Oxazinoindole-and thiazinoindole derivatives
    21.
    发明授权
    Oxazinoindole-and thiazinoindole derivatives 失效
    OXAZINOINDOLE-和THIAZINOINDOLE DERIVATIVES

    公开(公告)号:US3833575A

    公开(公告)日:1974-09-03

    申请号:US22628772

    申请日:1972-02-14

    IPC分类号: C07D209/08 C07D87/38

    CPC分类号: C07D209/08 Y10S514/925

    摘要: OXAZINOINDOLE DERIVATIVES CHARACTERIZED BY HAVING AN AMINO(LOWER)ALKYL RADICAL ATTACHED TO THE 1 POSITION OF A 1H-1,4-OXAZINO(4,3-A)INDOLE NUCLEUS ARE DISCLOSED. THE AMINO PORTION OF THE AMINO(LOWER)ALKYL RADICAL MAY BE FURTHER SUBSTITUTED WITH ONE OR TWO LOWER ALKYL GROUPS OR INCORPORATED IN A HETEROCYCLIC AMINE RADICAL. THE DERIVATIVES ARE SUBSTITUTED FURTHER AT POSITIONS 1 AND 10 AND MAY BE OPTIONALLY SUBSTITUTED AT POSITIONS 3. 4, 6, 7, 8 AND 9. THE OXAZINOINDOLE DERIVATIVES OF THIS INVENTION ARE USEFUL ANTIDEPRESSANT AND ANTIULCER AGENTS. METHODS FOR THE PREPARATION AND USE OF THESE DEIVATIVES ARE ALSO DISCLOSED.

    Oxoisoindoles
    22.
    发明授权
    Oxoisoindoles 失效
    OXOISOINDOLES

    公开(公告)号:US3715354A

    公开(公告)日:1973-02-06

    申请号:US3715354D

    申请日:1968-10-04

    申请人: ENDO LAB

    发明人: SCHOEN K PACHTER I

    IPC分类号: C07D209/44 C07D87/38

    CPC分类号: C07D209/44

    摘要: 5-AMINOMETHYL- AND 5-(SUBSTITUTED-AMINO)METHYL-4,5,6, 7-TETRAHYDROOXOISOINDOLES AND THE ACID ADDITION SALTS THEREOF ARE PREPARED BY QUATERNIZING 5-(DIMETHYLAMINO)METHYLOR 5-PIPERIDINOMETHYL-4,5,6,7-TETRAHYDROOXOISOINDOLES, AND REACTING THE QUATERNARY SALTS EITHER WITH A BASE AND AN AMINE, OR ALTERNATIVELY, WITH AN AMINE ONLY. COMPOUNDS OF THE INDICATED TYPES ARE USEFUL AS TRANQUILIZERS, ANTIDEPRESSANTS AND ANALGETICS.

    Cyclic diamides of 2-chloroethyl phosphonic acid
    27.
    发明授权
    Cyclic diamides of 2-chloroethyl phosphonic acid 失效
    2-氯乙基膦酸的环状二酰胺

    公开(公告)号:US3875157A

    公开(公告)日:1975-04-01

    申请号:US18489971

    申请日:1971-09-29

    申请人: GAF CORP

    IPC分类号: C07F9/44 C07D87/38

    CPC分类号: C07F9/44

    摘要: Plant growth regulating compounds are substituted 2chloroethylphosphonic diamides of the formula:

    WHEREIN R1 is cycloalkyl, R2 is hydrogen or cycloalkyl or R1 and R2 together form a heterocyclic ring such as morpholine, piperidine or pyrrolidine. They are prepared by the reaction of 2-chloroethylphosphonic dihalide with the appropriate amine or by the reaction of excess amine with a 2-chloroethyl dichlorophosphite followed by rearrangement of the chloroethyl ester intermediate.

    摘要翻译: 植物生长调节化合物是下式的取代的2-氯乙基膦酸二酰胺:

    4,5 polymethylene pyrimidine derivatives
    28.
    发明授权
    4,5 polymethylene pyrimidine derivatives 失效
    4,5聚甲基哌嗪衍生物

    公开(公告)号:US3757017A

    公开(公告)日:1973-09-04

    申请号:US3757017D

    申请日:1968-01-22

    申请人: MATHIEU J

    发明人: MATHIEU J

    摘要: NEW 4,5-POLYMETHYLENE-PYRIMIDINE DERIVATIVES OR THE GENERAL FORMULA

    2-R1,4,5-(-Z-),6-R2-PYRIMIDINE

    IN WHICH Z IS A POLYMETHYLENE CHAIN CONTAINING 3 TO 6 CARBON ATOMS R1 IS HYDROGEN, HALOGEN, ALKYL, HYDROXYALKYLAMINO OR MORPHOLINO, R2 IS HYDROGEN, HYDROXYALKYLAMINO, BIS(HYDROXYALKYL) AMINO, N-ALKYL-N-HYDROXYALKYLAMINO OR MORPHOLINO, WITH THE PROVISO THAT WHEN R2 IS HYDROGEN, R1 MUST BE A HYDROXYALKYLAMINO OR MORPHOLINO RADICAL, AS WELL AS THEIR SALTS WITH INORGANIC OR ORGANIC ACIDS. THE COMPOUNDS ARE HYPOTENSIVES, PERIPHERAL AND CORONARY VASODILATORS, DIURETICS, BRONCHODILATORS, SPASMOLYTICS AND CIRCULATORY AND RESPIRATORY ANALEPTICS.

    Aminodiphenyl-indolyl-methane dyestuffs
    30.
    发明授权
    Aminodiphenyl-indolyl-methane dyestuffs 失效
    氨基二苯甲酸甲酯试验

    公开(公告)号:US3652556A

    公开(公告)日:1972-03-28

    申请号:US3652556D

    申请日:1968-03-29

    申请人: BAYER AG

    CPC分类号: C09B11/26

    摘要: DYESTUFFS OF THE GENERAL FORMULA

    ((4-((-N-)>N-)PHENYL)-C(+)(-(2-R3-INDOL-3,1-YLENE)-R4)-)

    BENZENE X(-)

    ARE PREPARED WHICH ARE ADAPTED FOR USE IN DYEING AND PRINTING MATERIALS MADE OF LEATHER, TANNIN TREATED COTTON, CELLULOSE ACETATE, SYNTHETIC SUPER POLYAMIDES AND POLYURETHANES AND FOR THE DYEING OF LIGNIN-CONTAINING FIBERS AS WELL AS FOR USE IN PREPARING INK-TYPE MATERIALS. AS DYESTUFFS THE MATERIAL ARE CHARACTERIZED BY GOOD FASTNESS TO LIGHT, WET PROCESSING, RUBBING AND SUBLIMINATION, AND THEY ARE GENERALLY CHARACTERIZED BY GOOD AFFINITY TO THE SUBJECT FIBERS.