公开(公告)号：US20190225586A1

公开(公告)日：2019-07-25

申请号：US16335138

申请日：2017-09-18

Applicant: BAYER CROPSCIENCE AKTIENGESELLSCHAFT ,  CENTRE NATIONAL DE LA RECHERCHE SCIENTIFIQUE (CNRS)

Inventor： Sergii PAZENOK ,  Jean-Pierre VORS ,  Frédéric R. LEROUX ,  Etienne SCHMITT

IPC: C07D231/14 ,  C07C251/08

Abstract: The present invention relates to a novel process for preparing 3-fluoroalkyl-5-pyrazolecarboxylates from ketimines and oxalic acid derivatives which can be further transformed into 3-fluoroalkyl-5-pyrazolecarboxylic acids.

公开(公告)号：US20190029255A1

公开(公告)日：2019-01-31

申请号：US16054744

申请日：2018-08-03

Applicant: Bayer CropScience Aktiengesellschaft

Inventor： Pierre CRISTAU ,  Philippe DESBORDES ,  Julie GEIST ,  Lionel NICOLAS ,  Philippe RINOLFI ,  Jan-Peter SCHMIDT ,  Tomoki TSUCHIYA ,  Jean-Pierre VORS ,  Ulrike WACHENDORFF-NEUMANN

IPC: A01N43/56 ,  C07C47/575 ,  C07C47/55 ,  C07D231/16 ,  C07C25/18 ,  C07C47/546

Abstract: The present invention relates to fungicidal N-cycloalkyl-N-{[2-(1-substituted cycloalkyl)phenyl]methylene} carboxamide derivatives and their thiocarbonyl derivatives, their process of preparation and intermediate compounds for their preparation, their use as fungicides, particularly in the form of fungicidal compositions and methods for the control of phytopathogenic fungi of plants using these compounds or their compositions.

公开(公告)号：US20170150717A1

公开(公告)日：2017-06-01

申请号：US15320780

申请日：2015-06-22

Applicant: BAYER CROPSCIENCE AKTIENGESELLSCHAFT

Inventor： Christophe DUBOST ,  Philipp WINTER ,  Marco BRÜNJES ,  Mark James FORD ,  Ulrike WACHENDORFF-NEUMANN ,  Cyril MONTAGNE ,  Jean-Pierre VORS ,  Stephane BRUNET ,  Philippe RINOLFI

IPC: A01N43/40 ,  C07D213/82

CPC classification number: A01N43/40 ,  C07D213/82

Abstract: The present invention relates to novel difluoromethyl-nicotinic indanyl carboxamides, to processes for preparing these compounds, to compositions comprising these compounds, and to the use thereof as biologically active compounds, especially for control of harmful microorganisms in crop protection and in the protection of materials.

公开(公告)号：US20160108000A1

公开(公告)日：2016-04-21

申请号：US14892291

申请日：2014-05-19

Applicant: BAYER CROPSCIENCE AKTIENGESELLSCHAFT

Inventor： Sergii PAZENOK ,  Norbert LUI ,  Arnd NEEFF ,  Winfried ETZEL ,  Jean-Pierre VORS ,  Frederic R. LEROUX ,  Gregory LANDELLE ,  Mark James FORD

IPC: C07D231/12 ,  A01N43/56

CPC classification number: C07D231/12 ,  A01N43/56 ,  C07D231/14

Abstract: The present invention relates to a novel process for preparing 3,5-bis(fluoroalkyl)pyrazole derivatives from α,α-dihaloamines.

Abstract translation: 本发明涉及从α，α-二卤代胺制备3,5-双（氟代烷基）吡唑衍生物的新方法。

公开(公告)号：US20190082691A1

公开(公告)日：2019-03-21

申请号：US16190285

申请日：2018-11-14

Applicant: Bayer CropScience Aktiengesellschaft

Inventor： Sebastian HOFFMANN ,  Hendrik HELMKE ,  Peter DAHMEN ,  Ulrike WACHENDORFF-NEUMANN ,  David BERNIER ,  Ricarda MILLER ,  Pierre-Yves COQUERON ,  Pierre GENIX ,  Sven WITTROCK ,  Jean-Pierre VORS ,  Philippe KENNEL ,  Stephane BRUNET ,  Sebastien NAUD ,  Ruth MEISSNER

IPC: A01N43/50 ,  C07D233/58 ,  C07D233/60 ,  C07D233/68 ,  C07D233/61 ,  C07D233/84 ,  C07D233/92 ,  C07D401/06 ,  C07D233/74

Abstract: The present invention relates to novel 5-substituted imidazolylmethyl derivatives, to processes for preparing these compounds, to compositions comprising these compounds, and to the use thereof as biologically active compounds, especially for control of harmful microorganisms in crop protection and in the protection of materials and as plant growth regulators.

公开(公告)号：US20160340370A1

公开(公告)日：2016-11-24

申请号：US15114385

申请日：2015-01-23

Applicant: BAYER CROPSCIENCE AKTIENGESELLSCHAFT

Inventor： Mark James FORD ,  Jean-Pierre VORS ,  Olivier BAUDOIN ,  Simon JANODY

IPC: C07F7/08

CPC classification number: C07F7/081 ,  C07B2200/07 ,  C07C67/297 ,  C07C209/58 ,  C07C2602/08 ,  C07D209/48 ,  C07F7/1804 ,  C07F7/1872 ,  C07C211/42 ,  C07C69/24 ,  C07C69/63

Abstract: A description is given of a process for preparing 1-indanols and 1-indanamines by palladium-catalyzed arylation and of the use thereof as intermediates for the synthesis of fine chemicals and of active agrochemical ingredients.

Abstract translation: 给出了通过钯催化的芳基化制备1-茚满醇和1-茚满胺的方法及其作为合成精细化学品和活性农药成分的中间体的用途的描述。

公开(公告)号：US20160316752A1

公开(公告)日：2016-11-03

申请号：US15100966

申请日：2014-12-04

Applicant: BAYER CROPSCIENCE AKTIENGESELLSCHAFT

Inventor： Pierre CRISTAU ,  Philippe DESBORDES ,  Julie GEIST ,  Lionel NICOLAS ,  Philippe RINOLFI ,  Jan-Peter SCHMIDT ,  Tomoki TSUCHIYA ,  Jean-Pierre VORS ,  Ulrike WACHENDORFF-NEUMANN

IPC: A01N43/56 ,  C07C47/575 ,  C07D231/16 ,  C07C47/546 ,  C07C47/55 ,  C07C25/18

CPC classification number: A01N43/56 ,  C07C25/18 ,  C07C47/546 ,  C07C47/55 ,  C07C47/575 ,  C07C2601/02 ,  C07D231/16

Abstract: The present invention relates to fungicidal N-cycloalkyl-N-{[2-(1-substitutedcycloalkyl)phenyl]methylene} carboxamide derivatives and their thiocarbonyl derivatives, their process of preparation and intermediate compounds for their preparation, their use as fungicides, particularly in the form of fungicidal compositions and methods for the control of phytopathogenic fungi of plants using these compounds or their compositions

Abstract translation: 本发明涉及杀真菌N-环烷基-N - {[2-（1-取代环烷基）苯基]亚甲基}甲酰胺衍生物及其硫代羰基衍生物，其制备方法及其制备中间体化合物，它们用作杀真菌剂，特别是在 使用这些化合物或其组合物的杀真菌组合物和控制植物病原性真菌的方法

公开(公告)号：US20160264529A1

公开(公告)日：2016-09-15

申请号：US15031456

申请日：2014-10-28

Applicant: BAYER CROPSCIENCE AKTIENGESELLSCHAFT

Inventor： Christophe DUBOST ,  Ulrike WACHENDORFF-NEUMANN ,  Philipp WINTER ,  Stephane BRUNET ,  Jean-Pierre VORS ,  Cyril MONTAGNE

IPC: C07D231/16 ,  A01N43/56 ,  C07D213/82 ,  C07C25/22 ,  C07C209/62 ,  C07C17/23 ,  C07C17/275 ,  C07D231/14 ,  A01N43/40

CPC classification number: C07D231/16 ,  A01N43/40 ,  A01N43/56 ,  A01N45/00 ,  C07C17/23 ,  C07C17/275 ,  C07C25/22 ,  C07C209/62 ,  C07C211/60 ,  C07C211/61 ,  C07C2602/06 ,  C07C2603/94 ,  C07D213/82 ,  C07D231/14

Abstract: The present invention relates to novel benzocyclobutane(thio) carboxamides, to processes for preparing these compounds, to compositions comprising these compounds, and to the use thereof as biologically active compounds, especially for control of harmful microorganisms in crop protection and in the protection of materials.

Abstract translation: 本发明涉及新型苯并环丁烷（硫代）甲酰胺，制备这些化合物的方法，包含这些化合物的组合物，以及其作为生物活性化合物的用途，特别是用于控制作物保护和材料保护中的有害微生物 。

公开(公告)号：US20160031851A1

公开(公告)日：2016-02-04

申请号：US14783207

申请日：2014-04-09

Applicant: BAYER CROPSCIENCE AKTIENGESELLSCHAFT

Inventor： Sebastian HOFFMANN ,  Alexander SUDAU ,  Peter DAHMEN ,  Ulrike WACHENDORFF-NEUMANN ,  David BERNIER ,  Helene LACHAISE ,  Stephane BRUNET ,  Jacky VIDAL ,  Pierre GENIX ,  Pierre-Yves COQUERON ,  Julie GEIST ,  Jean-Pierre VORS ,  Philippe KENNEL ,  Ricarda MILLER

IPC: C07D401/06 ,  C07D405/14 ,  C07D401/14 ,  A01N43/653 ,  C07D403/06

CPC classification number: C07D401/06 ,  A01N43/653 ,  C07D213/42 ,  C07D401/14 ,  C07D403/06 ,  C07D405/14

Abstract: The present invention relates to novel triazolinthione derivatives, to processes for preparing these compounds, to compositions comprising these compounds, and to the use thereof as biologically active compounds, especially for control of harmful microorganisms in crop protection and in the protection of materials and as plant growth regulators.

Abstract translation: 本发明涉及新的三唑啉酮衍生物，制备这些化合物的方法，包含这些化合物的组合物及其作为生物活性化合物的用途，特别是用于控制作物保护中的有害微生物和作为植​​物的保护 生长调节剂

公开(公告)号：US20190023659A1

公开(公告)日：2019-01-24

申请号：US16070561

申请日：2017-01-13

Applicant: Bayer CropScience Aktiengesellschaft ,  CENTRE NATIONAL DE LA RECHERCHE SCIENTIFIQUE

Inventor： Sergii PAZENOK ,  Jean-Pierre VORS ,  Frédéric R LEROUX ,  Fallia ARIBI ,  Etienne SCHMITT ,  Armen PANOSSIAN

IPC: C07D215/18

Abstract: The invention relates to a novel process for preparing polyfluoroalkylated quinolines from ketimines in the presence of fluoroalkylamino reagents.