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75 条记录 (耗时 0.03 秒)

    1-Phenyl-4-amino-cyclohex-2-ene-1-carboxylic acid ethyl esters
    64.
    发明授权
    1-Phenyl-4-amino-cyclohex-2-ene-1-carboxylic acid ethyl esters 失效
    1-苯基-4-氨基 - 环己基-2-环己-1-羧酸乙酯

    公开(公告)号：US3957851A

    公开(公告)日：1976-05-18

    申请号：US226509

    申请日：1972-02-15

    申请人： Gerhard Satzinger ,  Manfred Franz Herrmann

    发明人： Gerhard Satzinger ,  Manfred Franz Herrmann

    IPC分类号： C07D211/14 ,  C07D211/34 ,  C07D211/46 ,  C07D295/155 ,  C07C101/38

    CPC分类号： C07D295/155 ,  C07D211/14 ,  C07D211/34 ,  C07D211/46

    摘要： The invention relates to 1-phenyl-4-amino-cyclohex-2-ene-1-carboxylic-acid-esters of the general formula I ##SPC1##wherein R.sub.1 and R.sub.2 may be the same or different and may be H, alkyl, hydroxyalkyl, alkenyl, preferably with 1 to 4 C-atoms, aralkyl which may be bonded to each other, in which connection the heterocyclic system formed may be substituted further by the OH-- group and where attachment takes place by an oxygen or a nitrogen atom, if desired, which in its turn carries an H, alkyl with 1 to 4 C-atoms, aryl which may be substituted by chlorine, preferably in 3 or 4-position, and by methoxy, preferably in 2 or 4-position, acyl, preferably alkanoyl with 1 to 4 C-atoms, and aroyl, or aralkyl, and R.sub.3 represents an alkyl radical with 1 to 4 C-atoms, the salts thereof and quarternary ammonium compounds, and a process for their preparation. These compounds have analgesic and neuroleptic properties.

    Benzo(b)thiophene derivatives
    67.
    发明授权
    Benzo(b)thiophene derivatives 失效
    BENZO（B）噻吩衍生物

    公开(公告)号：US4082770A

    公开(公告)日：1978-04-04

    申请号：US785809

    申请日：1977-04-08

    申请人： Peter Johannes Stoss ,  Manfred Franz Reinhold Herrmann ,  Gerhard Satzinger

    发明人： Peter Johannes Stoss ,  Manfred Franz Reinhold Herrmann ,  Gerhard Satzinger

    IPC分类号： C07D333/70 ,  C07D333/64

    CPC分类号： C07D333/70

    摘要： The present invention relates to novel benzo(b)thiophene derivatives of the general formula: ##STR1## wherein Y represents a hydrogen or halogen atom; A represents a hydrogen atom or a phenyl group which may be substituted with a halogen atom or a lower alkoxy group; B represents a radical of the formula OR' or NR.sup.2 R.sup.3, wherein R' is an alkyl radical of 1 to 5 carbon atoms which may be substituted with hydroxy, lower alkoxy, phenyl or phenoxy groups or a cycloalkyl or phenyl group which may be substituted by lower alkoxy or halogen atoms; R.sup.2 and R.sup.3, which may be identical or different, represent, if identical, hydrogen, alkyl radicals of 1 to 5 carbon atoms which may be substituted by hydroxy, lower alkoxy, phenoxy, di-lower alkylamino, or phenyl groups; or, if R.sup.2 is hydrogen, R.sup.3 represents either a hydroxyl or an amino group which may be substituted by lower alkyl, dialkyl, alkylidene, phenyl or acyl groups or a lower alkyl group which may be substituted by hydroxy, lower alkoxy, phenoxy, dialkylamino, pyrrolidino, piperidino or morpholino groups; R.sup.3 further is a cycloalkyl or phenyl group, which may be substituted by a halogen or a lower alkoxy radical; R.sup.2 and R.sup.3 together with the nitrogen atom to which they are attached, may form an aziridine, pyrrolidine, piperidine, morpholine or piperazine ring which may be substituted by lower alkyl, hydroxyalkyl, phenylalkyl, phenyl or acetyl groups; or A and B together with the C--N group may form a 5, 6, or 7-membered heterocyclic ring.The present invention further relates to the processes for the preparation of these derivatives and to the salts of these compounds with physiologically acceptable inorganic and organic acids such as hydrochloric acid, sulfuric acid, phosphoric acid, fumaric acid, oxalic acid, citric acid, etc., and the quaternary ammonium compounds.

    Certain dibenzothiacyclic-S-oximides
    69.
    发明授权
    Certain dibenzothiacyclic-S-oximides 失效
    某些二苯并硫代-S-锑酰亚胺

    公开(公告)号：US4076723A

    公开(公告)日：1978-02-28

    申请号：US769641

    申请日：1977-02-17

    申请人： Peter Stoss ,  Gerhard Satzinger

    发明人： Peter Stoss ,  Gerhard Satzinger

    IPC分类号： C07D333/76 ,  C07D337/14 ,  C07D335/12 ,  C07D335/16

    CPC分类号： C07D333/76

    摘要： The present invention is concerned with novel tricyclic sulphoximides and with the preparation thereof. This family of compounds has been found to possess antihistominic, antitussive, antiinflammatory, sedative, and diuretic properties.

    摘要翻译： 本发明涉及新型三环磺酰亚胺及其制备方法。 已经发现这种化合物家族具有抗真菌，止咳，抗炎，镇静和利尿的特性。

    Thianthrene and phenoxathiine s-oximides
    70.
    发明授权
    Thianthrene and phenoxathiine s-oximides 失效
    噻蒽和吩草酸S-锑酰亚胺

    公开(公告)号：US4033981A

    公开(公告)日：1977-07-05

    申请号：US663312

    申请日：1976-03-03

    申请人： Peter Stoss ,  Gerhard Satzinger

    发明人： Peter Stoss ,  Gerhard Satzinger

    IPC分类号： C07D333/76 ,  C07D339/08 ,  C07D327/08

    CPC分类号： C07D333/76

    摘要： The present invention is concerned with novel tricyclic sulphoximides and with the preparation thereof. This family of compounds has been found to possess antihistominic, antitussive, antiinflammatory, sedative, and diuretic properties.

    摘要翻译： 本发明涉及新型三环磺酰亚胺及其制备方法。 已经发现这种化合物家族具有抗真菌，止咳，抗炎，镇静和利尿的特性。