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公开(公告)号：US20130005968A1
公开(公告)日：2013-01-03
申请号：US13615894
申请日：2012-09-14
Applicant: I. Fraser Pickersgill , John E. Bishop , Christoph Koellner , Jean-Marc Gomez , Achim Geiser , Robert Hett , Vince Ammoscato , Stephen Munk , Young Lo , Fang-Ting Chiu , Vithalanand R. Kulkarni
Inventor： I. Fraser Pickersgill , John E. Bishop , Christoph Koellner , Jean-Marc Gomez , Achim Geiser , Robert Hett , Vince Ammoscato , Stephen Munk , Young Lo , Fang-Ting Chiu , Vithalanand R. Kulkarni
IPC: C07F5/04
CPC classification number: C07K5/06191 , C07F5/025 , C07F5/04 , Y02P20/55
Abstract: The invention relates to the synthesis of boronic ester and acid compounds. More particularly, the invention provides improved synthetic processes for the large-scale production of boronic ester and acid compounds, including the peptide boronic acid proteasome inhibitor bortezomib.
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公开(公告)号：US08283467B2
公开(公告)日：2012-10-09
申请号：US12706063
申请日：2010-02-16
Applicant: Vince Ammoscato , John E. Bishop , Fang-Ting Chiu , Achim Geiser , Jean-Marc Gomez , Robert Hett , Christoph Koellner , Vithalanand R. Kulkarni , Young Lo , Stephen Munk , I. Fraser Pickersgill
Inventor： Vince Ammoscato , John E. Bishop , Fang-Ting Chiu , Achim Geiser , Jean-Marc Gomez , Robert Hett , Christoph Koellner , Vithalanand R. Kulkarni , Young Lo , Stephen Munk , I. Fraser Pickersgill
IPC: C07F5/02
CPC classification number: C07K5/06191 , C07F5/025 , C07F5/04 , Y02P20/55
Abstract: The invention relates to the synthesis of boronic ester and acid compounds. More particularly, the invention provides improved synthetic processes for the large-scale production of boronic ester and acid compounds, including the peptide boronic acid proteasome inhibitor bortezomib.
Abstract translation: 本发明涉及硼酸酯和酸化合物的合成。 更具体地，本发明提供了用于大规模生产硼酸酯和酸化合物的改进的合成方法，包括肽硼酸蛋白酶体抑制剂硼替佐米。
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公开(公告)号：US20100174072A1
公开(公告)日：2010-07-08
申请号：US12706063
申请日：2010-02-16
Applicant: I. Fraser Pickersgill , John E. Bishop , Christoph Koellner , Jean-Marc Gomez , Achim Geiser , Robert Hett , Vince Ammoscato , Stephen Munk , Young Lo , Fang-Ting Chiu , Vithalanand R. Kulkarni
Inventor： I. Fraser Pickersgill , John E. Bishop , Christoph Koellner , Jean-Marc Gomez , Achim Geiser , Robert Hett , Vince Ammoscato , Stephen Munk , Young Lo , Fang-Ting Chiu , Vithalanand R. Kulkarni
IPC: C07F5/04
CPC classification number: C07K5/06191 , C07F5/025 , C07F5/04 , Y02P20/55
Abstract: The invention relates to the synthesis of boronic ester and acid compounds. More particularly, the invention provides improved synthetic processes for the large-scale production of boronic ester and acid compounds, including the peptide boronic acid proteasome inhibitor bortezomib.
Abstract translation: 本发明涉及硼酸酯和酸化合物的合成。 更具体地，本发明提供了用于大规模生产硼酸酯和酸化合物的改进的合成方法，包括肽硼酸蛋白酶体抑制剂硼替佐米。
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公开(公告)号：US20050240047A1
公开(公告)日：2005-10-27
申请号：US11088667
申请日：2005-03-24
Applicant: I. Pickersgill , John Bishop , Christoph Koellner , Jean-Marc Gomez , Achim Geiser , Robert Hett , Vince Ammoscato , Stephen Munk , Young Lo , Fang-Ting Chiu , Vithalanand Kulkarni
Inventor： I. Pickersgill , John Bishop , Christoph Koellner , Jean-Marc Gomez , Achim Geiser , Robert Hett , Vince Ammoscato , Stephen Munk , Young Lo , Fang-Ting Chiu , Vithalanand Kulkarni
CPC classification number: C07K5/06191 , C07F5/025 , C07F5/04 , Y02P20/55
Abstract: The invention relates to the synthesis of boronic ester and acid compounds. More particularly, the invention provides improved synthetic processes for the large-scale production of boronic ester and acid compounds, including the peptide boronic acid proteasome inhibitor bortezomib.
Abstract translation: 本发明涉及硼酸酯和酸化合物的合成。 更具体地，本发明提供了用于大规模生产硼酸酯和酸化合物的改进的合成方法，包括肽硼酸蛋白酶体抑制剂硼替佐米。
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