公开(公告)号：US20090036509A1

公开(公告)日：2009-02-05

申请号：US11628324

申请日：2005-06-11

申请人： Markus Gewehr ,  Bernd Muller ,  Thomas Grote ,  Wassilios Grammenos ,  Anja Schwogler ,  Joachim Rheinheimer ,  Carsten Blettner ,  Peter Schafer ,  Frank Schieweck ,  Oliver Wagner ,  Frank Werner ,  Jan Rether ,  Siegfried Strathmann ,  Reinhard Stierl ,  Maria Scherer

发明人： Markus Gewehr ,  Bernd Muller ,  Thomas Grote ,  Wassilios Grammenos ,  Anja Schwogler ,  Joachim Rheinheimer ,  Carsten Blettner ,  Peter Schafer ,  Frank Schieweck ,  Oliver Wagner ,  Frank Werner ,  Jan Rether ,  Siegfried Strathmann ,  Reinhard Stierl ,  Maria Scherer

IPC分类号： A01N43/56 ,  C07D231/14 ,  A01P3/00

CPC分类号： C07D231/14

摘要： The present invention relates to N-(ortho-phenyl)-1-methyl-3-trifluoromethylpyrazole-4-carboxanilides of the formula I in which the substituents are as defined below: R1 and R2 independently of one another are halogen, C1-C6-alkyl, C1-C6-haloalkyl, cyano, nitro, methoxy, trifluoromethoxy or difluoromethoxy; with the proviso that when R2 is chlorine in position 4, R1 is not trifluoromethyl in position 3.

摘要翻译： 本发明涉及式I的N-（邻 - 苯基）-1-甲基-3-三氟甲基吡唑-4-甲酰苯胺，其中取代基如下所定义：R 1和R 2彼此独立地为卤素，C 1 -C 6 烷基，C 1 -C 6卤代烷基，氰基，硝基，甲氧基，三氟甲氧基或二氟甲氧基; 条件是当R2在4位是氯时，R1不在3位是三氟甲基。

公开(公告)号：US20080171774A1

公开(公告)日：2008-07-17

申请号：US11885990

申请日：2006-03-15

申请人： Markus Gewehr ,  Jochen Dietz ,  Thomas Grote ,  Carsten Blettner ,  Wassilios Grammenos ,  Udo Hunger ,  Bernd Muller ,  Frank Schieweck ,  Anja Schwogler ,  Jan Klaas Lohmann ,  Joachim Rheinheimer ,  Peter Schafer ,  Siegfried Strathmann ,  Reinhard Stierl ,  Jan Rether ,  Karl Eicken

发明人： Markus Gewehr ,  Jochen Dietz ,  Thomas Grote ,  Carsten Blettner ,  Wassilios Grammenos ,  Udo Hunger ,  Bernd Muller ,  Frank Schieweck ,  Anja Schwogler ,  Jan Klaas Lohmann ,  Joachim Rheinheimer ,  Peter Schafer ,  Siegfried Strathmann ,  Reinhard Stierl ,  Jan Rether ,  Karl Eicken

IPC分类号： C07D213/63 ,  C07D213/56 ,  A61K31/4415 ,  A61K31/455

CPC分类号： C07D213/82

摘要： The present invention relates to nicotinanilides of the formula I in which: n=0, 1, 2; m=2, 3; X1=F, chlorine; X2=halogen; Y=CN, NO2, C1-C4-alkyl, C1-C4-haloalkyl, methoxy or methylthio; p=0, 1; R1=halogen, methyl, C1-C4-haloalkyl, methoxy, methylthio, methylsulfinyl or methylsulfonyl; R2=hydrogen, methyl or ethyl; W=O, S; processes for preparing these compounds, compositions and seed comprising them and also methods for controlling harmful fungi.

摘要翻译： 本发明涉及式I的烟酰苯胺，其中：n = 0,1,2; m = 2，3; X 1 = F，氯; X 2 =卤素; Y = CN，NO 2，C 1 -C 4 - 烷基，C 1 -C 3 - 4 - 卤代烷基，甲氧基或甲硫基; p = 0,1， R 1 =卤素，甲基，C 1 -C 4 - 卤代烷基，甲氧基，甲硫基，甲基亚磺酰基或甲基磺酰基; R 2 =氢，甲基或乙基; W = O，S; 制备这些化合物的方法，包含它们的组合物和种子以及控制有害真菌的方法。

公开(公告)号：US20080076785A1

公开(公告)日：2008-03-27

申请号：US11663982

申请日：2005-09-27

申请人： Carsten Blettner ,  Jordi Tormo i Blasco ,  Bernd Muller ,  Markus Gewehr ,  Wassilios Grammenos ,  Thomas Grote ,  Udo Hunger ,  Joachim Rheinheimer ,  Peter Schafer ,  Frank Schieweck ,  Anja Schwogler ,  Oliver Wagner ,  John-Bryan Speakman ,  Thorsten Jabs ,  Siegfried Strathmann ,  Ulrich Schofl ,  Maria Scherer ,  Reinhard Stierl

发明人： Carsten Blettner ,  Jordi Tormo i Blasco ,  Bernd Muller ,  Markus Gewehr ,  Wassilios Grammenos ,  Thomas Grote ,  Udo Hunger ,  Joachim Rheinheimer ,  Peter Schafer ,  Frank Schieweck ,  Anja Schwogler ,  Oliver Wagner ,  John-Bryan Speakman ,  Thorsten Jabs ,  Siegfried Strathmann ,  Ulrich Schofl ,  Maria Scherer ,  Reinhard Stierl

IPC分类号： A01N43/54 ,  A01P3/00 ,  C07D239/70

CPC分类号： A01N43/90 ,  C07D487/04

摘要： The invention relates to 7-aminomethyl-1,2,4-triazolo[1,5-a]pyrimidine compounds of general formula (I) and the agriculturally compatible salts of said compounds. In said formula: R1 and R2 represent hydrogen, alkyl, haloalkyl, alkoxy, cycloalkyl, bicycloalkyl, halocycloalkyl, alkenyl, alkadienyl, haloalkenyl, cycloalkenyl, halocycloalkenyl, alkynyl, haloalkynyl or phenyl, naphthyl, or a 5- or 6-membered saturated, partially unsaturated or aromatic heterocycle, containing 1 to 4 heteroatoms from the group containing O, N or S, or R1 and R2, together with the nitrogen atom to which they are bonded, can also form a five- or six-membered heterocyclyl or heteroaryl, which is bonded by means of N and can contain 1 to 3 additional heteroatoms from the group containing O, N and S as the ring member and can be substituted according to the description; R3 and R4 represent hydrogen, alkyl, haloalkyl, haloalkoxy, alkoxy, or alkoxyalkyl; X represents halogen, cyano, a 5- or 6-membered saturated, partially unsaturated or aromatic heterocycle, containing 1, 2 or 3 heteroatoms from the group containing O, N or S as the ring member, alkyl, alkoxy, alkenyl or alkynyl, whereby the latter 4 groups can be substituted according to the description; L is defined as cited in the claims and the description; and m represents 0, 1, 2, 3, 4 or 5. The invention also relates to the use of the triazolopyrimidine compounds of general formula (I) and their agriculturally compatible salts for controlling plant-pathogenic fungi, to a method for controlling plant-pathogenic fungi, containing at least one compound of general formula (I) and/or an agriculturally compatible salt of said compound and at least one liquid or solid carrier.

摘要翻译： 本发明涉及通式（I）的7-氨基甲基-1,2,4-三唑并[1,5-a]嘧啶化合物和所述化合物的农业上相容的盐。 在所述式中：R 1和R 2表示氢，烷基，卤代烷基，烷氧基，环烷基，二环烷基，卤代环烷基，烯基，链烯基，卤代烯基，环烯基，卤代环烯基，炔基，卤代炔基或苯基，萘基或5-或6-元饱和， 部分不饱和或芳族杂环，含有1至4个含有O，N或S的杂原子，或R 1和R 2与它们所键合的氮原子一起也可以形成五元或六元杂环基或杂芳基 ，其通过N键合并且可以含有来自含有O，N和S的基团的1至3个另外的杂原子作为环成员，并且可以根据描述进行取代; R3和R4代表氢，烷基，卤代烷基，卤代烷氧基，烷氧基或烷氧基烷基; X代表卤素，氰基，含有1,2或3个杂原子的5-或6-元饱和的部分不饱和或芳族杂环，所述杂环含有作为环成员的O，N或S，烷基，烷氧基，烯基或炔基， 由此后4个组可以根据描述被替代; L定义为权利要求书和说明书中引用的; 和m表示0,1,2,3,4或5.本发明还涉及通式（I）的三唑并嘧啶化合物及其农业上相容的盐用于控制植物致病真菌的用途，用于控制植物的方法 致病真菌，含有至少一种通式（I）的化合物和/或所述化合物的农业上相容的盐和至少一种液体或固体载体。

公开(公告)号：US20070105928A1

公开(公告)日：2007-05-10

申请号：US10582938

申请日：2004-12-14

申请人： Jordi Tormo I Blasco ,  Carsten Blettner ,  Bernd Muller ,  Markus Gewehr ,  Wassilios Grammenos ,  Thomas Grote ,  Joachim Rheinheimer ,  Peter Schafer ,  Frank Schieweck ,  Anja Schwogler ,  Oliver Wagner ,  Maria Scherer ,  Siegfried Strathmann ,  Ulrich Schofl ,  Reinhard Stierl

发明人： Jordi Tormo I Blasco ,  Carsten Blettner ,  Bernd Muller ,  Markus Gewehr ,  Wassilios Grammenos ,  Thomas Grote ,  Joachim Rheinheimer ,  Peter Schafer ,  Frank Schieweck ,  Anja Schwogler ,  Oliver Wagner ,  Maria Scherer ,  Siegfried Strathmann ,  Ulrich Schofl ,  Reinhard Stierl

IPC分类号： A61K31/41

CPC分类号： F02B43/04 ,  F02B19/14 ,  F02B43/10 ,  F02M25/10 ,  Y02T10/121 ,  Y02T10/125 ,  Y02T10/32

摘要： 6-Pentafluorophenyltriazolopyrimidines of the formula I in which the substituents are as defined below: R1 is alkyl, haloalkyl, cycloalkyl, halocycloalkyl, alkenyl, haloalkenyl, cycloalkenyl, halocycloalkenyl, alkinyl, haloalkinyl or phenyl, naphthyl, or a five- or six-membered saturated, partially unsaturated or aromatic heterocycle which contains one to four heteroatoms from the group consisting of O, N and S, R2 is hydrogen or one of the groups mentioned under R1, R1 and R2 together with the nitrogen atom to which they are attached may also form a five- or six-membered heterocyclyl or heteroaryl which is attached via N and may contain one to three further heteroatoms from the group consisting of O, N and S as ring members; R1 and/or R2 may be substituted as defined in the description; X is cyano, alkyl, alkoxy, alkenyloxy, haloalkoxy or haloalkenyloxy, processes for preparing these compounds, compositions comprising them and their use for controlling phytopathogenic harmful fungi.

摘要翻译： 式I的6-五氟苯基三唑并嘧啶，其中取代基如下：R 1是烷基，卤代烷基，环烷基，卤代环烷基，烯基，卤代烯基，环烯基，卤代环烯基，炔基，卤代炔基或苯基，萘基， 或五元或六元饱和，部分不饱和或芳族杂环，其含有一至四个由O，N和S组成的组的杂原子，R 2是氢或下述基团之一 R 1，R 1和R 2与它们所连接的氮原子一起也可以形成五元或六元杂环基 或杂芳基，其通过N连接并且可以含有一个至三个由O，N和S组成的组的另外的杂原子作为环成员; R 1和/或R 2可以如说明书中所定义的取代; X是氰基，烷基，烷氧基，烯氧基，卤代烷氧基或卤代烯氧基，制备这些化合物的方法，包含它们的组合物及其用于控制​​植物病原性有害真菌的用途。

公开(公告)号：US20070078149A1

公开(公告)日：2007-04-05

申请号：US10580416

申请日：2004-12-16

申请人： Jordi Tormo I Blasco ,  Carsten Blettner ,  Bernd Muller ,  Markus Gewehr ,  Wassilios Grammenos ,  Thomas Grote ,  Joachim Rheinheimer ,  Peter Schafer ,  Frank Schieweck ,  Anja Schwogler ,  Oliver Wagner ,  Maria Scherer ,  Siegfried Strathmann ,  Ulrich Schofl ,  Reinhard Stierl

发明人： Jordi Tormo I Blasco ,  Carsten Blettner ,  Bernd Muller ,  Markus Gewehr ,  Wassilios Grammenos ,  Thomas Grote ,  Joachim Rheinheimer ,  Peter Schafer ,  Frank Schieweck ,  Anja Schwogler ,  Oliver Wagner ,  Maria Scherer ,  Siegfried Strathmann ,  Ulrich Schofl ,  Reinhard Stierl

IPC分类号： A01N43/90 ,  C07D487/04

CPC分类号： C07D487/04 ,  A01N43/90

摘要： Triazolopyrimidines of the formula I in which the substituents are as defined below: R1, R2 are hydrogen, alkyl, haloalkyl, cycloalkyl, halocycloalkyl, alkenyl, haloalkenyl, cycloalkenyl, halocycloalkenyl, alkynyl, haloalkynyl or phenyl, naphthyl, or a five- or six-membered saturated, partially unsaturated or aromatic heterocycle which contains one to four heteroatoms from the group consisting of O, N and S, R1 and R2 together with the nitrogen atom to which they are attached may also form a five- or six-membered heterocyclyl or heteroaryl which is attached via N and may contain a further heteroatom from the group consisting of O, N and S as ring member and may be substituted as defined in the description; L1, L2 are hydrogen, cyano, haloalkyl, alkoxy, alkenyloxy or C(═O)A, where at least one group L1 or L2 is not hydrogen; A is hydrogen, hydroxyl, alkyl, alkoxy, haloalkoxy, C1-C8-alkylamino or dialkylamino; L3 is hydrogen, halogen, cyano, nitro, haloalkyl, alkoxy or alkoxycarbonyl; X is halogen, cyano, alkyl, haloalkyl, alkoxy or haloalkoxy; processes and intermediates for preparing these compounds, compositions comprising them and their use for controlling phytopathogenic harmful fungi.

摘要翻译： 其中取代基如下定义的式I的三唑并嘧啶：R 1，R 2是氢，烷基，卤代烷基，环烷基，卤代环烷基，烯基，卤代烯基，环烯基， 卤代环烯基，炔基，卤代炔基或苯基，萘基或五或六元饱和的部分不饱和或芳族杂环，其含有一至四个由O，N和S组成的组的杂原子，R 1 和R 2与它们所连接的氮原子一起也可以形成五元或六元杂环基或杂芳基，其通过N连接并且可以含有来自以下的另外的杂原子： O，N和S作为环成员，并且可以如说明书中所定义的取代; L 1，L 2是氢，氰基，卤代烷基，烷氧基，烯氧基或C（-O）A，其中至少一个基团L 1 >或L 2不是氢; A是氢，羟基，烷基，烷氧基，卤代烷氧基，C 1 -C 8烷基氨基或二烷基氨基; L 3是氢，卤素，氰基，硝基，卤代烷基，烷氧基或烷氧基羰基; X是卤素，氰基，烷基，卤代烷基，烷氧基或卤代烷氧基; 制备这些化合物的方法和中间体，包含它们的组合物及其用于控制​​植物病原性有害真菌的用途。

公开(公告)号：US20080280759A1

公开(公告)日：2008-11-13

申请号：US10582971

申请日：2004-12-14

申请人： Jordi Tormo i Blasco ,  Carsten Blettner ,  Bernd Muller ,  Markus Gewehr ,  Wassilios Grammenos ,  Thomas Grote ,  Joachim Rheinheimer ,  Peter Schafer ,  Frank Schieweck ,  Anja Schwogler ,  Oliver Wagner ,  Maria Scherer ,  Siegfried Strathmann ,  Ulrich Schofl ,  Reinhard Stierl

发明人： Jordi Tormo i Blasco ,  Carsten Blettner ,  Bernd Muller ,  Markus Gewehr ,  Wassilios Grammenos ,  Thomas Grote ,  Joachim Rheinheimer ,  Peter Schafer ,  Frank Schieweck ,  Anja Schwogler ,  Oliver Wagner ,  Maria Scherer ,  Siegfried Strathmann ,  Ulrich Schofl ,  Reinhard Stierl

IPC分类号： A01C1/06 ,  C07D487/04 ,  A61K31/519

CPC分类号： A01N43/90 ,  C07D487/04

摘要： 6-(2-Halo-4-alkoxyphenyl)triazolopyrimidines of the formula I in which the substituents are as defined below: R1 is alkyl, haloalkyl, cycloalkyl, halocycloalkyl, alkenyl, haloalkenyl, cycloalkenyl, halocycloalkenyl, alkynyl, haloalkynyl or phenyl, naphthyl, or a five- or six-membered saturated, partially unsaturated or aromatic heterocycle which contains one to four heteroatoms from the group consisting of O, N and S, R2 is hydrogen or one of the groups mentioned under R1, R1 and R2 together with the nitrogen atom to which they are attached may also form a five- or six-membered heterocyclyl or heteroaryl which is attached via N and may contain one to three further heteroatoms from the group consisting of O, N and S as ring members; R3 is alkyl, haloalkyl, alkenyl, haloalkenyl, alkynyl, haloalkynyl, phenylalkyl, mono- or dialkoxyalkyl; R1, R2 and/or R3 may be substituted as mentioned in the description; L is hydrogen, fluorine or chlorine; X is cyano, alkyl, alkoxy, alkenyloxy, haloalkoxy or haloalkenyloxy; processes for preparing these compounds, compositions comprising them and their use for controlling phytopathogenic harmful fungi.

摘要翻译： 其中取代基如下定义的式I的6-（2-卤代-4-烷氧基苯基）三唑并嘧啶：R 1是烷基，卤代烷基，环烷基，卤代环烷基，烯基，卤代烯基，环烯基，卤代环烯基 ，炔基，卤代炔基或苯基，萘基或五元或六元饱和的部分不饱和或芳族杂环，其含有一至四个由O，N和S组成的组的杂原子，R 2， 是氢或R 1，R 1和R 2所提及的基团之一与它们所连接的氮原子一起也可以 形成通过N连接的五元或六元杂环基或杂芳基，并且可以含有一个至三个由O，N和S组成的组的另外的杂原子作为环成员; R 3是烷基，卤代烷基，烯基，卤代烯基，炔基，卤代炔基，苯基烷基，单或二烷氧基烷基; R 1，R 2和/或R 3可以如说明书中所述被取代; L是氢，氟或氯; X是氰基，烷基，烷氧基，烯氧基，卤代烷氧基或卤代烯氧基; 制备这些化合物的方法，包含它们的组合物及其用于控制​​植物病原性有害真菌的用途。

公开(公告)号：US20080153707A1

公开(公告)日：2008-06-26

申请号：US11883957

申请日：2006-02-15

申请人： Markus Gewehr ,  Jochen Dietz ,  Thomas Grote ,  Carsten Blettner ,  Wassilios Grammenos ,  Udo Hunger ,  Bernd Muller ,  Frank Schieweck ,  Anja Schwogler ,  Jan Klaas Lohmann ,  Joachim Rheinheimer ,  Peter Schafer ,  Siegfried Strathmann ,  Reinhard Stierl

发明人： Markus Gewehr ,  Jochen Dietz ,  Thomas Grote ,  Carsten Blettner ,  Wassilios Grammenos ,  Udo Hunger ,  Bernd Muller ,  Frank Schieweck ,  Anja Schwogler ,  Jan Klaas Lohmann ,  Joachim Rheinheimer ,  Peter Schafer ,  Siegfried Strathmann ,  Reinhard Stierl

IPC分类号： A01N43/56 ,  C07D231/00 ,  A01N25/26

CPC分类号： C07D231/14 ,  A01N43/56

摘要： The present invention relates to pyrazolecarboxanilides I in which the variables are as defined below: n is zero or 2; m is 2 or 3; X1 is fluorine or chlorine; X2 is halogen; Y is CN, NO2, C1-C4-alkyl, C1-C4-haloalkyl, methoxy or methylthio; p is zero or 1; R1 is fluorine, chlorine, bromine, C1-C4-alkyl or C1-C4-haloalkyl; R2 is hydrogen or halogen; R3 is hydrogen, methyl or ethyl; W is O or S; with the proviso that, if a) W═O, R1=methyl and R3 is hydrogen, R2 is not fluorine, or b) W═O, n=0, m=2, p=0, R2 and R3 are hydrogen, R1 is not trifluoromethyl or difluoromethyl, to processes for preparing these compounds, to compositions comprising them and to methods for using them for controlling harmful fungi.

摘要翻译： 本发明涉及吡唑烷酰苯胺I，其中变量如下：n为0或2; m为2或3; X 1是氟或氯; X 2是卤素; Y是CN，NO 2，C 1 -C 4 - 烷基，C 1 -C 3 - 4 - 卤代烷基，甲氧基或甲硫基; p为零或1; R 1是氟，氯，溴，C 1 -C 4 - C 1-4烷基或C 1 -C 3 - 低级烷基; R 2是氢或卤素; R 3是氢，甲基或乙基; W为O或S; 条件是，如果a）WO，R 1 =甲基和R 3是氢，R 2不是氟，或b） WO，n = 0，m = 2，p = 0，R 2和R 3是氢，R 1不是三氟甲基或二氟甲基 ，制备这些化合物的方法，包含它们的组合物以及用于控制有害真菌的方法。

公开(公告)号：US20080119493A1

公开(公告)日：2008-05-22

申请号：US10590326

申请日：2005-03-08

申请人： Jordi Tormo i Blasco ,  Carsten Blettner ,  Bernd Muller ,  Markus Gewehr ,  Wassilios Grammenos ,  Thomas Grote ,  Joachim Rheinheimer ,  Peter Schafer ,  Frank Schieweck ,  Anja Schwogler ,  Oliver Wagner ,  Matthias Niedenbruck ,  Maria Scherer ,  Siegfried Strathmann ,  Ulrich Schofl ,  Reinhard Stierl ,  Udo Hunger

发明人： Jordi Tormo i Blasco ,  Carsten Blettner ,  Bernd Muller ,  Markus Gewehr ,  Wassilios Grammenos ,  Thomas Grote ,  Joachim Rheinheimer ,  Peter Schafer ,  Frank Schieweck ,  Anja Schwogler ,  Oliver Wagner ,  Matthias Niedenbruck ,  Maria Scherer ,  Siegfried Strathmann ,  Ulrich Schofl ,  Reinhard Stierl ,  Udo Hunger

IPC分类号： A01N43/90 ,  C07D487/04 ,  A01P3/00

CPC分类号： C07D487/04

摘要： The invention relates to 5,6-dialkyl-7-amino-triazolopyrimidines of formula (I), in which the substituents are defined as follows: R1 represents alkyl, alkoxyalkyl, alkenyl or alkynyl; R2 represents alkyl, alkoxyalkyl, alkenyl or alkynyl, R1 and/or R2 being substituted according to the description. The invention also relates to a method for producing said compounds, to agents containing the latter and to their use for controlling plant-pathogenic fungi.

摘要翻译： 本发明涉及式（I）的5,6-二烷基-7-氨基 - 三唑并嘧啶，其中取代基定义如下：R 1表示烷基，烷氧基烷基，烯基或炔基; R 2表示根据描述被取代的烷基，烷氧基烷基，烯基或炔基，R 1和/或R 2 2。 本发明还涉及一种生产所述化合物的方法，含有后者的药剂及其用于控制​​植物致病真菌的用途。

公开(公告)号：US20080039319A1

公开(公告)日：2008-02-14

申请号：US11596464

申请日：2005-05-11

申请人： Carsten Blettner ,  Markus Gewehr ,  Wassilios Grammenos ,  Thomas Grote ,  Udo Hunger ,  Bernd Muller ,  Matthias Niedenbruck ,  Joachim Rheinheimer ,  Peter Schafer ,  Frank Schieweck ,  Anja Schwogler ,  Oliver Wagner ,  Barbara Nave ,  Maria Scherer ,  Siegfried Strathmann ,  Ulrich Schofl ,  Reinhard Stierl

发明人： Carsten Blettner ,  Markus Gewehr ,  Wassilios Grammenos ,  Thomas Grote ,  Udo Hunger ,  Bernd Muller ,  Matthias Niedenbruck ,  Joachim Rheinheimer ,  Peter Schafer ,  Frank Schieweck ,  Anja Schwogler ,  Oliver Wagner ,  Barbara Nave ,  Maria Scherer ,  Siegfried Strathmann ,  Ulrich Schofl ,  Reinhard Stierl

IPC分类号： A01N43/90 ,  A01N25/34 ,  A01N59/20

CPC分类号： A01N43/90 ,  A01N59/06 ,  A01N59/02 ,  A01N57/12 ,  A01N47/38 ,  A01N47/34 ,  A01N47/24 ,  A01N47/04 ,  A01N43/50 ,  A01N43/76 ,  A01N43/653 ,  A01N43/36 ,  A01N43/40 ,  A01N43/32 ,  A01N37/48 ,  A01N37/46 ,  A01N37/38 ,  A01N37/34 ,  A01N2300/00

摘要： The invention relates to fungicidal mixtures containing in the form of active components 1) 5-methyl-7-amino-triazolopyrimidine of formula (I), wherein R1 is alkyl, halogenalkyl, alkenyl or cyclopentyl, R2 is hydrogen or alkyl, R1 and R2 together with the nitrogen atom to which they are bound may form a piperidinyl cycle substitutable by a methyl group, L1 is fluorine or chlorine, L2, L3 are independently from each other hydrogen, fluorine or chlorine and 2) at least one type of active substance selected from groups A) azoles, B) strobilurins, C) acyl alanines, D) amine derivatives, E) anilinopyrimidines; F) dicarboximides; G) cinnamic acid amides and analogues thereof, H) antibiotics, K) dithiocarbamates, L) heterocyclic compounds, M) sulphur and copper fungicides, N) nitrophenyl derivatives, O) phenylpyrroles, P) sulfenic acid derivatives, Q) other fungicides and R) growth retardants according to the descriptions, wherein said mixtures contain the compounds in a synergically efficient amount. Novel triazolopyrimidines, methods for controlling pathogenic fungi using the mixtures of the compound (1) with active substances of the groups A) and R), the use the compounds (I) with the active substances of the groups A) and R) for producing said mixtures and agents containing said mixtures are also disclosed.

摘要翻译： 本发明涉及含有活性组分形式的杀真菌混合物1）式（I）的5-甲基-7-氨基 - 三唑并嘧啶，其中R 1是烷基，卤代烷基，烯基或环戊基，R R 2是氢或烷基，R 1和R 2与它们所连接的氮原子一起可以形成可被 甲基，L 1是氟或氯，L 2，L 3，3彼此独立地为氢，氟或氯，以及2）在 至少一种活性物质选自A）唑类，B）嗜球果伞素，C）酰基丙氨酸，D）胺衍生物，E）苯胺基嘧啶; F）二羧酰亚胺; G）肉桂酸酰胺及其类似物，H）抗生素，K）二硫代氨基甲酸盐，L）杂环化合物，M）硫和铜杀真菌剂，N）硝基苯基衍生物，O）苯基吡咯，P）亚磺酸衍生物，Q）其他杀真菌剂和R ）生长阻滞剂，其中所述混合物包含协同有效量的化合物。 新型三唑并嘧啶，使用化合物（1）与A）和R）基团的活性物质的混合物来控制致病真菌的方法，将化合物（I）与A）和R）基团的活性物质一起用于生产 还公开了含有所述混合物的所述混合物和试剂。

公开(公告)号：US20070149588A1

公开(公告)日：2007-06-28

申请号：US10582984

申请日：2004-12-14

申请人： Jordi Tormo i Blasco ,  Carsten Blettner ,  Bernd Muller ,  Markus Gewehr ,  Wassilios Grammenos ,  Thomas Grote ,  Joachim Rheinheimer ,  Peter Schafer ,  Frank Schieweck ,  Anja Schwogler ,  Oliver Wagner ,  Maria Scherer ,  Siegfried Strathmann ,  Ulrich Schofl ,  Reinhard Stierl

发明人： Jordi Tormo i Blasco ,  Carsten Blettner ,  Bernd Muller ,  Markus Gewehr ,  Wassilios Grammenos ,  Thomas Grote ,  Joachim Rheinheimer ,  Peter Schafer ,  Frank Schieweck ,  Anja Schwogler ,  Oliver Wagner ,  Maria Scherer ,  Siegfried Strathmann ,  Ulrich Schofl ,  Reinhard Stierl

IPC分类号： A01N43/64

CPC分类号： C07D487/04

摘要： The invention relates to 6-(2,3,6-trifluorophenyl)-triazolopyrimidines of formula (I), in which the substituents are defined as follows: R1 represents alkyl, haloalkyl, cycloalkyl, halocycloalkyl, alkenyl, haloalkenyl, cycloalkenyl, halocycloalkenyl, alkynyl, haloalkynyl or phenyl, naphthyl, or a five- or six-membered saturated, partially unsaturated or aromatic heterocycle, containing one to four heteroatoms from the group O, N or S; R2 represents hydrogen or one of the groups cited for R1; R1 and R2, together with the nitrogen atom, to which they are bonded, can also form a five- or six-membered heterocyclyl or heteroaryl, which is bonded via N and can contain one to three additional heteroatoms from the groups O, N and S as a ring member; R1 and/or R2 can be substituted in accordance with the description; X represents cyano, alkyl, alkoxy, alkenyloxy, haloalkoxy or haloalkenyloxy. The invention also relates to methods for producing said compounds, to agents containing the latter and to their use for combating plant-pathogenic fungi.

摘要翻译： 本发明涉及式（I）的6-（2,3,6-三氟苯基） - 三唑并嘧啶，其中取代基定义如下：R 1表示烷基，卤代烷基，环烷基，卤代环烷基， 烯基，卤代烯基，环烯基，卤代环烯基，炔基，卤代炔基或苯基，萘基或含有一至四个O，N或S基的杂原子的五元或六元饱和的部分不饱和或芳族杂环; R 2表示氢或R 1所引用的基团之一; R 1和R 2与它们所键合的氮原子一起也可以形成五或六元杂环基或杂芳基，其通过 并且可以含有一个至三个作为环成员的来自基团O，N和S的另外的杂原子; R 1和/或R 2可以根据描述代替; X表示氰基，烷基，烷氧基，烯氧基，卤代烷氧基或卤代烯氧基。 本发明还涉及生产所述化合物的方法，含有后者的试剂和用于对抗植物致病性真菌的用途。