公开(公告)号：US09365495B2

公开(公告)日：2016-06-14

申请号：US14365822

申请日：2012-12-20

Applicant: Maximilian Dochnahl ,  Michael Rack ,  Michael Keil ,  Bernd Wolf ,  Uwe Josef Vogelbacher ,  Joachim Gebhardt ,  Timo Frassetto ,  Volker Maywald

Inventor： Maximilian Dochnahl ,  Michael Rack ,  Michael Keil ,  Bernd Wolf ,  Uwe Josef Vogelbacher ,  Joachim Gebhardt ,  Timo Frassetto ,  Volker Maywald

IPC: C07C231/24 ,  C07D413/04 ,  C07C231/12 ,  C07C235/20 ,  C07D207/06 ,  C07D211/06 ,  C07D295/185 ,  C07C235/34 ,  C07D207/16 ,  C07D211/16

CPC classification number: C07C231/24 ,  C07C231/12 ,  C07C235/20 ,  C07C235/34 ,  C07D207/06 ,  C07D207/16 ,  C07D211/16 ,  C07D295/185 ,  C07D413/04

Abstract: The present invention relates to a process for manufacturing aryloxyacetamides of formula (I), by reacting haloacetamides of formula (II) with a phenol of formula (III); wherein the variables are defined according to the description, and aryloxyacetamides of formula (I).

Abstract translation: 本发明涉及通过使式（II）的卤代乙酰胺与式（III）的苯酚反应制备式（I）的芳氧基乙酰胺的方法; 其中所述变量根据描述定义，和式（I）的芳氧基乙酰胺。

公开(公告)号：US20110130286A1

公开(公告)日：2011-06-02

申请号：US13056320

申请日：2009-07-23

Applicant: Liliana Parra Rapado ,  Eike Hupe ,  Matthias Witschel ,  Thomas Seitz ,  Anja Simon ,  Robert Reinhard ,  Bernd Sievernich ,  Klaus Grossmann ,  Thomas Ehrhardt ,  Trevor William Newton ,  Frank Stelzer ,  Tao Qu ,  William Karl Moberg ,  Dschun Song ,  Michael Rack ,  Timo Frassetto ,  Klaus Kreuz ,  Julia Major

Inventor： Liliana Parra Rapado ,  Eike Hupe ,  Matthias Witschel ,  Thomas Seitz ,  Anja Simon ,  Robert Reinhard ,  Bernd Sievernich ,  Klaus Grossmann ,  Thomas Ehrhardt ,  Trevor William Newton ,  Frank Stelzer ,  Tao Qu ,  William Karl Moberg ,  Dschun Song ,  Michael Rack ,  Timo Frassetto ,  Klaus Kreuz ,  Julia Major

IPC: A01N57/16 ,  C07D401/06 ,  A01N43/60 ,  A01P13/00 ,  C07D401/14 ,  A01N43/84 ,  C07D413/14 ,  C07D491/08 ,  C07F9/145

CPC classification number: C07D401/06 ,  A01N43/60 ,  A01N43/78 ,  A01N43/80 ,  A01N43/82 ,  A01N43/84 ,  A01N43/90 ,  C07D403/06 ,  A01N33/18 ,  A01N43/54 ,  A01N2300/00

Abstract: Piperazine compounds of the formula I in which the variables are defined according to the description, their agriculturally suitable salts, processes and intermediates for preparing the piperazine compounds of the formula I, compositions comprising them and their use as herbicides, i.e. for controlling harmful plants, and also a method for controlling unwanted vegetation which comprises allowing a herbicidally effective amount of at least one piperazine compound of the formula I to act on plants, their seed and/or their habitat.

Abstract translation: 根据描述定义变量的哌嗪化合物，其农业上合适的盐，用于制备式I的哌嗪化合物的方法和中间体，包含它们的组合物及其作为除草剂的用途，即用于防治有害植物， 以及用于控制不想要的植物的方法，其包括允许除草有效量的至少一种式I的哌嗪化合物作用于植物，其种子和/或其栖息地。

公开(公告)号：US09062012B2

公开(公告)日：2015-06-23

申请号：US14365774

申请日：2012-12-20

Applicant: Bernd Wolf ,  Joachim Gebhardt ,  Uwe Josef Vogelbacher ,  Maximilian Dochnahl ,  Michael Rack ,  Michael Keil ,  Timo Frassetto ,  Volker Maywald

Inventor： Bernd Wolf ,  Joachim Gebhardt ,  Uwe Josef Vogelbacher ,  Maximilian Dochnahl ,  Michael Rack ,  Michael Keil ,  Timo Frassetto ,  Volker Maywald

IPC: C07D265/36 ,  C07D413/04

CPC classification number: C07D265/36 ,  C07D413/04

Abstract: The present invention relates to a process for manufacturing 4-substituted amino-benzoxazinones of formula (I), by reacting a NH-benzoxazinone of formula (II) with a compound of formula (III); wherein the variables are defined according to the description.

Abstract translation: 本发明涉及式（I）的4-取代氨基 - 苯并恶嗪酮的制备方法，其中式（II）的N-苯并恶嗪酮与式（III）的化合物反应; 其中根据描述定义变量。

公开(公告)号：US20110144336A1

公开(公告)日：2011-06-16

申请号：US13058677

申请日：2009-07-30

Applicant: Thomas Zierke ,  Eike Hupe ,  Michael Rack ,  Liliana Parra Rapado ,  Timo Frassetto

Inventor： Thomas Zierke ,  Eike Hupe ,  Michael Rack ,  Liliana Parra Rapado ,  Timo Frassetto

IPC: C07D241/08

CPC classification number: C07D241/08

Abstract: A process for preparing piperazinedione derivatives of the formula I in which R1 is hydrogen, alkyl, alkenyl, alkynyl and alkylcarbonyl, R2 is hydrogen, alkyl, alkenyl, C3-C4-alkynyl and C(═O)R11, R3, R4 are each hydrogen, alkyl and haloalkyl, where the groups may be substituted, which comprises reacting amines of the formula II H2N—R1  II in which R1 is hydrogen and alkyl which may optionally be substituted with N-acylated amino acid derivatives of the formula III in which X is halogen, Y is halogen, alkoxy or phenyloxy which may be substituted and R2, R3 and R4 are each as defined at the outset, under basic conditions in an aqueous solvent.

Abstract translation: 其中R 1是氢，烷基，烯基，炔基和烷基羰基，R 2是氢，烷基，烯基，C 3 -C 4炔基和C（= O）R 11，R 3，R 4各自是式I的哌嗪二酮衍生物的方法 氢，烷基和卤代烷基，其中基团可以被取代，其包括使式II的其中R 1是氢的式IIH 2 N-R 1 II的烷基和可以被式III的N-酰化的氨基酸衍生物任选取代的烷基，其中 X是卤素，Y是可以被取代的卤素，烷氧基或苯氧基，R2，R3和R4各自在碱性条件下在水性溶剂中首先定义。

公开(公告)号：US20110207609A1

公开(公告)日：2011-08-25

申请号：US13126658

申请日：2009-10-26

Applicant: Liliana Parra Rapado ,  Frank Stelzer ,  Matthias Witschel ,  Thomas Seitz ,  Trevor William Newton ,  Julia Major ,  Tao Qu ,  William Karl Moberg ,  Dschun Song ,  Michael Rack ,  Timo Frassetto ,  Anja Simon ,  Robert Reinhard ,  Bernd Sievernich ,  Klaus Grossmann ,  Thomas Ehrhardt ,  Klaus Kreuz

Inventor： Liliana Parra Rapado ,  Frank Stelzer ,  Matthias Witschel ,  Thomas Seitz ,  Trevor William Newton ,  Julia Major ,  Tao Qu ,  William Karl Moberg ,  Dschun Song ,  Michael Rack ,  Timo Frassetto ,  Anja Simon ,  Robert Reinhard ,  Bernd Sievernich ,  Klaus Grossmann ,  Thomas Ehrhardt ,  Klaus Kreuz

IPC: A01N43/60 ,  C07D409/06 ,  C07D413/14 ,  A01N43/84 ,  C07D403/06 ,  C07D413/06 ,  A01N43/80 ,  A01P13/00

CPC classification number: C07D241/08

Abstract: Piperazine compounds of the formula I in which the variables are defined according to the description, their agriculturally suitable salts, processes and intermediates for preparing the piperazines of the formula I, compositions comprising them and their use as herbicides, i.e. for controlling harmful plants, and also a method for controlling unwanted vegetation which comprises allowing a herbicidally effective amount of at least one piperazine compound of the formula I to act on plants, their seed and/or their habitat.

Abstract translation: 式I的哌嗪化合物，其中根据描述定义变量，其农业上合适的盐，用于制备式I的哌嗪的方法和中间体，包含它们的组合物及其作为除草剂的用途，即用于防治有害植物，以及 还包括控制不需要的植物的方法，其包括允许除草有效量的式I的至少一种哌嗪化合物作用于植物，其种子和/或其栖息地。

公开(公告)号：US20110183848A1

公开(公告)日：2011-07-28

申请号：US13121976

申请日：2009-09-29

Applicant: Liliana Parra Rapado ,  Frank Stelzer ,  Matthias Witschel ,  Thomas Seitz ,  Anja Simon ,  Robert Reinhard ,  Bernd Sievernich ,  Klaus Grossmann ,  Thomas Ehrhardt ,  Trevor Wlliam Newton ,  Julia Major ,  Tao Qu ,  William Karl Moberg ,  Dschun Song ,  Michael Rack ,  Timo Frassetto ,  Klaus Kreuz

Inventor： Liliana Parra Rapado ,  Frank Stelzer ,  Matthias Witschel ,  Thomas Seitz ,  Anja Simon ,  Robert Reinhard ,  Bernd Sievernich ,  Klaus Grossmann ,  Thomas Ehrhardt ,  Trevor Wlliam Newton ,  Julia Major ,  Tao Qu ,  William Karl Moberg ,  Dschun Song ,  Michael Rack ,  Timo Frassetto ,  Klaus Kreuz

IPC: A01N43/70 ,  C07D241/08 ,  A01N43/60 ,  A01P13/00 ,  C07D401/06 ,  A01N55/10 ,  C07F7/08

CPC classification number: C07D401/06 ,  C07D403/06

Abstract: Piperazine compounds of the formula I in which the variables are defined according to the description, their agriculturally suitable salts, processes and intermediates for preparing the piperazine compounds of the formula I, compositions comprising them and their use as herbicides, i.e. for controlling harmful plants, and also a method for controlling unwanted vegetation which comprises allowing a herbicidally effective amount of at least one piperazine compound of the formula I to act on plants, their seed and/or their habitat.

Abstract translation: 根据描述定义变量的哌嗪化合物，其农业上合适的盐，用于制备式I的哌嗪化合物的方法和中间体，包含它们的组合物及其作为除草剂的用途，即用于防治有害植物， 以及用于控制不想要的植物的方法，其包括允许除草有效量的至少一种式I的哌嗪化合物作用于植物，其种子和/或其栖息地。

公开(公告)号：US08921572B2

公开(公告)日：2014-12-30

申请号：US13511093

申请日：2009-11-26

Applicant: Timo Frassetto

Inventor： Timo Frassetto

IPC: C07D261/04

CPC classification number: C07D261/04

Abstract: A process for preparing 5,5-disubstituted 4,5-dihydroisoxazole-3-thiocarboxamidine salts of the formula (I), wherein 3-unsubstituted 4,5-dihydroisoxazoles are first reacted with a chlorinating or brominating reagent to give 3-halogenated 4,5-dihydroisoxazoles and the latter then react with thiourea to give the compounds of the formula (I).

Abstract translation: 制备式（I）的5,5-二取代的4,5-二氢异恶唑-3-硫代甲脒盐的方法，其中3-未取代的4,5-二氢异恶唑首先与氯化或溴化试剂反应，得到3-卤代4 ，5-二氢异恶唑，然后与硫脲反应，得到式（I）化合物。

公开(公告)号：US20140357861A1

公开(公告)日：2014-12-04

申请号：US14365829

申请日：2012-12-20

Applicant: Maximilian Dochnahl ,  Michael Rack ,  Michael Keil ,  Bernd Wolf ,  Uwe Josef Vogelbacher ,  Joachim Gebhardt ,  Timo Frassetto ,  Volker Maywald

Inventor： Maximilian Dochnahl ,  Michael Rack ,  Michael Keil ,  Bernd Wolf ,  Uwe Josef Vogelbacher ,  Joachim Gebhardt ,  Timo Frassetto ,  Volker Maywald

IPC: C07D265/36 ,  C07C231/12

CPC classification number: C07D265/36 ,  C07C231/12 ,  C07D413/04

Abstract: The present invention relates to a process for manufacturing a benzoxazinone of formula (I), by reacting a nitro compound of formula (II) with a reducing agent to obtain an amino compound of formula (III), and then reacting the amino compound of formula (III) with an acid; wherein the variables are defined according to the description, and benzoxazinone of formula (I).

Abstract translation: 本发明涉及式（I）的苯并恶嗪酮的制备方法，通式（II）的硝基化合物与还原剂反应得到式（III）的氨基化合物，然后使式 （III）与酸反应; 其中根据描述定义变量，和式（I）的苯并嗪酮。

公开(公告)号：US20120238760A1

公开(公告)日：2012-09-20

申请号：US13511090

申请日：2009-11-26

Applicant: Timo Frassetto

Inventor： Timo Frassetto

IPC: C07D261/04

CPC classification number: C07D261/04

Abstract: The present invention relates to a process for preparing 5,5-disubstituted 2-isoxazolines of the formula (I) where R1, R2 are each independently C1-C6-alkyl or C1-C4-haloalkyl; or R1 and R2 together form a C2-C5-alkanediyl chain which may be mono- to tetrasubstituted by C1-C4-alkyl and/or interrupted by oxygen or by optionally C1-C4-alkyl-substituted nitrogen.

Abstract translation: 本发明涉及制备式（I）的5,5-二取代的2-异恶唑啉的方法，其中R 1，R 2各自独立地为C 1 -C 6 - 烷基或C 1 -C 4 - 卤代烷基; 或者R 1和R 2一起形成C 2 -C 5链烷二基链，其可以被C 1 -C 4烷基单取代和四取代，和/或被中间或被任选被C 1 -C 4烷基取代的氮所隔开。

公开(公告)号：US09359312B2

公开(公告)日：2016-06-07

申请号：US14365829

申请日：2012-12-20

Applicant: Maximilian Dochnahl ,  Michael Rack ,  Michael Keil ,  Bernd Wolf ,  Uwe Josef Vogelbacher ,  Joachim Gebhardt ,  Timo Frassetto ,  Volker Maywald

Inventor： Maximilian Dochnahl ,  Michael Rack ,  Michael Keil ,  Bernd Wolf ,  Uwe Josef Vogelbacher ,  Joachim Gebhardt ,  Timo Frassetto ,  Volker Maywald

IPC: C07D265/36 ,  C07D413/04 ,  C07C231/12

CPC classification number: C07D265/36 ,  C07C231/12 ,  C07D413/04

Abstract: The present invention relates to a process for manufacturing a benzoxazinone of formula (I), by reacting a nitro compound of formula (II) with a reducing agent to obtain an amino compound of formula (III), and then reacting the amino compound of formula (III) with an acid; wherein the variables are defined according to the description, and benzoxazinone of formula (I).

Abstract translation: 本发明涉及式（I）的苯并恶嗪酮的制备方法，通式（II）的硝基化合物与还原剂反应得到式（III）的氨基化合物，然后使式 （III）与酸反应; 其中根据描述定义变量，和式（I）的苯并嗪酮。