公开(公告)号：US20050256138A1

公开(公告)日：2005-11-17

申请号：US10513030

申请日：2003-04-30

申请人： Jordi Tormo i Blasco ,  Carsten Blettner ,  Bernd Muller ,  Markus Gewhr ,  Wassilios Grammenos ,  Thomas Grote ,  Andreas Gypser ,  Joachim Rheinheimer ,  Peter Schafer ,  Frank Schieweck ,  Anja Schwogler ,  Eberhard Ammermann ,  Siegfried Strathmann ,  Gisela Lorenz ,  Reinhard Stierl

发明人： Jordi Tormo i Blasco ,  Carsten Blettner ,  Bernd Muller ,  Markus Gewhr ,  Wassilios Grammenos ,  Thomas Grote ,  Andreas Gypser ,  Joachim Rheinheimer ,  Peter Schafer ,  Frank Schieweck ,  Anja Schwogler ,  Eberhard Ammermann ,  Siegfried Strathmann ,  Gisela Lorenz ,  Reinhard Stierl

IPC分类号： A01N43/90 ,  C07C69/65 ,  C07D487/04 ,  A61K31/519

CPC分类号： C07D487/04 ,  A01N43/90 ,  C07C69/65

摘要： Disclosed are a method for producing fungicidal triazolopyrimidine compounds, agents containing said compounds, and the use thereof for controlling harmful fungi. Also disclosed are triazolopyrimidines of formula (1), in which the substituents have the following meaning: L1 represents alkyl; L2 represents halogen; L3represents hydrogen or halogen; X represents halogen, cyano, alkyl, alkoxy, or haloalkoxy; R1, R2 represent hydrogen, alkyl, haloalkyl, cycloalkyl, alkenyl, alkadienyl, alkinyl, or cycloalkinyl, phenyl, naphthyl, or a five-unit to ten-unit saturated, partially unsaturated, or aromatic heterocycle containing one to four heteroatoms from the group O, N, or S. R1 and R2 can also form a five-unit or six-unit ring along with the nitrogen atom to which they are linked. Said ring can be interrupted and/or substituted by an atom from the group O, N, and S while R1 and/or R2 can be substituted according to the description. The invention also relates to methods and intermediate products for producing said compounds, agents containing said compounds, and the use thereof for controlling harmful fungi.

摘要翻译： 公开了生产杀真菌三唑并嘧啶化合物的方法，含有所述化合物的试剂及其用于控制​​有害真菌的用途。 还公开了式（1）的三唑并嘧啶，其中取代基具有以下含义：L 1表示烷基; L 2表示卤素; L 3表示氢或卤素; X表示卤素，氰基，烷基，烷氧基或卤代烷氧基; R 1，R 2代表氢，烷基，卤代烷基，环烷基，烯基，链二烯基，炔基或环炔基，苯基，萘基或五个单元至十个单元 饱和的，部分不饱和的或芳族杂环，其含有一至四个O，N或S的杂原子.R 1和R 2也可以形成五单元或 六单元环与它们所连接的氮原子一起。 所述环可以被O，N和S基团的原子中断和/或取代，而R 1和/或R 2可以根据描述被取代 。 本发明还涉及用于生产所述化合物的方法和中间产物，含有所述化合物的试剂及其用于控制​​有害真菌的用途。

公开(公告)号：US20080076785A1

公开(公告)日：2008-03-27

申请号：US11663982

申请日：2005-09-27

申请人： Carsten Blettner ,  Jordi Tormo i Blasco ,  Bernd Muller ,  Markus Gewehr ,  Wassilios Grammenos ,  Thomas Grote ,  Udo Hunger ,  Joachim Rheinheimer ,  Peter Schafer ,  Frank Schieweck ,  Anja Schwogler ,  Oliver Wagner ,  John-Bryan Speakman ,  Thorsten Jabs ,  Siegfried Strathmann ,  Ulrich Schofl ,  Maria Scherer ,  Reinhard Stierl

发明人： Carsten Blettner ,  Jordi Tormo i Blasco ,  Bernd Muller ,  Markus Gewehr ,  Wassilios Grammenos ,  Thomas Grote ,  Udo Hunger ,  Joachim Rheinheimer ,  Peter Schafer ,  Frank Schieweck ,  Anja Schwogler ,  Oliver Wagner ,  John-Bryan Speakman ,  Thorsten Jabs ,  Siegfried Strathmann ,  Ulrich Schofl ,  Maria Scherer ,  Reinhard Stierl

IPC分类号： A01N43/54 ,  A01P3/00 ,  C07D239/70

CPC分类号： A01N43/90 ,  C07D487/04

摘要： The invention relates to 7-aminomethyl-1,2,4-triazolo[1,5-a]pyrimidine compounds of general formula (I) and the agriculturally compatible salts of said compounds. In said formula: R1 and R2 represent hydrogen, alkyl, haloalkyl, alkoxy, cycloalkyl, bicycloalkyl, halocycloalkyl, alkenyl, alkadienyl, haloalkenyl, cycloalkenyl, halocycloalkenyl, alkynyl, haloalkynyl or phenyl, naphthyl, or a 5- or 6-membered saturated, partially unsaturated or aromatic heterocycle, containing 1 to 4 heteroatoms from the group containing O, N or S, or R1 and R2, together with the nitrogen atom to which they are bonded, can also form a five- or six-membered heterocyclyl or heteroaryl, which is bonded by means of N and can contain 1 to 3 additional heteroatoms from the group containing O, N and S as the ring member and can be substituted according to the description; R3 and R4 represent hydrogen, alkyl, haloalkyl, haloalkoxy, alkoxy, or alkoxyalkyl; X represents halogen, cyano, a 5- or 6-membered saturated, partially unsaturated or aromatic heterocycle, containing 1, 2 or 3 heteroatoms from the group containing O, N or S as the ring member, alkyl, alkoxy, alkenyl or alkynyl, whereby the latter 4 groups can be substituted according to the description; L is defined as cited in the claims and the description; and m represents 0, 1, 2, 3, 4 or 5. The invention also relates to the use of the triazolopyrimidine compounds of general formula (I) and their agriculturally compatible salts for controlling plant-pathogenic fungi, to a method for controlling plant-pathogenic fungi, containing at least one compound of general formula (I) and/or an agriculturally compatible salt of said compound and at least one liquid or solid carrier.

摘要翻译： 本发明涉及通式（I）的7-氨基甲基-1,2,4-三唑并[1,5-a]嘧啶化合物和所述化合物的农业上相容的盐。 在所述式中：R 1和R 2表示氢，烷基，卤代烷基，烷氧基，环烷基，二环烷基，卤代环烷基，烯基，链烯基，卤代烯基，环烯基，卤代环烯基，炔基，卤代炔基或苯基，萘基或5-或6-元饱和， 部分不饱和或芳族杂环，含有1至4个含有O，N或S的杂原子，或R 1和R 2与它们所键合的氮原子一起也可以形成五元或六元杂环基或杂芳基 ，其通过N键合并且可以含有来自含有O，N和S的基团的1至3个另外的杂原子作为环成员，并且可以根据描述进行取代; R3和R4代表氢，烷基，卤代烷基，卤代烷氧基，烷氧基或烷氧基烷基; X代表卤素，氰基，含有1,2或3个杂原子的5-或6-元饱和的部分不饱和或芳族杂环，所述杂环含有作为环成员的O，N或S，烷基，烷氧基，烯基或炔基， 由此后4个组可以根据描述被替代; L定义为权利要求书和说明书中引用的; 和m表示0,1,2,3,4或5.本发明还涉及通式（I）的三唑并嘧啶化合物及其农业上相容的盐用于控制植物致病真菌的用途，用于控制植物的方法 致病真菌，含有至少一种通式（I）的化合物和/或所述化合物的农业上相容的盐和至少一种液体或固体载体。

公开(公告)号：US20070105928A1

公开(公告)日：2007-05-10

申请号：US10582938

申请日：2004-12-14

申请人： Jordi Tormo I Blasco ,  Carsten Blettner ,  Bernd Muller ,  Markus Gewehr ,  Wassilios Grammenos ,  Thomas Grote ,  Joachim Rheinheimer ,  Peter Schafer ,  Frank Schieweck ,  Anja Schwogler ,  Oliver Wagner ,  Maria Scherer ,  Siegfried Strathmann ,  Ulrich Schofl ,  Reinhard Stierl

发明人： Jordi Tormo I Blasco ,  Carsten Blettner ,  Bernd Muller ,  Markus Gewehr ,  Wassilios Grammenos ,  Thomas Grote ,  Joachim Rheinheimer ,  Peter Schafer ,  Frank Schieweck ,  Anja Schwogler ,  Oliver Wagner ,  Maria Scherer ,  Siegfried Strathmann ,  Ulrich Schofl ,  Reinhard Stierl

IPC分类号： A61K31/41

CPC分类号： F02B43/04 ,  F02B19/14 ,  F02B43/10 ,  F02M25/10 ,  Y02T10/121 ,  Y02T10/125 ,  Y02T10/32

摘要： 6-Pentafluorophenyltriazolopyrimidines of the formula I in which the substituents are as defined below: R1 is alkyl, haloalkyl, cycloalkyl, halocycloalkyl, alkenyl, haloalkenyl, cycloalkenyl, halocycloalkenyl, alkinyl, haloalkinyl or phenyl, naphthyl, or a five- or six-membered saturated, partially unsaturated or aromatic heterocycle which contains one to four heteroatoms from the group consisting of O, N and S, R2 is hydrogen or one of the groups mentioned under R1, R1 and R2 together with the nitrogen atom to which they are attached may also form a five- or six-membered heterocyclyl or heteroaryl which is attached via N and may contain one to three further heteroatoms from the group consisting of O, N and S as ring members; R1 and/or R2 may be substituted as defined in the description; X is cyano, alkyl, alkoxy, alkenyloxy, haloalkoxy or haloalkenyloxy, processes for preparing these compounds, compositions comprising them and their use for controlling phytopathogenic harmful fungi.

摘要翻译： 式I的6-五氟苯基三唑并嘧啶，其中取代基如下：R 1是烷基，卤代烷基，环烷基，卤代环烷基，烯基，卤代烯基，环烯基，卤代环烯基，炔基，卤代炔基或苯基，萘基， 或五元或六元饱和，部分不饱和或芳族杂环，其含有一至四个由O，N和S组成的组的杂原子，R 2是氢或下述基团之一 R 1，R 1和R 2与它们所连接的氮原子一起也可以形成五元或六元杂环基 或杂芳基，其通过N连接并且可以含有一个至三个由O，N和S组成的组的另外的杂原子作为环成员; R 1和/或R 2可以如说明书中所定义的取代; X是氰基，烷基，烷氧基，烯氧基，卤代烷氧基或卤代烯氧基，制备这些化合物的方法，包含它们的组合物及其用于控制​​植物病原性有害真菌的用途。

公开(公告)号：US20070078149A1

公开(公告)日：2007-04-05

申请号：US10580416

申请日：2004-12-16

申请人： Jordi Tormo I Blasco ,  Carsten Blettner ,  Bernd Muller ,  Markus Gewehr ,  Wassilios Grammenos ,  Thomas Grote ,  Joachim Rheinheimer ,  Peter Schafer ,  Frank Schieweck ,  Anja Schwogler ,  Oliver Wagner ,  Maria Scherer ,  Siegfried Strathmann ,  Ulrich Schofl ,  Reinhard Stierl

发明人： Jordi Tormo I Blasco ,  Carsten Blettner ,  Bernd Muller ,  Markus Gewehr ,  Wassilios Grammenos ,  Thomas Grote ,  Joachim Rheinheimer ,  Peter Schafer ,  Frank Schieweck ,  Anja Schwogler ,  Oliver Wagner ,  Maria Scherer ,  Siegfried Strathmann ,  Ulrich Schofl ,  Reinhard Stierl

IPC分类号： A01N43/90 ,  C07D487/04

CPC分类号： C07D487/04 ,  A01N43/90

摘要： Triazolopyrimidines of the formula I in which the substituents are as defined below: R1, R2 are hydrogen, alkyl, haloalkyl, cycloalkyl, halocycloalkyl, alkenyl, haloalkenyl, cycloalkenyl, halocycloalkenyl, alkynyl, haloalkynyl or phenyl, naphthyl, or a five- or six-membered saturated, partially unsaturated or aromatic heterocycle which contains one to four heteroatoms from the group consisting of O, N and S, R1 and R2 together with the nitrogen atom to which they are attached may also form a five- or six-membered heterocyclyl or heteroaryl which is attached via N and may contain a further heteroatom from the group consisting of O, N and S as ring member and may be substituted as defined in the description; L1, L2 are hydrogen, cyano, haloalkyl, alkoxy, alkenyloxy or C(═O)A, where at least one group L1 or L2 is not hydrogen; A is hydrogen, hydroxyl, alkyl, alkoxy, haloalkoxy, C1-C8-alkylamino or dialkylamino; L3 is hydrogen, halogen, cyano, nitro, haloalkyl, alkoxy or alkoxycarbonyl; X is halogen, cyano, alkyl, haloalkyl, alkoxy or haloalkoxy; processes and intermediates for preparing these compounds, compositions comprising them and their use for controlling phytopathogenic harmful fungi.

摘要翻译： 其中取代基如下定义的式I的三唑并嘧啶：R 1，R 2是氢，烷基，卤代烷基，环烷基，卤代环烷基，烯基，卤代烯基，环烯基， 卤代环烯基，炔基，卤代炔基或苯基，萘基或五或六元饱和的部分不饱和或芳族杂环，其含有一至四个由O，N和S组成的组的杂原子，R 1 和R 2与它们所连接的氮原子一起也可以形成五元或六元杂环基或杂芳基，其通过N连接并且可以含有来自以下的另外的杂原子： O，N和S作为环成员，并且可以如说明书中所定义的取代; L 1，L 2是氢，氰基，卤代烷基，烷氧基，烯氧基或C（-O）A，其中至少一个基团L 1 >或L 2不是氢; A是氢，羟基，烷基，烷氧基，卤代烷氧基，C 1 -C 8烷基氨基或二烷基氨基; L 3是氢，卤素，氰基，硝基，卤代烷基，烷氧基或烷氧基羰基; X是卤素，氰基，烷基，卤代烷基，烷氧基或卤代烷氧基; 制备这些化合物的方法和中间体，包含它们的组合物及其用于控制​​植物病原性有害真菌的用途。

公开(公告)号：US20080176831A1

公开(公告)日：2008-07-24

申请号：US11596891

申请日：2005-05-17

申请人： Anja Schwogler ,  Frank Schieweck ,  Joachim Rheinheimer ,  Markus Gewehr ,  Bernd Muller ,  Thomas Grote ,  Wassilios Grammenos ,  Udo Hunger ,  Carsten Blettner ,  Peter Schafer ,  Oliver Wagner ,  Reinhard Stierl ,  Ulrich Schofl ,  Siegfried Strathmann ,  Maria Scherer

发明人： Anja Schwogler ,  Frank Schieweck ,  Joachim Rheinheimer ,  Markus Gewehr ,  Bernd Muller ,  Thomas Grote ,  Wassilios Grammenos ,  Udo Hunger ,  Carsten Blettner ,  Peter Schafer ,  Oliver Wagner ,  Reinhard Stierl ,  Ulrich Schofl ,  Siegfried Strathmann ,  Maria Scherer

IPC分类号： A01N43/46 ,  C07D403/04 ,  A01N43/54 ,  A01P7/00 ,  A01P3/00 ,  A01N43/58

CPC分类号： C07D401/04 ,  C07D403/04

摘要： The invention relates to 2-substituted pyrimidines of the formula I in which the index n and the substituents L and R1 to R3 are as defined in the description and X is a group —CH—Ra, —N— or —S—; R1 may be hydrogen, halogen, C1-C6-alkyl, C1-C6-alkoxy, cyano or C1-C6-alkoxycarbonyl; Rb is hydrogen, C1-C6-alkyl or C3-C6-cycloalkyl; T is a group —CH—Ra—; p is an integer from 1 to 4; Y is a group —CH—Ra— or —N—Rb o is 0 or 1; Z is O, S or a group N(Rc) Rc is hydrogen, C1-C6-alkyl or C1-C6-alkoxy, and to processes for their preparation, to pesticidal compositions comprising them and to their use as pesticides.

摘要翻译： 本发明涉及式I的2-取代嘧啶，其中指数n和取代基L和R 1至R 3如在说明书中所定义，X是 基团-CH-R a，N - 或-S-; R 1可以是氢，卤素，C 1 -C 6 - 烷基，C 1 -C 3 > 6个 - 烷氧基，氰基或C 1 -C 6 - 烷氧基羰基; R b是氢，C 1 -C 6 - 烷基或C 3 -C 6 - 环烷基; T是基团-CH-R a， p是1至4的整数; Y是基团-CH-R a - 或-N-R b是0或1; Z是O，S或基团N（R c）R c是氢，C 1 -C 6 烷基或C 1 -C 6 - 烷氧基，并且其制备方法，包含它们的杀虫组合物及其作为农药的用途。

公开(公告)号：US20080132522A1

公开(公告)日：2008-06-05

申请号：US11631006

申请日：2005-07-12

申请人： Joachim Rheinheimer ,  Frank Schieweck ,  Thomas Grote ,  Carsten Blettner ,  Anja Schwogler ,  Markus Gewehr ,  Wassilios Grammenos ,  Udo Hunger ,  Bernd Muller ,  Peter Schafer ,  Jochen Dietz ,  John-Bryan Speakman ,  Maria Scherer ,  Siegfried Strathmann ,  Ulrich Schofl ,  Reinhard Stierl

发明人： Joachim Rheinheimer ,  Frank Schieweck ,  Thomas Grote ,  Carsten Blettner ,  Anja Schwogler ,  Markus Gewehr ,  Wassilios Grammenos ,  Udo Hunger ,  Bernd Muller ,  Peter Schafer ,  Jochen Dietz ,  John-Bryan Speakman ,  Maria Scherer ,  Siegfried Strathmann ,  Ulrich Schofl ,  Reinhard Stierl

IPC分类号： A01N43/54 ,  C07D401/04 ,  A01P3/00 ,  A01P13/00 ,  A01P15/00

CPC分类号： C07D239/34 ,  C07D401/04 ,  C07D403/12

摘要： The invention relates to 2-substituted pyrimidines of the formula I in which the index n and the substituents R1 to R4, B and L are as defined in the description and Y is a group —O— or —S—, and to processes for their preparation, pesticidal compositions and methods for controlling harmful fungi and animal pests using the compounds according to the invention.

摘要翻译： 本发明涉及式I的2-取代嘧啶，其中指数n和取代基R 1至R 4，B和L如说明书中所定义，以及 Y是基团-O-或-S-，并且使用本发明的化合物进行制备，杀虫组合物和控制有害真菌和动物害虫的方法。

公开(公告)号：US20080058208A1

公开(公告)日：2008-03-06

申请号：US11547185

申请日：2005-03-26

申请人： Jordi Tormo i Blasco ,  Carsten Blettner ,  Bernd Muller ,  Markus Gewehr ,  Wassilios Grammenos ,  Thomas Grote ,  Joachim Rheinheimer ,  Peter Schafer ,  Frank Schieweck ,  Anja Schwogler ,  Oliver Wagner ,  Matthias Niedenbruck ,  Maria Scherer ,  Siegfried Strathmann ,  Ulrich Schofl ,  Reinhard Stierl

发明人： Jordi Tormo i Blasco ,  Carsten Blettner ,  Bernd Muller ,  Markus Gewehr ,  Wassilios Grammenos ,  Thomas Grote ,  Joachim Rheinheimer ,  Peter Schafer ,  Frank Schieweck ,  Anja Schwogler ,  Oliver Wagner ,  Matthias Niedenbruck ,  Maria Scherer ,  Siegfried Strathmann ,  Ulrich Schofl ,  Reinhard Stierl

IPC分类号： C07D487/04 ,  A01N25/34 ,  A01N43/90

CPC分类号： C07D487/04

摘要： The invention relates to 5,6-cycloalkyl-7-aminotriazolopyrimidines of formula (I), where X=alkylene or alkenylene, whereby the carbon chain can be interrupted by one or two heteroatoms selected from S, O or NR1, R1═H, alkyl or C(═O)alkyl, L=halogen, cyano, nitro, alkyl, haloalkyl, alkoxy, haloalkoxy, alkenyl, alkinyl or NR2R3; R2,R3=each one of the groups given for R1 and m=a whole number from 0 to 5, whereby the aliphatic groups can be substituted by one to three of the following groups: halogen, cyano, nitro, hydroxy, alkoxy, alkylthio, or NRaRb, where Ra, Rb═H or alkyl in which the carbon chains can be halogenated. The invention further relates to methods for production of said compounds, agents comprising the same and use thereof for the prevention of fungal pests harmful to plants.

摘要翻译： 本发明涉及式（I）的5,6-环烷基-7-氨基三唑并嘧啶，其中X =亚烷基或亚烯基，其中碳链可被一个或两个选自S，O或NR 1的杂原子中断， 卤素，氰基，硝基，烷基，卤代烷基，烷氧基，卤代烷氧基，烯基，炔基或NR 2（O） 3 3 R 2，R 3 =每个给定R 1的基团，m = 0至5的整数，由此脂族基 基团可以被一至三个以下基团取代：卤素，氰基，硝基，羟基，烷氧基，烷硫基或NR a R b，其中R 0， 或其中碳链可以被卤化的烷基。 本发明还涉及生产所述化合物的方法，包含该化合物的试剂及其用于预防对植物有害的真菌害虫的用途。

公开(公告)号：US20080280759A1

公开(公告)日：2008-11-13

申请号：US10582971

申请日：2004-12-14

申请人： Jordi Tormo i Blasco ,  Carsten Blettner ,  Bernd Muller ,  Markus Gewehr ,  Wassilios Grammenos ,  Thomas Grote ,  Joachim Rheinheimer ,  Peter Schafer ,  Frank Schieweck ,  Anja Schwogler ,  Oliver Wagner ,  Maria Scherer ,  Siegfried Strathmann ,  Ulrich Schofl ,  Reinhard Stierl

发明人： Jordi Tormo i Blasco ,  Carsten Blettner ,  Bernd Muller ,  Markus Gewehr ,  Wassilios Grammenos ,  Thomas Grote ,  Joachim Rheinheimer ,  Peter Schafer ,  Frank Schieweck ,  Anja Schwogler ,  Oliver Wagner ,  Maria Scherer ,  Siegfried Strathmann ,  Ulrich Schofl ,  Reinhard Stierl

IPC分类号： A01C1/06 ,  C07D487/04 ,  A61K31/519

CPC分类号： A01N43/90 ,  C07D487/04

摘要： 6-(2-Halo-4-alkoxyphenyl)triazolopyrimidines of the formula I in which the substituents are as defined below: R1 is alkyl, haloalkyl, cycloalkyl, halocycloalkyl, alkenyl, haloalkenyl, cycloalkenyl, halocycloalkenyl, alkynyl, haloalkynyl or phenyl, naphthyl, or a five- or six-membered saturated, partially unsaturated or aromatic heterocycle which contains one to four heteroatoms from the group consisting of O, N and S, R2 is hydrogen or one of the groups mentioned under R1, R1 and R2 together with the nitrogen atom to which they are attached may also form a five- or six-membered heterocyclyl or heteroaryl which is attached via N and may contain one to three further heteroatoms from the group consisting of O, N and S as ring members; R3 is alkyl, haloalkyl, alkenyl, haloalkenyl, alkynyl, haloalkynyl, phenylalkyl, mono- or dialkoxyalkyl; R1, R2 and/or R3 may be substituted as mentioned in the description; L is hydrogen, fluorine or chlorine; X is cyano, alkyl, alkoxy, alkenyloxy, haloalkoxy or haloalkenyloxy; processes for preparing these compounds, compositions comprising them and their use for controlling phytopathogenic harmful fungi.

摘要翻译： 其中取代基如下定义的式I的6-（2-卤代-4-烷氧基苯基）三唑并嘧啶：R 1是烷基，卤代烷基，环烷基，卤代环烷基，烯基，卤代烯基，环烯基，卤代环烯基 ，炔基，卤代炔基或苯基，萘基或五元或六元饱和的部分不饱和或芳族杂环，其含有一至四个由O，N和S组成的组的杂原子，R 2， 是氢或R 1，R 1和R 2所提及的基团之一与它们所连接的氮原子一起也可以 形成通过N连接的五元或六元杂环基或杂芳基，并且可以含有一个至三个由O，N和S组成的组的另外的杂原子作为环成员; R 3是烷基，卤代烷基，烯基，卤代烯基，炔基，卤代炔基，苯基烷基，单或二烷氧基烷基; R 1，R 2和/或R 3可以如说明书中所述被取代; L是氢，氟或氯; X是氰基，烷基，烷氧基，烯氧基，卤代烷氧基或卤代烯氧基; 制备这些化合物的方法，包含它们的组合物及其用于控制​​植物病原性有害真菌的用途。

公开(公告)号：US20080119493A1

公开(公告)日：2008-05-22

申请号：US10590326

申请日：2005-03-08

申请人： Jordi Tormo i Blasco ,  Carsten Blettner ,  Bernd Muller ,  Markus Gewehr ,  Wassilios Grammenos ,  Thomas Grote ,  Joachim Rheinheimer ,  Peter Schafer ,  Frank Schieweck ,  Anja Schwogler ,  Oliver Wagner ,  Matthias Niedenbruck ,  Maria Scherer ,  Siegfried Strathmann ,  Ulrich Schofl ,  Reinhard Stierl ,  Udo Hunger

发明人： Jordi Tormo i Blasco ,  Carsten Blettner ,  Bernd Muller ,  Markus Gewehr ,  Wassilios Grammenos ,  Thomas Grote ,  Joachim Rheinheimer ,  Peter Schafer ,  Frank Schieweck ,  Anja Schwogler ,  Oliver Wagner ,  Matthias Niedenbruck ,  Maria Scherer ,  Siegfried Strathmann ,  Ulrich Schofl ,  Reinhard Stierl ,  Udo Hunger

IPC分类号： A01N43/90 ,  C07D487/04 ,  A01P3/00

CPC分类号： C07D487/04

摘要： The invention relates to 5,6-dialkyl-7-amino-triazolopyrimidines of formula (I), in which the substituents are defined as follows: R1 represents alkyl, alkoxyalkyl, alkenyl or alkynyl; R2 represents alkyl, alkoxyalkyl, alkenyl or alkynyl, R1 and/or R2 being substituted according to the description. The invention also relates to a method for producing said compounds, to agents containing the latter and to their use for controlling plant-pathogenic fungi.

摘要翻译： 本发明涉及式（I）的5,6-二烷基-7-氨基 - 三唑并嘧啶，其中取代基定义如下：R 1表示烷基，烷氧基烷基，烯基或炔基; R 2表示根据描述被取代的烷基，烷氧基烷基，烯基或炔基，R 1和/或R 2 2。 本发明还涉及一种生产所述化合物的方法，含有后者的药剂及其用于控制​​植物致病真菌的用途。

公开(公告)号：US20080039319A1

公开(公告)日：2008-02-14

申请号：US11596464

申请日：2005-05-11

申请人： Carsten Blettner ,  Markus Gewehr ,  Wassilios Grammenos ,  Thomas Grote ,  Udo Hunger ,  Bernd Muller ,  Matthias Niedenbruck ,  Joachim Rheinheimer ,  Peter Schafer ,  Frank Schieweck ,  Anja Schwogler ,  Oliver Wagner ,  Barbara Nave ,  Maria Scherer ,  Siegfried Strathmann ,  Ulrich Schofl ,  Reinhard Stierl

发明人： Carsten Blettner ,  Markus Gewehr ,  Wassilios Grammenos ,  Thomas Grote ,  Udo Hunger ,  Bernd Muller ,  Matthias Niedenbruck ,  Joachim Rheinheimer ,  Peter Schafer ,  Frank Schieweck ,  Anja Schwogler ,  Oliver Wagner ,  Barbara Nave ,  Maria Scherer ,  Siegfried Strathmann ,  Ulrich Schofl ,  Reinhard Stierl

IPC分类号： A01N43/90 ,  A01N25/34 ,  A01N59/20

CPC分类号： A01N43/90 ,  A01N59/06 ,  A01N59/02 ,  A01N57/12 ,  A01N47/38 ,  A01N47/34 ,  A01N47/24 ,  A01N47/04 ,  A01N43/50 ,  A01N43/76 ,  A01N43/653 ,  A01N43/36 ,  A01N43/40 ,  A01N43/32 ,  A01N37/48 ,  A01N37/46 ,  A01N37/38 ,  A01N37/34 ,  A01N2300/00

摘要： The invention relates to fungicidal mixtures containing in the form of active components 1) 5-methyl-7-amino-triazolopyrimidine of formula (I), wherein R1 is alkyl, halogenalkyl, alkenyl or cyclopentyl, R2 is hydrogen or alkyl, R1 and R2 together with the nitrogen atom to which they are bound may form a piperidinyl cycle substitutable by a methyl group, L1 is fluorine or chlorine, L2, L3 are independently from each other hydrogen, fluorine or chlorine and 2) at least one type of active substance selected from groups A) azoles, B) strobilurins, C) acyl alanines, D) amine derivatives, E) anilinopyrimidines; F) dicarboximides; G) cinnamic acid amides and analogues thereof, H) antibiotics, K) dithiocarbamates, L) heterocyclic compounds, M) sulphur and copper fungicides, N) nitrophenyl derivatives, O) phenylpyrroles, P) sulfenic acid derivatives, Q) other fungicides and R) growth retardants according to the descriptions, wherein said mixtures contain the compounds in a synergically efficient amount. Novel triazolopyrimidines, methods for controlling pathogenic fungi using the mixtures of the compound (1) with active substances of the groups A) and R), the use the compounds (I) with the active substances of the groups A) and R) for producing said mixtures and agents containing said mixtures are also disclosed.

摘要翻译： 本发明涉及含有活性组分形式的杀真菌混合物1）式（I）的5-甲基-7-氨基 - 三唑并嘧啶，其中R 1是烷基，卤代烷基，烯基或环戊基，R R 2是氢或烷基，R 1和R 2与它们所连接的氮原子一起可以形成可被 甲基，L 1是氟或氯，L 2，L 3，3彼此独立地为氢，氟或氯，以及2）在 至少一种活性物质选自A）唑类，B）嗜球果伞素，C）酰基丙氨酸，D）胺衍生物，E）苯胺基嘧啶; F）二羧酰亚胺; G）肉桂酸酰胺及其类似物，H）抗生素，K）二硫代氨基甲酸盐，L）杂环化合物，M）硫和铜杀真菌剂，N）硝基苯基衍生物，O）苯基吡咯，P）亚磺酸衍生物，Q）其他杀真菌剂和R ）生长阻滞剂，其中所述混合物包含协同有效量的化合物。 新型三唑并嘧啶，使用化合物（1）与A）和R）基团的活性物质的混合物来控制致病真菌的方法，将化合物（I）与A）和R）基团的活性物质一起用于生产 还公开了含有所述混合物的所述混合物和试剂。