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公开(公告)号:US09545106B2
公开(公告)日:2017-01-17
申请号:US14118573
申请日:2012-05-30
申请人: Jerome Yves Cassayre , Peter Renold , Myriem El Qacemi , Thomas Pitterna , Julie Clementine Toueg
发明人: Jerome Yves Cassayre , Peter Renold , Myriem El Qacemi , Thomas Pitterna , Julie Clementine Toueg
IPC分类号: C07D413/00 , A01N43/80 , C07D261/02 , C07D327/02 , C07D413/14 , C07D411/12 , C07D413/12
CPC分类号: A01N43/80 , C07D261/02 , C07D327/02 , C07D411/12 , C07D413/12 , C07D413/14
摘要: The present invention provides compounds of formula (I): wherein A1, A2, A3 and A4 are independently of one another C—H, C—R5, or nitrogen; B1—B2—B3—B4 is —CH2—C═N—CH2—, —CH2—N—CH2—CH2—, —CH2—C═CH-0- or —CH═C—CH2-0-; G1 is oxygen or sulfur; L is a single bond or C1-C8alkylene; R1 is hydrogen, C1-C8alkyl, C1-C8alkylcarbonyl-, C1-C8alkoxy, C2-C8alkenyl, C2-C8alkynyl, C1-C8alkoxy-C1-C8alkyl, aryl or aryl substituted by one to three R6, or R1 is heterocyclyl or heterocyclyl substituted by one to three R6 or C1-C8alkoxycarbonyl-; R2 is hydrogen, C1-C8haloalkyl or C1-C8alkyl; R3 is C1-C8haloalkyl; R4 is aryl or aryl substituted by one to three R6, or R4 is heterocyclyl or heterocyclyl substituted by one to three R6; Y1 is CR7R8, C═O or C═S; Y2, Y3 and Y4 are independently CR7R8, C=0, C═S, N—R9, O, S, SO or SO2; wherein at least two adjacent ring atoms in the ring formed by Y1, Y2, Y3 and Y4 are heteroatoms; each R7 and R8 is independently hydrogen, halogen, C1-C8alkyl, or C1-C8haloalkyl; and R5, R6, R7, R8 and R9 are as defined in the claims. The invention also relates to processes and intermediates for preparing these compounds, to insecticidal, acaricidal, nematicidal and molluscicidal compositions comprising these compounds and to methods of using these compounds to control insect, acarine, nematode and mollusc pests.
摘要翻译: 本发明提供式(I)化合物:其中A1,A2,A3和A4彼此独立地为C-H,C-R5或氮; B1-B2-B3-B4是-CH2-C≡N-CH2-,-CH2-N-CH2-CH2-,-CH2-C≡CH-O-或-CH = C-CH2-O-; G1是氧或硫; L是单键或C1-C8亚烷基; R 1是氢,C 1 -C 8烷基,C 1 -C 8烷基羰基 - ,C 1 -C 8烷氧基,C 2 -C 8烯基,C 2 -C 8炔基,C 1 -C 8烷氧基-C 1 -C 8烷基,被1至3个R 6取代的芳基或芳基,或R 1是杂环基或杂环基取代 一至三个R6或C1-C8烷氧基羰基 - ; R2是氢,C1-C8卤代烷基或C1-C8烷基; R3是C1-C8卤代烷基; R4是被一至三个R6取代的芳基或芳基,或R4是被一至三个R6取代的杂环基或杂环基; Y1是CR7R8,C = O或C = S; Y2,Y3和Y4独立地为CR7R8,C = 0,C = S,N-R9,O,S,SO或SO2; 其中由Y1,Y2,Y3和Y4形成的环中至少两个相邻的环原子是杂原子; 每个R 7和R 8独立地是氢,卤素,C 1 -C 8烷基或C 1 -C 8卤代烷基; 且R 5,R 6,R 7,R 8和R 9如权利要求中所定义。 本发明还涉及制备这些化合物的方法和中间体,包含这些化合物的杀虫,杀螨,杀线虫和杀软体动物的组合物,以及使用这些化合物来控制昆虫,螨虫,线虫和软体动物害虫的方法。
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公开(公告)号:US20140235869A1
公开(公告)日:2014-08-21
申请号:US14240541
申请日:2012-08-24
IPC分类号: A01N43/80 , C07D331/04
CPC分类号: C07D413/12 , A01N43/36 , A01N43/80 , C07D331/04 , C07D409/12
摘要: The present invention relates to processes for the preparation of thietane derivatives of the formula (IA) and thietane derivatives of the formula (IB) wherein R1, R2, A1, A2, A3, A4, B, and n are as defined in the claims. The invention also relates to intermediates useful in the processes, as well as the compounds of formula (IA) and (IB) and their use as pesticides.
摘要翻译: 本发明涉及制备式(IA)的硫杂环丁烷衍生物和式(IB)的硫杂环丁烷衍生物的方法,其中R1,R2,A1,A2,A3,A4,B和n如权利要求中所定义 。 本发明还涉及可用于该方法的中间体以及式(IA)和(IB)的化合物及其作为农药的用途。
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公开(公告)号:US08686014B2
公开(公告)日:2014-04-01
申请号:US13062420
申请日:2009-07-24
IPC分类号: A01N43/80 , C07D413/12
CPC分类号: A01N43/80 , C07D413/12
摘要: A compound of Formula (I): where A1, A2, A3, A4, A5, A6, G1, L, R1, R2, R3, R4, Y1, Y2 and Y3 are as defined in claim 1; or a sail or N-oxide thereof. Furthermore, the present invention relates to processes and intermediates for preparing compounds of formula (I), to insecticidal, acaricidal, molluscicidal and nematicidal compositions comprising compounds of formula (I) and to methods of using compounds of formula (I) to combat and control insect, acarine, mollusc and nematode pests.
摘要翻译: 式(I)的化合物:其中A1,A2,A3,A4,A5,A6,G1,L,R1,R2,R3,R4,Y1,Y2和Y3如权利要求1所定义; 或其帆或N-氧化物。 此外,本发明涉及制备式(I)化合物的方法和中间体,其包含式(I)化合物的杀虫,杀螨,杀软体动物和杀线虫组合物,以及使用式(I)化合物来对抗和控制的方法 昆虫,螨虫,软体动物和线虫害虫。
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公开(公告)号:US20120316124A1
公开(公告)日:2012-12-13
申请号:US13579637
申请日:2011-02-17
IPC分类号: C07D261/04 , C07D413/12 , A01N43/84 , C07D417/12 , A01N43/824 , A01P9/00 , A01N43/90 , A01N47/44 , A01P7/04 , A01P7/02 , A01P5/00 , A01N43/80 , C07D473/34
CPC分类号: C07D261/04 , A01N43/80 , C07D413/10 , C07D413/12 , C07D417/12
摘要: The present invention relates to compounds formula (I), wherein P is P1, P2, heterocyclyl or heterocyclyl substituted by one to five Z; and wherein A1, A2, A3, A4, G1, R1, R2, R3, R4, R5, R6, R17, R18, R19 and R20 are as defined in claim 1; or a salt or N-oxide thereof. Furthermore, the present invention relates to processes and intermediates for preparing compounds of formula (I), to insecticidal, acaricidal, nematicidal and molluscicidal compositions comprising the compounds of formula (I) and to methods of using the compounds of formula (I) to control insect, acarine, nematode and mollusc pests.
摘要翻译: 本发明涉及式(I)化合物,其中P为P1,P2,被1至5个Z取代的杂环基或杂环基; 并且其中A1,A2,A3,A4,G1,R1,R2,R3,R4,R5,R6,R17,R18,R19和R20如权利要求1中所定义; 或其盐或N-氧化物。 此外,本发明涉及制备式(I)化合物的方法和中间体,其包含式(I)化合物的杀虫,杀螨,杀线虫和杀软体动物的组合物和使用式(I)化合物控制的方法 昆虫,螨虫,线虫和软体动物害虫。
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公开(公告)号:US08895587B2
公开(公告)日:2014-11-25
申请号:US14118037
申请日:2012-05-15
IPC分类号: C07D307/28 , A01N43/10 , A01N43/36 , A01N43/40 , A01N43/78 , A01N43/80 , C07D207/20 , C07D261/04 , C07D405/12 , C07D407/12 , C07D409/12 , C07D413/04 , C07D413/12 , C07D417/12 , A01N43/08
CPC分类号: C07D307/28 , A01N43/08 , A01N43/10 , A01N43/36 , A01N43/40 , A01N43/78 , A01N43/80 , C07D207/20 , C07D261/04 , C07D405/12 , C07D407/12 , C07D409/12 , C07D413/04 , C07D413/12 , C07D417/12
摘要: The present invention provides compounds of formula (I) wherein R1, R2, R3, R4, G1, n, A1, A2, A3, A4, Y1, Y2, and Y3 are as defined in the claims. The invention also relates to processes and intermediates for preparing these compounds, to insecticidal, acaricidal, nematicidal and molluscicidal compositions comprising these compounds and to methods of using these compounds to control insect, acarine, nematode and mollusc pests.
摘要翻译: 本发明提供式(I)化合物,其中R1,R2,R3,R4,G1,n,A1,A2,A3,A4,Y1,Y2和Y3如权利要求中所定义。 本发明还涉及制备这些化合物的方法和中间体,包含这些化合物的杀虫,杀螨,杀线虫和杀软体动物的组合物,以及使用这些化合物来控制昆虫,螨虫,线虫和软体动物害虫的方法。
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公开(公告)号:US08957058B2
公开(公告)日:2015-02-17
申请号:US13878118
申请日:2011-10-03
IPC分类号: A61K31/43 , C07D207/00 , C07D295/00 , A01N43/78 , C07D207/08 , C07D401/04 , C07D409/10 , C07D409/14 , A01N43/36 , A01N43/40 , A01N43/50 , A01N43/60
CPC分类号: A01N43/78 , A01N43/36 , A01N43/40 , A01N43/50 , A01N43/60 , C07D207/08 , C07D401/04 , C07D409/10 , C07D409/14
摘要: The invention relates to compounds of formula (I): where A1, A2, A3, A4, G1, R1, R2, R3 and R4 are as defined in claim 1; or a salt or N-oxide thereof. Furthermore, the present invention relates to processes and intermediates for preparing compounds of formula (I), to insecticidal, acaricidal, nematicidal and molluscicidal compositions comprising the compounds of formula (I) and to methods of using the compounds of formula (I) to control insect, acarine, nematode and mollusc pests.
摘要翻译: 本发明涉及式(I)化合物:其中A1,A2,A3,A4,G1,R1,R2,R3和R4如权利要求1所定义; 或其盐或N-氧化物。 此外,本发明涉及制备式(I)化合物的方法和中间体,其包含式(I)化合物的杀虫,杀螨,杀线虫和杀软体动物的组合物和使用式(I)化合物控制的方法 昆虫,螨虫,线虫和软体动物害虫。
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公开(公告)号:US20110224079A1
公开(公告)日:2011-09-15
申请号:US13130721
申请日:2009-11-30
申请人: Michel Muehlebach , Thomas Pitterna , Andre Jeanguenat , Myriem El Qacemi , Roger Graham Hall , Andrew Edmunds , Camilla Corsi , Andre Stoller , Christopher Richard Godfrey , Jurgen Harry Schaetzer , Olivier Loiseleur , Peter Maienfisch , Jerome Yves Cassayre
发明人: Michel Muehlebach , Thomas Pitterna , Andre Jeanguenat , Myriem El Qacemi , Roger Graham Hall , Andrew Edmunds , Camilla Corsi , Andre Stoller , Christopher Richard Godfrey , Jurgen Harry Schaetzer , Olivier Loiseleur , Peter Maienfisch , Jerome Yves Cassayre
IPC分类号: A01N25/32 , A01N43/40 , C07D471/10 , C07D211/98 , C07D405/12 , C07D211/56 , C07D409/12 , C07D401/12 , A01P3/00 , A01P13/00 , A01P15/00 , A01P21/00
CPC分类号: C07D471/10 , A01N43/90 , A01N47/06 , C07D211/94
摘要: Novel compounds of the formula (I), wherein the substituents are as defined in claim 1; compositions containing them and their use as insecticides, acaricides, nematicides or molluscicides.
摘要翻译: 新的式(I)化合物,其中取代基如权利要求1所定义; 含有它们的组合物及其作为杀虫剂,杀螨剂,杀线虫剂或杀软体动物剂的用途。
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公开(公告)号:US20140107161A1
公开(公告)日:2014-04-17
申请号:US14118037
申请日:2012-05-12
IPC分类号: C07D307/28 , A01N43/80 , C07D207/20 , A01N43/36 , C07D413/04 , C07D413/12 , C07D417/12 , A01N43/78 , A01N43/08 , C07D407/12 , C07D409/12 , A01N43/10 , C07D405/12 , A01N43/40 , C07D261/04
CPC分类号: C07D307/28 , A01N43/08 , A01N43/10 , A01N43/36 , A01N43/40 , A01N43/78 , A01N43/80 , C07D207/20 , C07D261/04 , C07D405/12 , C07D407/12 , C07D409/12 , C07D413/04 , C07D413/12 , C07D417/12
摘要: The present invention provides compounds of formula (I) wherein R1, R2, R2, R3, R4, G1, n, A1, A2, A3, A4, Y1, Y2, and Y3 are as defined in the claims. The invention also relates to processes and intermediates for preparing these compounds, to insecticidal, acaricidal, nematicidal and molluscicidal compositions comprising these compounds and to methods of using these compounds to control insect, acarine, nematode and mollusc pests.
摘要翻译: 本发明提供式(I)化合物,其中R1,R2,R2,R3,R4,G1,n,A1,A2,A3,A4,Y1,Y2和Y3如权利要求中所定义。 本发明还涉及制备这些化合物的方法和中间体,包含这些化合物的杀虫,杀螨,杀线虫和杀软体动物的组合物,以及使用这些化合物来控制昆虫,螨虫,线虫和软体动物害虫的方法。
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公开(公告)号:US09067892B2
公开(公告)日:2015-06-30
申请号:US13133754
申请日:2009-12-09
申请人: Michel Muehlebach , Thomas Pitterna , Jerome Yves Cassayre , Andrew Edmunds , Camilla Corsi , Myriem El Qacemi , Roger Graham Hall , Andre Jeanguenat , Andre Stoller , Christopher Richard Godfrey , Jurgen Harry Schaetzer , Olivier Loiseleur , Peter Maienfisch , Neil Brian Carter
发明人: Michel Muehlebach , Thomas Pitterna , Jerome Yves Cassayre , Andrew Edmunds , Camilla Corsi , Myriem El Qacemi , Roger Graham Hall , Andre Jeanguenat , Andre Stoller , Christopher Richard Godfrey , Jurgen Harry Schaetzer , Olivier Loiseleur , Peter Maienfisch , Neil Brian Carter
IPC分类号: A01N25/32 , C07D211/32 , A01N43/40 , C07D211/94 , A01N43/90 , C07D471/10
CPC分类号: C07D471/10 , A01N43/90 , A01N47/06 , C07D211/94 , C07D405/12
摘要: A compound of the formula (I), wherein the substituents are as defined in claim 1, are useful as a pesticides.
摘要翻译: 式(I)的化合物,其中取代基如权利要求1中所定义,可用作农药。
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公开(公告)号:US09867375B2
公开(公告)日:2018-01-16
申请号:US14418213
申请日:2012-07-31
IPC分类号: A01N43/653 , A01N43/56 , A01N43/80 , A01N53/00 , A01N43/08 , A01N43/36 , C07D207/09 , C07D207/20 , C07D261/04 , C07D403/10 , G06Q30/00
CPC分类号: A01N53/00 , A01N43/08 , A01N43/36 , A01N43/56 , A01N43/653 , A01N43/80 , C07D207/09 , C07D207/20 , C07D261/04 , C07D403/10 , G06Q30/018
摘要: The present invention provides methods comprising applying to a crop of soybean plants, the locus thereof, or propagation material thereof, a compound of formula (I) wherein —B1—B2—B3— is —C═N—O—, —C═N—CH2—, —N—CH2—CH2—, or —C═C—O—; R1 is trifluoromethyl, difluoromethyl or chlorodifluoromethyl; R2 is group (X) wherein X2 is C—X6 or nitrogen; X1, X3 and X6 are independently hydrogen, halogen or trihalomethyl, wherein at least one of X1, X3 and X6 is not hydrogen; A is selected from group (A1) to (A4) and Y1, Y2, Y3, R5 and R8 are as defined in claim 1. The methods are preferably for the control of stinkbugs, in particular Euschistus.
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