公开(公告)号：US20070197556A1

公开(公告)日：2007-08-23

申请号：US11579048

申请日：2005-05-11

申请人： Jordi Tormo i Blasco ,  Thomas Grote ,  Maria Scherer ,  Reinhard Stierl ,  Siegfried Strathmann ,  Ulrich Schofl ,  Markus Gewehr

发明人： Jordi Tormo i Blasco ,  Thomas Grote ,  Maria Scherer ,  Reinhard Stierl ,  Siegfried Strathmann ,  Ulrich Schofl ,  Markus Gewehr

IPC分类号： A01N43/76 ,  A01N43/64 ,  A01N43/26 ,  A01N43/90 ,  A01N43/78 ,  A01N43/50

CPC分类号： A01N43/90 ,  A01N43/78 ,  A01N43/56 ,  A01N43/32 ,  A01N43/08 ,  A01N2300/00

摘要： Fungicidal mixtures, comprising, as active components, 1) the triazolopyrimidine derivative of the formula I and 2) at least one biphenylamide of the formula II in which the variables are as defined below: A is oxathiinyl or 5-membered heteroaryl which contains one to four nitrogen atoms or one to three nitrogen atoms and/or one sulfur or oxygen atom, where A may be substituted according to the description; R1 is hydrogen, alkyl, alkylcarbonyl or a group A which is attached via carbonyl; Ra, Rb are halogen, cyano, alkyl, haloalkyl, alkoxycarbonyl, alkoxy, haloalkoxy, alkylthio, alkylcarbonyl, formyl, alkylene or alkenylene which links two adjacent carbon atoms; m is 0, 1, 2, 3, 4 or 5; n is 0, 1 or 2; in a synergistically effective amount, methods for controlling harmful fungi using mixtures of the compound I with compound II and the use of the compound I with compounds II for preparing such mixtures, and also compositions comprising these mixtures.

摘要翻译： 包含作为活性成分的杀真菌混合物，1）式I的三唑并嘧啶衍生物和2）至少一种式II的联苯酰胺，其中变量如下所定义：A是氧亚硫代基或5元杂芳基，其含有1至 四个氮原子或一至三个氮原子和/或一个硫或氧原子，其中A可以根据描述被取代; R 1是氢，烷基，烷基羰基或通过羰基连接的基团A; R 2是卤素，氰基，烷基，卤代烷基，烷氧基羰基，烷氧基，卤代烷氧基，烷硫基，烷基羰基，甲酰基，亚烷基或亚链烯基，其连接两个相邻的碳原子; m为0,1,2,3,4或5; n为0,1或2; 在协同有效量的情况下，使用化合物I与化合物II的混合物控制有害真菌的方法以及化合物I与化合物II用于制备此类混合物的用途，以及包含这些混合物的组合物。

公开(公告)号：US20070105928A1

公开(公告)日：2007-05-10

申请号：US10582938

申请日：2004-12-14

申请人： Jordi Tormo I Blasco ,  Carsten Blettner ,  Bernd Muller ,  Markus Gewehr ,  Wassilios Grammenos ,  Thomas Grote ,  Joachim Rheinheimer ,  Peter Schafer ,  Frank Schieweck ,  Anja Schwogler ,  Oliver Wagner ,  Maria Scherer ,  Siegfried Strathmann ,  Ulrich Schofl ,  Reinhard Stierl

发明人： Jordi Tormo I Blasco ,  Carsten Blettner ,  Bernd Muller ,  Markus Gewehr ,  Wassilios Grammenos ,  Thomas Grote ,  Joachim Rheinheimer ,  Peter Schafer ,  Frank Schieweck ,  Anja Schwogler ,  Oliver Wagner ,  Maria Scherer ,  Siegfried Strathmann ,  Ulrich Schofl ,  Reinhard Stierl

IPC分类号： A61K31/41

CPC分类号： F02B43/04 ,  F02B19/14 ,  F02B43/10 ,  F02M25/10 ,  Y02T10/121 ,  Y02T10/125 ,  Y02T10/32

摘要： 6-Pentafluorophenyltriazolopyrimidines of the formula I in which the substituents are as defined below: R1 is alkyl, haloalkyl, cycloalkyl, halocycloalkyl, alkenyl, haloalkenyl, cycloalkenyl, halocycloalkenyl, alkinyl, haloalkinyl or phenyl, naphthyl, or a five- or six-membered saturated, partially unsaturated or aromatic heterocycle which contains one to four heteroatoms from the group consisting of O, N and S, R2 is hydrogen or one of the groups mentioned under R1, R1 and R2 together with the nitrogen atom to which they are attached may also form a five- or six-membered heterocyclyl or heteroaryl which is attached via N and may contain one to three further heteroatoms from the group consisting of O, N and S as ring members; R1 and/or R2 may be substituted as defined in the description; X is cyano, alkyl, alkoxy, alkenyloxy, haloalkoxy or haloalkenyloxy, processes for preparing these compounds, compositions comprising them and their use for controlling phytopathogenic harmful fungi.

摘要翻译： 式I的6-五氟苯基三唑并嘧啶，其中取代基如下：R 1是烷基，卤代烷基，环烷基，卤代环烷基，烯基，卤代烯基，环烯基，卤代环烯基，炔基，卤代炔基或苯基，萘基， 或五元或六元饱和，部分不饱和或芳族杂环，其含有一至四个由O，N和S组成的组的杂原子，R 2是氢或下述基团之一 R 1，R 1和R 2与它们所连接的氮原子一起也可以形成五元或六元杂环基 或杂芳基，其通过N连接并且可以含有一个至三个由O，N和S组成的组的另外的杂原子作为环成员; R 1和/或R 2可以如说明书中所定义的取代; X是氰基，烷基，烷氧基，烯氧基，卤代烷氧基或卤代烯氧基，制备这些化合物的方法，包含它们的组合物及其用于控制​​植物病原性有害真菌的用途。

公开(公告)号：US20070078149A1

公开(公告)日：2007-04-05

申请号：US10580416

申请日：2004-12-16

申请人： Jordi Tormo I Blasco ,  Carsten Blettner ,  Bernd Muller ,  Markus Gewehr ,  Wassilios Grammenos ,  Thomas Grote ,  Joachim Rheinheimer ,  Peter Schafer ,  Frank Schieweck ,  Anja Schwogler ,  Oliver Wagner ,  Maria Scherer ,  Siegfried Strathmann ,  Ulrich Schofl ,  Reinhard Stierl

发明人： Jordi Tormo I Blasco ,  Carsten Blettner ,  Bernd Muller ,  Markus Gewehr ,  Wassilios Grammenos ,  Thomas Grote ,  Joachim Rheinheimer ,  Peter Schafer ,  Frank Schieweck ,  Anja Schwogler ,  Oliver Wagner ,  Maria Scherer ,  Siegfried Strathmann ,  Ulrich Schofl ,  Reinhard Stierl

IPC分类号： A01N43/90 ,  C07D487/04

CPC分类号： C07D487/04 ,  A01N43/90

摘要： Triazolopyrimidines of the formula I in which the substituents are as defined below: R1, R2 are hydrogen, alkyl, haloalkyl, cycloalkyl, halocycloalkyl, alkenyl, haloalkenyl, cycloalkenyl, halocycloalkenyl, alkynyl, haloalkynyl or phenyl, naphthyl, or a five- or six-membered saturated, partially unsaturated or aromatic heterocycle which contains one to four heteroatoms from the group consisting of O, N and S, R1 and R2 together with the nitrogen atom to which they are attached may also form a five- or six-membered heterocyclyl or heteroaryl which is attached via N and may contain a further heteroatom from the group consisting of O, N and S as ring member and may be substituted as defined in the description; L1, L2 are hydrogen, cyano, haloalkyl, alkoxy, alkenyloxy or C(═O)A, where at least one group L1 or L2 is not hydrogen; A is hydrogen, hydroxyl, alkyl, alkoxy, haloalkoxy, C1-C8-alkylamino or dialkylamino; L3 is hydrogen, halogen, cyano, nitro, haloalkyl, alkoxy or alkoxycarbonyl; X is halogen, cyano, alkyl, haloalkyl, alkoxy or haloalkoxy; processes and intermediates for preparing these compounds, compositions comprising them and their use for controlling phytopathogenic harmful fungi.

摘要翻译： 其中取代基如下定义的式I的三唑并嘧啶：R 1，R 2是氢，烷基，卤代烷基，环烷基，卤代环烷基，烯基，卤代烯基，环烯基， 卤代环烯基，炔基，卤代炔基或苯基，萘基或五或六元饱和的部分不饱和或芳族杂环，其含有一至四个由O，N和S组成的组的杂原子，R 1 和R 2与它们所连接的氮原子一起也可以形成五元或六元杂环基或杂芳基，其通过N连接并且可以含有来自以下的另外的杂原子： O，N和S作为环成员，并且可以如说明书中所定义的取代; L 1，L 2是氢，氰基，卤代烷基，烷氧基，烯氧基或C（-O）A，其中至少一个基团L 1 >或L 2不是氢; A是氢，羟基，烷基，烷氧基，卤代烷氧基，C 1 -C 8烷基氨基或二烷基氨基; L 3是氢，卤素，氰基，硝基，卤代烷基，烷氧基或烷氧基羰基; X是卤素，氰基，烷基，卤代烷基，烷氧基或卤代烷氧基; 制备这些化合物的方法和中间体，包含它们的组合物及其用于控制​​植物病原性有害真菌的用途。

公开(公告)号：US20070054929A1

公开(公告)日：2007-03-08

申请号：US10555894

申请日：2004-05-10

申请人： Jordi Tormo i Blasco ,  Carsten Blettner ,  Bernd Muller ,  Markus Gewehr ,  Wassilios Grammenos ,  Thomas Grote ,  Andreas Gypser ,  Joachim Rheinheimer ,  Peter Schafer ,  Frank Schieweck ,  Anja Schwogler ,  Oliver Wagner ,  Siegfried Strathmann ,  Ulrich Schofl ,  Maria Scherer ,  Reinhard Stierl

发明人： Jordi Tormo i Blasco ,  Carsten Blettner ,  Bernd Muller ,  Markus Gewehr ,  Wassilios Grammenos ,  Thomas Grote ,  Andreas Gypser ,  Joachim Rheinheimer ,  Peter Schafer ,  Frank Schieweck ,  Anja Schwogler ,  Oliver Wagner ,  Siegfried Strathmann ,  Ulrich Schofl ,  Maria Scherer ,  Reinhard Stierl

IPC分类号： A61K31/506 ,  C07D403/04

CPC分类号： C07D239/48 ,  A01N43/56 ,  C07D403/04

摘要： The present invention relates to pyrimidines of the formula I in which the index n and the substituents L, R1-R3 are as defined in the description and R4 corresponds to one of the formulae and to processes and intermediates for preparing these compounds, to compositions comprising them and to their use for controlling phytopathogenic harmful fungi.

摘要翻译： 本发明涉及式I的嘧啶，其中指数n和取代基L，R 1〜R 3如说明书中所定义， 4对应于一个公式，以及制备这些化合物的方法和中间体，包含它们的组合物及其用于控制​​植物病原性有害真菌的用途。

公开(公告)号：US20070004759A1

公开(公告)日：2007-01-04

申请号：US10573988

申请日：2004-10-02

申请人： Jordi Tormo i Blasco ,  Thomas Grote ,  Maria Scherer ,  Reinhard Stierl ,  Siegfried Strathmann ,  Ulrich Schofl

发明人： Jordi Tormo i Blasco ,  Thomas Grote ,  Maria Scherer ,  Reinhard Stierl ,  Siegfried Strathmann ,  Ulrich Schofl

IPC分类号： A01N43/90 ,  A01N37/18

CPC分类号： A01N43/90 ,  A01N37/22 ,  A01N2300/00

摘要： The invention relates to fungicidal mixtures for combating rice pathogens containing in the form of active agents 1) a triazolopyrimidine derivative of formula (I) and 2) fenhexamid of formula (II) at a synergistically effective quantity and to a method for combating rice pathogens by the compound of formula (1) and the compound of formula (1) mixtures and the use the compound of formula (I) with the compound of formula (II) for producing such mixtures and agents containing said mixtures.

摘要翻译： 本发明涉及用于防治含有活性剂形式的水稻病原体的杀真菌混合物1）式（I）的三氮代嘧啶衍生物和2）协同有效量的式（II）的十六酰胺和通过以下方式对抗水稻病原体的方法： 式（1）化合物和式（1）化合物的混合物，以及将式（I）化合物与式（II）化合物用于制备含有所述混合物的混合物和试剂。

公开(公告)号：US20060264447A1

公开(公告)日：2006-11-23

申请号：US10574083

申请日：2004-10-07

申请人： Jordi Blasco ,  Thomas Grote ,  Maria Scherer ,  Reinhard Stierl ,  Siegfried Strathmann ,  Ulrich Schofl

发明人： Jordi Blasco ,  Thomas Grote ,  Maria Scherer ,  Reinhard Stierl ,  Siegfried Strathmann ,  Ulrich Schofl

IPC分类号： A01N43/90 ,  A01N43/40

CPC分类号： A01N43/90 ,  A01N43/40 ,  A01N2300/00

摘要： Fungicidal mixtures for controlling rice pathogens, which mixtures comprise, as active components, 1) the triazolopyrimidine derivative of the formula I, and 2) fluazinam of the formula II, in a synergistically effective amount, methods for controlling rice pathogens using mixtures of the compound I with the compound II, the use of the compound I with the compound II for preparing such mixtures and compositions comprising these mixtures are described.

摘要翻译： 用于控制水稻病原体的杀真菌混合物，其混合物包含作为活性组分的1）式I的三唑并嘧啶衍生物和2）协同有效量的式II的氟啶胺，使用化合物的混合物控制水稻病原体的方法 I与化合物II，描述了化合物I与化合物II用于制备这种混合物的用途和包含这些混合物的组合物。

公开(公告)号：US20060258685A1

公开(公告)日：2006-11-16

申请号：US10558251

申请日：2004-05-27

申请人： Olivier Wagner ,  Thomas Grote ,  Carsten Blettner ,  Markus Gewehr ,  Wassilios Grammenos ,  Andreas Gypser ,  Bernd Muller ,  Joachim Rheinheimer ,  Peter Schafer ,  Frank Schieweck ,  Anja Schwogler ,  Jordi Blasco ,  Alan Akers ,  John-Bryan Speakman ,  Michael Rack ,  Reinhard Stierl ,  Maria Scherer ,  Ulrich Schofl ,  Siegfried Strathmann

发明人： Olivier Wagner ,  Thomas Grote ,  Carsten Blettner ,  Markus Gewehr ,  Wassilios Grammenos ,  Andreas Gypser ,  Bernd Muller ,  Joachim Rheinheimer ,  Peter Schafer ,  Frank Schieweck ,  Anja Schwogler ,  Jordi Blasco ,  Alan Akers ,  John-Bryan Speakman ,  Michael Rack ,  Reinhard Stierl ,  Maria Scherer ,  Ulrich Schofl ,  Siegfried Strathmann

IPC分类号： A61K31/519 ,  C07D487/04

CPC分类号： C07D487/04 ,  A01N43/90

摘要： The invention relates to substituted pyrazolopyrimidines of formula (I) wherein the substituents have the following designations: L represents halogen, alkyl, halogenalkyl, alkenyl, alkoxy, amino, NHR, NR2, cyano, S(═O)nA1 or C(═O)A2, R representing alkyl or alkylcarbonyl, A1 representing hydrogen, hydroxy, alkyl, alkylamino or dialkylamino, n representing 0, 1 or 2, and A2 representing alkenyl, alkoxy, halogenalkoxy or one of the groups cited for A1; m represents 0 or 1 to 5; R1 represents alkyl, halogenalkyl, cycloalkyl, halogencycloalkyl, alkenyl, alkadienyl, halogenalkenyl, cycloalkenyl, alkinyl, halogenalkinyl or cycloalkinyl, phenyl, naphthyl, or a five-membered to ten-membered saturated, partially unsaturated or aromatic heterocycle containing between one and four heteroatoms from the group O, N or S; and R2 represents hydrogen or one of the groups cited for R1. Together with the nitrogen atom to which they are bonded, R1 and R2 can form a five-membered to six-membered ring that can be interrupted by an atom from the groups O, N and S, and R1 and/or R2 can also be substituted according to the description. Furthermore, in formula (I): X represents halogen, cyano, OH, alkyl, alkoxy or halogenalkoxy; Y represents a five-membered to ten-membered saturated, partially unsaturated or aromatic heterocycle according to the description, or a group X or another group according to the description; p represents 1 or 2, the groups Y being potentially different when p=2; and p represents 0, when X is according to the description. The invention also relates to methods and intermediate products for producing said compounds, agents containing the same, and the use thereof for controlling phytopathogenic fungi.

公开(公告)号：US20060128727A1

公开(公告)日：2006-06-15

申请号：US10559461

申请日：2004-06-08

申请人： Jordi Tormo I Blasco ,  Thomas Grote ,  Maria Scherer ,  Reinhard Stierl ,  Siegfried Strathmann ,  Ulrich Schofl

发明人： Jordi Tormo I Blasco ,  Thomas Grote ,  Maria Scherer ,  Reinhard Stierl ,  Siegfried Strathmann ,  Ulrich Schofl

IPC分类号： A01N43/54 ,  A01N43/90

CPC分类号： A01N43/90 ,  A01N43/54 ,  A01N2300/00

摘要： Fungicidal mixtures, comprising, as active components: 1) the triazolopyrimidine derivative of the formula I, 2) a pyrimidineanilide of the formula II, in which R is methyl, cyclopropyl or 1-propynyl, in a synergistically effective amount, methods for controlling harmful fungi from the class of the Oomycetes using mixtures of the compound I with one of the compounds II, and the use of the compound I with one of the compounds II for preparing such mixtures and compositions comprising these mixtures are described.

摘要翻译： 包含作为活性成分的杀真菌混合物：1）式I的三唑并嘧啶衍生物，2）式Ⅱ的嘧啶酰苯胺，其中R是甲基，环丙基或1-丙炔基，协同有效量，用于控制有害的 描述了使用化合物I与化合物II之一的混合物从卵菌纲类中获得的真菌，以及化合物I与化合物II之一用于制备这些混合物和包含这些混合物的组合物的用途。

公开(公告)号：US20080280759A1

公开(公告)日：2008-11-13

申请号：US10582971

申请日：2004-12-14

申请人： Jordi Tormo i Blasco ,  Carsten Blettner ,  Bernd Muller ,  Markus Gewehr ,  Wassilios Grammenos ,  Thomas Grote ,  Joachim Rheinheimer ,  Peter Schafer ,  Frank Schieweck ,  Anja Schwogler ,  Oliver Wagner ,  Maria Scherer ,  Siegfried Strathmann ,  Ulrich Schofl ,  Reinhard Stierl

发明人： Jordi Tormo i Blasco ,  Carsten Blettner ,  Bernd Muller ,  Markus Gewehr ,  Wassilios Grammenos ,  Thomas Grote ,  Joachim Rheinheimer ,  Peter Schafer ,  Frank Schieweck ,  Anja Schwogler ,  Oliver Wagner ,  Maria Scherer ,  Siegfried Strathmann ,  Ulrich Schofl ,  Reinhard Stierl

IPC分类号： A01C1/06 ,  C07D487/04 ,  A61K31/519

CPC分类号： A01N43/90 ,  C07D487/04

摘要： 6-(2-Halo-4-alkoxyphenyl)triazolopyrimidines of the formula I in which the substituents are as defined below: R1 is alkyl, haloalkyl, cycloalkyl, halocycloalkyl, alkenyl, haloalkenyl, cycloalkenyl, halocycloalkenyl, alkynyl, haloalkynyl or phenyl, naphthyl, or a five- or six-membered saturated, partially unsaturated or aromatic heterocycle which contains one to four heteroatoms from the group consisting of O, N and S, R2 is hydrogen or one of the groups mentioned under R1, R1 and R2 together with the nitrogen atom to which they are attached may also form a five- or six-membered heterocyclyl or heteroaryl which is attached via N and may contain one to three further heteroatoms from the group consisting of O, N and S as ring members; R3 is alkyl, haloalkyl, alkenyl, haloalkenyl, alkynyl, haloalkynyl, phenylalkyl, mono- or dialkoxyalkyl; R1, R2 and/or R3 may be substituted as mentioned in the description; L is hydrogen, fluorine or chlorine; X is cyano, alkyl, alkoxy, alkenyloxy, haloalkoxy or haloalkenyloxy; processes for preparing these compounds, compositions comprising them and their use for controlling phytopathogenic harmful fungi.

摘要翻译： 其中取代基如下定义的式I的6-（2-卤代-4-烷氧基苯基）三唑并嘧啶：R 1是烷基，卤代烷基，环烷基，卤代环烷基，烯基，卤代烯基，环烯基，卤代环烯基 ，炔基，卤代炔基或苯基，萘基或五元或六元饱和的部分不饱和或芳族杂环，其含有一至四个由O，N和S组成的组的杂原子，R 2， 是氢或R 1，R 1和R 2所提及的基团之一与它们所连接的氮原子一起也可以 形成通过N连接的五元或六元杂环基或杂芳基，并且可以含有一个至三个由O，N和S组成的组的另外的杂原子作为环成员; R 3是烷基，卤代烷基，烯基，卤代烯基，炔基，卤代炔基，苯基烷基，单或二烷氧基烷基; R 1，R 2和/或R 3可以如说明书中所述被取代; L是氢，氟或氯; X是氰基，烷基，烷氧基，烯氧基，卤代烷氧基或卤代烯氧基; 制备这些化合物的方法，包含它们的组合物及其用于控制​​植物病原性有害真菌的用途。

公开(公告)号：US20080255158A1

公开(公告)日：2008-10-16

申请号：US10590925

申请日：2005-03-14

申请人： Jordi Tormo I Blasco ,  Thomas Grote ,  Maria Scherer ,  Reinhard Stierl ,  Siegfried Strathmann ,  Ulrich Schofl

发明人： Jordi Tormo I Blasco ,  Thomas Grote ,  Maria Scherer ,  Reinhard Stierl ,  Siegfried Strathmann ,  Ulrich Schofl

IPC分类号： A01N43/90 ,  A01P3/00

CPC分类号： A01N47/38 ,  A01N47/34 ,  A01N43/90 ,  A01N2300/00

摘要： The invention relates to fungicidal mixtures containing in the form of active agents: a triazolopyrimidine derivative of formula (I) and thiophanate-methyl of formula (II) in synergistically active quantity and to a method for controlling harmful fungi by means of the mixture of the compounds I and II, thereby making it possible to produce said mixtures and the products containing them.

摘要翻译： 本发明涉及含有活性剂形式的杀真菌混合物：具有协同活性的式（I）三唑并嘧啶衍生物和式（II）的甲基托布津 - 甲基和通过混合物的混合物控制有害真菌的方法 化合物I和II，从而使得可以生产所述混合物和含有它们的产物。