公开(公告)号：US06482984B2

公开(公告)日：2002-11-19

申请号：US09760710

申请日：2001-01-17

申请人： Wassilios Grammenos ,  Hubert Sauter ,  Andreas Gypser ,  Markus Gewehr ,  Jordi Tormo i Blasco ,  Arne Ptock ,  Bernd Müller ,  Oliver Cullmann ,  Thomas Grote ,  Eberhard Ammermann ,  Siegfried Strathmann ,  Gisela Lorenz

发明人： Wassilios Grammenos ,  Hubert Sauter ,  Andreas Gypser ,  Markus Gewehr ,  Jordi Tormo i Blasco ,  Arne Ptock ,  Bernd Müller ,  Oliver Cullmann ,  Thomas Grote ,  Eberhard Ammermann ,  Siegfried Strathmann ,  Gisela Lorenz

IPC分类号： C07C23305

CPC分类号： C07C251/48 ,  A01N37/50

摘要： Iminooxy-substituted benzyl phenyl ethers of the formula I in which the substituents and the index are as defined below: Y is H, CH3, F or Cl; Q is C(═CHOCH3)—COOCH3, C(═CHCH3)—COOCH3, C(═NOCH3)—COOCH3, C(═NOCH3)—CONHCH3 or N(—OCH3)—COOCH3; X is hydrogen, halogen, alkyl, alkoxy or CF3; m is 1 or 2, where the radicals X may be different if m=2; R1 is alkyl and R2 is hydrogen or alkyl; or R1 and R2 together are cyclopropyl, cyclopentyl or cyclohexyl; R3 is alkyl or CF3; and R4 is alkyl, alkenyl, alkynyl, haloalkyl, haloalkenyl or haloalkynyl; processes and intermediates for their preparation, compositions comprising them, and their use, are described.

摘要翻译： 取代基和指数如下定义的式Iin的亚氨氧基取代的苄基苯基醚：Y是H，CH 3，F或Cl; Q是C（= CHOCH 3）-COOCH 3，C（= CHCH 3）-COOCH 3，C （= NOCH 3）-COOCH 3，C（= NOCH 3）-CONHCH 3或N（-OCH 3）-COOCH 3; X是氢，卤素，烷基，烷氧基或CF 3; m是1或2，其中基团X可以不同，如果m = 2; R 1是烷基，R 2是氢或烷基; 或者R 1和R 2一起是环丙基，环戊基或环己基; R 3是烷基或CF 3; 和R 4是烷基，烯基，炔基，卤代烷基，卤代烯基或卤代炔基;其制备方法和中间体，包含它们的组合物及其用途。

公开(公告)号：US06451790B1

公开(公告)日：2002-09-17

申请号：US09889164

申请日：2001-07-11

申请人： Markus Gewehr ,  Hubert Sauter ,  Bernd Müller ,  Wassilios Grammenos ,  Andreas Gypser ,  Arne Ptock ,  Oliver Cullmann ,  Jordi Tormo i Blasco ,  Eberhard Ammermann ,  Siegfried Strathmann ,  Gisela Lorenz ,  Volker Harries ,  Roland Götz ,  Thomas Grote

发明人： Markus Gewehr ,  Hubert Sauter ,  Bernd Müller ,  Wassilios Grammenos ,  Andreas Gypser ,  Arne Ptock ,  Oliver Cullmann ,  Jordi Tormo i Blasco ,  Eberhard Ammermann ,  Siegfried Strathmann ,  Gisela Lorenz ,  Volker Harries ,  Roland Götz ,  Thomas Grote

IPC分类号： C07D41312

CPC分类号： C07D413/12 ,  A01N43/82 ,  A01N43/88 ,  C07D231/20 ,  C07D249/12 ,  C07D413/14

摘要： Compounds of formula I wherein W is optionally substituted alkylene; Y is N or CRa; Ra is hydrogen, halogen or alkyl; R1n represents hydrogen or 1 to 4 substituents; R2 is hydrogen, nitro, cyano, halogen, alkyl, haloalkyl, alkoxy, alkylthio or alkoxycarbonyl; R3 is optionally substituted alkyl, cycloalkyl, aryl or hetaryl; A is N—OR4, CH—OR4, CH—SR4 or CHR5; R4 is alkyl or haloalkyl; R5 is halogen, alkyl or haloalkyl; methods and intermediates for their preparation. The compounds and compositions comprising them are useful for combating animal pests and harmful fungi.

摘要翻译： 式I的化合物，其中W是任选取代的亚烷基; Y是N或CR a; R a是氢，卤素或烷基; R 11代表氢或1-4个取代基; R 2是氢，硝基，氰基，卤素，烷基，卤代烷基，烷氧基，烷硫基或 烷氧基羰基; R3是任选取代的烷基，环烷基，芳基或杂芳基; A是N-OR4，CH-OR4，CH-SR4或CHR5; R4是烷基或卤代烷基; R5是卤素，烷基或卤代烷基;其制备方法和中间体 。 包含它们的化合物和组合物可用于对抗动物害虫和有害真菌。

公开(公告)号：US20060211711A1

公开(公告)日：2006-09-21

申请号：US10550571

申请日：2004-03-30

申请人： Jordi Blasco ,  Carsten Blettner ,  Bernd Müller ,  Markus Gewehr ,  Wassilios Grammenos ,  Thomas Grote ,  Andreas Gypser ,  Joachim Rheinheimer ,  Peter Schäfer ,  Frank Schieweck ,  Anja Schwögler ,  Maria Scherer ,  Siegfried Strathmann ,  Ulrich Schöfl ,  Reinhard Stierl

发明人： Jordi Blasco ,  Carsten Blettner ,  Bernd Müller ,  Markus Gewehr ,  Wassilios Grammenos ,  Thomas Grote ,  Andreas Gypser ,  Joachim Rheinheimer ,  Peter Schäfer ,  Frank Schieweck ,  Anja Schwögler ,  Maria Scherer ,  Siegfried Strathmann ,  Ulrich Schöfl ,  Reinhard Stierl

IPC分类号： A61K31/519 ,  C07D487/04 ,  A01N43/90

CPC分类号： C07D487/04 ,  A01N43/90

摘要： 7-alkinylamino-triazolopyrimidins of formula (I), wherein the substituents have the following meanings: L=halogen, alkyl, halogenalkyl, alkoxy, amino, NHR, NR2, cyano, S(O)nA1 or C(O)A2; R=alkyl or alkylcarbonyl, A1=hydrogen, hydroxy, alkyl, alkylamino or aialkylamino; n=0, 1 or 2; A2=alkenyl, alkoxy, halogenalkoxy or one of the groups cited in A1; m=1, 2, 3, 4 or 5, whereby at least one group L is present in an ortho-position to the bond with the triazolopyrimidine skeleton; X=halogen, cyano, alkyl, halogenalkyl or alkoxy; R1=hydrogen or alkyl; R2=alkinyl which can be unsubstituted or substituted according to the description. The invention also relates to methods for the production of said compounds, agents containing said compounds and the use thereof to combat harmful phytopathogenic fungi.

摘要翻译： 式（I）的7-烷基氨基 - 三唑并嘧啶类，其中取代基具有以下含义：L =卤素，烷基，卤代烷基，烷氧基，氨基，NHR，NR 2，氰基，S（O） 或者C（O）A 2 O 2。 R =烷基或烷基羰基，A 1〜H 2，羟基，烷基，烷基氨基或亚烷基氨基; n = 0,1或2; 链烯基，烷氧基，卤代烷氧基或A 1中引用的基团之一; m = 1,2,3,4或5，其中至少一个基团L存在于与三唑并嘧啶骨架的键的邻位; X =卤素，氰基，烷基，卤代烷基或烷氧基; R 1 =氢或烷基; R 2 =炔基，其可以是未取代的或根据描述取代的。 本发明还涉及生产所述化合物的方法，含有所述化合物的试剂及其用于对抗有害植物病原真菌的用途。

公开(公告)号：US06696607B2

公开(公告)日：2004-02-24

申请号：US10297287

申请日：2002-12-04

申请人： Wassilios Grammenos ,  Hubert Sauter ,  Oliver Cullmann ,  Markus Gewehr ,  Bernd Müller ,  Jordi Tormo i Blasco ,  Norbert Götz ,  Thorsten Volk ,  Gisela Lorenz ,  Eberhard Ammermann ,  Reinhard Stierl ,  Siegfried Strathmann

发明人： Wassilios Grammenos ,  Hubert Sauter ,  Oliver Cullmann ,  Markus Gewehr ,  Bernd Müller ,  Jordi Tormo i Blasco ,  Norbert Götz ,  Thorsten Volk ,  Gisela Lorenz ,  Eberhard Ammermann ,  Reinhard Stierl ,  Siegfried Strathmann

IPC分类号： C07C23309

CPC分类号： A01N37/36 ,  A01N37/18 ,  A01N37/38 ,  C07C231/02 ,  C07C233/22

摘要： Use of phenethylacrylamides of the formula I: in which the substituents have the following meanings: X is halogen, alkyl, haloalkyl, alkoxy, haloalkoxy and —O—C(Ra,Rb)—C≡C—R6; Ra,Rb and Rc have the meanings given in the description; m,n independently of one another are 1 to 4, it being possible for the radicals X or Y to be different if m or n is greater than 1; Y is halogen, nitro, cyano, alkyl, CF3, alkoxy and phenyl; R1,R2 independently of one another are hydrogen, halogen, alkyl, alkoxy, haloalkoxy and CF3; R3,R4,R5,R6 independently of one another are hydrogen, halogen, alkyl, alkoxy, or R3 and R4 together form a cyclopropyl ring, it being possible for the C—R5— and C—R6 bonds can be in the E- or Z-position relative to each other; for controlling phytopathogenic fungal pests, novel phenethylacrylamides, their preparation, and compositions comprising them.

摘要翻译： 使用式I的苯乙基丙烯酰胺：其中取代基具有以下含义：X是卤素，烷基，卤代烷基，烷氧基，卤代烷氧基和-OC（R a，R b）-C = CR 6; R a，R b和R c具有说明书中给出的含义; m，n彼此独立地为1至4，如果m或n可以使基团X或Y不同 大于1; Y是卤素，硝基，氰基，烷基，CF 3，烷氧基和苯基; R 1，R 2彼此独立地是氢，卤素，烷基，烷氧基，卤代烷氧基和CF 3; R 3 R 4，R 5，R 6彼此独立地是氢，卤素，烷基，烷氧基或R 3和R 4一起形成环丙基环，其中CR <5> - 和CR 6键可以相对于彼此位于E-或Z-位;用于控制植物病原性真菌害虫，新型苯乙基丙烯酰胺，它们的制备和包含它们的组合物。

公开(公告)号：US20100286175A1

公开(公告)日：2010-11-11

申请号：US12840392

申请日：2010-07-21

申请人： Wassilios Grammenos ,  Thomas Grote ,  Carsten Blettner ,  Markus Gewehr ,  Udo Hünger ,  Bernd Müller ,  Joachim Rheinheimer ,  Peter Schäfer ,  Frank Schieweck ,  Anja Schwögler ,  Ulrich Schöfl ,  Harald Köhle ,  Siegfried Strathmann ,  Maria Scherer ,  Reinhard Stierl ,  Jan Rether

发明人： Wassilios Grammenos ,  Thomas Grote ,  Carsten Blettner ,  Markus Gewehr ,  Udo Hünger ,  Bernd Müller ,  Joachim Rheinheimer ,  Peter Schäfer ,  Frank Schieweck ,  Anja Schwögler ,  Ulrich Schöfl ,  Harald Köhle ,  Siegfried Strathmann ,  Maria Scherer ,  Reinhard Stierl ,  Jan Rether

IPC分类号： A01N43/54 ,  C07D401/04 ,  A01P3/00

CPC分类号： C07D401/04

摘要： The invention relates to 2-(pyridin-2-yl)-pyrimidine compounds of general formula (I) and their use for controlling pathogenic fungi and as plant protection products that, as an active constituent, contain compounds of this type: In general formula (I), k represents 0, 1, 2, 3; m represents 0, 1, 2, 3, 4 or 5; n represents 1, 2, 3, 4 or 5; R1, independent of one another, represents halogen, OH, CN, NO2, C1-C4 alkyl, C1-C4 alkyl halide, C1-C4 alkoxy, C1-C4 alkoxy halide, C2-C4 alkenyl, C2-C4 alkynyl, C3-C8 cycloalkyl, C1-C4 alkoxy-C1-C4 alkyl, amino, phenoxy, which is optionally substituted by halogen or C1-C4 alkyl, NHR, NR2, C(Ra)═N—ORb, S(═O)pA1 or C(═O)A2, or two radicals R1 bound to adjacent carbon atoms can, together, also represent a group —O-Alk-O—, wherein Alk represents a linear or branched C1-C4 alkylene, and 1, 2, 3 or 4 hydrogen atoms can also be replaced by halogen; R2 represents C1-C4 alkyl halide, C1-C4 alkoxy, C1-C4 alkoxy halide, hydroxy, halogen, CN or NO2; whereby R2 can also represent hydrogen or C1-C4 alkyl when at least one of the three following conditions is fulfilled: n represents 3, 4 or 5; k represents 1, 2 or 3; if m is not equal to 0, at least one of the radicals R1 represents a radical that differs from halogen, C1-C4 alkyl, C1-C4 alkoxy and C1-C4 alkyl halide, and; R3 represents C1-C4 alkyl.

摘要翻译： 本发明涉及通式（I）的2-（吡啶-2-基） - 嘧啶化合物及其用于控制​​致病真菌的用途，作为作为活性成分的植物保护产品含有这种化合物：通式 （I）中，k表示0,1,2,3; m表示0,1,2,3,4或5; n表示1,2,3,4或5; R 1彼此独立地表示卤素，OH，CN，NO 2，C 1 -C 4烷基，C 1 -C 4烷基卤，C 1 -C 4烷氧基，C 1 -C 4烷氧基卤化物，C 2 -C 4烯基，C 2 -C 4炔基， C8环烷基，C1-C4烷氧基-C1-C4烷基，氨基，苯氧基，其任选被卤素或C 1 -C 4烷基取代，NHR，NR 2，C（R a）= N-OR b，S（= O）p A1或C （ΟO）A2或与相邻碳原子结合的两个基团R1一起也可以代表基团-O-Alk-O-，其中Alk表示直链或支链C 1 -C 4亚烷基，和1,2,3或 4个氢原子也可以被卤素取代; R2代表C1-C4烷基卤，C1-C4烷氧基，C1-C4烷氧基卤化物，羟基，卤素，CN或NO2; 其中当满足以下三个条件中的至少一个时，R2还可以表示氢或C1-C4烷基：n表示3,4或5; k表示1,2或3; 如果m不等于0，则基团R1中的至少一个表示与卤素，C 1 -C 4烷基，C 1 -C 4烷氧基和C 1 -C 4烷基卤化物不同的基团， R3表示C1-C4烷基。

公开(公告)号：US07820647B2

公开(公告)日：2010-10-26

申请号：US11596891

申请日：2005-05-17

申请人： Anja Schwögler ,  Frank Schieweck ,  Joachim Rheinheimer ,  Markus Gewehr ,  Bernd Müller ,  Thomas Grote ,  Wassilios Grammenos ,  Udo Hünger ,  Carsten Blettner ,  Peter Schäfer ,  Oliver Wagner ,  Reinhard Stierl ,  Ulrich Schöfl ,  Siegfried Strathmann ,  Maria Scherer

发明人： Anja Schwögler ,  Frank Schieweck ,  Joachim Rheinheimer ,  Markus Gewehr ,  Bernd Müller ,  Thomas Grote ,  Wassilios Grammenos ,  Udo Hünger ,  Carsten Blettner ,  Peter Schäfer ,  Oliver Wagner ,  Reinhard Stierl ,  Ulrich Schöfl ,  Siegfried Strathmann ,  Maria Scherer

IPC分类号： C07D239/48 ,  C07D403/04 ,  A01N43/54 ,  A01N43/58 ,  A01N43/34 ,  A01P3/00

CPC分类号： C07D401/04 ,  C07D403/04

摘要： The invention relates to 2-substituted pyrimidines of the formula I in which the index n and the substituents L and R1 to R3 are as defined in the description and X is a group —CH—Ra, —N—Rb—, —O— or —S—; Ra may be hydrogen, halogen, C1-C6-alkyl, C1-C6-alkoxy, cyano or C1-C6-alkoxycarbonyl; Rb is hydrogen, C1-C6-alkyl or C3-C6-cycloalkyl; T is a group —CH—Ra—; p is an integer from 1 to 4; Y is a group —CH—Ra— or —N—Rb—, o is 0 or 1; Z is O, S or a group N(Rc) Rc is hydrogen, C1-C6-alkyl or C1-C6-alkoxy, and to processes for their preparation, to pesticidal compositions comprising them and to their use as pesticides.

摘要翻译： 本发明涉及式I的2-取代嘧啶，其中指数n和取代基L和R1至R3如说明书中所定义，X为基团-CH-Ra，-N-Rb-，-O- 或-S-; R a可以是氢，卤素，C 1 -C 6 - 烷基，C 1 -C 6 - 烷氧基，氰基或C 1 -C 6 - 烷氧基羰基; R b是氢，C 1 -C 6 - 烷基或C 3 -C 6 - 环烷基; T是基团-CH-R a; p是1至4的整数; Y是基团-CH-R a或-N-R b - ，o是0或1; Z是O，S或基团N（R c）R c是氢，C 1 -C 6烷基或C 1 -C 6 - 烷氧基，并且其制备方法，包含它们的杀虫组合物和它们作为农药的用途。

公开(公告)号：US07786043B2

公开(公告)日：2010-08-31

申请号：US11632342

申请日：2005-07-22

申请人： Wassilios Grammenos ,  Thomas Grote ,  Carsten Blettner ,  Markus Gewehr ,  Udo Hünger ,  Bernd Müller ,  Joachim Rheinheimer ,  Peter Schäfer ,  Frank Schieweck ,  Anja Schwögler ,  Ulrich Schöfl ,  Harald Köhle ,  Siegfried Strathmann ,  Maria Scherer ,  Reinhard Stierl ,  Jan Rether

发明人： Wassilios Grammenos ,  Thomas Grote ,  Carsten Blettner ,  Markus Gewehr ,  Udo Hünger ,  Bernd Müller ,  Joachim Rheinheimer ,  Peter Schäfer ,  Frank Schieweck ,  Anja Schwögler ,  Ulrich Schöfl ,  Harald Köhle ,  Siegfried Strathmann ,  Maria Scherer ,  Reinhard Stierl ,  Jan Rether

IPC分类号： C07D239/74 ,  C07D239/70 ,  C07D401/04 ,  C07D403/04 ,  A01N43/54 ,  C07D213/16 ,  C07D213/84 ,  C07D213/53 ,  C07D213/61 ,  C07D213/26

CPC分类号： C07D401/04

摘要： The invention relates to 2-(pyridin-2-yl)-pyrimidine compounds of general formula (I) and their use for controlling pathogenic fungi and as plant protection products that, as an active constituent, contain compounds of this type: In general formula (I), k represents 0, 1, 2, 3; m represents 0, 1, 2, 3, 4 or 5; n represents 1, 2, 3, 4 or 5; R1, independent of one another, represents halogen, OH, CN, NO2, C1-C4 alkyl, C1-C4 alkyl halide, C1-C4 alkoxy, C1-C4 alkoxy halide, C2-C4 alkenyl, C2-C4 alkynyl, C3-C8 cycloalkyl, C1-C4 alkoxy-C1-C4 alkyl, amino, phenoxy, which is optionally substituted by halogen or C1-C4 alkyl, NHR, NR2, C(Ra)═N—ORb, S(═O)pA1 or C(═O)A2, or two radicals R1 bound to adjacent carbon atoms can, together, also represent a group —O-Alk-O—, wherein Alk represents a linear or branched C1-C4 alkylene, and 1, 2, 3 or 4 hydrogen atoms can also be replaced by halogen; R2 represents C1-C4 alkyl halide, C1-C4 alkoxy, C1-C4 alkoxy halide, hydroxy, halogen, CN or NO2; whereby R2 can also represent hydrogen or C1-C4 alkyl when at least one of the three following conditions is fulfilled: n represents 3, 4 or 5; k represents 1, 2 or 3; if m is not equal to 0, at least one of the radicals R1 represents a radical that differs from halogen, C1-C4 alkyl, C1-C4 alkoxy and C1-C4 alkyl halide, and; R3 represents C1-C4 alkyl.

摘要翻译： 本发明涉及通式（I）的2-（吡啶-2-基） - 嘧啶化合物及其用于控制​​致病真菌的用途，作为作为活性成分的植物保护产品含有这种化合物：通式 （I）中，k表示0,1,2,3; m表示0,1,2,3,4或5; n表示1,2,3,4或5; R 1彼此独立地表示卤素，OH，CN，NO 2，C 1 -C 4烷基，C 1 -C 4烷基卤，C 1 -C 4烷氧基，C 1 -C 4烷氧基卤化物，C 2 -C 4烯基，C 2 -C 4炔基， C8环烷基，C1-C4烷氧基-C1-C4烷基，氨基，苯氧基，其任选被卤素或C 1 -C 4烷基取代，NHR，NR 2，C（R a）= N-OR b，S（= O）p A1或C （ΟO）A2或与相邻碳原子结合的两个基团R1一起也可以代表基团-O-Alk-O-，其中Alk表示直链或支链C 1 -C 4亚烷基，和1,2,3或 4个氢原子也可以被卤素取代; R2代表C1-C4烷基卤，C1-C4烷氧基，C1-C4烷氧基卤化物，羟基，卤素，CN或NO2; 其中当满足以下三个条件中的至少一个时，R2还可以表示氢或C1-C4烷基：n表示3,4或5; k表示1,2或3; 如果m不等于0，则基团R1中的至少一个表示与卤素，C 1 -C 4烷基，C 1 -C 4烷氧基和C 1 -C 4烷基卤化物不同的基团， R3表示C1-C4烷基。

公开(公告)号：US08008232B2

公开(公告)日：2011-08-30

申请号：US11883957

申请日：2006-02-15

申请人： Markus Gewehr ,  Jochen Dietz ,  Thomas Grote ,  Carsten Blettner ,  Wassilios Grammenos ,  Udo Hünger ,  Bernd Müller ,  Frank Schieweck ,  Anja Schwögler ,  Jan Klaas Lohmann ,  Joachim Rheinheimer ,  Peter Schäfer ,  Siegfried Strathmann ,  Reinhard Stierl

发明人： Markus Gewehr ,  Jochen Dietz ,  Thomas Grote ,  Carsten Blettner ,  Wassilios Grammenos ,  Udo Hünger ,  Bernd Müller ,  Frank Schieweck ,  Anja Schwögler ,  Jan Klaas Lohmann ,  Joachim Rheinheimer ,  Peter Schäfer ,  Siegfried Strathmann ,  Reinhard Stierl

IPC分类号： A01N43/56 ,  C07D231/10

CPC分类号： C07D231/14 ,  A01N43/56

摘要： The present invention relates to pyrazolecarboxanilides I in which the variables are as defined below: n is zero or 2; m is 2 or 3; X1 is fluorine or chlorine; X2 is halogen; Y is CN, NO2, C1-C4-alkyl, C1-C4-haloalkyl, methoxy or methylthio; p is zero or 1; R1 is fluorine, chlorine, bromine, C1-C4-alkyl or C1-C4-haloalkyl; R2 is hydrogen or halogen; R3 is hydrogen, methyl or ethyl; W is O or S; with the proviso that, if a) W=O, R1=methyl and R3 is hydrogen, R2 is not fluorine, or b) W=O, n=0, m=2, p=0, R2 and R3 are hydrogen, R1 is not trifluoromethyl or difluoromethyl, to processes for preparing these compounds, to compositions comprising them and to methods for using them for controlling harmful fungi.

摘要翻译： 本发明涉及吡唑烷酰苯胺I，其中变量如下：n为0或2; m为2或3; X1是氟或氯; X2是卤素; Y是CN，NO 2，C 1 -C 4烷基，C 1 -C 4卤代烷基，甲氧基或甲硫基; p为零或1; R1是氟，氯，溴，C1-C4-烷基或C1-C4卤代烷基; R2是氢或卤素; R3是氢，甲基或乙基; W为O或S; 条件是，如果a）W = O，则R1 =甲基且R3为氢，R2不为氟，或b）W = O，n = 0，m = 2，p = 0，R2和R3为氢， R1不是三氟甲基或二氟甲基，制备这些化合物的方法，包含它们的组合物以及用于控制有害真菌的方法。

公开(公告)号：US07695728B2

公开(公告)日：2010-04-13

申请号：US11630569

申请日：2005-06-18

申请人： Joachim Rheinheimer ,  Frank Schieweck ,  Thomas Grote ,  Carsten Blettner ,  Anja Schwögler ,  Markus Gewehr ,  Wassilios Grammenos ,  Udo Hünger ,  Bernd Müller ,  Peter Schäfer ,  John-Bryan Speakman ,  Maria Scherer ,  Siegfried Strathmann ,  Ulrich Schöfl ,  Reinhard Stierl

发明人： Joachim Rheinheimer ,  Frank Schieweck ,  Thomas Grote ,  Carsten Blettner ,  Anja Schwögler ,  Markus Gewehr ,  Wassilios Grammenos ,  Udo Hünger ,  Bernd Müller ,  Peter Schäfer ,  John-Bryan Speakman ,  Maria Scherer ,  Siegfried Strathmann ,  Ulrich Schöfl ,  Reinhard Stierl

IPC分类号： C07D401/04 ,  C07D213/61 ,  C07D417/04 ,  C07D213/70 ,  C07D213/86 ,  C07D213/78 ,  A01N43/40

CPC分类号： C07D401/04 ,  A01N43/40 ,  A01N43/54 ,  A01N43/56 ,  A01N43/653 ,  A01N43/78 ,  C07D213/61 ,  C07D213/70 ,  C07D213/74 ,  C07D213/78 ,  C07D213/84 ,  C07D213/86 ,  C07D417/04

摘要： The invention relates to 2-substituted pyridines of the formula I in which the index n and the substituents R1 to R4 and L are as defined in the description and in each case one of the two ring members X1, X2 is N, the other is C—H or C-halogen; Y is a group —CH—R1—, —N—R1—, —O— or —S— and is five- or six-membered hetaryl comprising 1 to 3 heteroatoms selected from the group consisting of O, N and S or is phenyl, and to processes for their preparation, intermediates for their preparation, pesticidal compositions and methods for controlling harmful fungi and animal pests using the compounds according to the invention.

摘要翻译： 本发明涉及式I中的2-取代吡啶，其中指数n和取代基R 1至R 4和L如说明书中所定义，并且在每种情况下，两个环成员X1，X2中的一个为N，另一个为 C-H或C-卤素; Y是基团-CH-R 1，-N-R 1，-O-或-S-，是包含1至3个选自O，N和S的杂原子的五元或六元杂芳基，或者是 苯基，及其制备方法，其制备中间体，杀虫组合物和使用本发明化合物控制有害真菌和动物害虫的方法。

公开(公告)号：US06562833B1

公开(公告)日：2003-05-13

申请号：US09701859

申请日：2000-12-05

申请人： Bernd Müller ,  Hubert Sauter ,  Herbert Bayer ,  Oliver Cullmann ,  Markus Gewehr ,  Wassilios Grammenos ,  Andreas Gypser ,  Arne Ptock ,  Norbert Götz ,  Thomas Grote ,  Michael Rack ,  Eberhard Ammermann ,  Gisela Lorenz ,  Siegfried Strathmann ,  John-Bryan Speakman

发明人： Bernd Müller ,  Hubert Sauter ,  Herbert Bayer ,  Oliver Cullmann ,  Markus Gewehr ,  Wassilios Grammenos ,  Andreas Gypser ,  Arne Ptock ,  Norbert Götz ,  Thomas Grote ,  Michael Rack ,  Eberhard Ammermann ,  Gisela Lorenz ,  Siegfried Strathmann ,  John-Bryan Speakman

IPC分类号： C07D23942

CPC分类号： C07D239/42 ,  A01N43/54

摘要： 2-(N-phenylamino)pyrimidines of the formula I, where: R1, R3 independently of one another are cyano, C1-C8-alkyl, C2-C6-alkenyl, C2-C6-alkynyl, where the radicals alkyl, alkenyl and alkynyl may be substituted by cyano, halogen, C1-C4-alkoxy or C1-C4-alkoxycarbonyl, or are C3-C8-cycloalkyl or a group C(═NORx)Ry R2 is halogen, C1-C8-alkyl, C2-C6-alkenyl, C2-C6-alkynyl, where the radicals alkyl, alkenyl and alkynyl may be substituted by cyano, halogen, C1-C4-alkoxy or C1-C4-alkoxycarbonyl, or R1 and R2 together with the two linking carbon atoms form a fused-on partially unsaturated 4- to 8-membered ring which may be up to trisubstituted by identical or different substituents selected from the group consisting of C1-C4-alkyl, halogen and C1-C4-alkoxy-carbonyl, which may contain a carbonyl group and/or, in addition to the multiple bond of the pyrimidine ring, a double bond and/or which may be interrupted by O, S or N—(C1-C4-alkyl); the substituents R4 to R8, Rx, Ry, Ra and Rb are as defined in the description; are used as fungicides.

摘要翻译： 式I的2-（N-苯基氨基）嘧啶，其中：R 1，R 3彼此独立地是氰基，C 1 -C 8 - 烷基，C 2 -C 6 - 烯基，C 2 -C 6 - 炔基，其中基团烷基，烯基和 炔基可以被氰基，卤素，C 1 -C 4 - 烷氧基或C 1 -C 4 - 烷氧基羰基取代，或者是C 3 -C 8 - 环烷基或C（= NOR x）R 1 R 2是卤素，C 1 -C 8烷基，C 2 -C 6 - 烯基，C 2 -C 6 - 炔基，其中基团烷基，烯基和炔基可以被氰基，卤素，C 1 -C 4 - 烷氧基或C 1 -C 4 - 烷氧基羰基取代，或者R 1和R 2与两个连接碳原子一起形成稠合 - 部分不饱和的4-至8-元环，其可以由可以含有羰基的C 1 -C 4 - 烷基，卤素和C 1 -C 4 - 烷氧基 - 羰基的相同或不同取代基取代三取代， /或除了嘧啶环的多重键之外，可以被O，S或N-（C 1 -C 4 - 烷基）中断的双键和/或被中间的取代基取代基R4至R8，Rx，Ry，Ra 和Rb如t所定义 他的描述;被用作杀真菌剂。