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公开(公告)号:US07960310B2
公开(公告)日:2011-06-14
申请号:US12063869
申请日:2006-08-02
申请人: Anthony Cornelius O'Sullivan , Jürgen Harry Schaetzer , Christoph Lüthy , Alison Clare Elliott , Christopher John Mathews
发明人: Anthony Cornelius O'Sullivan , Jürgen Harry Schaetzer , Christoph Lüthy , Alison Clare Elliott , Christopher John Mathews
IPC分类号: A01N43/78
CPC分类号: A01N43/78 , C07D277/18 , C07D417/12
摘要: The use of a compound of formula (I) wherein X is (i), (ii) or (iii), formula (i), formula (ii), formula (iii) Y is O, S(O)m, NR3, CR5R6, CR5R6—CR7R8, O—CR7R8, S(O)m—CR7R8, NR3—CR7R8, CR5R6—O, CR5R6—S(O)m, CR5R6—NR3, SO2—NR3, NR3—SO2, NR3—O or O—NR3; m is 0, 1, or 2; the ring (T) formula (T) is a 5- or 6-membered aromatic or heteroaromatic ring; R1 to R10 are specified organic groups and n and is 0, 1, 2, 3 or 4; or salts or N-oxides thereof or compositions containing them in controlling insects, acarines, nematodes or molluscs. Novel compounds are also provided.
摘要翻译: 其中X为(i),(ii)或(iii),式(i),式(ii),式(iii)Y的式(I)化合物的使用为O,S(O)m,NR 3 ,CR5R6,CR5R6-CR7R8,O-CR7R8,S(O)m-CR7R8,NR3-CR7R8,CR5R6-O,CR5R6-S(O)m,CR5R6-NR3,SO2-NR3,NR3-SO2,NR3-O 或O-NR3; m为0,1或2; 环(T)式(T)是5或6元芳族或杂芳族环; R1至R10为指定的有机基团,n为0,1,2,3或4; 或其盐或N-氧化物或含有它们的组合物来控制昆虫,螨类,线虫或软体动物。 还提供了新的化合物。
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公开(公告)号:US20110218341A1
公开(公告)日:2011-09-08
申请号:US13105596
申请日:2011-05-11
申请人: Anthony Cornelius O'Sullivan , Jürgen Harry Schaetzer , Christoph Lüthy , Alison Clare Elliott , Christopher John Mathews
发明人: Anthony Cornelius O'Sullivan , Jürgen Harry Schaetzer , Christoph Lüthy , Alison Clare Elliott , Christopher John Mathews
IPC分类号: C07D277/18
CPC分类号: A01N43/78 , C07D277/18 , C07D417/12
摘要: The use of a compound of formula I wherein X is (i), (ii) or (iii) Y is O, S(O)m, NR3, CR5R6, CR5R6—CR7R8, O—CR7R8, S(O)m—CR7R8, NR3—CR7R8, CR5R6—O, CR5R6—S(O)m, CR5R6—NR3, SO2—NR3, NR3—SO2, NR3—O or O—NR3; m is 0, 1, or 2; the ring (T) is a 5- or 6-membered aromatic or heteroaromatic ring; R1 to R10 are specified organic groups and n and is 0, 1, 2, 3 or 4; or salts or N-oxides thereof or compositions containing them in controlling insects, acarines, nematodes or molluscs. Novel compounds are also provided.
摘要翻译: 其中X是(i),(ii)或(iii)Y的式I化合物是O,S(O)m,NR 3,CR 5 R 6,CR 5 R 6 -CR 7 R 8,O-CR 7 R 8,S(O) CR7R8,NR3-CR7R8,CR5R6-O,CR5R6-S(O)m,CR5R6-NR3,SO2-NR3,NR3-SO2,NR3-O或O-NR3; m为0,1或2; 环(T)是5或6元芳族或杂芳族环; R1至R10为指定的有机基团,n为0,1,2,3或4; 或其盐或N-氧化物或含有它们的组合物来控制昆虫,螨类,线虫或软体动物。 还提供了新的化合物。
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公开(公告)号:US20080300285A1
公开(公告)日:2008-12-04
申请号:US12063869
申请日:2006-08-02
申请人: Anthony Cornelius O'Sullivan , Jurgen Harry Schaetzer , Christophe Luthy , Alison Clare Elliott , Christopher John Mathews
发明人: Anthony Cornelius O'Sullivan , Jurgen Harry Schaetzer , Christophe Luthy , Alison Clare Elliott , Christopher John Mathews
IPC分类号: A01N43/78 , C07D417/12 , C07D277/18 , A01P9/00 , A01P7/04 , A01P7/02
CPC分类号: A01N43/78 , C07D277/18 , C07D417/12
摘要: The use of a compound of formula (I) wherein X is (i), (ii) or (iii), formula (i), formula (ii), formula (iii) Y is O, S(O)m, NR3, CR5R6, CR5R6—CR7R8, O—CR7R8, S(O)m—CR7R8, NR3—CR7R8, CR5R6—O, CR5R6—S(O)m, CR5R6—NR3, SO2—NR3, NR3—SO2, NR3—O or O—NR3; m is 0, 1, or 2; the ring (T) formula (T) is a 5- or 6-membered aromatic or heteroaromatic ring; R1 to R10 are specified organic groups and n and is 0, 1, 2, 3 or 4; or salts or N-oxides thereof or compositions containing them in controlling insects, acarines, nematodes or molluscs. Novel compounds are also provided.
摘要翻译: 其中X为(i),(ii)或(iii),式(i),式(ii),式(iii)Y的式(I)化合物的使用为O,S(O)m,NR 3 ,CR5R6,CR5R6-CR7R8,O-CR7R8,S(O)m-CR7R8,NR3-CR7R8,CR5R6-O,CR5R6-S(O)m,CR5R6-NR3,SO2-NR3,NR3-SO2,NR3-O 或O-NR3; m为0,1或2; 环(T)式(T)是5或6元芳族或杂芳族环; R1至R10为指定的有机基团,n为0,1,2,3或4; 或其盐或N-氧化物或含有它们的组合物来控制昆虫,螨类,线虫或软体动物。 还提供了新的化合物。
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公开(公告)号:US08455663B2
公开(公告)日:2013-06-04
申请号:US12677825
申请日:2008-09-09
IPC分类号: C07D233/22 , C07C255/13
CPC分类号: C07D233/16 , A01N43/50
摘要: The present invention relates to novel imidazoline derivatives and their use as insecticidal, acaricidal, molluscicidal and nematocidal agents. The invention also extends to insecticidal, acaricidal, molluscicidal and nematicidal compositions comprising such imidazoline derivatives, and to methods of using such derivatives and/or compositions to combat and control insect, acarine, mollusc and nematode pests. A compound of formula (I) and salts and N-oxides thereof, wherein: R1 is C1-10 alkyl; R2 is chloro, bromo or iodo; R3 is C2-5 alkyl, C1-5 haloalkyl, C1-6 hydroxyalkyl, C1-5alkoxy-(C1-3)-alkyl, di-(C1-5 alkoxy)-(C1-3)-alkyl, C1-5alkylthio-(C1-3)-alkyl; C1-5 alkylsulfinyl-(C1-3)alkyl; C2-5 alkenyl, C1-5 haloalkenyl, C2-5 alkinyl, C3-6 cycloalkyl, C3-6 cycloalkenyl, hydroxy, C1-5 alkoxy, C1-5haloalkoxy, C1-5alkylthio, C1-5 haloalkylthio, formyl, cyano, bromo, or iodo; Z is hydrogen, hydroxy, nitro cyano, rhodano, formyl, G-, G-S—, G-S—S—, G-A-, R7R8N—, R7R8N—S—, R7R8N-A-, G-O-A-, G-S-A-, (R10O)(R11O)P(X)—, (R10O)(R11S)P(X)—, (R10O)(R11)P(X)—, (R10S)(R11S)P(X)—, (R10O)(R14R15N)P(X)—, (R11)(R14R15N)P(X)—, (R14R15N)(R16R17N)P(X)—, G-N═CH—, G-O—N═CH—, N≡C—N═CH—, or Z is a group of formula (II), wherein B is S—, S—S—, S(O)—, C(O)—, or (CH2)n—; n is an integer from 1 to 6; and R1, R2, and R3 are as defined above; and G is optionally substituted C1-10alkyl, optionally substituted C2-10 alkenyl, optionally substituted C2-10 alkynyl, optionally substituted C3-7 cycloalkyl, optionally substituted C3-7 cycloalkenyl, optionally substituted aryl, optionally substituted heteroaryl or optionally substituted heterocyclyl; A is S(O), SO2, C(O) or C(S).
摘要翻译: 本发明涉及新的咪唑啉衍生物及其作为杀虫,杀螨,杀软体动物和杀线虫剂的用途。 本发明还延伸到包含这种咪唑啉衍生物的杀虫,杀螨,杀软体动物和杀线虫组合物,以及使用这些衍生物和/或组合物来对抗和控制昆虫,螨虫,软体动物和线虫的害虫的方法。 式(I)化合物及其盐和N-氧化物,其中:R1为C1-10烷基; R2是氯,溴或碘; R3是C2-5烷基,C1-5卤代烷基,C1-6羟基烷基,C1-5烷氧基 - (C1-3) - 烷基,二 - (C1-5烷氧基) - (C1-3) - 烷基,C1-5烷硫基 - (C 1-3) - 烷基; C 1-5烷基亚磺酰基 - (C 1-3)烷基; C2-5烯基,C1-5卤代烯基,C2-5炔基,C3-6环烷基,C3-6环烯基,羟基,C1-5烷氧基,C1-5卤代烷氧基,C1-5烷硫基,C1-5卤代烷硫基,甲酰基,氰基,溴 ,或碘; Z是氢,羟基,硝基氰基,罗丹明,甲酰基,G-,GS-,GSS-,GA-,R7R8N-,R7R8N-S-,R7R8N-A-,GOA-,GSA-,(R10O) P(X) - ,(R10O)(R11S)P(X) - ,(R10O)(R11)P(X) - ,(R10S)(R11S)P(X) - ,(R10O)(R14R15N) X) - ,(R11)(R14R15N)P(X) - ,(R14R15N)(R16R17N)P(X) - ,GN = CH-,GON = CH-,N = CN = CH-,或Z为基团 其中B为S-,SS-,S(O) - ,C(O) - 或(CH 2)n - )的式(II) n是1至6的整数; 并且R 1,R 2和R 3如上所定义; 任选取代的C 2-10炔基,任选取代的C 3-7环烷基,任选取代的C 3-7环烯基,任选取代的芳基,任选取代的杂芳基或任选取代的杂环基; A是S(O),SO 2,C(O)或C(S)。
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5.
公开(公告)号:US20100120882A1
公开(公告)日:2010-05-13
申请号:US12527213
申请日:2008-01-28
IPC分类号: A01N43/50 , C07D233/22
CPC分类号: C07D233/22 , C07C255/16
摘要: The present invention relates to imidazoline derivatives and their use as insecticidal, acaricidal, molluscicidal and nematocidal agents. The invention also extends to insecticidal, acaricidal, molluscicidal and nematicidal compositions comprising such imidazoline derivatives, and to methods of using such derivatives and/or compositions to combat and control insect, acarine, mollusc and nematode pests. In particular the present invention relates to imidazolines with alkyl and fluoro substituents.
摘要翻译: 本发明涉及咪唑啉衍生物及其作为杀虫,杀螨,杀软体动物和杀线虫剂的用途。 本发明还延伸到包含这种咪唑啉衍生物的杀虫,杀螨,杀软体动物和杀线虫组合物,以及使用这些衍生物和/或组合物来对抗和控制昆虫,螨虫,软体动物和线虫的害虫的方法。 特别地,本发明涉及具有烷基和氟取代基的咪唑啉。
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公开(公告)号:US08309739B2
公开(公告)日:2012-11-13
申请号:US13105596
申请日:2011-05-11
申请人: Anthony Cornelius O'Sullivan , Juergen Harry Schaetzer , Christoph Luethy , Allison Clare Elliott , Christopher John Mathews
发明人: Anthony Cornelius O'Sullivan , Juergen Harry Schaetzer , Christoph Luethy , Allison Clare Elliott , Christopher John Mathews
IPC分类号: C07D277/18
CPC分类号: A01N43/78 , C07D277/18 , C07D417/12
摘要: The use of a compound of formula I wherein X is (i), (ii) or (iii) Y is O, S(O)m, NR3, CR5R6, CR5R6—CR7R8, O—CR7R8, S(O)m—CR7R8, NR3—CR7R8, CR5R6—O, CR5R6—S(O)m, CR5R6—NR3, SO2—NR3, NR3—SO2, NR3—O or O—NR3; m is 0, 1, or 2; the ring (T) is a 5- or 6-membered aromatic or heteroaromatic ring; R1 to R10 are specified organic groups and n and is 0, 1, 2, 3 or 4; or salts or N-oxides thereof or compositions containing them in controlling insects, acarines, nematodes or molluscs. Novel compounds are also provided.
摘要翻译: 其中X是(i),(ii)或(iii)Y的式I化合物是O,S(O)m,NR 3,CR 5 R 6,CR 5 R 6 -CR 7 R 8,O-CR 7 R 8,S(O) CR7R8,NR3-CR7R8,CR5R6-O,CR5R6-S(O)m,CR5R6-NR3,SO2-NR3,NR3-SO2,NR3-O或O-NR3; m为0,1或2; 环(T)是5或6元芳族或杂芳族环; R1至R10为指定的有机基团,n为0,1,2,3或4; 或其盐或N-氧化物或含有它们的组合物来控制昆虫,螨类,线虫或软体动物。 还提供了新的化合物。
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7.
公开(公告)号:US08497293B2
公开(公告)日:2013-07-30
申请号:US12741896
申请日:2008-10-24
IPC分类号: A01N43/50 , A01N33/18 , C07D233/14 , C07C43/188 , A01P3/00 , A01P5/00 , A01P7/00 , A01P7/04
CPC分类号: C07D233/22 , A01N43/50 , C07D401/12
摘要: The present invention relates to novel imidazoline derivatives and their use as insecticidal, acaricidal, molluscicidal and nematocidal agents. The invention also extends to insecticidal, acaricidal, molluscicidal and nematicidal compositions comprising such imidazoline derivatives, and to methods of using such derivatives and/or compositions to combat and control insect, acarine, mollusc and nematode pests. A compound of formula (I): and the salts and N-oxides thereof.
摘要翻译: 本发明涉及新的咪唑啉衍生物及其作为杀虫,杀螨,杀软体动物和杀线虫剂的用途。 本发明还延伸到包含这种咪唑啉衍生物的杀虫,杀螨,杀软体动物和杀线虫组合物,以及使用这些衍生物和/或组合物来对抗和控制昆虫,螨虫,软体动物和线虫的害虫的方法。 式(I)的化合物及其盐和N-氧化物。
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公开(公告)号:US08106075B2
公开(公告)日:2012-01-31
申请号:US11576950
申请日:2005-10-10
申请人: Anthony Cornelius O'Sullivan , David John Hughes , André Jeanguenat , Michel Muehlebach , Olivier Loiseleur
发明人: Anthony Cornelius O'Sullivan , David John Hughes , André Jeanguenat , Michel Muehlebach , Olivier Loiseleur
IPC分类号: A61K31/336 , A61K31/4156 , A61K31/4427 , A61K31/4439
CPC分类号: C07D405/14 , A01N43/56 , C07D401/04 , C07D409/14
摘要: Compounds of formula I wherein the substituents are as defined in claim 1, and the agrochemically acceptable salts and all stereoisomers and tautomeric forms of the compounds of formula I can be used as agrochemical active ingredients and can be prepared in a manner known per se.
摘要翻译: 其中取代基如权利要求1所定义的式I化合物,以及式I化合物的农业化学上可接受的盐和所有立体异构体和互变异构形式可以用作农业化学活性成分,并且可以以本身已知的方式制备。
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9.
公开(公告)号:US07732416B2
公开(公告)日:2010-06-08
申请号:US11319686
申请日:2005-12-28
摘要: What is described are a compound of the formula in which R1 is C1-C12alkyl, C3-C8cycloalkyl or C2-C12alkenyl; R2 is H, unsubstituted or mono- to pentasubstituted C1-C12alkyl or unsubstituted or mono- to pentasubstituted C1-C12alkenyl; R3 is C2-C12alkyl, mono- to pentasubstituted C1-C12alkyl, unsubstituted or mono- to pentasubstituted C1-C6alkoxy-C1-C6alkyl, unsubstituted or mono- to pentasubstituted C3-C12cycloalkyl, C2-C12alkenyl, C2-C12alkynyl; or R2 and R3 together are an alkylene or alkenylene bridge; with the proviso that R1 is not sec-butyl or isopropyl if R2 is H and R3 is 2-hydroxyethyl, isopropyl, n-octyl or benzyl; or, if appropriate, in E/Z isomer, an E/Z isomer mixture and/or a tautomer thereof; a process for preparing and using these compounds and their tautomers; pesticides whose active compound is selected from these compounds and their tautomers; and a process for preparing these compounds and compositions, and the use of these compounds and compositions.
摘要翻译: 描述的是下式的化合物,其中R 1是C 1 -C 12烷基,C 3 -C 8环烷基或C 2 -C 12链烯基; R 2为H,未取代或单价至五价取代的C 1 -C 12烷基或未取代或单价至五价取代的C 1 -C 12烯基; R 3是C 2 -C 12烷基,未被取代的或被一或五取代的C 1 -C 6烷氧基-C 1 -C 6烷基,未取代的或一至五取代的C 3 -C 12环烷基,C 2 -C 12链烯基,C 2 -C 12炔基; 或者R 2和R 3一起是亚烷基或亚烯基桥; 条件是R1不是仲丁基或异丙基,如果R2是H,R3是2-羟乙基,异丙基,正辛基或苄基; 或者如果合适的话,在E / Z异构体中,E / Z异构体混合物和/或其互变异构体; 一种制备和使用这些化合物及其互变异构体的方法; 活性化合物选自这些化合物及其互变异构体的农药; 以及制备这些化合物和组合物的方法,以及这些化合物和组合物的用途。
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公开(公告)号:US07161011B2
公开(公告)日:2007-01-09
申请号:US10400826
申请日:2003-03-27
申请人: Thomas Pitterna , Henry Szczepanski , Peter Maienfisch , Ottmar Franz Hüter , Thomas Rapold , Marcel Senn , Thomas Göbel , Anthony Cornelius O'Sullivan
发明人: Thomas Pitterna , Henry Szczepanski , Peter Maienfisch , Ottmar Franz Hüter , Thomas Rapold , Marcel Senn , Thomas Göbel , Anthony Cornelius O'Sullivan
IPC分类号: C07D277/36
CPC分类号: C07D277/32 , C07D277/16 , C07D277/36 , C07D277/70 , C07D277/74
摘要: Described is a process for the preparation of a compound of the formula wherein R is unsubstituted or substituted C1–C12alkyl, C2–C4alkenyl, C2–C4alkynyl, C3–C6cycloalkyl, aryl or heteroaryl, or —SR1; R1 is unsubstituted or substituted C1–C12alkyl, C2–C4alkenyl, C2–C4alkenyl, C2–C4alkynyl, cycloalkyl, aryl or heteroaryl; and X is a leaving group; which comprises a) reacting a compound of the formula wherein R is as defined for formula (I), with a water removing reagent.
摘要翻译: 描述了制备下式化合物的方法,其中R是未取代的或取代的C 1 -C 12烷基,C 2 - C 4链烯基,C 2 -C 4炔基,C 3 -C 6亚烷基,C 3 -C 4炔基,C 3 -C 4炔基,C 3 -C 6亚烷基, >环烷基,芳基或杂芳基,或-SR 1 N; R 1是未取代的或取代的C 1 -C 12烷基,C 2 -C 4烷基, /亚烷基,C 2 -C 4链烯基,C 2 -C 4 - 炔基,环烷基,芳基 或杂芳基; X为离去群; 其包括a)使式(I)化合物与式(I)所定义的化合物与除水试剂反应。
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