Thiochromanoylpyrazolone derivatives
    32.
    发明授权
    Thiochromanoylpyrazolone derivatives 失效
    硫代色酰基吡唑啉酮衍生物

    公开(公告)号:US06352959B1

    公开(公告)日:2002-03-05

    申请号:US09857053

    申请日:2001-05-31

    IPC分类号: A01N4384

    CPC分类号: C07D409/06 C07D409/14

    摘要: Thiochromanoylpyrazolone derivatives of the formula I where: A is an unsubstituted or substituted, saturated or unsaturated alkyl chain; R1 is cyano, thiocyanato, nitro, OR4, SR5, SOR6, S02R6, ONR6NR7, ON═CR6R8, NR9R10, P(O)R11R12, P(S)R11R12, COR, CO2R6, unsubstituted or substituted phenyl or heterocyclyl; R2 is alkyl, haloalkyl, alkoxy or haloalkoxy; R3 is hydrogen, alkyl or halogen; X is oxygen, sulfur, S═O, S(═O)2, CR13R14, C═O or C═NR15; m is 0, 1 or 2; n is 0, 1, 2, 3 or 4; R16 is substituted pyrazol-4-yl-carbonyl or substituted (4,5-dihydro-5-oxo-pyrazol-4-yl)methylidene; and their agriculturally useful salts; Processes for preparing the thiochromanoylpyrazolone derivatives, compositions comprising them, and the use of these derivatives or of the compositions comprising them for controlling undesirable plants are described.

    摘要翻译: 其中:A为未取代或取代的饱和或不饱和烷基链; R1为氰基,氰硫基,硝基,OR4,SR5,SOR6,SO2R6,ONR6NR7,ON = CR6R8,NR9R10,P(O)R11R12, P(S)R 11 R 12,COR,CO 2 R 6,未取代或取代的苯基或杂环基; R 2是烷基,卤代烷基,烷氧基或卤代烷氧基; R 3是氢,烷基或卤素; X是氧,硫,S = O,S(= O) 2,CR 13 R 14,C = O或C = NR 15; m为0,1或2; n为0,1,2,3或4; R 16为取代的吡唑-4-基 - 羰基或取代的(4,5-二氢 描述了制备硫代色满酰基吡唑啉酮衍生物的方法,包含它们的组合物,以及这些衍生物或包含它们的组合物用于防治不期望的植物的用途。

    TRICYCLIC BENZOYLPYRAZOLE DERIVATIVES
    33.
    发明申请
    TRICYCLIC BENZOYLPYRAZOLE DERIVATIVES 审中-公开
    三苯甲酰基吡唑衍生物

    公开(公告)号:US20070197393A1

    公开(公告)日:2007-08-23

    申请号:US11461491

    申请日:2006-08-01

    摘要: Tricyclic benzoylpyrazole derivatives of the formula I where: X is oxygen, sulfur, S═O, S(═O)2, CR6R7, NR8 or a bond; Y together with the two carbons to which it is attached forms a saturated, partially saturated or unsaturated 5- or 6-membered heterocycle; R1, R2, R6, R7 are hydrogen, alkyl, haloalkyl, alkoxy or haloalkoxy; R3 is halogen, alkyl, haloalkyl, alkoxy or haloalkoxy; R4 is hydrogen, nitro, halogen, cyano, alkyl, haloalkyl, alkoxy, haloalkoxy, alkylthio, haloalkylthio, alkylsulfinyl, haloalkylsulfinyl, alkylsulfonyl, haloalkylsulfonyl, unsubstituted or substituted aminosulfonyl or unsubstituted or substituted sulfonylamino; R5 is hydrogen, alkyl or halogen; l is 0, 1 or 2; R8 is hydrogen, alkyl, haloalkyl, alkylcarbonyl, formyl, alkoxycarbonyl, haloalkoxycarbonyl, alkylsulfonyl or haloalkylsulfonyl; R9 is substituted pyrazol-4-ylcarbonyl or substituted 5-oxopyrazolin-4-ylmethylidene; and their agriculturally useful salts; processes and intermediates for preparing the tricyclic benzoylpyrazole derivatives; compositions comprising them and the use of these derivatives or of the compositions comprising them for controlling undesirable plants are described.

    摘要翻译: 式I的三环苯甲酰基吡唑衍生物其中:X是氧,硫,SO,S(-O)2,CR 6,R 7, NR 8或键; Y与连接的两个碳一起形成饱和的,部分饱和的或不饱和的5-或6-元杂环; R 1,R 2,R 6,R 7是氢,烷​​基,卤代烷基,烷氧基或卤代烷氧基; R 3是卤素,烷基,卤代烷基,烷氧基或卤代烷氧基; R 4是氢,硝基,卤素,氰基,烷基,卤代烷基,烷氧基,卤代烷氧基,烷硫基,卤代烷硫基,烷基亚磺酰基,卤代烷基亚磺酰基,烷基磺酰基,卤代烷基磺酰基,未取代或取代的氨基磺酰基或未取代或取代的磺酰基氨基; R 5是氢,烷基或卤素; l为0,1或2; R 8是氢,烷基,卤代烷基,烷基羰基,甲酰基,烷氧基羰基,卤代烷氧基羰基,烷基磺酰基或卤代烷基磺酰基; R 9是取代的吡唑-4-基羰基或取代的5-氧代吡唑啉-4-基亚甲基; 及其农业用盐; 制备三环苯甲酰基吡唑衍生物的方法和中间体; 描述了包含它们的组合物以及这些衍生物或包含它们的组合物用于防治不期望的植物的用途。