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公开(公告)号:US07855291B2
公开(公告)日:2010-12-21
申请号:US11647517
申请日:2006-12-28
申请人: Hugh Alfred Burgoon, Jr. , Ramanaiah C. Kanamarlapudi , Iain Fraser Pickersgill , Zhi-Cai Shi , Wenxue Wu , Haiming Zhang
发明人: Hugh Alfred Burgoon, Jr. , Ramanaiah C. Kanamarlapudi , Iain Fraser Pickersgill , Zhi-Cai Shi , Wenxue Wu , Haiming Zhang
IPC分类号: C07D239/34 , C07D403/12 , A61K31/506 , A61K31/505 , A61P9/02
CPC分类号: A61K31/505 , C07D239/47
摘要: Intermediates and synthetic processes for the preparation of substituted phenylalanine-based compounds (e.g., of Formula I) are disclosed:
摘要翻译: 公开了用于制备取代的苯丙氨酸类化合物(例如式I)的中间体和合成方法:
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2.Methods of preparing 4-phenyl-6-(2,2,2-trifluoro-1-phenylethoxy)pyrimidine-based compounds 有权
标题翻译: 制备4-苯基-6-(2,2,2-三氟-1-苯基乙氧基)嘧啶类化合物的方法公开(公告)号:US08575362B2
公开(公告)日:2013-11-05
申请号:US13160678
申请日:2011-06-15
申请人: Mark S. Bednarz , Hugh Alfred Burgoon, Jr. , Shinya Iimura , Ramanaiah C. Kanamarlapudi , Qiuling Song , Wenxue Wu , Jie Yan , Haiming Zhang
发明人: Mark S. Bednarz , Hugh Alfred Burgoon, Jr. , Shinya Iimura , Ramanaiah C. Kanamarlapudi , Qiuling Song , Wenxue Wu , Jie Yan , Haiming Zhang
IPC分类号: C07D231/12
CPC分类号: C07D403/12 , C07D231/12
摘要: Methods useful for preparing compounds of formula I: and salts thereof are disclosed. Also disclosed are intermediates useful in the preparation of such compounds.
摘要翻译: 公开了可用于制备式I化合物及其盐的方法。 还公开了可用于制备这些化合物的中间体。
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3.METHODS OF PREPARING 4-PHENYL-6-(2,2,2-TRIFLUORO-1-PHENYLETHOXY)PYRIMIDINE-BASED COMPOUNDS 有权
标题翻译: 制备4-苯基-6-(2,2,2-三氟-1-苯基乙基)吡啶基化合物的方法公开(公告)号:US20110301349A1
公开(公告)日:2011-12-08
申请号:US13160678
申请日:2011-06-15
申请人: Mark S. Bednarz , Hugh Alfred Burgoon, JR. , Shinya Iimura , Ramanaiah C. Kanamarlapudi , Qiuling Song , Wenxue Wu , Jie Yan , Haiming Zhang
发明人: Mark S. Bednarz , Hugh Alfred Burgoon, JR. , Shinya Iimura , Ramanaiah C. Kanamarlapudi , Qiuling Song , Wenxue Wu , Jie Yan , Haiming Zhang
IPC分类号: C07D239/42 , C07D231/12
CPC分类号: C07D403/12 , C07D231/12
摘要: Methods useful for preparing compounds of formula I: and salts thereof are disclosed. Also disclosed are intermediates useful in the preparation of such compounds.
摘要翻译: 公开了可用于制备式I化合物及其盐的方法。 还公开了可用于制备这些化合物的中间体。
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公开(公告)号:US07968729B2
公开(公告)日:2011-06-28
申请号:US12732311
申请日:2010-03-26
申请人: Mark S. Bednarz , Hugh Alfred Burgoon, Jr. , Shinya Iimura , Ramanaiah C. Kanamarlapudi , Qiuling Song , Wenxue Wu , Jie Yan , Haiming Zhang
发明人: Mark S. Bednarz , Hugh Alfred Burgoon, Jr. , Shinya Iimura , Ramanaiah C. Kanamarlapudi , Qiuling Song , Wenxue Wu , Jie Yan , Haiming Zhang
IPC分类号: C07D231/10
CPC分类号: C07D403/12 , C07D231/12
摘要: Methods useful for preparing compounds of formula I: and salts thereof are disclosed. Also disclosed are intermediates useful in the preparation of such compounds.
摘要翻译: 公开了可用于制备式I化合物及其盐的方法。 还公开了可用于制备这些化合物的中间体。
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5.METHODS OF PREPARING 4-PHENYL-6-(2,2,2-TRIFLUORO-1-PHENYLETHOXY)PYRIMIDINE-BASED COMPOUNDS 审中-公开
标题翻译: 制备4-苯基-6-(2,2,2-三氟-1-苯基乙基)吡啶基化合物的方法公开(公告)号:US20090062540A1
公开(公告)日:2009-03-05
申请号:US12196341
申请日:2008-08-22
申请人: Mark S. Bednarz , Hugh Alfred Burgoon, JR. , Shinya Iimura , Ramanaiah C. Kanamarlapudi , Qiuling Song , Wenxue Wu , Jie Yan , Haiming Zhang
发明人: Mark S. Bednarz , Hugh Alfred Burgoon, JR. , Shinya Iimura , Ramanaiah C. Kanamarlapudi , Qiuling Song , Wenxue Wu , Jie Yan , Haiming Zhang
IPC分类号: C07D403/12 , C07D231/12
CPC分类号: C07D403/12 , C07D231/12
摘要: Methods useful for preparing compounds of formula I: and salts thereof are disclosed. Also disclosed are intermediates useful in the preparation of such compounds.
摘要翻译: 公开了可用于制备式I化合物及其盐的方法。 还公开了可用于制备这些化合物的中间体。
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公开(公告)号:US20090048280A1
公开(公告)日:2009-02-19
申请号:US11647517
申请日:2006-12-28
申请人: Hugh Alfred Burgoon, JR. , Ramanaiah C. Kanamarlapudi , Iain Fraser Pickersgill , Zhi-Cai Shi , Wenxue Wu , Haiming Zhang
发明人: Hugh Alfred Burgoon, JR. , Ramanaiah C. Kanamarlapudi , Iain Fraser Pickersgill , Zhi-Cai Shi , Wenxue Wu , Haiming Zhang
IPC分类号: A61K31/513 , C07D239/46
CPC分类号: A61K31/505 , C07D239/47
摘要: Intermediates and synthetic processes for the preparation of substituted phenylalanine-based compounds (e.g., of Formula I) are disclosed:
摘要翻译: 公开了用于制备取代的苯丙氨酸类化合物(例如式I)的中间体和合成方法:
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公开(公告)号:US07919618B2
公开(公告)日:2011-04-05
申请号:US11832738
申请日:2007-08-02
IPC分类号: C07D401/04 , C07D401/14 , C07D403/04 , C07D403/14
CPC分类号: C07D401/04
摘要: Novel methods of synthesizing piperazines, piperidines and related compounds are disclosed, as are compounds useful for their preparation.
摘要翻译: 公开了合成哌嗪,哌啶和相关化合物的新方法,以及可用于其制备的化合物。
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公开(公告)号:US20100240906A1
公开(公告)日:2010-09-23
申请号:US12732311
申请日:2010-03-26
申请人: Mark S. Bednarz , Hugh Alfred Burgoon, JR. , Shinya Iimura , Ramanaiah C. Kanamarlapudi , Qiuling Song , Wenxue Wu , Jie Yan , Haiming Zhang
发明人: Mark S. Bednarz , Hugh Alfred Burgoon, JR. , Shinya Iimura , Ramanaiah C. Kanamarlapudi , Qiuling Song , Wenxue Wu , Jie Yan , Haiming Zhang
IPC分类号: C07D233/60
CPC分类号: C07D403/12 , C07D231/12
摘要: Methods useful for preparing compounds of formula I: and salts thereof are disclosed. Also disclosed are intermediates useful in the preparation of such compounds.
摘要翻译: 公开了可用于制备式I化合物及其盐的方法。 还公开了可用于制备这些化合物的中间体。
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