ,  Thomas Grote ,  Andreas Gypser ,  Joachim Rheinheimer ,  Peter Schäfer ,  Frank Schieweck ,  Anja Schwögler ,  Eberhard Ammermann ,  Siegfried Strathmann ,  Ulrich Schöfl ,  Reinhard Stierl

发明人： Jordi Tormo i Blasco ,  Carsten Blettner ,  Bernd Müller ,  Markus Gewehr ,  Wassilios Grammenos ,  Thomas Grote ,  Andreas Gypser ,  Joachim Rheinheimer ,  Peter Schäfer ,  Frank Schieweck ,  Anja Schwögler ,  Eberhard Ammermann ,  Siegfried Strathmann ,  Ulrich Schöfl ,  Reinhard Stierl

IPC分类号： A01N43/90 ,  A61K31/519 ,  C07D487/00

CPC分类号： C07D487/04

摘要： The invention relates to 5-alkyl-7-aminotriazolopyrimidines of the formula (I) and to the salts thereof. In said formula substituents have the following meanings: R1 and R2 each is a hydrogen atom or a group of alkyl, alcenyl, haloalkyl, cycloalky, phenyl or naphtyle, saturated, unstaturated or aromatic heterocycle having from five to six members which contain from one to four nitrogen atoms or one to three nitrogen atoms and one sulfur or oxygen atom, or R1 and R2 can from together with a connecting them nitrogen atom a cycle of 5 to 6 members containing from one to four nitrogen atoms or from one to three nitrogen atoms and one sulfur or oxygen atom, R3 is a cycloalkyl or bicycloalkyl group, R1, R2 and R3 can be substituted in conformity with a description, and X is an alkyl or alkyl halide group. The inventive methods and intermediary products necessary for producing said compounds, agents containing them and the use therefore for fighting against harmful mushroom are also disclosed.

摘要翻译： 本发明涉及式（I）的5-烷基-7-氨基三唑并嘧啶及其盐。 在所述式中，取代基具有以下含义：R 1和R 2各自为氢原子或具有5至6个成员的烷基，烯基，卤代烷基，环烷基，苯基或萘杂，饱和的，不饱和的或芳族杂环的基团， 四个氮原子或一个至三个氮原子和一个硫或氧原子，或者R 1和R 2可以连同它们的氮原子一起包含5至6个含有1-4个氮原子或1-3个氮原子的成员 和一个硫或氧原子，R 3为环烷基或双环烷基，R 1，R 2和R 3可以根据说明书进行取代，X为烷基或卤代烷基。 还公开了生产所述化合物所需的创造性方法和中间产物，含有它们的试剂和用于防止有害蘑菇的用途。

公开(公告)号：US07763622B2

公开(公告)日：2010-07-27

申请号：US10532719

申请日：2003-11-04

申请人： Jordi Tormo i Blasco ,  Carsten Blettner ,  Bernd Müller ,  Markus Gewehr ,  Wassilios Grammenos ,  Thomas Grote ,  Andreas Gypser ,  Joachim Rheinheimer ,  Peter Schäfer ,  Frank Schieweck ,  Anja Schwögler ,  Eberhard Ammermann ,  Siegfried Strathmann ,  Ulrich Schöfl ,  Reinhard Stierl

发明人： Jordi Tormo i Blasco ,  Carsten Blettner ,  Bernd Müller ,  Markus Gewehr ,  Wassilios Grammenos ,  Thomas Grote ,  Andreas Gypser ,  Joachim Rheinheimer ,  Peter Schäfer ,  Frank Schieweck ,  Anja Schwögler ,  Eberhard Ammermann ,  Siegfried Strathmann ,  Ulrich Schöfl ,  Reinhard Stierl

IPC分类号： A01N43/90 ,  A61K31/519 ,  C07D471/00 ,  C07D487/00 ,  C07D491/00

CPC分类号： C07C69/65 ,  A01N43/90 ,  C07D487/04

摘要： Substituted 6-(2-halogenphenyl)-triazolopyrimidines of formula I in which R1 denote alkyl, alkenyl, alkynyl, alkadienyl, haloalkyl, haloalkenyl, cycloalkyl, phenyl, naphthyl, or a 5- or 6-membered saturated, unsaturated, or aromatic heterocycle, containing one to four nitrogen atoms or one to three nitrogen atoms and one sulfur or oxygen atom, wherein R1 and R2 radicals may be substituted as defined in the description, R2 denote hydrogen, or a group mentioned for R1; or R1 and R2 together with the interjacent nitrogen atom represent a 5- or 6-membered heterocycle, containing one to four nitrogen atoms or one to three nitrogen atoms and one sulfur or oxygen atom, which ring may be substituted as defined in the description; Hal is halogen; L1, L3 independently denote hydrogen, halogen, or alkyl; L2 is hydrogen, halogen, haloalkyl, or NH2, NHRb, or N(Rb)2, wherein Rb is as defined in the description, wherein at least one from L1, L2, and L3 is not hydrogen; X is halogen, cyano, alkyl, alkoxy, haloalkoxy or alkenyloxy. processes for their preparation, compositions containing them and to their use for combating phytopathogenic fungi.

摘要翻译： 取代的式I的6-（2-卤代苯基） - 三唑并嘧啶，其中R 1表示烷基，烯基，炔基，链二烯基，卤代烷基，卤代烯基，环烷基，苯基，萘基或5-或6-元饱和，不饱和或芳族杂环 含有一至四个氮原子或一至三个氮原子和一个硫或氧原子，其中R 1和R 2基团可以如说明书中所定义而被取代，R 2表示氢或R 1所提及的基团; 或R1和R2与相邻的氮原子一起表示含有1-4个氮原子或一至三个氮原子和一个硫或氧原子的5-或6-元杂环，该环可以如说明书中所定义而被取代; 卤素是卤素; L 1，L 3独立地表示氢，卤素或烷基; L2是氢，卤素，卤代烷基或NH2，NHRb或N（Rb）2，其中Rb如说明书中所定义，其中L1，L2和L3中的至少一个不是氢; X是卤素，氰基，烷基，烷氧基，卤代烷氧基或烯氧基。 其制备方法，含有它们的组合物及其用于对抗植物病原真菌的用途。

公开(公告)号：US07388018B2

公开(公告)日：2008-06-17

申请号：US10570893

申请日：2004-09-10

申请人： Wassilios Grammenos ,  Carsten Blettner ,  Bernd Müller ,  Markus Gewehr ,  Jordi Tormo i Blasco ,  Thomas Grote ,  Joachim Rheinheimer ,  Peter Schäfer ,  Frank Schieweck ,  Anja Schwögler ,  Oliver Wagner ,  Norbert Götz ,  Siegfried Strathmann ,  Ulrich Schöfl ,  Maria Scherer ,  Reinhard Stierl

发明人： Wassilios Grammenos ,  Carsten Blettner ,  Bernd Müller ,  Markus Gewehr ,  Jordi Tormo i Blasco ,  Thomas Grote ,  Joachim Rheinheimer ,  Peter Schäfer ,  Frank Schieweck ,  Anja Schwögler ,  Oliver Wagner ,  Norbert Götz ,  Siegfried Strathmann ,  Ulrich Schöfl ,  Maria Scherer ,  Reinhard Stierl

IPC分类号： A61K31/541 ,  A61K31/496 ,  C07D417/02 ,  C07D403/02

CPC分类号： C04B35/632 ,  C07D213/42 ,  C07D215/12 ,  C07D401/12 ,  C07D409/12

摘要： Sulfonamides of the formula I where the substituents are as follows: R1 is hydrogen, alkyl, alkoxy, alkenyl or alkynyl; and R2, R3, R4, R5 are hydrogen, halogen, alkyl, alkoxy or halomethyl; R2 and R3 together may also form a phenyl, cyclopentyl or cyclohexyl ring, it being possible for these rings to carry two groups R2, and R3, R2, R3, are hydrogen, halogen, alkyl, alkoxy or halomethyl; in case a), if R2, R3, R4 and R5 are hydrogen: X is phenyl substituted by a group —C(R6)═NOR7, where R6 is alkyl and R7 is alkyl, benzyl, alkenyl, haloalkyl, haloalkenyl, alkynyl or haloalkynyl; and in case b), if at least one of the groups R2, R3, R4 and R5 is not hydrogen: X is phenyl, naphthyl or a five- or six-membered saturated, or partially unsaturated or aromatic heterocycle which is attached via a carbon atom and contains one to four heteroatoms from the group consisting of O, N and S, where X may be substituted according to the description; Processes for preparing these compounds, compositions comprising them and their use for controlling phytopathogenic harmful fungi.

摘要翻译： 式I的磺酰胺，其中取代基如下：R 1是氢，烷基，烷氧基，烯基或炔基; R 2，R 3，R 4，R 5是氢，卤素，烷基，烷氧基或卤代甲基 ; R 2和R 3一起也可以形成苯基，环戊基或环己基环，这些环可以携带两个基团R 2， R 3，R 2，R 3，R 3，R 3，R 3，R 3，R 3，R 3，R 3，R 3， 在a）情况下，如果R 2，R 3，R 4和R 5是氢：X是 由基团-C（R 6） - NOR 7取代的苯基，其中R 6为烷基，R 7为H 烷基，苄基，烯基，卤代烷基，卤代烯基，炔基或卤代炔基; 并且在情况b）中，如果R 2，R 3，R 4和R 5中的至少一个， SUP>不是氢：X是苯基，萘基或五或六元饱和或部分不饱和或芳族杂环，其通过碳原子连接并含有一至四个由O，N和S组成的组的杂原子 ，其中X可以根据描述被替代; 制备这些化合物的方法，包含它们的组合物及其用于控制​​植物病原性有害真菌的用途。

公开(公告)号：US06730680B2

公开(公告)日：2004-05-04

申请号：US10314595

申请日：2002-12-10

申请人： Klaus Jüergen Pees ,  Jordi Tormo i Blasco ,  Hubert Sauter ,  Oliver Cullman ,  Markus Gewehr ,  Wassilios Grammenos ,  Bernd Müller ,  Thomas Grote ,  Andreas Gypser ,  Joachim Rheinheimer ,  Peter Schäfer ,  Frank Schieweck ,  Eberhard Ammermann ,  Siegried Strathmann ,  Gisela Lorenz ,  Rheinhard Stierl

发明人： Klaus Jüergen Pees ,  Jordi Tormo i Blasco ,  Hubert Sauter ,  Oliver Cullman ,  Markus Gewehr ,  Wassilios Grammenos ,  Bernd Müller ,  Thomas Grote ,  Andreas Gypser ,  Joachim Rheinheimer ,  Peter Schäfer ,  Frank Schieweck ,  Eberhard Ammermann ,  Siegried Strathmann ,  Gisela Lorenz ,  Rheinhard Stierl

IPC分类号： A01N4354

CPC分类号： C07D487/04

摘要： 6-Phenyl-Pyrazolopyrimidines of formula I wherein R1 is alkyl, alkenyl, alkynyl, alkadienyl or haloalkyl, cycloalkyl, bicycloalkyl, phenyl, naphthyl, or 5- or 6-membered heterocyclyl, containing one to four nitrogen atoms or one to three nitrogen atoms and one sulfur or oxygen atom, or 5- or 6-membered heteroaryl, containing one to four nitrogen atoms or one to three nitrogen atoms and one sulfur or oxygen atom,  where these radicals may be unsubstituted or substituted as defined in the specification, Y is oxygen, sulfur, NR2 or a single bond; wherein R2 is defined in the specification; and R1 and R2 together with the interjacent nitrogen atom may represent a 5- or 6-membered heterocyclic ring, containing one to four nitrogen atoms or one to three nitrogen atoms and one sulfur or oxygen atom, which may be substituted by one or more Rc radicals; m is 0 or an integer from 1 to 4; L each independently is halogen, nitro, alkyl, alkoxy, and X is halogen; processes and intermediates for preparing these compounds, compositions comprising them and their use for controlling phytopathogenic fungi are described.

摘要翻译： 式I的6-苯基 - 吡唑并嘧啶，其中R 1是含有1-4个氮原子或一至三个氮的烷基，烯基，炔基，链二烯基或卤代烷基，环烷基，二环烷基，苯基，萘基或5-或6-元杂环基 原子和一个硫或氧原子，或含有一至四个氮原子或一至三个氮原子和一个硫或氧原子的5-或6-元杂芳基，其中这些基团可以未被取代或如说明书中所定义的取代， Y是氧，硫，NR 2或单键; 其中R 2在说明书中定义; 和R 1和R 2与中间的氮原子一起可以表示含有1-4个氮原子或1-3个氮原子和一个硫或氧原子的5或6元杂环，其可被取代 由一个或多个R c基团取代; m为0或1至4的整数; L各自独立地为卤素，硝基，烷基，烷氧基和X为卤素;制备这些化合物的方法和中间体， 描述了用于控制植物病原真菌的用途。

公开(公告)号：US06552026B2

公开(公告)日：2003-04-22

申请号：US09735033

申请日：2000-12-12

申请人： Klaus Jüergen Pees ,  Jordi Tormo i Blasco ,  Hubert Sauter ,  Oliver Cullman ,  Markus Gewehr ,  Wassilios Grammenos ,  Bernd Müller ,  Thomas Grote ,  Andreas Gypser ,  Joachim Rheinheimer ,  Peter Schäfer ,  Frank Schieweck ,  Eberhard Ammermann ,  Siegried Strathmann ,  Gisela Lorenz ,  Rheinhard Stierl

发明人： Klaus Jüergen Pees ,  Jordi Tormo i Blasco ,  Hubert Sauter ,  Oliver Cullman ,  Markus Gewehr ,  Wassilios Grammenos ,  Bernd Müller ,  Thomas Grote ,  Andreas Gypser ,  Joachim Rheinheimer ,  Peter Schäfer ,  Frank Schieweck ,  Eberhard Ammermann ,  Siegried Strathmann ,  Gisela Lorenz ,  Rheinhard Stierl

IPC分类号： C07D48704

CPC分类号： C07D487/04

摘要： 6-Phenyl-Pyrazolopyrimidines of formula I wherein R1 is alkyl, alkenyl, alkynyl, alkadienyl or haloalkyl, cycloalkyl, bicycloalkyl, phenyl, naphthyl, or 5- or 6-membered heterocyclyl, containing one to four nitrogen atoms or one to three nitrogen atoms and one sulfur or oxygen atom, or 5- or 6-membered heteroaryl, containing one to four nitrogen atoms or one to three nitrogen atoms and one sulfur or oxygen atom,  where these radicals may be unsubstituted or substituted as defined in the specification, Y is oxygen, sulfur, NR2 or a single bond; wherein R2is defined in the specification; and R1 and R 2 together with the interjacent nitrogen atom may represent a 5- or 6-membered heterocyclic ring, containing one to four nitrogen atoms or one to three nitrogen atoms and one sulfur or oxygen atom, which may be substituted by one or more Rc radicals; m is 0 or an integer from 1 to 4; L each independently is halogen, nitro, alkyl, alkoxy, and X is halogen; processes and intermediates for preparing these compounds, compositions comprising them and their use for controlling phytopathogenic fungi are described.

摘要翻译： 式I的6-苯基 - 吡唑并嘧啶，其中R1是具有1-4个氮原子或1-3个氮原子的烷基，烯基，炔基，链二烯基或卤代烷基，环烷基，双环烷基，苯基，萘基或5-或6-元杂环基， 硫或氧原子，或含有一至四个氮原子或一至三个氮原子和一个硫或氧原子的5-或6-元杂芳基，其中这些基团可以未被取代或如说明书中所定义取代，Y是氧 ，硫，NR 2或单键; 其中R2在说明书中定义; 并且R 1和R 2与中间的氮原子一起可以表示含有1-4个氮原子或1-3个氮原子和一个硫或氧原子的5或6元杂环，其可被一个或多个R c 基团; m为0或1至4的整数; L各自独立地为卤素，硝基，烷基，烷氧基和X为卤素;制备这些化合物的方法和中间体，包含它们的组合物及其用于防治植物病原真菌的用途。

公开(公告)号：US20050256138A1

公开(公告)日：2005-11-17

申请号：US10513030

申请日：2003-04-30

申请人： Jordi Tormo i Blasco ,  Carsten Blettner ,  Bernd Muller ,  Markus Gewhr ,  Wassilios Grammenos ,  Thomas Grote ,  Andreas Gypser ,  Joachim Rheinheimer ,  Peter Schafer ,  Frank Schieweck ,  Anja Schwogler ,  Eberhard Ammermann ,  Siegfried Strathmann ,  Gisela Lorenz ,  Reinhard Stierl

发明人： Jordi Tormo i Blasco ,  Carsten Blettner ,  Bernd Muller ,  Markus Gewhr ,  Wassilios Grammenos ,  Thomas Grote ,  Andreas Gypser ,  Joachim Rheinheimer ,  Peter Schafer ,  Frank Schieweck ,  Anja Schwogler ,  Eberhard Ammermann ,  Siegfried Strathmann ,  Gisela Lorenz ,  Reinhard Stierl

IPC分类号： A01N43/90 ,  C07C69/65 ,  C07D487/04 ,  A61K31/519

CPC分类号： C07D487/04 ,  A01N43/90 ,  C07C69/65

摘要： Disclosed are a method for producing fungicidal triazolopyrimidine compounds, agents containing said compounds, and the use thereof for controlling harmful fungi. Also disclosed are triazolopyrimidines of formula (1), in which the substituents have the following meaning: L1 represents alkyl; L2 represents halogen; L3represents hydrogen or halogen; X represents halogen, cyano, alkyl, alkoxy, or haloalkoxy; R1, R2 represent hydrogen, alkyl, haloalkyl, cycloalkyl, alkenyl, alkadienyl, alkinyl, or cycloalkinyl, phenyl, naphthyl, or a five-unit to ten-unit saturated, partially unsaturated, or aromatic heterocycle containing one to four heteroatoms from the group O, N, or S. R1 and R2 can also form a five-unit or six-unit ring along with the nitrogen atom to which they are linked. Said ring can be interrupted and/or substituted by an atom from the group O, N, and S while R1 and/or R2 can be substituted according to the description. The invention also relates to methods and intermediate products for producing said compounds, agents containing said compounds, and the use thereof for controlling harmful fungi.

摘要翻译： 公开了生产杀真菌三唑并嘧啶化合物的方法，含有所述化合物的试剂及其用于控制​​有害真菌的用途。 还公开了式（1）的三唑并嘧啶，其中取代基具有以下含义：L 1表示烷基; L 2表示卤素; L 3表示氢或卤素; X表示卤素，氰基，烷基，烷氧基或卤代烷氧基; R 1，R 2代表氢，烷基，卤代烷基，环烷基，烯基，链二烯基，炔基或环炔基，苯基，萘基或五个单元至十个单元 饱和的，部分不饱和的或芳族杂环，其含有一至四个O，N或S的杂原子.R 1和R 2也可以形成五单元或 六单元环与它们所连接的氮原子一起。 所述环可以被O，N和S基团的原子中断和/或取代，而R 1和/或R 2可以根据描述被取代 。 本发明还涉及用于生产所述化合物的方法和中间产物，含有所述化合物的试剂及其用于控制​​有害真菌的用途。

公开(公告)号：US09487519B2

公开(公告)日：2016-11-08

申请号：US10589953

申请日：2005-03-08

申请人： Jordi Tormo i Blasco ,  Carsten Blettner ,  Bernd Müller ,  Markus Gewehr ,  Wassilios Grammenos ,  Thomas Grote ,  Joachim Rheinheimer ,  Peter Schäfer ,  Frank Schieweck ,  Anja Schwögler ,  Oliver Wagner ,  Matthias Niedenbrück ,  Maria Scherer ,  Siegfried Strathmann ,  Ulrich Schöfl ,  Reinhard Stierl

发明人： Jordi Tormo i Blasco ,  Carsten Blettner ,  Bernd Müller ,  Markus Gewehr ,  Wassilios Grammenos ,  Thomas Grote ,  Joachim Rheinheimer ,  Peter Schäfer ,  Frank Schieweck ,  Anja Schwögler ,  Oliver Wagner ,  Matthias Niedenbrück ,  Maria Scherer ,  Siegfried Strathmann ,  Ulrich Schöfl ,  Reinhard Stierl

IPC分类号： C07D487/04

CPC分类号： C07D487/04

摘要： 5,6-Dialkyl-7-aminotriazolopyrimidines of the formula I in which the substituents are as defined below: R1 is alkyl or alkoxyalkyl, where the aliphatic groups may be substituted as defined in the description; R2 is CHR3CH3, cyclopropyl, CH═CH2 or CH2CH═CH2; R3 is hydrogen, CH3 or CH2CH3; processes for preparing these compounds, compositions comprising them and their use for controlling phytopathogenic harmful fungi.

公开(公告)号：US07488732B2

公开(公告)日：2009-02-10

申请号：US10549936

申请日：2004-03-30

申请人： Jordi Tormo i Blasco ,  Carsten Blettner ,  Bernd Müller ,  Markus Gewehr ,  Wassilios Grammenos ,  Thomas Grote ,  Andreas Gypser ,  Joachim Rheinheimer ,  Peter Schäfer ,  Frank Schieweck ,  Anja Schwögler ,  Oliver Wagner ,  Maria Scherer ,  Siegfried Strathmann ,  Ulrich Schöfl ,  Reinhard Stierl

发明人： Jordi Tormo i Blasco ,  Carsten Blettner ,  Bernd Müller ,  Markus Gewehr ,  Wassilios Grammenos ,  Thomas Grote ,  Andreas Gypser ,  Joachim Rheinheimer ,  Peter Schäfer ,  Frank Schieweck ,  Anja Schwögler ,  Oliver Wagner ,  Maria Scherer ,  Siegfried Strathmann ,  Ulrich Schöfl ,  Reinhard Stierl

IPC分类号： C07D239/28 ,  C07D239/34 ,  C07D239/42 ,  C07D239/46 ,  A01N43/54

CPC分类号： A01N43/54 ,  C07D239/28 ,  C07D239/30

摘要： 2-Substituted pyrimidines of the formula I in which the index n and the substituents L, Ra, Rb, Rc, Rz, Ru, Rv, A′, A″ and A′″ are as defined in the description and: R1 is C3-C10-alkyl, C3-C10-alkenyl, C3-C10-alkynyl, C3-C12-cycloalkyl, C3-C10-cycloalkenyl or a five- to ten-membered saturated, partially unsaturated or aromatic heterocycle which is attached via carbon and contains one to four heteroatoms from the group consisting of O, N and S, R2 is halogen, cyano, C1-C4-alkyl, C2-C4-alkenyl, C2-C4-alkynyl, C1-C4-alkoxy, C3-C4-alkenyloxy or C3-C4-alkynyloxy, where the alkyl, alkenyl and alkynyl radicals of R2 may be substituted by halogen, cyano, nitro, C1-C2-alkoxy or C1-C4-alkoxycarbonyl, and R3 is cyano, CO2Ra, C(═O)NRzRb, C(═O)—N—ORb, C(═S)—NRaRb, C(═NORa)NRzRb, C(═NRa)NRzRb, C(═O)NRa—NRzRb, C(═N—NRzRc)NRaRb, C(═O)Ra, C(═NORb)Ra, C(═N—NRzRb)Ra, CRaRb—ORz, CRaRb—NRzRc, ON(═CRaRb), O—C(═O)Ra, NRaRb′, NRa(C(═O)Rb), NRa(C(═O)ORb), NRa(C(═O)—NRzRb), NRa(C(═NRc)Rb), NRa(N═CRcRb), NRa—NRzRb, NRz—ORa, NRa(C(═NRc)—NRzRb), NRa(C(═NORc)Rb), processes for preparing these compounds, compositions comprising these compounds and their pesticidal use are described.

摘要翻译： 其中指数n和取代基L，Ra，Rb，Rc，Rz，Ru，Rv，A'，A“和A”'如说明书中所定义的式I的2-取代的嘧啶：R1 C 3 -C 10 - 烷基，C 3 -C 10 - 烯基，C 3 -C 10 - 炔基，C 3 -C 12 - 环烷基，C 3 -C 10 - 环烯基或五至十元饱和的部分不饱和或芳族杂环，其通过碳 并且含有一至四个由O，N和S组成的组的杂原子，R2是卤素，氰基，C1-C4-烷基，C2-C4-烯基，C2-C4-炔基，C1-C4-烷氧基，C3-C4 - 烯氧基或C 3 -C 4 - 炔氧基，其中R 2的烷基，烯基和炔基可以被卤素，氰基，硝基，C 1 -C 2 - 烷氧基或C 1 -C 4 - 烷氧基羰基取代，并且R 3是氰基，CO 2 R a，C（ -O）NR z R b，C（-O）-N-OR b，C（-S）-NR a R b，C（-NOR a）NR z R b，C（-NR a）NR z R b，C（O）NR a -NR b R b，C -NRaRb，C（-O）Ra，C（-NORb）Ra，C（-N-NRzRb）Ra，CRaRb-ORz，CRaRb-NRzRc，ON（-CRaRb），OC（-O）Ra，NRaRb ，NR a（C（-O）R b），NR a（C（-O）R b），NR a（C（-O）OR b） NRa-N RzRb，NRz-ORa，NRa（C（-NRc）-NRzRb），NRa（C（-NORc）Rb），制备这些化合物的方法，包含这些化合物的组合物及其杀虫剂用途。

公开(公告)号：US07375108B2

公开(公告)日：2008-05-20

申请号：US10564013

申请日：2004-07-15

申请人： Anja Schwögler ,  Markus Gewehr ,  Bernd Müller ,  Thomas Grote ,  Wassilios Grammenos ,  Jordi Tormo i Blasco ,  Andreas Gypser ,  Joachim Rheinheimer ,  Carsten Blettner ,  Peter Schäfer ,  Frank Schieweck ,  Oliver Wagner ,  Reinhard Stierl ,  Ulrich Schöfl ,  Siegfried Strathmann ,  Maria Scherer

发明人： Anja Schwögler ,  Markus Gewehr ,  Bernd Müller ,  Thomas Grote ,  Wassilios Grammenos ,  Jordi Tormo i Blasco ,  Andreas Gypser ,  Joachim Rheinheimer ,  Carsten Blettner ,  Peter Schäfer ,  Frank Schieweck ,  Oliver Wagner ,  Reinhard Stierl ,  Ulrich Schöfl ,  Siegfried Strathmann ,  Maria Scherer

IPC分类号： C07D239/42 ,  A01N43/54

CPC分类号： C07D239/42

摘要： The invention relates to 2-substituted pyrimidines of the formula I in which the index n and the substituents R1 to R3 and L are as defined in the description and R4 corresponds to one of the formulae in which Ra, X and Rb are as defined in the description; and also to processes for preparing these compounds, to pesticidal compositions comprising these compounds and to their use as pesticides.

摘要翻译： 本发明涉及式I的2-取代嘧啶，其中指数n和取代基R 1至R 3和L如说明书中所定义， SUP> 4 对应于其中R a，S，X和R b的定义之一如说明书中所定义; 以及制备这些化合物的方法，包括这些化合物的农药组合物及其作为农药的用途。