2-Substituted 7-Aminoazolopyrimidines, Processes For Their Preparation And Their Use For Controlling Harmful Fungi, And Compositions Comprising These Compounds
    1.
    发明申请
    2-Substituted 7-Aminoazolopyrimidines, Processes For Their Preparation And Their Use For Controlling Harmful Fungi, And Compositions Comprising These Compounds 审中-公开
    2-取代的7-氨基偶氮嘧啶,其制备方法及其用于控制​​有害真菌和包含这些化合物的组合物

    公开(公告)号:US20080139581A1

    公开(公告)日:2008-06-12

    申请号:US11885536

    申请日:2006-03-02

    IPC分类号: A01N43/90 A01P3/00 C07D487/04

    CPC分类号: C07D487/04

    摘要: 2-Substituted 7-aminoazolopyrimidines of the formula I in which the substituents are as defined below: R1 is hydrogen, halogen, cyano, alkyl, haloalkyl, alkenyl, alkynyl, cycloalkyl, alkoxy, alkoxyalkyl, benzyloxyalkyl, alkoxyalkenyl or alkoxyalkynyl; R2 is hydrogen, halogen, cyano, alkyl, haloalkyl, alkenyl, alkynyl, cycloalkyl, alkoxy, alkoxyalkyl and alkylthioalkyl, where the carbon chains in R1 and/or R2 may be substituted according to the description; R3 is halogen, cyano, NRARB, hydroxyl, mercapto, alkyl, haloalkyl, cycloalkyl, alkoxy, alkylthio, cycloalkoxy, cycloalkylthio, carboxyl, formyl, alkylcarbonyl, alkoxycarbonyl, alkenyloxycarbonyl, alkynyloxycarbonyl, phenyl, phenoxy, phenylthio, benzyloxy, benzylthio, alkyl-S(O)m—; A is N and CRx; Rx is hydrogen or one of the groups mentioned under R3; processes and intermediates for preparing these compounds, compositions comprising them and their use for controlling phytopathogenic harmful fungi.

    摘要翻译: 2-取代的式I的7-氨基偶氮嘧啶,其中取代基如下:R 1是氢,卤素,氰基,烷基,卤代烷基,烯基,炔基,环烷基,烷氧基,烷氧基烷基,苄氧基烷基 ,烷氧基烯基或烷氧基炔基; R 2是氢,卤素,氰基,烷基,卤代烷基,烯基,炔基,环烷基,烷氧基,烷氧基烷基和烷硫基烷基,其中R 1和/或R 2可以根据描述代替; R 3是卤素,氰基,NR B,B,羟基,巯基,烷基,卤代烷基,环烷基,烷氧基,烷硫基,环烷氧基,环烷硫基 ,羧基,甲酰基,烷基羰基,烷氧基羰基,烯氧基羰基,炔氧基羰基,苯基,苯氧基,苯硫基,苄氧基,苄硫基,烷基-S(O) A是N和CR R x是氢或R 3中提到的基团之一; 制备这些化合物的方法和中间体,包含它们的组合物及其用于控制​​植物病原性有害真菌的用途。

    Use Of 5-Alkyl-6-Phenylalkyl-7-Aminoazolopyrimidines, Novel Azolopyrimidines, Processes For Their Preparation And Compositions Comprising Them
    2.
    发明申请
    Use Of 5-Alkyl-6-Phenylalkyl-7-Aminoazolopyrimidines, Novel Azolopyrimidines, Processes For Their Preparation And Compositions Comprising Them 审中-公开
    5-烷基-6-苯基烷基-7-氨基偶氮嘧啶,新型二唑嘧啶,其制备方法及其组合物的应用

    公开(公告)号:US20080188494A1

    公开(公告)日:2008-08-07

    申请号:US11912335

    申请日:2006-04-24

    IPC分类号: A01N43/90 C07D487/04 A01P3/00

    CPC分类号: A01N43/90 C07D487/04

    摘要: The use of 5-alkyl-6-phenylalkyl-7-aminoazolopyrimidines of the formula I in which the variables are as defined below: Y is alkylene, alkenylene or alkynylene, optionally substituted by alkyl groups; R1 is halogen, cyano, nitro, hydroxyl, mercapto, alkyl, haloalkyl, alkenyl, cycloalkyl, cycloalkenyl, alkoxy, haloalkoxy, alkenyloxy, alkynyloxy, alkylthio, NRARB, alkylcarbonyl, phenyl, naphthyl, or a five- or six-membered saturated, partially unsaturated or aromatic heterocycle which contains one to four heteroatoms from the group consisting of O, N and S; RA, RB is hydrogen, alkyl or alkylcarbonyl; n is zero, 1, 2, 3 or 4; R2 is alkyl, alkenyl, cycloalkyl, alkoxyalkyl or alkylthioalkyl; R3 is hydrogen, halogen, cyano, NRARB, hydroxyl, mercapto, alkyl, haloalkyl, cycloalkyl, alkoxy, alkylthio, cycloalkoxy, cycloalkylthio, carboxyl, formyl, alkylcarbonyl, alkoxycarbonyl, alkenyloxycarbonyl, alkynyloxycarbonyl, phenyl, phenoxy, phenylthio, benzyloxy, benzylthio, alkyl-S(O)m—; m is 0, 1 or 2; A is N or C—Ra; Ra is hydrogen or alkyl; where the carbon atoms in Y, R1, R2, R3 and Ra may be substituted according to the description; for controlling phytopathogenic harmful fungi; novel 5-alkyl-6-phenylalkyl-7-amino-azolopyrimidines, processes for their preparation and compositions comprising them.

    摘要翻译: 使用式I的5-烷基-6-苯基烷基-7-氨基偶氮嘧啶,其中变量如下所定义:Y是任选被烷基取代的亚烷基,亚烯基或亚炔基; R 1是卤素,氰基,硝基,羟基,巯基,烷基,卤代烷基,烯基,环烷基,环烯基,烷氧基,卤代烷氧基,烯氧基,炔氧基,烷硫基,NR 或含有一至四个由O,N和S组成的组的杂原子的五元或六元饱和的部分不饱和或芳族杂环; R A,B B是氢,烷基或烷基羰基; n为零,1,2,3或4; R 2是烷基,烯基,环烷基,烷氧基烷基或烷硫基烷基; R 3是氢,卤素,氰基,NR B,B,羟基,巯基,烷基,卤代烷基,环烷基,烷氧基,烷硫基,环烷氧基 烷氧基羰基,烷氧羰基,烷氧基羰基,苯氧基,苯硫基,苄氧基,苄硫基,烷基-S(O)m - m为0,1或2; A是N或C-R a a R a是氢或烷基; 其中Y,R 1,R 2,R 3和R a中的碳原子可以根据 描述; 用于控制植物病原性有害真菌; 新的5-烷基-6-苯基烷基-7-氨基 - 偶氮嘧啶,其制备方法和包含它们的组合物。