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1.BIARYL HETEROCYCLIC COMPOUNDS AND METHODS OF MAKING AND USING THE SAME 有权
Title translation: 二元杂环化合物及其制备和使用方法公开(公告)号:US20090118502A1
公开(公告)日:2009-05-07
申请号:US12275941
申请日:2008-11-21
Applicant: Jiacheng Zhou , Ashoke Bhattacharjee , Shili Chen , Yi Chen , Jay J. Farmer , Joel A. Goldberg , Roger Hanselmann , Rongliang Lou , Alia Orbin , Adegboyega K. Oyelere , Josseph M. Salvino , Dane M. Springer , Jennifer Tran , Deping Wang , Yusheng Wu
Inventor: Jiacheng Zhou , Ashoke Bhattacharjee , Shili Chen , Yi Chen , Jay J. Farmer , Joel A. Goldberg , Roger Hanselmann , Rongliang Lou , Alia Orbin , Adegboyega K. Oyelere , Josseph M. Salvino , Dane M. Springer , Jennifer Tran , Deping Wang , Yusheng Wu
IPC: C07D413/02 , C07D401/02
CPC classification number: C07D487/04 , C07D263/20 , C07D263/24 , C07D263/26 , C07D263/32 , C07D413/10 , C07D413/12 , C07D413/14 , C07D417/10 , C07D417/12 , C07D417/14 , C07D453/02 , C07D471/04 , C07D473/00 , C07D473/34
Abstract: The present invention relates generally to the field of anti-infective, anti-proliferative, anti-inflammatory, and prokinetic agents. More particularly, the invention relates to a family of compounds having both a biaryl moiety and at least one heterocylic moiety that are useful as such agents.
Abstract translation: 本发明一般涉及抗感染,抗增殖,抗炎和促动力的领域。 更具体地,本发明涉及具有联芳基部分和至少一个可用作这种试剂的杂环部分的化合物族。
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公开(公告)号:US20060264426A1
公开(公告)日:2006-11-23
申请号:US11486769
申请日:2006-07-14
Applicant: Jiacheng Zhou , Ashoke Bhattacharjee , Shili Chen , Yi Chen , Jay Farmer , Joel Goldberg , Roger Hanselmann , Rongliang Lou , Alia Orbin , Adegboyega Oyelere , Joseph Salvino , Dane Springer , Jennifer Tran , Deping Wang , Yusheng Wu
Inventor: Jiacheng Zhou , Ashoke Bhattacharjee , Shili Chen , Yi Chen , Jay Farmer , Joel Goldberg , Roger Hanselmann , Rongliang Lou , Alia Orbin , Adegboyega Oyelere , Joseph Salvino , Dane Springer , Jennifer Tran , Deping Wang , Yusheng Wu
IPC: A61K31/541 , A61K31/5377 , A61K31/52 , A61K31/498 , A61K31/496 , A61K31/454 , A61K31/4709 , A61K31/422 , C07D473/02 , C07D417/02 , C07D403/02
CPC classification number: C07D487/04 , C07D263/20 , C07D263/24 , C07D263/26 , C07D263/32 , C07D413/10 , C07D413/12 , C07D413/14 , C07D417/10 , C07D417/12 , C07D417/14 , C07D453/02 , C07D471/04 , C07D473/00 , C07D473/34
Abstract: The present invention relates generally to the field of anti-infective, anti-proliferative, anti-inflammatory, and prokinetic agents. More particularly, the invention relates to a family of compounds having both a biaryl moiety and at least one heterocylic moiety that are useful as such agents.
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公开(公告)号:US08497378B2
公开(公告)日:2013-07-30
申请号:US13120278
申请日:2009-09-23
Applicant: Roger Hanselmann , Maxwell M. Reeve , Graham Johnson
Inventor: Roger Hanselmann , Maxwell M. Reeve , Graham Johnson
IPC: C07D215/38
CPC classification number: C07D401/14
Abstract: The present invention relates to the field of synthesizing anti-infective compounds. More particularly, the invention relates to synthesizing a family of quinolone compounds useful as anti-infective agents. The invention includes a process for preparing a quinolone compound wherein less than about 0.40% of dimeric impurity of the quinolone is produced.
Abstract translation: 本发明涉及抗感染化合物的合成领域。 更具体地,本发明涉及合成可用作抗感染剂的喹诺酮化合物家族。 本发明包括一种喹诺酮化合物的制备方法,其中产生小于约0.40%的喹诺酮二聚体杂质。
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4.Biaryl Heterocyclic Compounds And Methods Of Making And Using The Same 审中-公开
Title translation: 二芳基杂环化合物及其制备和使用方法公开(公告)号:US20120010200A1
公开(公告)日:2012-01-12
申请号:US13240297
申请日:2011-09-22
Applicant: Jiacheng Zhou , Ashoke Bhattacharjee , Shili Chen , Yi Chen , Jay J. Farmer , Joel A. Goldberg , Roger Hanselmann , Rongliang Lou , Alia Orbin , Adegboyega K. Oyelere , Joseph M. Salvino , Dane M. Springer , Jennifer Tran , Deping Wang , Yusheng Wu
Inventor: Jiacheng Zhou , Ashoke Bhattacharjee , Shili Chen , Yi Chen , Jay J. Farmer , Joel A. Goldberg , Roger Hanselmann , Rongliang Lou , Alia Orbin , Adegboyega K. Oyelere , Joseph M. Salvino , Dane M. Springer , Jennifer Tran , Deping Wang , Yusheng Wu
IPC: A61K31/541 , C07D413/10 , C07D271/06 , C07D471/04 , C07D279/10 , A61K31/422 , A61K31/497 , A61K31/4245 , A61K31/519 , A61K31/5377 , A61P31/04 , A61P31/12 , A61P33/00 , A61P31/10 , A61P1/00 , A61P35/00 , C07D263/22
CPC classification number: C07D487/04 , C07D263/20 , C07D263/24 , C07D263/26 , C07D263/32 , C07D413/10 , C07D413/12 , C07D413/14 , C07D417/10 , C07D417/12 , C07D417/14 , C07D453/02 , C07D471/04 , C07D473/00 , C07D473/34
Abstract: The present invention relates generally to the field of anti-infective, anti-proliferative, anti-inflammatory, and prokinetic agents. More particularly, the invention relates to a family of compounds having both a biaryl moiety and at least one heterocylic moiety that are useful as such agents.
Abstract translation: 本发明一般涉及抗感染,抗增殖,抗炎和促动力的领域。 更具体地,本发明涉及具有联芳基部分和至少一个可用作这种试剂的杂环部分的化合物族。
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公开(公告)号:US20100234615A1
公开(公告)日:2010-09-16
申请号:US11921838
申请日:2006-06-08
Applicant: Shili Chen , Rongliang Lou , Yusheng Wu , Jiacheng Zhou , Roger Hanselmann
Inventor: Shili Chen , Rongliang Lou , Yusheng Wu , Jiacheng Zhou , Roger Hanselmann
IPC: C07D403/12
CPC classification number: C07D249/04 , C07D413/06 , C07D413/12 , C07D413/14 , C07F7/0814
Abstract: The present invention relates to processes for the preparation of triazoles. These compounds are useful as anti-infective, anti-proliferative, anti-inflammatory, and prokinetic agents.
Abstract translation: 本发明涉及制备三唑的方法。 这些化合物可用作抗感染,抗增殖,抗炎和促动力。
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公开(公告)号:US20100022772A1
公开(公告)日:2010-01-28
申请号:US10566150
申请日:2004-07-28
Applicant: Yusheng Wu , Chen Shili , Yi Chen , Roger Hanselmann , Rongliang Lou , Jiacheng Zhou
Inventor: Yusheng Wu , Chen Shili , Yi Chen , Roger Hanselmann , Rongliang Lou , Jiacheng Zhou
IPC: C07D417/12 , C07D413/12 , C07D413/10 , C07D263/20 , C07D413/14
CPC classification number: C07D263/20 , C07D263/32 , C07D413/06 , C07D413/10 , C07D413/12 , C07D413/14 , C07D417/10 , C07D417/12 , C07D417/14 , C07D453/02 , C07D473/00 , C07D487/04
Abstract: The present invention relates to processes for the preparation of biaryl oxazolidinones. These compounds are useful as anti-infective, anti-proliferative, anti-inflammatory, and prokinetic agents.
Abstract translation: 本发明涉及制备联芳基恶唑烷酮的方法。 这些化合物可用作抗感染,抗增殖,抗炎和促动力。
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7.Biaryl heterocyclic compounds and methods of making and using the same 有权
Title translation: 二芳基杂环化合物及其制备和使用方法公开(公告)号:US20050203147A1
公开(公告)日:2005-09-15
申请号:US11118808
申请日:2005-04-29
Applicant: Jiacheng Zhou , Ashoke Bhattacharjee , Shili Chen , Yi Chen , Jay Farmer , Joel Goldberg , Roger Hanselmann , Rongliang Lou , Alia Orbin , Adegboyega Oyelere , Joseph Salvino , Dane Springer , Jennifer Tran , Deping Wang , Yusheng Wu
Inventor: Jiacheng Zhou , Ashoke Bhattacharjee , Shili Chen , Yi Chen , Jay Farmer , Joel Goldberg , Roger Hanselmann , Rongliang Lou , Alia Orbin , Adegboyega Oyelere , Joseph Salvino , Dane Springer , Jennifer Tran , Deping Wang , Yusheng Wu
IPC: A61K31/421 , A61K31/4439 , A61K31/497 , A61K31/501 , C07D255/02 , C07D257/04 , C07D263/20 , C07D263/32 , C07D263/38 , C07D403/10 , C07D413/02 , C07D413/10 , C07D413/12 , C07D413/14 , C07D417/10 , C07D417/12 , C07D417/14 , C07D453/02 , C07D473/00 , C07D487/04
CPC classification number: C07D487/04 , C07D263/20 , C07D263/24 , C07D263/26 , C07D263/32 , C07D413/10 , C07D413/12 , C07D413/14 , C07D417/10 , C07D417/12 , C07D417/14 , C07D453/02 , C07D471/04 , C07D473/00 , C07D473/34
Abstract: The present invention relates generally to the field of anti-infective, anti-proliferative, anti-inflammatory, and prokinetic agents. More particularly, the invention relates to a family of compounds having both a biaryl moiety and at least one heterocylic moiety that are useful as such agents.
Abstract translation: 本发明一般涉及抗感染,抗增殖,抗炎和促动力的领域。 更具体地,本发明涉及具有联芳基部分和至少一个可用作这种试剂的杂环部分的化合物族。
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公开(公告)号:US20050043317A1
公开(公告)日:2005-02-24
申请号:US10859476
申请日:2004-06-02
Applicant: Jiacheng Zhou , Ashoke Bhattacharjee , Shili Chen , Yi Chen , Jay Farmer , Joel Goldberg , Roger Hanselmann , Rongliang Lou , Alia Orbin , Adegboyega Oyelere , Joseph Salvino , Dane Springer , Jennifer Tran , Deping Wang , Yusheng Wu
Inventor: Jiacheng Zhou , Ashoke Bhattacharjee , Shili Chen , Yi Chen , Jay Farmer , Joel Goldberg , Roger Hanselmann , Rongliang Lou , Alia Orbin , Adegboyega Oyelere , Joseph Salvino , Dane Springer , Jennifer Tran , Deping Wang , Yusheng Wu
IPC: A61K31/421 , A61K31/4439 , A61K31/497 , A61K31/501 , C07D255/02 , C07D257/04 , C07D263/20 , C07D263/32 , C07D263/38 , C07D403/10 , C07D413/02 , C07D413/10 , C07D413/12 , C07D413/14 , C07D417/10 , C07D417/12 , C07D417/14 , C07D453/02 , C07D473/00 , C07D487/04
CPC classification number: C07D487/04 , C07D263/20 , C07D263/24 , C07D263/26 , C07D263/32 , C07D413/10 , C07D413/12 , C07D413/14 , C07D417/10 , C07D417/12 , C07D417/14 , C07D453/02 , C07D471/04 , C07D473/00 , C07D473/34
Abstract: The present invention relates generally to the field of anti-infective, anti-proliferative, anti-inflammatory, and prokinetic agents. More particularly, the invention relates to a family of compounds having both a biaryl moiety and at least one heterocylic moiety that are useful as such agents.
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公开(公告)号:US08895741B2
公开(公告)日:2014-11-25
申请号:US13618091
申请日:2012-09-14
Applicant: Yusheng Wu , Shili Chen , Yi Chen , Roger Hanselmann , Rongliang Lou , Jiacheng Zhou
Inventor: Yusheng Wu , Shili Chen , Yi Chen , Roger Hanselmann , Rongliang Lou , Jiacheng Zhou
IPC: C07D263/20 , C07D263/32 , C07D413/06 , C07D417/14 , C07D453/02 , C07D413/12 , C07D417/10 , C07D487/04 , C07D417/12 , C07D473/00 , C07D413/10 , C07D413/14
CPC classification number: C07D263/20 , C07D263/32 , C07D413/06 , C07D413/10 , C07D413/12 , C07D413/14 , C07D417/10 , C07D417/12 , C07D417/14 , C07D453/02 , C07D473/00 , C07D487/04
Abstract: The present invention relates to processes for the preparation of biaryl oxazolidinones. These compounds are useful as anti-infective, anti-proliferative, anti-inflammatory, and prokinetic agents.
Abstract translation: 本发明涉及制备联芳基恶唑烷酮的方法。 这些化合物可用作抗感染,抗增殖,抗炎和促动力。
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公开(公告)号:US08399660B2
公开(公告)日:2013-03-19
申请号:US11921838
申请日:2006-06-08
Applicant: Shili Chen , Rongliang Lou , Yusheng Wu , Jiacheng Zhou , Roger Hanselmann
Inventor: Shili Chen , Rongliang Lou , Yusheng Wu , Jiacheng Zhou , Roger Hanselmann
IPC: A61K31/541 , A61P25/24 , C07D413/10
CPC classification number: C07D249/04 , C07D413/06 , C07D413/12 , C07D413/14 , C07F7/0814
Abstract: The present invention relates to processes for the preparation of triazoles. These compounds are useful as anti-infective, anti-proliferative, anti-inflammatory, and prokinetic agents.
Abstract translation: 本发明涉及制备三唑的方法。 这些化合物可用作抗感染,抗增殖,抗炎和促动力。
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