Substituted 5-Hetaryl-4-Aminopyrimidines
    82.
    发明申请

    公开(公告)号:US20110201496A1

    公开(公告)日:2011-08-18

    申请号:US12293432

    申请日:2007-03-26

    CPC分类号: A01N43/54

    摘要: The present invention relates to the use of 5-hetaryl-4-aminopyrimidines of the formula I and their salts for controlling plant-damaging fungi. The invention also relates to novel 5-hetaryl-4-aminopyrimidines and to crop protection compositions comprising at least one such compound as active component. Het is an optionally substituted 5- or 6-membered aromatic heterocycle which has 1, 2, 3 or 4 heteroatoms selected from the group consisting of nitrogen, oxygen and sulfur as ring members, where the 5- or 6-membered heteroaromatic radical may have 1, 2, 3 or 4 identical or different substituents L, R1, R2 are inter alia hydrogen, C1-C8-alkyl, C3-C8-cycloalkyl, C5-C10-bicycloalkyl, C2-C8-alkenyl, C4-C10-alkadienyl, C3-C6-cycloalkenyl, C2-C8-alkynyl, phenyl, naphthyl or a five- or six-membered saturated, partially unsaturated or aromatic heterocycle which has one, two, three or four heteroatoms from the group consisting of O, N or S as ring members; or together form a ring; R3 is inter alia hydrogen, OH, halogen, cyano, NR31R32, C1-C8-alkyl, C1-C8-alkoxy, C1-C8-alkylthio, C1-C8-alkylsulfinyl, C1-C8-alkylsulfonyl, C2-C8-alkenyl or C2-C8-alkynyl, and R4 is halogen, cyano, hydroxyl, mercapto, N3, C1-C6-alkyl, C2-C8-alkenyl, C2-C8-alkynyl, C1-C6-haloalkyl, C1-C6-alkoxy, C3-C8-alkenyloxy, C3-C8-alkynyloxy, C1-C6-haloalkoxy, C1-C6-alkylthio, C3-C8-alkenylthio, C3-C8-alkinylthio, C1-C6-haloalkylthio, or is a radical of the formula C(═Z)OR41, C(═Z)NR42R43, C(═Z)NR44—NR42R43, C(═Z)R45, CR46R47—OR48, CR46R47—NR42R43, ON(═CR49R50), O—C(═Z)R45, NR42R43a, NR51(C(═Z)R45), NR51(C(═Z)OR41), NR51(C(═Z)—NR42R43), NR52a(N═CR49R50), NR52NR42R43, NR52OR41 or C(═N—X—R45)SR41.

    2-Substituted 7-Aminoazolopyrimidines, Processes For Their Preparation And Their Use For Controlling Harmful Fungi, And Compositions Comprising These Compounds
    89.
    发明申请
    2-Substituted 7-Aminoazolopyrimidines, Processes For Their Preparation And Their Use For Controlling Harmful Fungi, And Compositions Comprising These Compounds 审中-公开
    2-取代的7-氨基偶氮嘧啶,其制备方法及其用于控制​​有害真菌和包含这些化合物的组合物

    公开(公告)号:US20080139581A1

    公开(公告)日:2008-06-12

    申请号:US11885536

    申请日:2006-03-02

    IPC分类号: A01N43/90 A01P3/00 C07D487/04

    CPC分类号: C07D487/04

    摘要: 2-Substituted 7-aminoazolopyrimidines of the formula I in which the substituents are as defined below: R1 is hydrogen, halogen, cyano, alkyl, haloalkyl, alkenyl, alkynyl, cycloalkyl, alkoxy, alkoxyalkyl, benzyloxyalkyl, alkoxyalkenyl or alkoxyalkynyl; R2 is hydrogen, halogen, cyano, alkyl, haloalkyl, alkenyl, alkynyl, cycloalkyl, alkoxy, alkoxyalkyl and alkylthioalkyl, where the carbon chains in R1 and/or R2 may be substituted according to the description; R3 is halogen, cyano, NRARB, hydroxyl, mercapto, alkyl, haloalkyl, cycloalkyl, alkoxy, alkylthio, cycloalkoxy, cycloalkylthio, carboxyl, formyl, alkylcarbonyl, alkoxycarbonyl, alkenyloxycarbonyl, alkynyloxycarbonyl, phenyl, phenoxy, phenylthio, benzyloxy, benzylthio, alkyl-S(O)m—; A is N and CRx; Rx is hydrogen or one of the groups mentioned under R3; processes and intermediates for preparing these compounds, compositions comprising them and their use for controlling phytopathogenic harmful fungi.

    摘要翻译: 2-取代的式I的7-氨基偶氮嘧啶,其中取代基如下:R 1是氢,卤素,氰基,烷基,卤代烷基,烯基,炔基,环烷基,烷氧基,烷氧基烷基,苄氧基烷基 ,烷氧基烯基或烷氧基炔基; R 2是氢,卤素,氰基,烷基,卤代烷基,烯基,炔基,环烷基,烷氧基,烷氧基烷基和烷硫基烷基,其中R 1和/或R 2可以根据描述代替; R 3是卤素,氰基,NR B,B,羟基,巯基,烷基,卤代烷基,环烷基,烷氧基,烷硫基,环烷氧基,环烷硫基 ,羧基,甲酰基,烷基羰基,烷氧基羰基,烯氧基羰基,炔氧基羰基,苯基,苯氧基,苯硫基,苄氧基,苄硫基,烷基-S(O) A是N和CR R x是氢或R 3中提到的基团之一; 制备这些化合物的方法和中间体,包含它们的组合物及其用于控制​​植物病原性有害真菌的用途。