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公开(公告)号：US20090182058A1
公开(公告)日：2009-07-16
申请号：US12087790
申请日：2007-01-15
IPC分类号： A61K31/12 , C07C49/255 , A61P35/00 , A61P37/00
CPC分类号： C07C49/835 , C07C45/74 , C07C49/84 , C07C225/22
摘要： The present invention relates to novel chalcone derivatives of formula (I): wherein X, Y, Z, W, RI, R2, R3, R4 and R5 are as defined, said derivatives having antimitotic activity, as well as to pharmaceutical compositions containing such compounds and to their use for making drugs.
摘要翻译： 本发明涉及式（I）的新型查耳酮衍生物：其中X，Y，Z，W，R 1，R 2，R 3，R 4和R 5如上所定义，所述衍生物具有抗有丝分裂活性， 化合物及其用于制造药物的用途。
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2.发明授权Para-coumaric acid or para-hydroxycinnamic acid derivatives and their use in cosmetic or dermatological compositions 有权对香豆酸或对羟基肉桂酸衍生物及其在化妆品或皮肤病学组合物中的用途公开(公告)号：US08481593B2
公开(公告)日：2013-07-09
申请号：US13152718
申请日：2011-06-03
IPC分类号： A61K31/216 , A61K31/165 , C07C69/76 , C07C233/00
CPC分类号： A61K8/55 , A61K8/37 , A61K8/375 , A61K8/42 , A61K8/463 , A61K2800/782 , A61Q1/06 , A61Q1/10 , A61Q5/02 , A61Q17/00 , A61Q19/00 , A61Q19/02 , A61Q19/10
摘要： The invention relates to the use of para-coumaric acid or para-hydroxycinnamic acid derivatives in cosmetic or dermatological compositions, specifically to the use of at least one compound derived from para-coumaric acid having a general formula (I) below: in which, especially, Z represents an oxygen or an —NH— group; X and Y are identical and each represent a CH or CH2 group, as an active principle with depigmenting, free-radical-scavenging and/or antiinflammatory activity. The invention also relates to the use of the above compounds for cosmetic care or for the preparation of a pharmaceutical composition, especially for depigmenting an area of skin, having antiradical and/or antiinflammatory activity.
摘要翻译： 本发明涉及对香草酸或对羟基肉桂酸衍生物在化妆品或皮肤病学组合物中的用途，具体涉及使用至少一种衍生自下列通式（I）的对 - 香豆酸的化合物：其中， 特别地，Z表示氧或-NH-基团; X和Y是相同的，并且各自表示CH或CH 2基团，作为具有脱色素，自由基清除和/或抗炎活性的活性成分。 本发明还涉及上述化合物用于化妆品护理或制备药物组合物，特别是用于脱色皮肤区域的具有抗原和/或抗炎活性的用途。
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3.发明申请Para-coumaric acid or para-hydroxycinnamic acid derivatives and their use in cosmetic or dermatological compositions 审中-公开对香豆酸或对羟基肉桂酸衍生物及其在化妆品或皮肤病学组合物中的用途公开(公告)号：US20070183996A1
公开(公告)日：2007-08-09
申请号：US11594440
申请日：2006-11-08
IPC分类号： A61K31/21 , A61K31/216 , A61Q19/02
CPC分类号： A61K8/55 , A61K8/37 , A61K8/375 , A61K8/42 , A61K8/463 , A61K2800/782 , A61Q1/06 , A61Q1/10 , A61Q5/02 , A61Q17/00 , A61Q19/00 , A61Q19/02 , A61Q19/10
摘要： The invention relates to the use of para-coumaric acid or para-hydroxycinnamic acid derivatives in cosmetic or dermatological compositions, specifically to the use of at least one compound derived from para-coumaric acid having a general formula (I) below: in which, especially, Z represents an oxygen or an —NH— group; X and Y are identical and each represent a CH or CH2 group, as an active principle with depigmenting, free-radical-scavenging and/or antiinflammatory activity. The invention also relates to the use of the above compounds for cosmetic care or for the preparation of a pharmaceutical composition, especially for depigmenting an area of skin, having antiradical and/or antiinflammatory activity.
摘要翻译： 本发明涉及对香草酸或对羟基肉桂酸衍生物在化妆品或皮肤病学组合物中的用途，具体涉及使用至少一种衍生自下列通式（I）的对 - 香豆酸的化合物：其中， 特别地，Z表示氧或-NH-基团; X和Y是相同的，并且各自表示CH或CH 2 CO 2基团，作为具有脱色素，自由基清除和/或抗炎活性的活性成分。 本发明还涉及上述化合物用于化妆品护理或制备药物组合物，特别是用于脱色皮肤区域的具有抗原和/或抗炎活性的用途。
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4.发明申请Para-Coumaric Acid or Para-Hydroxycinnamic Acid Derivatives and Their Use in Cosmetic or Dermatological Compositions 有权对 - 香豆酸或对羟基肉桂酸衍生物及其在化妆品或皮肤病学组合物中的应用公开(公告)号：US20110237551A1
公开(公告)日：2011-09-29
申请号：US13152718
申请日：2011-06-03
IPC分类号： A61K31/6615 , C07C69/734 , A61K31/216 , A61K8/37 , C07C233/29 , A61K31/165 , A61K8/42 , C07F9/12 , A61K8/55 , C07C305/24 , A61K31/255 , A61K8/46 , A61Q19/00 , A61P17/00
CPC分类号： A61K8/55 , A61K8/37 , A61K8/375 , A61K8/42 , A61K8/463 , A61K2800/782 , A61Q1/06 , A61Q1/10 , A61Q5/02 , A61Q17/00 , A61Q19/00 , A61Q19/02 , A61Q19/10
摘要： The invention relates to the use of para-coumaric acid or para-hydroxycinnamic acid derivatives in cosmetic or dermatological compositions, specifically to the use of at least one compound derived from para-coumaric acid having a general formula (I) below: in which, especially, Z represents an oxygen or an —NH— group; X and Y are identical and each represent a CH or CH2 group, as an active principle with depigmenting, free-radical-scavenging and/or antiinflammatory is activity.The invention also relates to the use of the above compounds for cosmetic care or for the preparation of a pharmaceutical composition, especially for depigmenting an area of skin, having antiradical and/or antiinflammatory activity.
摘要翻译： 本发明涉及对香草酸或对羟基肉桂酸衍生物在化妆品或皮肤病学组合物中的用途，具体涉及使用至少一种衍生自下列通式（I）的对 - 香豆酸的化合物：其中， 特别地，Z表示氧或-NH-基团; X和Y是相同的，并且各自表示CH或CH 2基团，作为具有脱色素，自由基清除和/或抗炎活性的活性成分。 本发明还涉及上述化合物用于化妆品护理或制备药物组合物，特别是用于脱色皮肤区域的具有抗原和/或抗炎活性的用途。
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5.发明申请Method of cosmetic depigmentation care by applying at least one aurone 审中-公开应用至少一种of of的化妆品色素沉着护理方法公开(公告)号：US20060228313A1
公开(公告)日：2006-10-12
申请号：US11127594
申请日：2005-05-12
CPC分类号： C07D307/83 , A61K8/35 , A61K8/49 , A61K8/4973 , A61Q5/02 , A61Q19/02 , A61Q19/10 , C07D405/06 , C07D407/06 , C07D409/06
摘要： at least one aurone or a natural or synthetic derivative of aurone, or an analogue of aurone, in which the independent phenyl ring can be substituted by a heterocycle of pyrrole, imidazole, triazole, pyridine, furan, or thiophene type, is disclosed as a cosmetic agent, or as an active substance, for the manufacture either of a cosmetic composition, or of a pharmaceutical composition, notably a dermatological composition, having a melanogenesis-inhibiting activity or a depigmenting activity, or an anti-tyrosinase activity.
摘要翻译： 公开了至少一种鸢尾醇或天然或合成的鸢尾醇衍生物，或其中独立苯环可以被吡咯，咪唑，三唑，吡啶，呋喃或噻吩类型的杂环取代的噢an的类似物。 化妆品或作为活性物质，用于制造具有黑素生成抑制活性或脱色素活性或抗酪氨酸酶活性的化妆品组合物或药物组合物，特别是皮肤病学组合物。
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公开(公告)号：US06471973B2
公开(公告)日：2002-10-29
申请号：US09828986
申请日：2001-04-10
IPC分类号： A61K900
CPC分类号： A61K8/498 , A61Q1/06 , A61Q5/02 , A61Q19/06 , A61Q19/08 , A61Q19/10 , C07D311/30 , C07D311/32 , C07H17/07 , Y10S514/844 , Y10S514/886 , Y10S514/887 , Y10S514/969
摘要： The invention relates to a flavonoid ester. This flavonoid ester results from the reaction product of at least one flavonoid selected from the group consisting of a flavonoid with a ketone group in the 4-position, a salt, ester or ether of such a flavonoid, and a C-heteroside and/or O-heteroside derivative of such a flavonoid, with the proviso that this flavonoid contains at least one free alcohol group, with an organic monoacid having from 3 to 30 carbon atoms. These flavonoid esters constitute useful active principles for the manufacture of cosmetic, dermopharmaceutical, pharmaceutical, dietetic or agri-foodstuff compositions.
摘要翻译： 本发明涉及类黄酮酯。 该类黄酮酯是由选自4-位的类黄酮与酮基的至少一种类黄酮，这种类黄酮的盐，酯或醚，以及C-杂苷和/或 这种类黄酮的O-杂苷衍生物，条件是该类黄酮含有至少一个游离醇基，具有3至30个碳原子的有机一元酸。 这些类黄酮酯构成用于制造化妆品，皮肤药物，药物，饮食或农产品组合物的有用的活性成分。
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公开(公告)号：US06235294B1
公开(公告)日：2001-05-22
申请号：US09113158
申请日：1998-07-10
IPC分类号： A61K600
CPC分类号： A61K8/498 , A61Q1/06 , A61Q5/02 , A61Q19/06 , A61Q19/08 , A61Q19/10 , C07D311/30 , C07D311/32 , C07H17/07 , Y10S514/844 , Y10S514/886 , Y10S514/887 , Y10S514/969
摘要： The invention relates to a flavonoid ester. This flavonoid ester results from the reaction product of at least one flavonoid selected from the group consisting of a flavonoid with a ketone group in the 4-position, a salt, ester or ether of such a flavonoid, and a C-heteroside and/or O-heteroside derivative of such a flavonoid, with the proviso that this flavonoid contains at least one free alcohol group, with an organic monoacid having from 3 to 30 carbon atoms. These flavonoid esters constitute useful active principles for the manufacture of cosmetic, dermopharmaceutical, pharmaceutical, dietetic or agri-foodstuff compositions.
摘要翻译： 本发明涉及类黄酮酯。 该类黄酮酯是由选自4-位的类黄酮与酮基的至少一种类黄酮，这种类黄酮的盐，酯或醚，以及C-杂苷和/或 这种类黄酮的O-杂苷衍生物，条件是该类黄酮含有至少一个游离醇基，具有3至30个碳原子的有机一元酸。 这些类黄酮酯构成用于制造化妆品，皮肤药物，药物，饮食或农产品组合物的有用的活性成分。
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