Substituted 3-phenylpyrazoles
    61.
    发明授权
    Substituted 3-phenylpyrazoles 失效
    取代的3-苯基吡唑

    公开(公告)号:US06197973B1

    公开(公告)日:2001-03-06

    申请号:US09230838

    申请日:1999-02-01

    IPC分类号: C07D23114

    摘要: 3-phenylpyrazoles of formula I wherein R1 is cyano, alkyl or haloalkyl; R2 is cyano or is optionally halogenated alkyl, alkoxy, alkylthio, alkylsulfinyl or alkylsulfonyl; R3 is hydrogen, cyano, halogen, alkyl or haloalkyl; R4 is hydrogen or halogen; R5 is cyano, halogen, or is optionally halogenated alkyl or alkoxy; R6, R7 independently of one another are optionally substituted alkyl, alkenyl, alkynyl, cycloalkyl, heterocyclyl or phenyl, optionally substituted alkylcarbonyl, alkoxycarbonyl, aminocarbonyl, alkylaminocarbonyl, dialkylaminocarbonyl or optionally halogenated alkylsulfonyl; X is a chemical bond, —C≡C—, —CH2—CH(R8)— or —CH═C(R8)—, wherein R8 is hydrogen, cyano, nitro, halogen, alkyl or haloalkyl; Y is oxygen or sulfur; their preparation and their use for controlling undesirable vegetation.

    摘要翻译: 式I的3-苯基吡唑,其中R1是氰基,烷基或卤代烷基; R2是氰基或任选被卤代烷基,烷氧基,烷硫基,烷基亚磺酰基或烷基磺酰基; R3是氢,氰基,卤素,烷基或卤代烷基; R4是氢或卤素; R5是 氰基,卤素或任选卤代烷基或烷氧基; R 6,R 7彼此独立地是任选取代的烷基,烯基,炔基,环烷基,杂环基或苯基,任选取代的烷基羰基,烷氧基羰基,氨基羰基,烷基氨基羰基,二烷基氨基羰基或任选卤代烷基磺酰基; X是化学键,-C = C-,-CH 2 -CH(R 8) - 或-CH = C(R 8) - ,其中R 8是氢,氰基,硝基,卤素,烷基或卤代烷基; Y是氧或硫 ;他们的准备和用于控制不良植被的用途。

    Substituted 2-phenylpyridines useful as herbicides
    62.
    发明授权
    Substituted 2-phenylpyridines useful as herbicides 失效
    用作除草剂的取代的2-苯基吡啶

    公开(公告)号:US5968874A

    公开(公告)日:1999-10-19

    申请号:US983288

    申请日:1998-01-20

    摘要: Substituted 2-phenylpyridines I ##STR1## where n is 0, 1;R.sup.1 is halogen, C.sub.1 -C.sub.6 -haloalkyl;R.sup.2 and R.sup.3 are H, halogen;R.sup.4 is cyano, halogen;X and Y are --O--, --S--;R.sup.5 and R.sup.6 are H, C.sub.1 -C.sub.4 -alkyl or together are a 1,2-ethylene, 1,3-propylene, 1,4-tetramethylene or 1,5-pentamethylene chain;R.sup.7 is C.sub.1 -C.sub.6 -haloalkyl, C.sub.3 -C.sub.6 -haloalkenyl, C.sub.2 -C.sub.6 -alkenyloxy-C.sub.1 -C.sub.4 -alkyl, C.sub.2 -C.sub.6 -alkenyloxy-C.sub.1 -C.sub.4 -alkoxy-C.sub.1 -C.sub.4 -alkyl, C.sub.3 -C.sub.6 -alkenyl, C.sub.3 -C.sub.6 -alkadienyl, C.sub.3 -C.sub.6 -alkynyl, C.sub.3 -C.sub.6 -cycloalkyl, C.sub.5 -C.sub.6 -cycloalkenyl, 3-oxetanyl, 3-thietanyl, phenyl, phenyl-C.sub.1 -C.sub.4 -alkyl or 5/6-membered heteroaryl having 1 to 3 hetero atoms selected from the group consisting of two oxygen atoms, two sulfur atoms and 3 nitrogen atoms, orR.sup.6 and R.sup.7 together are a 1,2-ethylene or 1,3-propylene chain which can have attached to it one or two C.sub.1 -C.sub.4 -alkyl substituents are used as herbicides and for the desiccation/defoliation of plants.

    摘要翻译: PCT No.PCT / EP96 / 03243 Sec。 371日期1998年1月20日 102(e)1998年1月20日PCT PCT 1996年7月23日PCT公布。 公开号WO97 / 06143 日期1997年2月20日取代的2-苯基吡啶I,其中n为0,1; R1是卤素,C1-C6-卤代烷基; R2和R3是H,卤素; R4是氰基,卤素; X和Y是-O - , - S- R5和R6是H,C1-C4-烷基或一起是1,2-亚乙基,1,3-丙烯,1,4-四亚甲基或1,5-五亚甲基链; R 7是C 1 -C 6卤代烷基,C 3 -C 6卤代链烯基,C 2 -C 6 - 烯氧基-C 1 -C 4 - 烷基,C 2 -C 6 - 烯氧基-C 1 -C 4 - 烷氧基-C 1 -C 4烷基,C 3 -C 6 - 烯基, C 3 -C 6 - 链烯基,C 3 -C 6 - 炔基,C 3 -C 6 - 环烷基,C 5 -C 6 - 环烯基,3-氧杂环丁烷基,3-硫杂环丁基,苯基,苯基-C 1 -C 4烷基或5 至3个选自两个氧原子,两个硫原子和3个氮原子的杂原子,或者R6和R7一起是可以连接至一个或两个的1,2-亚乙基或1,3-亚丙基链 C1-C4烷基取代基用作除草剂和用于植物的干燥/脱叶。

    Substituted (4-brompyrazole-3-yl) benzazoles

    公开(公告)号:US06482774B1

    公开(公告)日:2002-11-19

    申请号:US09673996

    申请日:2000-10-25

    IPC分类号: C07D41704

    摘要: Substituted (4-bromopyrazol-3-yl)benzazoles I and their salts where R1=H, C1-C4-alkyl, C1-C4-haloalkyl; R2=CN, Cl-C4-alkyl, C1-C4-haloalkyl, C1-C4-alkoxy, C1-C4-haloalkoxy, C1-C4-alkylthio, C1-C4-haloalkylthio, C1-C4-alkylsulfinyl, C1-C4-haloalkylsulfinyl, C1-C4-alkylsulfonyl, C1-C4-haloalkylsulfonyl; R4=H, halogen; R5=H, CN, halogen, C1-C4-alkyl, C1-C4-haloalkyl, C1-C4-alkoxy or C1-C4-haloalkoxy; Z=—N═C(XR6)—O— or —N═C(XR6)—S—, attached to &agr; via the nitrogen, oxygen or sulfur; X=a chemical bond, oxygen, sulfur, —S(O)—, —SO2—, —NH— or —N(R7)—; R6, R7=Cl-C6-alkyl, Cl-C6-haloalkyl, cyano-Cl-C4-alkyl, hydroxy-C1-C4-alkyl, C3-C6-alkenyl, cyano-C3-C6-alkenyl, C3-C6-haloalkenyl, C3-C6-alkynyl, cyano-C3-C6-alkynyl, C3-C6-haloalkynyl, C1-C4-alkoxy-C1-C4-alkyl, C1-C4-haloalkoxy-C1-C4-alkyl, C3-C4-alkenyloxy-C1-C4-alkyl, C3-C4-alkynyloxy-C1-C4-alkyl, C3-C8-cycloalkyloxy-C1-C4-alkyl, amino-Cl-C4-alkyl, C1-C4-alkylamino-C1-C4-alkyl, di(C1-C4-alkyl)amino-C1-C4-alkyl, Cl-C4-alkylthio-C1-C4-alkyl, C1-C4-haloalkylthio-C1-C4-alkyl, C3-C4-alkenylthio-C1-C4-alkyl, C3-C4-alkynylthio-C1-C4-alkyl, C1-C4-alkylsulfinyl-Cl-C4-alkyl, C1-C4-haloalkylsulfinyl-C1-C4-alkyl, C3-C4-alkenylsulfinyl-C1-C4-alkyl, C3-C4-alkynylsulfinyl-C1-C4-alkyl, C1-C4-alkylsulfonyl-C1-C4-alkyl, C1-C4-haloalkylsulfonyl-C1-C4-alkyl, C3-C4-alkenylsulfonyl-C1-C4-alkyl, C3-C4-alkynylsulfonyl-C1-C4-alkyl, hydroxycarbonyl-C1-C4-alkyl, C1-C4-alkoxycarbonyl-C1-C4-alkyl, which may carry a CN or C1-C4-alkoxycarbonyl group, C1-C4-alkylthiocarbonyl-C1-C4-alkyl, aminocarbonyl-C1-C4-alkyl, C1-C4-alkylaminocarbonyl-C1-C4-alkyl, di(C1-C4-alkyl)aminocarbonyl-C1-C4-alkyl, di(C1-C4-alkyl)-phosphonyl-C1-C4-alkyl, C1-C4-alkoxyimino-C1-C4-alkyl, C3-C4-alkenyloxyimino-C1-C4-alkyl, unsubstituted or substituted C3-C8-cycloalkyl, C3-C8-cycloalkyl-C1-C4-alkyl, phenyl, phenyl-C1-C4-alkyl, 3- to 7-membered heterocyclyl or heterocyclyl-C1-C4-alkyl, where each cycloalkyl and each heterocyclyl ring may contain a CO or CS ring member; if X=a chemical bond, —O—, —S—, —NH— or —N(R7)—, R6 may also be C1-C4-alkylcarbonyl, C1-C4-haloalkylcarbonyl, C1-C4-alkoxycarbonyl, C1-C4-alkylsulfonyl or C1-C4-haloalkylsulfonyl; if X=a chemical bond, R6 may furthermore be CN, SH, NH2, halogen, —CH2—CH(halogen)-R8, —CH═CH—R8 or —CH═C(halogen)-R8, where R8=COOH, C1-C4-alkoxycarbonyl, C1-C4-alkylthiocarbonyl, CONH2, C1-C4-alkylaminocarbonyl, di(C1-C4-alkyl)aminocarbonyl or di(C1-C4-alkyl)phosphonyl; or R6+R7=an unsubstituted or substituted 1,3-propylene, tetramethylene, pentamethylene or ethyleneoxyethylene chain. Use: As herbicides; for the desiccation/defoliation of plants.

    Substituted 2-phenyl-3(2H)-pyridazinones
    70.
    发明授权
    Substituted 2-phenyl-3(2H)-pyridazinones 失效
    取代的2-苯基-3(2H) - 哒嗪酮

    公开(公告)号:US06225313B1

    公开(公告)日:2001-05-01

    申请号:US09508781

    申请日:2000-03-16

    IPC分类号: C07D23718

    摘要: Substituted 2-phenyl-3(2H)-pyridazinones I and salts thereof, where n=0, 1, 2; R1=C1-C4-alkyl, C1-C4-haloalkyl; R2=H, halogen; R3=halogen, CN; R4=H, NO2, CN, CHO, NH—OH, C1-C4-alkyl, C1-C4-halogenalkyl, —OR5, —CH═N—OR6, —CH═C(R7)—CO—OR8, —CO—OR9, C1-C6-alkyl-SO2—NH, di(C1-C6-alkylsulfonyl)amino or R5=C1-C6-alkyl, C3-C6-alkenyl, C3-C6-alkynyl, (C1-C6-alkoxy)carbonyl-C1-C4-alkyl, (C3-C6-alkenyloxy)carbonyl-C1-C4-alkyl, (C3-C6-alkynyloxy)carbonyl-C1-C4-alkyl, C1-C4-alkoxy(C1-C4-alkoxy)carbonyl-C1-C4-alkyl; R6=H, C1-C4-alkyl, hydroxycarbonyl-C1-C4-alkyl, (C1-C4-alkoxy)carbonyl-C1-C4-alkyl; R7=H, halogen, C1-C4-alkyl; R8=H, C1-C6-alkyl; R9=H, C1-C6-alkyl, C3-C6-alkenyl, C3-C6-alkynyl, C1-C4-alkoxy-C1-C4-alkoxy, hydroxycarbonyl-C1-C4-alkyl, (C1-C6-alkoxy)carbonyl-C1-C4-alkyl, (C3-C6-alkenyloxy)carbonyl-C1-C4-alkyl, (C3-C6-alkynyloxy)carbonyl-C1-C4-alkyl, C1-C4-alkoxy-(C1-C4-alkoxy)carbonyl-C1-C4-alkyl; R10=H, C1-C6-alkyl, COOH, (C1-C6-alkoxy)carbonyl; and their use as herbicides and for the desiccation/defoliation of plants are described.

    摘要翻译: 取代的2-苯基-3(2H) - 哒嗪酮I和其盐,其中n = 0,1,2; R1 = C1-C4-烷基,C1-C4卤代烷基; R2 = H,卤素; R3 =卤素,CN; R4 = H,NO2,CN,CHO,NH-OH,C1-C4-烷基,C1-C4-卤代烷基,-OR5,-CH = N-OR6,-CH = C(R7) CO-OR 8,-CO-OR 9,C 1 -C 6烷基-SO 2 -NH,二(C 1 -C 6烷基磺酰基)氨基或R 5 = C 1 -C 6烷基,C 3 -C 6 - 烯基,C 3 -C 6炔基,(C 1 C 3-6 - 烷氧基)羰基-C 1 -C 4烷基,(C 3 -C 6 - 烯氧基)羰基-C 1 -C 4 - 烷基,(C 3 -C 6 - 炔氧基)羰基-C 1 -C 4烷基,C 1 -C 4 - C 1 -C 4 - 烷氧基)羰基-C 1 -C 4 - 烷基; R 6 = H,C 1 -C 4 - 烷基,羟基羰基-C 1 -C 4 - 烷基,(C 1 -C 4 - 卤素,C 1 -C 4 - 烷基; R8 = H,C1-C6-烷基; R9 = H,C1-C6-烷基,C3-C6-烯基,C3-C6-炔基,C1-C4-烷氧基-C1-C4-烷氧基,羟基羰基C1-C4- 烷基,(C 1 -C 6 - 烷氧基)羰基-C 1 -C 4 - 烷基,(C 3 -C 6 - 烯氧基)羰基-C 1 -C 4烷基,(C 3 -C 6 - 炔氧基)羰基-C 1 -C 4烷基,C 1 -C 4 - 烷氧基 - (C 1 -C 4 - 烷氧基)羰基-C 1 -C 4烷基; R 10 = H,C 1 -C 6烷基,COOH,(C 1 -C 6 - 烷氧基)羰基;及其作为除草剂和干燥/ 的植物被描述。