公开(公告)号：US20160316752A1

公开(公告)日：2016-11-03

申请号：US15100966

申请日：2014-12-04

Applicant: BAYER CROPSCIENCE AKTIENGESELLSCHAFT

Inventor： Pierre CRISTAU ,  Philippe DESBORDES ,  Julie GEIST ,  Lionel NICOLAS ,  Philippe RINOLFI ,  Jan-Peter SCHMIDT ,  Tomoki TSUCHIYA ,  Jean-Pierre VORS ,  Ulrike WACHENDORFF-NEUMANN

IPC: A01N43/56 ,  C07C47/575 ,  C07D231/16 ,  C07C47/546 ,  C07C47/55 ,  C07C25/18

CPC classification number: A01N43/56 ,  C07C25/18 ,  C07C47/546 ,  C07C47/55 ,  C07C47/575 ,  C07C2601/02 ,  C07D231/16

Abstract: The present invention relates to fungicidal N-cycloalkyl-N-{[2-(1-substitutedcycloalkyl)phenyl]methylene} carboxamide derivatives and their thiocarbonyl derivatives, their process of preparation and intermediate compounds for their preparation, their use as fungicides, particularly in the form of fungicidal compositions and methods for the control of phytopathogenic fungi of plants using these compounds or their compositions

Abstract translation: 本发明涉及杀真菌N-环烷基-N - {[2-（1-取代环烷基）苯基]亚甲基}甲酰胺衍生物及其硫代羰基衍生物，其制备方法及其制备中间体化合物，它们用作杀真菌剂，特别是在 使用这些化合物或其组合物的杀真菌组合物和控制植物病原性真菌的方法

公开(公告)号：US20160244433A1

公开(公告)日：2016-08-25

申请号：US15028004

申请日：2014-10-07

Applicant: BAYER CROPSCIENCE AKTIENGESELLSCHAFT

Inventor： Philippe DESBORDES ,  Philippe RINOLFI ,  Tomoki TSUCHIYA

IPC: C07D403/06 ,  A01N61/00 ,  C07D405/14 ,  A01N43/56 ,  C07D401/06 ,  A01N43/36 ,  C07D405/06 ,  C07D417/06 ,  A01N43/78 ,  A01N43/647 ,  C07D409/06

CPC classification number: C07D403/06 ,  A01N43/36 ,  A01N43/56 ,  A01N43/647 ,  A01N43/78 ,  A01N61/00 ,  C07D207/06 ,  C07D211/12 ,  C07D401/06 ,  C07D405/04 ,  C07D405/06 ,  C07D405/14 ,  C07D409/06 ,  C07D417/06

Abstract: The present invention relates to fungicidal N-hetarylcarbonyl-2-(benzocycloalken-1-yl)piperidines or pyrrolidines of formula (I), and their thiocarbonyl derivatives, wherein A represents a carbo-linked, unsaturated or partially saturated, 5-membered heterocyclyl group that can be substituted by up to four groups R that can be the same or different; T represents 0 or S; n represents 1 or 2; m represents 1, 2 or 3; p represents 1, 2, 3 or 4, L1 and L2 independently represent CZ4Z5, NZ6, 0, S, S(O) or S(0)2; and R and Z1-Z6 are as defined in the claims; their process of preparation and intermediate compounds for their preparation, their use as fungicides, particularly in the form of fungicidal compositions and methods for the control of phytopathogenic fungi of plants using these compounds or their compositions.

Abstract translation: 本发明涉及式（I）的杀真菌N-叔丁基羰基-2-（苯并环烯烃-1-基）哌啶或吡咯烷及其硫代羰基衍生物，其中A表示碳连接的不饱和或部分饱和的5元杂环基 可以被最多四个可以相同或不同的R基团取代的基团; T表示0或S; n表示1或2; m表示1,2或3; p表示1,2,3或4，L1和L2独立地表示CZ4Z5，NZ6,0，S，S（O）或S（0）2; 并且R和Z1-Z6如权利要求中所定义; 它们的制备方法和用于其制备的中间体化合物，它们用作杀真菌剂，特别是以杀真菌剂的形式和用于使用这些化合物或其组合物控制植物病原性真菌的方法。

公开(公告)号：US20200323211A1

公开(公告)日：2020-10-15

申请号：US16913862

申请日：2020-06-26

Applicant: Bayer CropScience Aktiengesellschaft

Inventor： Philippe DESBORDES ,  Christophe DUBOST ,  Jeremy DUFOUR ,  Mathieu GOURGUES ,  Philipp HOLSTEIN ,  Virginie LEMPEREUR ,  Frederic MIEGE ,  Philippe RINOLFI ,  Vincent RODESCHINI ,  Valerie TOQUIN ,  Francois VILLALBA ,  Ulrike WACHENDORFF-NEUMANN

IPC: A01N43/84 ,  A01N43/72 ,  C07D281/06 ,  C07D417/10

Abstract: The present disclosure relates to fungicidal active compounds, more specifically to benzosultams and analogues thereof, processes and, intermediates for their preparation and use thereof as fungicidal active compound, particularly in the form of fungicide compositions. The present disclosure also relates to methods for the control of phytopathogenic fungi of plants using these compounds or compositions comprising thereof.

公开(公告)号：US20190233444A1

公开(公告)日：2019-08-01

申请号：US15771846

申请日：2016-10-28

Applicant: Bayer CropScience Aktiengesellschaft

Inventor： Jérémy DUFOUR ,  Philippe DESBORDES ,  Christophe DUBOST ,  Mathieu GOURGUES ,  Ruth MEISSNER ,  Andrew PETTINGER ,  Philippe RINOLFI ,  Valérie TOQUIN ,  Ulrike WACHENDORFF-NEUMANN

IPC: C07F7/08 ,  C07F7/18 ,  C07D241/18 ,  C07D413/12 ,  A61P31/00

Abstract: The present disclosure relates to fungicidal active compounds, more specifically to trisubstitutedsilylphenoxyhetero-cycles and analogues thereof, processes and, intermediates for their preparation and use thereof as fungicidal active compound, particularly in the form of fungicide compositions. The present disclosure also relates to methods for the control of phytopathogenic fungi of plants using these compounds or compositions comprising thereof.

公开(公告)号：US20180139962A1

公开(公告)日：2018-05-24

申请号：US15575064

申请日：2016-05-19

Applicant: Bayer CropScience Aktiengesellschaft

Inventor： Pierre CRISTAU ,  Philippe DESBORDES ,  Julie GEIST ,  Lionel NICOLAS ,  Philippe RINOLFI ,  Jan Peter SCHMIDT ,  Tomoki TSUCHIYA

IPC: A01N43/56 ,  C07D333/12 ,  C07D333/16 ,  C07D333/20 ,  C07D333/22 ,  C07D333/24 ,  C07D401/12 ,  C07D409/12 ,  C07D409/14

CPC classification number: A01N43/56 ,  C07D333/12 ,  C07D333/16 ,  C07D333/20 ,  C07D333/22 ,  C07D333/24 ,  C07D401/12 ,  C07D409/12 ,  C07D409/14

Abstract: The invention relates to fungicidal N-cycloalkyl-N-{[ortho-(1-substituted-cycloalkyl)heteroaryl]methyl}carboxamides and their thiocarbonyl derivatives of formula (I), their process of preparation and intermediate compounds for their preparation, their use as fungicides, particularly in the form of fungicidal compositions, and methods for the control of phytopathogenic fungi of plants using these compounds or their compositions.

公开(公告)号：US20160326120A1

公开(公告)日：2016-11-10

申请号：US15101380

申请日：2014-12-04

Applicant: BAYER CROPSCIENCE AKTIENGESELLSCHAFT

Inventor： Pierre CRISTAU ,  Philippe DESBORDES ,  Julie GEIST ,  Lionel NICOLAS ,  Philippe RINOLFI ,  Jan-Peter SCHMIDT ,  Tomoki TSUCHIYA ,  Jean-Pierre VORS ,  Ulrike WACHENDORFF-NEUMANN

IPC: C07D231/12 ,  C07D249/06 ,  C07D307/38 ,  C07D263/32 ,  C07C211/27 ,  C07C217/48 ,  C07F7/08 ,  C07C255/46 ,  C07C47/54 ,  C07C47/55 ,  C07C47/575 ,  C07C22/04 ,  A01N43/56 ,  A01N43/647 ,  A01N43/10 ,  A01N43/76 ,  A01N33/04 ,  A01N55/00 ,  A01N37/34 ,  A01N35/04 ,  C07D307/54

CPC classification number: C07D231/12 ,  A01N33/04 ,  A01N35/04 ,  A01N37/34 ,  A01N43/10 ,  A01N43/56 ,  A01N43/647 ,  A01N43/76 ,  A01N55/00 ,  C07C22/04 ,  C07C47/54 ,  C07C47/55 ,  C07C47/575 ,  C07C211/27 ,  C07C217/48 ,  C07C255/46 ,  C07C2601/02 ,  C07D231/14 ,  C07D231/16 ,  C07D233/28 ,  C07D249/06 ,  C07D263/32 ,  C07D307/38 ,  C07D307/54 ,  C07F7/0803

Abstract: The present invention relates to fungicidal N-cycloalkyl-N-{[2-(1-substitutedcycloalkyl)phenyl]methylene} carboxamide derivatives and their thiocarbonyl derivatives, their process of preparation and intermediate compounds for their preparation, their use as fungicides, particularly in the form of fungicidal compositions and methods for the control of phytopathogenic fungi of plants using these compounds or their compositions.

Abstract translation: 本发明涉及杀真菌N-环烷基-N - {[2-（1-取代环烷基）苯基]亚甲基]甲酰胺衍生物及其硫代羰基衍生物，其制备方法及其制备中间体化合物，它们用作杀真菌剂，特别是在 使用这些化合物或其组合物的杀真菌组合物和控制植物病原性真菌的方法。

公开(公告)号：US20180146670A1

公开(公告)日：2018-05-31

申请号：US15575292

申请日：2016-05-19

Applicant: Bayer CropScience Aktiengesellschaft

Inventor： Pierre CRISTAU ,  Philippe DESBORDES ,  Julie GEIST ,  Lionel NICOLAS ,  Philippe RINOLFI ,  Jan Peter SCHMIDT ,  Tomoki TSUCHIYA

IPC: A01N43/56 ,  C07D409/12 ,  C07D401/12

CPC classification number: A01N43/56 ,  C07D401/12 ,  C07D409/12

Abstract: The invention relates to fungicidal N-cycloalkyl-N-{[ortho-(1-substituted-cycloalkyl)heteroaryl]methyl}carboxamides and their thiocarbonyl analogs of formula (I), their process of preparation, their use as fungicides, particularly in the form of fungicidal compositions, and methods for the control of phytopathogenic fungi of plants using these compounds or their compositions. A represents a carbo-linked, unsaturated or partially saturated, optionally substituted 5-membered heterocyclyl group; T represents O or S; Z1 represents an optionally substituted C3-C7-cycloalkyl; p represents 1-5; B1 represents a carbo-linked, unsaturated, monocyclic or fused bicyclic 5-, 6-, 8-, 9-, 10-membered heterocyclyl ring, wherein the dotted line between the two adjacent carbons represents a single bond, a double bond or an aromatic bond.

公开(公告)号：US20160255836A1

公开(公告)日：2016-09-08

申请号：US15029220

申请日：2014-10-15

Applicant: BAYER CROPSCIENCE AKTIENGESELLSCHAFT

Inventor： Philippe DESBORDES ,  Philippe RINOLFI ,  Tomoki TSUCHIYA ,  Julie GEIST ,  Lionel NICOLAS

IPC: A01N43/56 ,  C07D403/14 ,  C07D405/14 ,  C07D417/14 ,  A01N43/54 ,  A01N43/647 ,  A01N43/10 ,  A01N43/36 ,  C07D401/14 ,  C07D409/14 ,  A01N43/78

CPC classification number: A01N43/56 ,  A01N43/10 ,  A01N43/36 ,  A01N43/54 ,  A01N43/647 ,  A01N43/78 ,  C07D333/18 ,  C07D333/38 ,  C07D401/14 ,  C07D403/14 ,  C07D405/14 ,  C07D409/14 ,  C07D417/14

Abstract: The present invention relates to fungicidal N-cycloalkyl-N-(biheterocyclylmethylene)carboxamide derivatives and their thiocarbonyl derivatives, their process of preparation and intermediate compounds for their preparation, their use as fungicides, particularly in the form of fungicidal compositions and methods for the control of phytopathogenic fungi of plants using these compounds or their compositions.

Abstract translation: 本发明涉及杀真菌N-环烷基-N-（双杂环亚甲基）甲酰胺衍生物及其硫代羰基衍生物，其制备方法及其制备中间体化合物，其用作杀真菌剂，特别是杀真菌组合物和控制方法 使用这些化合物或其组合物的植物致病真菌。

公开(公告)号：US20200178532A1

公开(公告)日：2020-06-11

申请号：US16627983

申请日：2018-06-28

Applicant: Bayer CropScience Aktiengesellschaft

Inventor： Jullien REY ,  Joerg TIEBES ,  Marc MOSRIN ,  Thomas DROEGE ,  Hansjoerg DIETRICH ,  Anu Bheemaiah MACHETTIRA ,  Elmar GATZWEILER ,  Christopher Hugh ROSINGER ,  Dirk SCHMUTZLER ,  Daniela PORTZ ,  Kerstin ILG ,  Philippe RINOLFI

IPC: A01N43/90 ,  C07D513/04

Abstract: The invention relates to the technical field of the herbicides and/or plant growth regulators. Specifically, the invention primarily relates to novel substituted isothiazolopyridones, and compositions comprising said novel substituted isothiazolopyridones. Further, the present invention relates to processes for the preparation said novel substituted isothiazolopyridones and their use as herbicides and/or plant growth regulators.

公开(公告)号：US20190335753A1

公开(公告)日：2019-11-07

申请号：US16314641

申请日：2017-07-03

Applicant: Bayer CropScience Aktiengesellschaft

Inventor： Philippe DESBORDES ,  Christophe DUBOST ,  Jeremy DUFOUR ,  Mathieu GOURGUES ,  Phillip HOLSTEIN ,  Virginie LEMPEREUR ,  Frederic MIEGE ,  Philippe RINOLFI ,  Vincent RODESCHINI ,  Valerie TOQUIN ,  Francois VILLALBA ,  Ulrike WACHENDORFF-NEUMANN

IPC: A01N43/84 ,  C07D417/10 ,  C07D281/06 ,  A01N43/72

Abstract: The present disclosure relates to fungicidal active compounds, more specifically to benzosultams and analogues thereof, processes and, intermediates for their preparation and use thereof as fungicidal active compound, particularly in the form of fungicide compositions. The present disclosure also relates to methods for the control of phytopathogenic fungi of plants using these compounds or compositions comprising thereof.