公开(公告)号：US20060160811A1

公开(公告)日：2006-07-20

申请号：US10563222

申请日：2004-07-15

申请人： Oliver Wagner ,  Thomas Grote ,  Carsten Blettner ,  Markus Gewehr ,  Wassilios Grammenos ,  Andreas Gypser ,  Bernd Muller ,  Joachim Rheinheimer ,  Peter Schafer ,  Frank Schieweck ,  Anja Schwogler ,  Jordi Blasco ,  Alan Akers ,  John-Bryan Speakman ,  Michael Rack ,  Reinhard Stierl ,  Maria Scherer ,  Siegfried Strathmann ,  Ulrich Schofl

发明人： Oliver Wagner ,  Thomas Grote ,  Carsten Blettner ,  Markus Gewehr ,  Wassilios Grammenos ,  Andreas Gypser ,  Bernd Muller ,  Joachim Rheinheimer ,  Peter Schafer ,  Frank Schieweck ,  Anja Schwogler ,  Jordi Blasco ,  Alan Akers ,  John-Bryan Speakman ,  Michael Rack ,  Reinhard Stierl ,  Maria Scherer ,  Siegfried Strathmann ,  Ulrich Schofl

IPC分类号： C07D487/02 ,  C07D471/02 ,  A61K31/53 ,  A61K31/519

CPC分类号： C07D471/04 ,  A01N43/90

摘要： The present invention relates to bicyclic compounds of general formula I, in which X, Y independently of one another are N or C—R4; n is 1, 2, 3, 4 or 5; Ra is halogen, cyano, C1-C6-alkyl, C1-C6-alkoxy, C1-C6-haloalkyl, C1-C6-haloalkoxy, C2-C6-alkenyl, C2-C6-alkenyloxy or C(O)R5; R1 is halogen, cyano, C1-C6-alkyl, C1-C6-haloalkyl, C2-C6-alkenyl, C2-C6-alkynyl, C3-C8-cycloalkyl which is optionally mono- or polysubstituted by alkyl and/or halogen, C5-C8-cycloalkenyl which is optionally mono- or polysubstituted by alkyl and/or halogen, OR6, SR6 or NR7R8; R2 is halogen, cyano, C1-C6-alkyl, C1-C6-haloalkyl, C2-C6-alkenyl, C2-C6-alkynyl, C3-C8-cycloalkyl which is optionally mono- or polysubstituted by alkyl and/or halogen, C5-C8-cycloalkenyl which is optionally mono- or polysubstituted by alkyl and/or halogen, OR6, SR6 or NR7R8; R3 is hydrogen, C1-C6-alkyl, C1-C6-haloalkyl or C3-C6-cycloalkyl which is optionally mono- or polysubstituted by alkyl and/or halogen; and the agriculturally acceptable salts of compounds I, plant protection agents, containing at least one compound of general formula I and/or one agriculturally-acceptable salt of I and at least one liquid or solid carrier substance, as well as a method for controlling phytopathogenic fungi.

公开(公告)号：US20070149400A1

公开(公告)日：2007-06-28

申请号：US10582934

申请日：2004-12-15

申请人： Jordi Tormo i Blasco ,  Carsten Biettner ,  Bernd Muller ,  Markus Gewehr ,  Wassilios Grammenos ,  Thomas Grote ,  Joachim Rheinheimer ,  Peter Schafer ,  Frank Schieweck ,  Anja Schwogler ,  Oliver Wagner ,  Maria Scherer ,  Siegfried Strathmann ,  Ulrich Schofl ,  Reinhard Stierl

发明人： Jordi Tormo i Blasco ,  Carsten Biettner ,  Bernd Muller ,  Markus Gewehr ,  Wassilios Grammenos ,  Thomas Grote ,  Joachim Rheinheimer ,  Peter Schafer ,  Frank Schieweck ,  Anja Schwogler ,  Oliver Wagner ,  Maria Scherer ,  Siegfried Strathmann ,  Ulrich Schofl ,  Reinhard Stierl

IPC分类号： A01N43/90 ,  C07D487/04

CPC分类号： C07D487/04 ,  A01N43/90

摘要： Substituted triazolopyrimidines of the formula I in which the substituents are as defined below: L is hydrogen, chlorine or bromine; R1, R2 are hydrogen, alkyl, haloalkyl, cycloalkyl, halocycloalkyl, alkenyl, haloalkenyl, cycloalkenyl, halocycloalkenyl, alkynyl, haloalkynyl or phenyl, naphthyl or a five- or six-membered saturated, partially unsaturated or aromatic heterocycle which contains one to four heteroatoms from the group consisting of O, N and S, R1 and R2 together with the nitrogen atom to which they are attached may also form a five- or six-membered heterocyclyl or heteroaryl which is attached via N and may contain a further heteroatom from the group consisting of O, N and S as ring member and/or may be substituted as defined in the description; R3 is alkyl, haloalkyl, alkenyl, haloalkenyl, alkynyl, haloalkynyl, cycloalkyl, halocycloalkyl or phenylalkyl; R1, R2 and/or R3 may be substituted as defined in the description; X is halogen, cyano, alkyl, haloalkyl, alkoxy or haloalkoxy; processes and intermediates for preparing these compounds, compositions comprising them and their use for controlling phytopathogenic harmful fungi.

摘要翻译： 取代基如下定义的式I的取代三唑并嘧啶：L是氢，氯或溴; R 1，R 2是氢，烷基，卤代烷基，环烷基，卤代环烷基，烯基，卤代烯基，环烯基，卤代环烯基，炔基，卤代炔基或苯基，萘基或五或 含有一至四个由O，N和S杂原子组成的组的六元饱和，部分不饱和或芳族杂环，R 1和R 2连同氮 它们所连接的原子也可以形成通过N连接的五元或六元杂环基或杂芳基，并且可以含有作为环成员的O，N和S中的另外的杂原子和/或可被取代为 在说明书中定义; R 3是烷基，卤代烷基，烯基，卤代烯基，炔基，卤代炔基，环烷基，卤代环烷基或苯基烷基; R 1，R 2和/或R 3可以如说明书中所定义的取代; X是卤素，氰基，烷基，卤代烷基，烷氧基或卤代烷氧基; 制备这些化合物的方法和中间体，包含它们的组合物及其用于控制​​植物病原性有害真菌的用途。

公开(公告)号：US20060293314A1

公开(公告)日：2006-12-28

申请号：US10570893

申请日：2004-09-10

申请人： Wassilos Grammenos ,  Carsten Blettner ,  Bernd Müller ,  Marker Gewehr ,  Jordi Blasco ,  Thomas Grote ,  Joachim Rheinheimer ,  Peter Schafer ,  Frank Schieweck ,  Anja Schwögler ,  Oliver Wagner ,  Norbert Gotz ,  Siegfried Strathmann ,  Ulrich Schöfl ,  Maria Scherer ,  Reinhard Stierl

发明人： Wassilos Grammenos ,  Carsten Blettner ,  Bernd Müller ,  Marker Gewehr ,  Jordi Blasco ,  Thomas Grote ,  Joachim Rheinheimer ,  Peter Schafer ,  Frank Schieweck ,  Anja Schwögler ,  Oliver Wagner ,  Norbert Gotz ,  Siegfried Strathmann ,  Ulrich Schöfl ,  Maria Scherer ,  Reinhard Stierl

IPC分类号： A61K31/541 ,  A61K31/5377 ,  A61K31/496 ,  A61K31/4439 ,  A61K31/44 ,  C07D417/02 ,  C07D403/02 ,  C07D413/02

CPC分类号： C04B35/632 ,  C07D213/42 ,  C07D215/12 ,  C07D401/12 ,  C07D409/12

摘要： Sulfonamides of the formula I where the substituents are as follows: R1 is hydrogen, alkyl, alkoxy, alkenyl or alkynyl; and R2, R3, R4, R5 are hydrogen, halogen, alkyl, alkoxy or halomethyl; R2 and R3 together may also form a phenyl, cyclopentyl or cyclohexyl ring, it being possible for these rings to carry two groups R2, and R3,, R2,, R3, are hydrogen, halogen, alkyl, alkoxy or halomethyl; in case a), if R2, R3, R4 and R5 are hydrogen: X is phenyl substituted by a group —C(R6)═NOR7, where R6 is alkyl and R7 is alkyl, benzyl, alkenyl, haloalkyl, haloalkenyl, alkynyl or haloalkynyl; and in case b), if at least one of the groups R2, R3, R4 and R5 is not hydrogen: X is phenyl, naphthyl or a five- or six-membered saturated, or partially unsaturated or aromatic heterocycle which is attached via a carbon atom and contains one to four heteroatoms from the group consisting of O, N and S, where X may be substituted according to the description; Processes for preparing these compounds, compositions comprising them and their use for controlling phytopathogenic harmful fungi.

摘要翻译： 式I的磺酰胺，其中取代基如下：R 1是氢，烷基，烷氧基，烯基或炔基; R 2，R 3，R 4，R 5是氢，卤素，烷基，烷氧基或卤代甲基 ; R 2和R 3一起也可以形成苯基，环戊基或环己基环，这些环可以携带两个基团R 2， R 3，R 3，R 3，R 3，R 3，R 3和R 3分别为氢，卤素，烷基，烷氧基或卤代甲基; 在a）情况下，如果R 2，R 3，R 4和R 5是氢：X是 由基团-C（R 6） - NOR 7取代的苯基，其中R 6为烷基，R 7为H 烷基，苄基，烯基，卤代烷基，卤代烯基，炔基或卤代炔基; 并且在情况b）中，如果R 2，R 3，R 4和R 5中的至少一个， SUP>不是氢：X是苯基，萘基或五或六元饱和或部分不饱和或芳族杂环，其通过碳原子连接并含有一至四个由O，N和S组成的组的杂原子 ，其中X可以根据描述被替代; 制备这些化合物的方法，包含它们的组合物及其用于控制​​植物病原性有害真菌的用途。

公开(公告)号：US07709637B2

公开(公告)日：2010-05-04

申请号：US11548864

申请日：2006-10-12

申请人： Thomas Grote ,  Andreas Gypser ,  Joachim Rheinheimer ,  Ingo Rose ,  Peter Schäfer ,  Frank Schieweck ,  Hubert Sauter ,  Markus Gewehr ,  Bernd Müller ,  Jordi Tormo i Blasco ,  Eberhard Ammermann ,  Siegfried Strathmann ,  Gisela Lorenz ,  Reinhard Stierl

发明人： Thomas Grote ,  Andreas Gypser ,  Joachim Rheinheimer ,  Ingo Rose ,  Peter Schäfer ,  Frank Schieweck ,  Hubert Sauter ,  Markus Gewehr ,  Bernd Müller ,  Jordi Tormo i Blasco ,  Eberhard Ammermann ,  Siegfried Strathmann ,  Gisela Lorenz ,  Reinhard Stierl

IPC分类号： C07D403/04 ,  C07D239/38

CPC分类号： C07D239/42 ,  A01N43/54 ,  A01N43/56 ,  A01N43/60 ,  A01N43/647 ,  A01N43/653 ,  A01N43/713 ,  A01N43/90 ,  C07D231/12 ,  C07D233/56 ,  C07D249/08 ,  C07D403/04 ,  C07D473/06 ,  C07D487/04

摘要： 5-Phenylpyrimidines of the formula I, in which the substituents have the following meanings: R1 is a five- to ten-membered saturated, partially unsaturated or aromatic mono- or bicyclic heterocycle comprising one to four hetero atoms selected from the group consisting of O, N or S, which heterocycle can be substituted as defined in the description, R2 is hydrogen, halogen, cyano, alkyl, haloalkyl or alkoxy; R3, R4 are hydrogen, alkyl, haloalkyl, cycloalkyl, halocycloalkyl, alkenyl, haloalkenyl, cycloalkenyl, alkynyl, haloalkynyl or cycloalkynyl, R3 and R4 together with the nitrogen atom to which they are bonded may also form a five- or six-membered ring which can be interrupted by a hetero atom and have attached to it one or more substituents; R5, R6 are hydrogen, halogen, alkyl, haloalkyl or alkoxy; R7, R8 are hydrogen, halogen, alkyl or haloalkyl; R9 is hydrogen, halogen, alkyl, alkoxy, cycloalkoxy, haloalkoxy or alkoxycarbonyl, Processes and intermediates for the preparation of these compounds, and their use for controlling harmful fungi.

摘要翻译： 式I的5-苯基嘧啶，其中取代基具有以下含义：R 1是5至10元饱和的，部分不饱和的或芳族的单环或双环杂环，其包含一至四个选自O ，N或S，该杂环可以如描述中所定义而被取代，R 2是氢，卤素，氰基，烷基，卤代烷基或烷氧基; R3，R4是氢，烷基，卤代烷基，环烷基，卤代环烷基，烯基，卤代烯基，环烯基，炔基，卤代炔基或环炔基，R3和R4与它们所键合的氮原子一起也可以形成五元或六元环 其可以被杂原子中断并且与其连接一个或多个取代基; R5，R6是氢，卤素，烷基，卤代烷基或烷氧基; R 7，R 8为氢，卤素，烷基或卤代烷基; R9是氢，卤素，烷基，烷氧基，环烷氧基，卤代烷氧基或烷氧羰基。用于制备这些化合物的方法和中间体及其用于控制​​有害真菌的用途。

公开(公告)号：US07153860B2

公开(公告)日：2006-12-26

申请号：US10471532

申请日：2002-03-13

申请人： Thomas Grote ,  Andreas Gypser ,  Joachim Rheinheimer ,  Ingo Rose ,  Peter Schäfer ,  Frank Schieweck ,  Hubert Sauter ,  Markus Gewehr ,  Bernd Müller ,  Jordi Tormo i Blasco ,  Eberhard Ammermann ,  Siegfried Strathmann ,  Gisela Lorenz ,  Reinhard Stierl

发明人： Thomas Grote ,  Andreas Gypser ,  Joachim Rheinheimer ,  Ingo Rose ,  Peter Schäfer ,  Frank Schieweck ,  Hubert Sauter ,  Markus Gewehr ,  Bernd Müller ,  Jordi Tormo i Blasco ,  Eberhard Ammermann ,  Siegfried Strathmann ,  Gisela Lorenz ,  Reinhard Stierl

IPC分类号： C07D239/42 ,  A01N43/54 ,  C07D239/47

CPC分类号： C07D239/42 ,  A01N43/54 ,  A01N43/56 ,  A01N43/60 ,  A01N43/647 ,  A01N43/653 ,  A01N43/713 ,  A01N43/90 ,  C07D231/12 ,  C07D233/56 ,  C07D249/08 ,  C07D403/04 ,  C07D473/06 ,  C07D487/04

摘要： The invention relates to 5-phenylpyrimidine of formula (I) wherein the substituents have the following designations: R1 represents a five to ten-membered saturated, partially unsaturated or aromatic monocyclic or bicyclic heterocycle which contains between one and four heteroatoms from the group O, N or S, and which can be substituted as defined in the description; R2 represents hydrogen, halogen, cyano, alkyl, halogenalkyl or alkoxy; R3 and R4 represent hydrogen, alkyl, halogenalkyl, cycloalkyl, halogencycloalkyl, alkenyl, halogenalkenyl, cycloalkenyl, alkinyl, halogenalkinyl or cycloalkinyl; together with the nitrogen atom to which they are bonded, R3 and R4 can also form a five or six-membered ring which can be split by a heteroatom and can carry at least one substituent; R5 and R6 represent hydrogen, halogen, alkyl, halogenalkyl or alkoxy; R1 and R8 represent hydrogen, halogen, alkyl or halogenalkyl; and R9 represents hydrogen, halogen, alkyl, alkoxy, cycloalkoxy, halogenalkoxy or alkoxycarbonyl. The invention also relates to methods and intermediate products for producing said compounds and the use of the same for controlling pathogenic fungi

摘要翻译： 本发明涉及式（I）的5-苯基嘧啶，其中取代基具有以下指定：R 1表示5至10元饱和，部分不饱和或芳族单环或双环杂环，其含有一个 和来自O，N或S基团的四个杂原子，并且可以如说明书中定义的那样被取代; R 2表示氢，卤素，氰基，烷基，卤代烷基或烷氧基; R 3和R 4代表氢，烷基，卤代烷基，环烷基，卤代烷基，烯基，卤代烯基，环烯基，炔基，卤代炔基或环炔基; 与它们所键合的氮原子一起，R 3和R 4还可以形成五元或六元环，其可以被杂原子分解并且可以携带 至少一个取代基; R 5和R 6代表氢，卤素，烷基，卤代烷基或烷氧基; R 1和R 8代表氢，卤素，烷基或卤代烷基; R 9表示氢，卤素，烷基，烷氧基，环烷氧基，卤代烷氧基或烷氧基羰基。 本发明还涉及用于生产所述化合物的方法和中间产物及其用于控制​​致病真菌的用途

公开(公告)号：US20050256138A1

公开(公告)日：2005-11-17

申请号：US10513030

申请日：2003-04-30

申请人： Jordi Tormo i Blasco ,  Carsten Blettner ,  Bernd Muller ,  Markus Gewhr ,  Wassilios Grammenos ,  Thomas Grote ,  Andreas Gypser ,  Joachim Rheinheimer ,  Peter Schafer ,  Frank Schieweck ,  Anja Schwogler ,  Eberhard Ammermann ,  Siegfried Strathmann ,  Gisela Lorenz ,  Reinhard Stierl

发明人： Jordi Tormo i Blasco ,  Carsten Blettner ,  Bernd Muller ,  Markus Gewhr ,  Wassilios Grammenos ,  Thomas Grote ,  Andreas Gypser ,  Joachim Rheinheimer ,  Peter Schafer ,  Frank Schieweck ,  Anja Schwogler ,  Eberhard Ammermann ,  Siegfried Strathmann ,  Gisela Lorenz ,  Reinhard Stierl

IPC分类号： A01N43/90 ,  C07C69/65 ,  C07D487/04 ,  A61K31/519

CPC分类号： C07D487/04 ,  A01N43/90 ,  C07C69/65

摘要： Disclosed are a method for producing fungicidal triazolopyrimidine compounds, agents containing said compounds, and the use thereof for controlling harmful fungi. Also disclosed are triazolopyrimidines of formula (1), in which the substituents have the following meaning: L1 represents alkyl; L2 represents halogen; L3represents hydrogen or halogen; X represents halogen, cyano, alkyl, alkoxy, or haloalkoxy; R1, R2 represent hydrogen, alkyl, haloalkyl, cycloalkyl, alkenyl, alkadienyl, alkinyl, or cycloalkinyl, phenyl, naphthyl, or a five-unit to ten-unit saturated, partially unsaturated, or aromatic heterocycle containing one to four heteroatoms from the group O, N, or S. R1 and R2 can also form a five-unit or six-unit ring along with the nitrogen atom to which they are linked. Said ring can be interrupted and/or substituted by an atom from the group O, N, and S while R1 and/or R2 can be substituted according to the description. The invention also relates to methods and intermediate products for producing said compounds, agents containing said compounds, and the use thereof for controlling harmful fungi.

摘要翻译： 公开了生产杀真菌三唑并嘧啶化合物的方法，含有所述化合物的试剂及其用于控制​​有害真菌的用途。 还公开了式（1）的三唑并嘧啶，其中取代基具有以下含义：L 1表示烷基; L 2表示卤素; L 3表示氢或卤素; X表示卤素，氰基，烷基，烷氧基或卤代烷氧基; R 1，R 2代表氢，烷基，卤代烷基，环烷基，烯基，链二烯基，炔基或环炔基，苯基，萘基或五个单元至十个单元 饱和的，部分不饱和的或芳族杂环，其含有一至四个O，N或S的杂原子.R 1和R 2也可以形成五单元或 六单元环与它们所连接的氮原子一起。 所述环可以被O，N和S基团的原子中断和/或取代，而R 1和/或R 2可以根据描述被取代 。 本发明还涉及用于生产所述化合物的方法和中间产物，含有所述化合物的试剂及其用于控制​​有害真菌的用途。

公开(公告)号：US20060211573A1

公开(公告)日：2006-09-21

申请号：US10548690

申请日：2004-03-24

申请人： Jordi Blasco ,  Carsten Blettner ,  Bernd Muller ,  Markus Gewehr ,  Wassilios Grammenos ,  Thomas Grote ,  Andreas Gypser ,  Joachim Rheinheimer ,  Peter Schalfer ,  Frank Schieweck ,  Anja Schwogler ,  Maria Scherer ,  Siegfried Strathmann ,  Ulrich Schofl ,  Reinhard Stierl

发明人： Jordi Blasco ,  Carsten Blettner ,  Bernd Muller ,  Markus Gewehr ,  Wassilios Grammenos ,  Thomas Grote ,  Andreas Gypser ,  Joachim Rheinheimer ,  Peter Schalfer ,  Frank Schieweck ,  Anja Schwogler ,  Maria Scherer ,  Siegfried Strathmann ,  Ulrich Schofl ,  Reinhard Stierl

IPC分类号： A01N43/90 ,  C07D487/04

CPC分类号： C07D487/04 ,  A01N43/90

摘要： 7-(Alkenylamino)triazolopyrimidines of the formula I wherein the substituents have the following meanings: L is halogen, alkyl, haloalkyl, alkoxy, amino, NHR or NR2; R is alkyl or alkyl-carbonyl; m is 1, 2, 3, 4 or 5; X is halogen, cyano, alkyl, haloalkyl or alkoxy; R1 is alkyl or haloalkyl; R2 is hydrogen, alkyl or haloalkyl; R3 is alkenyl, which can be unsubstituted or partially or completely halogenated or can be substituted according to the Description; R4 is hydrogen or alkyl, R3 and R4 can also, together with the nitrogen atom to which they are bonded, form a five- or six-membered unsaturated ring which can be interrupted by an atom from the group consisting of O, N and S and/or can carry one or more sub-stituents. Processes for the preparation of these compounds, preparations comprising them and their use in the control of harmful phytopathogenic fungi.

摘要翻译： 式（I）的7-（烯基氨基）三唑并嘧啶，其中取代基具有以下含义：L是卤素，烷基，卤代烷基，烷氧基，氨基，NHR或NR 2。 R是烷基或烷基 - 羰基; m为1,2,3,4或5; X是卤素，氰基，烷基，卤代烷基或烷氧基; R 1是烷基或卤代烷基; R 2是氢，烷基或卤代烷基; R 3是烯基，其可以是未取代的或部分的或完全卤化的或可以根据描述被取代; R 4是氢或烷基，R 3和R 4也可以与它们所键合的氮原子一起形成五元环 - 或六元不饱和环，其可以被来自O，N和S的原子中断，和/或可以携带一个或多个亚取代基。 制备这些化合物的方法，包含它们的制剂及其在控制有害植物病原真菌中的用途。

公开(公告)号：US06593315B2

公开(公告)日：2003-07-15

申请号：US09896971

申请日：2001-07-02

申请人： Andreas Gypser ,  Thomas Grote ,  Joachim Rheinheimer ,  Ingo Rose ,  Oliver Cullmann ,  Markus Gewehr ,  Wassilios Grammenos ,  Jordi Tormo i Blasco ,  Bernd Müller ,  Hubert Sauter ,  Eberhard Ammermann ,  Siegfried Strathmann ,  Gisela Lorenz ,  Reinhard Stierl

发明人： Andreas Gypser ,  Thomas Grote ,  Joachim Rheinheimer ,  Ingo Rose ,  Oliver Cullmann ,  Markus Gewehr ,  Wassilios Grammenos ,  Jordi Tormo i Blasco ,  Bernd Müller ,  Hubert Sauter ,  Eberhard Ammermann ,  Siegfried Strathmann ,  Gisela Lorenz ,  Reinhard Stierl

IPC分类号： A01N3736

CPC分类号： C07C251/86 ,  A01N37/50

摘要： Salicylic acid derivatives of the formula I, where the index and the substituents have the following meanings: X is halogen, NO2, cyano, alkyl or alkoxy; m is 0, 1, 2 or 3, it being possible for the substituents X to be different from each other if n is greater than 1; A is OH, alkoxy, NH2, NHCH3 or N(CH3)2; R1 is phenyl, naphthyl, cycloalkyl, 5-membered or 6-membered hetaryl or 5-membered or 6-membered heterocyclyl, comprising one to three N atoms and/or one O or S atom or one or two O and/or S atoms, the ring systems being unsubstituted or substituted; R2 is hydrogen, cyano, alkyl, alkenyl, alkynyl, haloalkyl, alkoxy or alkylthio, processes for the preparation of these compounds, compositions comprising them, and their use for controlling harmful fungi.

摘要翻译： 式I的水杨酸衍生物，其中指数和取代基具有以下含义：X是卤素，NO 2，氰基，烷基或烷氧基; m是0,1,2或3，取代基X可以是 如果n大于1，A是不同的; A是OH，烷氧基，NH2，NHCH3或N（CH3）2; R1是苯基，萘基，环烷基，5元或6元杂芳基或5元或6- 包括一至三个N原子和/或一个O或S原子或一个或两个O和/或S原子，所述环系是未取代或取代的; R2是氢，氰基，烷基，烯基，炔基，卤代烷基， 烷氧基或烷硫基，制备这些化合物的方法，包含它们的组合物及其用于控制​​有害真菌的用途。

公开(公告)号：US20060258685A1

公开(公告)日：2006-11-16

申请号：US10558251

申请日：2004-05-27

申请人： Olivier Wagner ,  Thomas Grote ,  Carsten Blettner ,  Markus Gewehr ,  Wassilios Grammenos ,  Andreas Gypser ,  Bernd Muller ,  Joachim Rheinheimer ,  Peter Schafer ,  Frank Schieweck ,  Anja Schwogler ,  Jordi Blasco ,  Alan Akers ,  John-Bryan Speakman ,  Michael Rack ,  Reinhard Stierl ,  Maria Scherer ,  Ulrich Schofl ,  Siegfried Strathmann

发明人： Olivier Wagner ,  Thomas Grote ,  Carsten Blettner ,  Markus Gewehr ,  Wassilios Grammenos ,  Andreas Gypser ,  Bernd Muller ,  Joachim Rheinheimer ,  Peter Schafer ,  Frank Schieweck ,  Anja Schwogler ,  Jordi Blasco ,  Alan Akers ,  John-Bryan Speakman ,  Michael Rack ,  Reinhard Stierl ,  Maria Scherer ,  Ulrich Schofl ,  Siegfried Strathmann

IPC分类号： A61K31/519 ,  C07D487/04

CPC分类号： C07D487/04 ,  A01N43/90

摘要： The invention relates to substituted pyrazolopyrimidines of formula (I) wherein the substituents have the following designations: L represents halogen, alkyl, halogenalkyl, alkenyl, alkoxy, amino, NHR, NR2, cyano, S(═O)nA1 or C(═O)A2, R representing alkyl or alkylcarbonyl, A1 representing hydrogen, hydroxy, alkyl, alkylamino or dialkylamino, n representing 0, 1 or 2, and A2 representing alkenyl, alkoxy, halogenalkoxy or one of the groups cited for A1; m represents 0 or 1 to 5; R1 represents alkyl, halogenalkyl, cycloalkyl, halogencycloalkyl, alkenyl, alkadienyl, halogenalkenyl, cycloalkenyl, alkinyl, halogenalkinyl or cycloalkinyl, phenyl, naphthyl, or a five-membered to ten-membered saturated, partially unsaturated or aromatic heterocycle containing between one and four heteroatoms from the group O, N or S; and R2 represents hydrogen or one of the groups cited for R1. Together with the nitrogen atom to which they are bonded, R1 and R2 can form a five-membered to six-membered ring that can be interrupted by an atom from the groups O, N and S, and R1 and/or R2 can also be substituted according to the description. Furthermore, in formula (I): X represents halogen, cyano, OH, alkyl, alkoxy or halogenalkoxy; Y represents a five-membered to ten-membered saturated, partially unsaturated or aromatic heterocycle according to the description, or a group X or another group according to the description; p represents 1 or 2, the groups Y being potentially different when p=2; and p represents 0, when X is according to the description. The invention also relates to methods and intermediate products for producing said compounds, agents containing the same, and the use thereof for controlling phytopathogenic fungi.

公开(公告)号：US20080032889A1

公开(公告)日：2008-02-07

申请号：US11630558

申请日：2005-06-14

申请人： Carsten Blettner ,  Markus Gewehr ,  Wassilios Grammenos ,  Thomas Grote ,  Udo Hunger ,  Bernd Muller ,  Matthias Niedenbruck ,  Joachim Rheinheimer ,  Peter Schafer ,  Frank Schieweck ,  Anja Schwogler ,  Oliver Wagner ,  Barbara Nave ,  Maria Scherer ,  Siegfried Strathmann ,  Ulrich Schofl ,  Reinhard Stierl

发明人： Carsten Blettner ,  Markus Gewehr ,  Wassilios Grammenos ,  Thomas Grote ,  Udo Hunger ,  Bernd Muller ,  Matthias Niedenbruck ,  Joachim Rheinheimer ,  Peter Schafer ,  Frank Schieweck ,  Anja Schwogler ,  Oliver Wagner ,  Barbara Nave ,  Maria Scherer ,  Siegfried Strathmann ,  Ulrich Schofl ,  Reinhard Stierl

IPC分类号： A01N43/90 ,  A01C1/06 ,  C07D487/04

CPC分类号： A01N43/90 ,  C07D487/04

摘要： Substituted triazolopyrimidines of the formula I in which the substituents are as defined below: R1 is alkyl, halocycloalkyl, alkenyl, cycloalkyl, cycloalkenyl, halocycloalkenyl, alkynyl, haloalkynyl or naphthyl, or a five- or six-membered saturated, partially unsaturated or aromatic heterocycle comprising one to four heteroatoms from the group consisting of O, N and S, R2 is hydrogen, alkyl or one of the groups mentioned under R1; R1 and/or R2 may carry one to four identical or different groups Ra: Ra is chlorine, bromine, iodine, cyano, nitro, hydroxyl, alkyl, alkylcarbonyl, cycloalkyl, alkoxy, haloalkoxy, alkoxycarbonyl, alkylthio, alkylamino, dialkyl-amino, alkenyl, cycloalkenyl, alkenyloxy, haloalkenyloxy, alkynyl, halo-alkynyl, alkynyloxy, haloalkynyloxy, cycloalkoxy, cycloalkenyloxy, oxyalkylenoxy, naphthyl, a five- to ten-membered saturated, partially unsaturated or aromatic heterocycle comprising one to four heteroatoms from the group consisting of O, N and S, where these aliphatic, alicyclic or aromatic groups for their part may be substituted according to the description; and X is halogen; processes for preparing these compounds, compositions comprising them and their use for controlling phytopathogenic harmful fungi.

摘要翻译： 取代基如下定义的式I的取代三唑并嘧啶：R 1是烷基，卤代环烷基，烯基，环烷基，环烯基，卤代环烯基，炔基，卤代炔基或萘基，或五或六元环， 包含一至四个由O，N和S组成的组的杂原子的2-元饱和的，部分不饱和的或芳族的杂环，R 2是氢，烷基或R 1上提到的基团之一， / SUP>; R 1和/或R 2可以携带一至四个相同或不同的基团R a是：R a是 氯，溴，碘，氰基，硝基，羟基，烷基，烷基羰基，环烷基，烷氧基，卤代烷氧基，烷氧基羰基，烷硫基，烷基氨基，二烷基氨基，烯基，环烯基，烯氧基，卤代烯氧基，炔基，卤代炔基，炔氧基，卤代炔氧基， 环烷氧基，环烯氧基，氧亚烷基氧基，萘基，五至十元饱和的部分不饱和或芳族杂环，其包含一至四个由O，N和S组成的组的杂原子，其中这些脂族，脂环族或芳族基团可以 根据描述进行替代; X为卤素; 制备这些化合物的方法，包含它们的组合物及其用于控制​​植物病原性有害真菌的用途。